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—— (7R)-2-[(2-chlorophenyl)methylsulfanyl]-7-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H20ClN5O2S
(7R)-2-[(2-chlorophenyl)methylsulfanyl]-7-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-methoxy-4-phenylmethoxyphenyl)-5-methyl-N-pyridin-3-yl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H23N7O3
(7R)-7-(3-methoxy-4-phenylmethoxyphenyl)-5-methyl-N-pyridin-3-yl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-cyanophenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H24N6OS
(7S)-2-benzylsulfanyl-7-(4-cyanophenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-7-(4-phenylmethoxyphenyl)-N-pyridin-3-yl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H21N7O2
(7R)-5-methyl-7-(4-phenylmethoxyphenyl)-N-pyridin-3-yl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H25N7O4
(7R)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-methoxyphenyl)-5-methyl-7-[2-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N6O3
(7R)-N-(2-methoxyphenyl)-5-methyl-7-[2-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H24N6O2
(7S)-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2,4-dimethoxyphenyl)-5-(3,4-dimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C21H22N4O4
(7S)-7-(2,4-dimethoxyphenyl)-5-(3,4-dimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7S)-5-methyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C15H18N6O2
(7S)-5-methyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromo-2-butoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25BrN6O2
(7S)-7-(5-bromo-2-butoxyphenyl)-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-7-[2-[(2-methylphenyl)methoxy]phenyl]-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H24N6O2
(7R)-5-methyl-7-[2-[(2-methylphenyl)methoxy]phenyl]-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-N-(2-methylphenyl)-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N6O2
(7S)-5-methyl-N-(2-methylphenyl)-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromo-2-butoxyphenyl)-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23BrN6O2
(7S)-7-(5-bromo-2-butoxyphenyl)-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24FN5O4S
(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-5-methyl-7-[4-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H28N6O2
(7R)-N-(2,4-dimethylphenyl)-5-methyl-7-[4-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-7-[4-[(2,4,5-trimethylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H24N6O2
(7S)-5-methyl-7-[4-[(2,4,5-trimethylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[5-bromo-2-[(4-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C20H19BrN6O2
(7S)-7-[5-bromo-2-[(4-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H21ClN6O2
(7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2,4-dichlorophenyl)-5-methyl-N-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H14Cl2N6O
(7S)-7-(2,4-dichlorophenyl)-5-methyl-N-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[2-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C30H32N6O2
(7S)-7-[2-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H17ClN6O2
(7R)-7-[2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22Cl2N6O2
(7S)-7-[2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H21ClN6O2
(7R)-7-[2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(3-propoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C23H26N6O2
(7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(3-propoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(2-phenylmethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N6O2
(7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(2-phenylmethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25ClN6O2
(7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-fluorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H17FN6O2
(7R)-7-(4-fluorophenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-7-(3-propoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C15H18N6O2
(7R)-5-methyl-7-(3-propoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-methoxyphenyl)-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N6O3
(7S)-N-(2-methoxyphenyl)-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[2-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C29H30N6O2
(7R)-7-[2-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-N-(2-methylphenyl)-7-[2-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N6O2
(7S)-5-methyl-N-(2-methylphenyl)-7-[2-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H21ClN6O2
(7S)-7-[2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N7O4
(7S)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-N-(2,4-dimethylphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H15BrCl2N6O2
(7S)-7-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(S)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H25FN6O3
7-[(S)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-(4-methylpiperidin-1-yl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-5-methyl-N-phenyl-7-[4-[(2,4,5-trimethylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H28N6O2
(7S)-5-methyl-N-phenyl-7-[4-[(2,4,5-trimethylphenyl)methoxy]phenyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-pyrrolidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C23H21FN6O3
7-[(R)-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]-pyrrolidin-1-ylmethyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-7-[5-bromo-2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H16BrClN6O2
(7R)-7-[5-bromo-2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H15BrCl2N6O2
(7R)-7-[5-bromo-2-[(2,4-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N7O5
(7R)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2-butoxyphenyl)-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H24N6O2
(7R)-7-(2-butoxyphenyl)-5-methyl-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-butoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C23H26N6O3
(7S)-7-(3-butoxyphenyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-N-(2-methylphenyl)-7-(3-propoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H24N6O2
(7S)-5-methyl-N-(2-methylphenyl)-7-(3-propoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-7-[4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H25N7O4
(7S)-5-methyl-7-[4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-N-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7,8-dimethyl-3-[[[(2S)-oxolan-2-yl]methyl-[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C24H32N6O3
7,8-dimethyl-3-[[[(2S)-oxolan-2-yl]methyl-[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— (7R)-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23ClN6O2
(7R)-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-N-(2-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-(2-methylphenyl)-7-(3-propoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H24N6O2
(7R)-5-methyl-N-(2-methylphenyl)-7-(3-propoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[2-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H17ClN6O2
(7R)-7-[2-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C19H17ClN6O2
(7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(R)-azepan-1-yl-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H25FN6O3
7-[(R)-azepan-1-yl-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one