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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-[(4-ethoxy-3-methoxyphenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C23H26N4O3
7-[(4-ethoxy-3-methoxyphenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[1-[(2R)-2-(4-ethoxyphenoxy)propanoyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C24H27N3O4
7-[1-[(2R)-2-(4-ethoxyphenoxy)propanoyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(3-Ethoxy-4-prop-2-ynoxyphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N4O3
7-[(3-Ethoxy-4-prop-2-ynoxyphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3-ethoxy-4-hydroxyphenyl)methyl]-2-[(2S)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N4O3
7-[(3-ethoxy-4-hydroxyphenyl)methyl]-2-[(2S)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(5-propylfuran-2-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H23N5O2
7-[(5-propylfuran-2-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-propanoyl-2-[(2S)-1-(1-propylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N6O3
7-propanoyl-2-[(2S)-1-(1-propylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C21H26N6O
7-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3R)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]-5-methylimidazo[5,1-b][1,3]thiazole —— C17H23N5O2S2
7-[(3R)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]-5-methylimidazo[5,1-b][1,3]thiazole
—— 7-[(1-ethylpyrazol-4-yl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C17H25N5O
7-[(1-ethylpyrazol-4-yl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3S)-1-[(1-ethylpyrazol-4-yl)methyl]piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C21H24F3N5O
7-[(3S)-1-[(1-ethylpyrazol-4-yl)methyl]piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[1-(1-Ethylpyrazol-4-yl)sulfonylpiperidin-4-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole —— C17H23N5O2S2
7-[1-(1-Ethylpyrazol-4-yl)sulfonylpiperidin-4-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole
—— 7-[(3R)-1-(1-ethylpyrazole-4-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H20F3N5O2
7-[(3R)-1-(1-ethylpyrazole-4-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-acetyl-2-[(2S)-1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O4
7-acetyl-2-[(2S)-1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclohexylmethyl)-2-[(2S)-1-(1-ethylpyrazole-4-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H34N6O2
7-(cyclohexylmethyl)-2-[(2S)-1-(1-ethylpyrazole-4-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C19H20N4O3
7-[(3S)-1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-cyclopentyl-2-[(2R)-1-(1-ethylpyrazole-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H32N6O2
7-cyclopentyl-2-[(2R)-1-(1-ethylpyrazole-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H22N4O3
7-[(3S)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-(3,5-diethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-2-(dimethylamino)-6H-pyrido[4,3-d]pyrimidin-5-one —— C22H28N6O3
7-[1-(3,5-diethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-2-(dimethylamino)-6H-pyrido[4,3-d]pyrimidin-5-one
—— 7-[(3S)-1-(3,5-diethyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H22N4O3
7-[(3S)-1-(3,5-diethyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-cyclopentyl-2-[(2S)-1-(5-ethyl-4-methyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H34N6O2
7-cyclopentyl-2-[(2S)-1-(5-ethyl-4-methyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-ethyl-1-benzofuran-3-yl)methyl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C16H18N4O
7-[(2-ethyl-1-benzofuran-3-yl)methyl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(3R)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H22N4O3
7-[(3R)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-ethylsulfonyl-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H24N4O4S2
7-ethylsulfonyl-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O4S
7-ethylsulfonyl-2-[(2S)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2R)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O4S
7-ethylsulfonyl-2-[(2R)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2S)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H25FN4O4S
7-ethylsulfonyl-2-[(2S)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-amino-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]heptanamide —— C16H33N3O
7-amino-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]heptanamide
—— 7-ethylsulfonyl-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O4S
7-ethylsulfonyl-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-butyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C22H34N6O
7-[(1-butyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-butanoyl-2-[(2R)-1-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H32N6O3
7-butanoyl-2-[(2R)-1-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-butanoyl-2-[(2S)-1-(1-propylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H32N6O3
7-butanoyl-2-[(2S)-1-(1-propylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-butanoyl-2-[(2R)-1-(1-propylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H32N6O3
7-butanoyl-2-[(2R)-1-(1-propylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-butanoyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H27FN4O3
7-butanoyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-butanoyl-2-[(2R)-1-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H32N6O3
7-butanoyl-2-[(2R)-1-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-methoxyphenyl)methyl]-2-[(3S)-1-[(2S)-2-methylbutanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H32N4O3
7-[(4-methoxyphenyl)methyl]-2-[(3S)-1-[(2S)-2-methylbutanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-acetyl-2-[(3S)-1-(2-ethylbutanoyl)pyrrolidin-3-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H28N4O3
7-acetyl-2-[(3S)-1-(2-ethylbutanoyl)pyrrolidin-3-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclohexylmethyl)-2-[(2S)-1-[(2S)-2-methylbutanoyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H36N4O2
7-(cyclohexylmethyl)-2-[(2S)-1-[(2S)-2-methylbutanoyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-acetyl-2-[(3R)-1-(2-ethylbutanoyl)pyrrolidin-3-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H28N4O3
7-acetyl-2-[(3R)-1-(2-ethylbutanoyl)pyrrolidin-3-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-[(2S)-2-methylbutanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H27FN4O3
7-(2-fluorobenzoyl)-2-[(3S)-1-[(2S)-2-methylbutanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2S)-1-propanoylpiperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C16H24N4O4S
7-methylsulfonyl-2-[(2S)-1-propanoylpiperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-4'-[(3S,4S)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O4
7-chloro-4'-[(3S,4S)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one —— C22H26N6O3
7-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one
—— 7-chloro-4'-[(3S)-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O3
7-chloro-4'-[(3S)-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-chloro-4'-[(3R)-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O3
7-chloro-4'-[(3R)-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-chloro-N-[(1R,2S)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H29ClN2O3
7-chloro-N-[(1R,2S)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-(cyclohexylmethyl)-2-[(2R)-1-[(2R)-2-methylbutanoyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H36N4O2
7-(cyclohexylmethyl)-2-[(2R)-1-[(2R)-2-methylbutanoyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-4'-[(3R,4R)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O4
7-chloro-4'-[(3R,4R)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— (7S)-3-[[4-hydroxy-1-(thiophen-2-ylmethyl)piperidin-4-yl]methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S2
(7S)-3-[[4-hydroxy-1-(thiophen-2-ylmethyl)piperidin-4-yl]methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-chloro-4'-[(2R)-2-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O3
7-chloro-4'-[(2R)-2-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— (7S)-3-[[1-(cyclopropanecarbonyl)-4-hydroxypiperidin-4-yl]methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H27N3O3S
(7S)-3-[[1-(cyclopropanecarbonyl)-4-hydroxypiperidin-4-yl]methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one