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—— (7R)-7-methyl-N-[(2R)-4-phenylbutan-2-yl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C22H26N4O
(7R)-7-methyl-N-[(2R)-4-phenylbutan-2-yl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7S)-7-methyl-N-(thiophen-2-ylmethyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C17H18N4OS
(7S)-7-methyl-N-(thiophen-2-ylmethyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7R)-N-(furan-2-ylmethyl)-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C17H18N4O2
(7R)-N-(furan-2-ylmethyl)-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7R)-7-methyl-N-(4-methylcyclohexyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C19H26N4O
(7R)-7-methyl-N-(4-methylcyclohexyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7S)-7-methyl-N-[(2R)-4-phenylbutan-2-yl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C22H26N4O
(7S)-7-methyl-N-[(2R)-4-phenylbutan-2-yl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7R)-7-methyl-N-[[(2S)-oxolan-2-yl]methyl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C17H22N4O2
(7R)-7-methyl-N-[[(2S)-oxolan-2-yl]methyl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7R)-N-[(4-ethylphenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C21H24N4O
(7R)-N-[(4-ethylphenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— 7-[(2,4-dichlorophenyl)methyl]-8-[4-[(E)-[3-(2,4-dimethylphenyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-2-methoxyphenoxy]-1,3-dimethylpurine-2,6-dione —— C33H27Cl2N5O5S2
7-[(2,4-dichlorophenyl)methyl]-8-[4-[(E)-[3-(2,4-dimethylphenyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]-2-methoxyphenoxy]-1,3-dimethylpurine-2,6-dione
—— (7R)-7-methyl-N-(3-propylsulfanylpropyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C18H26N4OS
(7R)-7-methyl-N-(3-propylsulfanylpropyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7R)-7-methyl-N-[(2S)-4-phenylbutan-2-yl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C22H26N4O
(7R)-7-methyl-N-[(2S)-4-phenylbutan-2-yl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7R)-N-[(2-methoxyphenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C20H22N4O2
(7R)-N-[(2-methoxyphenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7S)-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C22H24N4O3
(7S)-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7S)-7-methyl-N-(4-methylcyclohexyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C19H26N4O
(7S)-7-methyl-N-(4-methylcyclohexyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7R)-7-methyl-N-(pyridin-3-ylmethyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C18H19N5O
(7R)-7-methyl-N-(pyridin-3-ylmethyl)-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7S)-N-(1,3-benzodioxol-5-ylmethyl)-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C20H20N4O3
(7S)-N-(1,3-benzodioxol-5-ylmethyl)-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7S)-N-[2-(3,4-diethoxyphenyl)ethyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C24H30N4O3
(7S)-N-[2-(3,4-diethoxyphenyl)ethyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7R)-N-[2-(3,4-dimethoxyphenyl)ethyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C22H26N4O3
(7R)-N-[2-(3,4-dimethoxyphenyl)ethyl]-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— (7Z)-7-(4-methylpent-3-enylidene)-3,4a,5,6,8,8a-hexahydro-2H-phthalazine-1,4-dione —— C14H20N2O2
(7Z)-7-(4-methylpent-3-enylidene)-3,4a,5,6,8,8a-hexahydro-2H-phthalazine-1,4-dione
—— (7R)-7-methyl-N-propyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C15H20N4O
(7R)-7-methyl-N-propyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— 7-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-4,6-dimethyl-2,3-dihydro-1,4-benzoxazine —— C17H26N2O3S
7-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-4,6-dimethyl-2,3-dihydro-1,4-benzoxazine
—— (7-methoxy-2-oxochromen-4-yl)methyl (2S)-2-acetamido-3-(1H-indol-3-yl)propanoate —— C24H22N2O6
(7-methoxy-2-oxochromen-4-yl)methyl (2S)-2-acetamido-3-(1H-indol-3-yl)propanoate
—— 7-chloro-3-methyl-N-[(1R,2R)-2-methylcyclohexyl]-1-benzofuran-2-carboxamide —— C17H20ClNO2
7-chloro-3-methyl-N-[(1R,2R)-2-methylcyclohexyl]-1-benzofuran-2-carboxamide
—— 7-[[2-amino-2-(4-hydroxyphenyl)acetyl]amino]-3-[(E)-but-1-enyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C19H21N3O5S
7-[[2-amino-2-(4-hydroxyphenyl)acetyl]amino]-3-[(E)-but-1-enyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 7-tert-butyl-5-[(2S)-2-hydroxy-3-naphthalen-2-yloxypropyl]sulfanyl-1,3-dimethylpyrimido[4,5-d]pyrimidine-2,4-dione —— C25H28N4O4S
7-tert-butyl-5-[(2S)-2-hydroxy-3-naphthalen-2-yloxypropyl]sulfanyl-1,3-dimethylpyrimido[4,5-d]pyrimidine-2,4-dione
—— (7S)-7-methyl-N-(2-methyl-2-morpholin-4-ylpropyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C19H28N4OS
(7S)-7-methyl-N-(2-methyl-2-morpholin-4-ylpropyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 7-[4-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-nitrophenoxy]chromen-2-one —— C21H20N2O7S
7-[4-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-nitrophenoxy]chromen-2-one
—— 7-chloro-2-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-3-prop-2-enylquinazolin-4-one —— C19H22ClN3O3S
7-chloro-2-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-3-prop-2-enylquinazolin-4-one
—— [(7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-[1-(4-chlorophenyl)sulfonylpyrrolidin-2-yl]methanone —— C31H30ClN3O3S
[(7E)-7-benzylidene-3-phenyl-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-[1-(4-chlorophenyl)sulfonylpyrrolidin-2-yl]methanone
—— 7-chloro-3-(2-methoxyethyl)-2-[(2S)-1-oxo-1-phenylpropan-2-yl]sulfanylquinazolin-4-one —— C20H19ClN2O3S
7-chloro-3-(2-methoxyethyl)-2-[(2S)-1-oxo-1-phenylpropan-2-yl]sulfanylquinazolin-4-one
—— (7S)-2-(2-methylpropyl)-5-oxo-N-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C16H19N5O2
(7S)-2-(2-methylpropyl)-5-oxo-N-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-chloro-N-[4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-3-methyl-1-benzofuran-2-carboxamide —— C22H23ClN2O5S
7-chloro-N-[4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonylphenyl]-3-methyl-1-benzofuran-2-carboxamide
—— (7R)-N-(4-chlorophenyl)-2-(4-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C19H16ClN5O2
(7R)-N-(4-chlorophenyl)-2-(4-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-2-(4-methylphenyl)-5-oxo-N-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C19H17N5O2
(7S)-2-(4-methylphenyl)-5-oxo-N-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(4-fluorophenyl)-2-(2-methylpropyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C16H18FN5O2
(7S)-N-(4-fluorophenyl)-2-(2-methylpropyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-5-oxo-2-phenyl-N-[3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C19H14F3N5O2
(7S)-5-oxo-2-phenyl-N-[3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(3-methylphenyl)-2-(4-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C20H19N5O2
(7R)-N-(3-methylphenyl)-2-(4-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— [(7E)-7-(4-chlorobenzylidene)-3-(4-chlorophenyl)-5-methyl-3,3a,4,5,6,7-hexahydro-2H-indazol-2-yl](2,4-dinitrophenyl)methanone —— C28H22Cl2N4O5
[(7E)-7-(4-chlorobenzylidene)-3-(4-chlorophenyl)-5-methyl-3,3a,4,5,6,7-hexahydro-2H-indazol-2-yl](2,4-dinitrophenyl)methanone
—— 7-chloro-2-[[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]pyrido[1,2-a]pyrimidin-4-one —— C17H17ClN4O
7-chloro-2-[[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-methoxy-N-[(1R)-1-phenylethyl]-2H-chromene-3-carboxamide —— C19H19NO3
7-methoxy-N-[(1R)-1-phenylethyl]-2H-chromene-3-carboxamide
—— 7-[[(2S)-2-(4-methoxyphenyl)pyrrolidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H19N3O2S
7-[[(2S)-2-(4-methoxyphenyl)pyrrolidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-ethyl-9a-[(E)-2-(4-methoxyphenyl)ethenyl]-9,9-dimethyl-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one —— C23H26N2O2
7-ethyl-9a-[(E)-2-(4-methoxyphenyl)ethenyl]-9,9-dimethyl-9,9a-dihydro-1H-imidazo[1,2-a]indol-2(3H)-one
—— 7-[[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl-methylamino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C17H17N3O3S
7-[[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl-methylamino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— [(7-methyl-5-nitro-2-oxoindol-3-yl)amino]thiourea —— C10H9N5O3S
[(7-methyl-5-nitro-2-oxoindol-3-yl)amino]thiourea
—— (7R,8S,8aS)-5-chloro-3-[(1E,3E,5S)-3,5-dimethylhepta-1,3-dienyl]-7,8-dihydroxy-7-methyl-8,8a-dihydro-1H-isochromen-6-one —— C19H25ClO4
(7R,8S,8aS)-5-chloro-3-[(1E,3E,5S)-3,5-dimethylhepta-1,3-dienyl]-7,8-dihydroxy-7-methyl-8,8a-dihydro-1H-isochromen-6-one
—— (7S)-7-(4-methoxyphenyl)-1,4-thiazepane —— C12H17NOS
(7S)-7-(4-methoxyphenyl)-1,4-thiazepane
—— 7-[2-(3,4-dimethoxyphenyl)ethyl]-6-imino-11-methyl-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C28H31N5O5
7-[2-(3,4-dimethoxyphenyl)ethyl]-6-imino-11-methyl-2-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 7-methyl-3-{(Z)-[3-(4-methylbenzyl)-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene]methyl}-2-(morpholin-4-yl)-4H-pyrido[1,2-a]pyrimidin-4-one —— C25H24N4O3S2
7-methyl-3-{(Z)-[3-(4-methylbenzyl)-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene]methyl}-2-(morpholin-4-yl)-4H-pyrido[1,2-a]pyrimidin-4-one
—— [(7E)-7-(4-bromobenzylidene)-3-(4-bromophenyl)-3,3a,4,5,6,7-hexahydro-2H-indazol-2-yl](2-phenylquinolin-4-yl)methanone —— C36H27Br2N3O
[(7E)-7-(4-bromobenzylidene)-3-(4-bromophenyl)-3,3a,4,5,6,7-hexahydro-2H-indazol-2-yl](2-phenylquinolin-4-yl)methanone
—— 7-methyl-3-{(Z)-[3-(4-methylbenzyl)-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene]methyl}-2-(4-methylpiperidin-1-yl)-4H-pyrido[1,2-a]pyrimidin-4-one —— C27H28N4O2S2
7-methyl-3-{(Z)-[3-(4-methylbenzyl)-4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene]methyl}-2-(4-methylpiperidin-1-yl)-4H-pyrido[1,2-a]pyrimidin-4-one
—— 7-benzyl-8-[(2Z)-2-[(4-bromophenyl)methylidene]hydrazinyl]-1,3-dimethylpurine-2,6-dione —— C21H19BrN6O2
7-benzyl-8-[(2Z)-2-[(4-bromophenyl)methylidene]hydrazinyl]-1,3-dimethylpurine-2,6-dione