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—— (7S)-N-(3-chloro-4-fluorophenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C24H24ClFN2O2S
(7S)-N-(3-chloro-4-fluorophenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7S)-3-ethyl-2-methyl-N-(4-methylphenyl)-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C24H26N2OS
(7S)-3-ethyl-2-methyl-N-(4-methylphenyl)-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7R)-N-(3,4-dimethylphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C25H28N2OS
(7R)-N-(3,4-dimethylphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C26H30N2O2S
(7R)-N-(2,4-dimethylphenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7S)-N-(2,4-dimethoxyphenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C26H30N2O4S
(7S)-N-(2,4-dimethoxyphenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7R)-3-ethyl-2-methyl-N-(2-methylphenyl)-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C24H26N2OS
(7R)-3-ethyl-2-methyl-N-(2-methylphenyl)-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7R)-N-(3,5-dimethylphenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C26H30N2O2S
(7R)-N-(3,5-dimethylphenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— 7-benzyl-3-cyclohexyl-2-[(2Z)-2-(4-fluorobenzylidene)hydrazinyl]-5,6,7,8-tetrahydropyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4(3H)-one —— C29H30FN5OS
7-benzyl-3-cyclohexyl-2-[(2Z)-2-(4-fluorobenzylidene)hydrazinyl]-5,6,7,8-tetrahydropyrido[4',3':4,5]thieno[2,3-d]pyrimidin-4(3H)-one
—— 7-[(E)-3-chlorobut-2-enyl]-1,3-dimethyl-8-[(2Z)-2-[1-(4-nitrophenyl)ethylidene]hydrazinyl]purine-2,6-dione —— C19H20ClN7O4
7-[(E)-3-chlorobut-2-enyl]-1,3-dimethyl-8-[(2Z)-2-[1-(4-nitrophenyl)ethylidene]hydrazinyl]purine-2,6-dione
—— (7-methyl-4,5-dihydrothieno[2,3-e][1]benzothiol-2-yl)-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methanone —— C24H26N2OS2
(7-methyl-4,5-dihydrothieno[2,3-e][1]benzothiol-2-yl)-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methanone
—— 7-[(4-chlorophenyl)methyl]-8-[(2Z)-2-[[4-(dimethylamino)phenyl]methylidene]hydrazinyl]-3-methylpurine-2,6-dione —— C22H22ClN7O2
7-[(4-chlorophenyl)methyl]-8-[(2Z)-2-[[4-(dimethylamino)phenyl]methylidene]hydrazinyl]-3-methylpurine-2,6-dione
—— 7-[(E)-3-chlorobut-2-enyl]-1,3-dimethyl-8-[(2Z)-2-[(E)-4-phenylbut-3-en-2-ylidene]hydrazinyl]purine-2,6-dione —— C21H23ClN6O2
7-[(E)-3-chlorobut-2-enyl]-1,3-dimethyl-8-[(2Z)-2-[(E)-4-phenylbut-3-en-2-ylidene]hydrazinyl]purine-2,6-dione
—— 7-(4-chlorobenzyl)-1,3-dimethyl-8-[(2E)-2-(3-methylcyclohexylidene)hydrazinyl]-3,7-dihydro-1H-purine-2,6-dione —— C21H25ClN6O2
7-(4-chlorobenzyl)-1,3-dimethyl-8-[(2E)-2-(3-methylcyclohexylidene)hydrazinyl]-3,7-dihydro-1H-purine-2,6-dione
—— 7-(2-hydroxyethyl)-3-methyl-8-[2-[(4-oxocyclohexa-2,5-dien-1-ylidene)methyl]hydrazinyl]purine-2,6-dione —— C15H16N6O4
7-(2-hydroxyethyl)-3-methyl-8-[2-[(4-oxocyclohexa-2,5-dien-1-ylidene)methyl]hydrazinyl]purine-2,6-dione
—— (7E)-7-(4-chlorobenzylidene)-3-(4-chlorophenyl)-2-(4,5-diphenyl-1,3-thiazol-2-yl)-3,3a,4,5,6,7-hexahydro-2H-indazole —— C35H27Cl2N3S
(7E)-7-(4-chlorobenzylidene)-3-(4-chlorophenyl)-2-(4,5-diphenyl-1,3-thiazol-2-yl)-3,3a,4,5,6,7-hexahydro-2H-indazole
—— (7R)-2-benzylsulfanyl-7-(4-ethylphenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2S
(7R)-2-benzylsulfanyl-7-(4-ethylphenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-chlorophenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24ClN5O2S
(7R)-2-benzylsulfanyl-7-(4-chlorophenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-hydroxy-4,8-dimethyl-3-[3-oxo-3-(piperidin-1-yl)propyl]-2H-chromen-2-one —— C19H23NO4
7-hydroxy-4,8-dimethyl-3-[3-oxo-3-(piperidin-1-yl)propyl]-2H-chromen-2-one
—— 7-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C14H20N4O2S
7-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 7-hydroxy-4,8-dimethyl-3-[3-(morpholin-4-yl)-3-oxopropyl]-2H-chromen-2-one —— C18H21NO5
7-hydroxy-4,8-dimethyl-3-[3-(morpholin-4-yl)-3-oxopropyl]-2H-chromen-2-one
—— 7-hydroxy-4-methyl-3-[3-oxo-3-(piperidin-1-yl)propyl]-2H-chromen-2-one —— C18H21NO4
7-hydroxy-4-methyl-3-[3-oxo-3-(piperidin-1-yl)propyl]-2H-chromen-2-one
—— (7S)-2-benzylsulfanyl-7-(4-ethylphenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2S
(7S)-2-benzylsulfanyl-7-(4-ethylphenyl)-N-(4-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(E)-3-chlorobut-2-enyl]-8-[(2Z)-2-[(4-fluorophenyl)methylidene]hydrazinyl]-1,3-dimethylpurine-2,6-dione —— C18H18ClFN6O2
7-[(E)-3-chlorobut-2-enyl]-8-[(2Z)-2-[(4-fluorophenyl)methylidene]hydrazinyl]-1,3-dimethylpurine-2,6-dione
—— 7-hydroxy-4,8-dimethyl-3-[3-oxo-3-(pyrrolidin-1-yl)propyl]-2H-chromen-2-one —— C18H21NO4
7-hydroxy-4,8-dimethyl-3-[3-oxo-3-(pyrrolidin-1-yl)propyl]-2H-chromen-2-one
—— (7S)-7-(2-methoxyphenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H27N5O3
(7S)-7-(2-methoxyphenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— 7-Hydroxy-4-methyl-3-(3-morpholin-4-yl-3-oxopropyl)chromen-2-one —— C17H19NO5
7-Hydroxy-4-methyl-3-(3-morpholin-4-yl-3-oxopropyl)chromen-2-one
—— 7-hydroxy-4,8-dimethyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-2H-chromen-2-one —— C17H19NO5
7-hydroxy-4,8-dimethyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-2H-chromen-2-one
—— 7-[(3S)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C23H31N3O6S
7-[(3S)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— (7S)-5-methyl-3-N-(3-methylphenyl)-7-(2-nitrophenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H24N6O4
(7S)-5-methyl-3-N-(3-methylphenyl)-7-(2-nitrophenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-N-(3,5-dimethylphenyl)-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide —— C21H23NOS2
(7S)-N-(3,5-dimethylphenyl)-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide
—— 7-Hydroxy-4,8-dimethyl-3-(2-oxo-2-piperidin-1-ylethyl)chromen-2-one —— C18H21NO4
7-Hydroxy-4,8-dimethyl-3-(2-oxo-2-piperidin-1-ylethyl)chromen-2-one
—— 7-[[5-(4-chlorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C19H17ClN6OS2
7-[[5-(4-chlorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 7-Hydroxy-3-(4-hydroxyphenyl)-2-[4-(2-piperazin-1-ylethoxy)benzoyl]chromen-4-one —— C28H26N2O6
7-Hydroxy-3-(4-hydroxyphenyl)-2-[4-(2-piperazin-1-ylethoxy)benzoyl]chromen-4-one
—— 7-[(3R)-3-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C26H32N4O4S
7-[(3R)-3-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(3S)-3-(azepane-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C22H31N3O4S
7-[(3S)-3-(azepane-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— (7S)-3-N-(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H26FN5O3
(7S)-3-N-(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— 7-hydroxy-8-(morpholin-4-ylmethyl)-4-phenyl-6-propyl-2H-chromen-2-one —— C23H25NO4
7-hydroxy-8-(morpholin-4-ylmethyl)-4-phenyl-6-propyl-2H-chromen-2-one
—— 7-Hydroxy-3-(4-methoxyphenyl)-2-[4-(2-piperazin-1-ylethoxy)benzoyl]chromen-4-one —— C29H28N2O6
7-Hydroxy-3-(4-methoxyphenyl)-2-[4-(2-piperazin-1-ylethoxy)benzoyl]chromen-4-one
—— (7S)-N-(2,5-dimethylphenyl)-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide —— C21H23NOS2
(7S)-N-(2,5-dimethylphenyl)-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide
—— (7R)-N-(3,4-dimethylphenyl)-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide —— C21H23NOS2
(7R)-N-(3,4-dimethylphenyl)-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide
—— (7S)-N-[(2S)-butan-2-yl]-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide —— C17H23NOS2
(7S)-N-[(2S)-butan-2-yl]-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide
—— (7R)-3-N-(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H26FN5O3
(7R)-3-N-(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-7-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-7-(4-chlorophenyl)-6-N-(4-methoxyphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H24ClN5O3
(7R)-7-(4-chlorophenyl)-6-N-(4-methoxyphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— 7-[(3S)-3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C22H31N3O4S
7-[(3S)-3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— 7-[(3R)-3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one —— C22H31N3O4S
7-[(3R)-3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]sulfonyl-1,3,4,5-tetrahydro-1-benzazepin-2-one
—— (7R)-3-N,7-bis(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H23F2N5O3
(7R)-3-N,7-bis(4-fluorophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(2-chlorophenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C28H24ClN5O2
(7S)-7-(2-chlorophenyl)-5-methyl-3-N-(4-methylphenyl)-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-N-(2,5-dimethylphenyl)-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide —— C21H23NOS2
(7R)-N-(2,5-dimethylphenyl)-7-methyl-6,7,8,9-tetrahydro-1H-thiopyrano[4,3-b][1]benzothiole-3-carboxamide
—— 7-[(2R)-4-(4-cyclohexylpiperazin-1-yl)-4-oxobutan-2-yl]sulfonyl-6-methyl-4H-1,4-benzoxazin-3-one —— C23H33N3O5S
7-[(2R)-4-(4-cyclohexylpiperazin-1-yl)-4-oxobutan-2-yl]sulfonyl-6-methyl-4H-1,4-benzoxazin-3-one
—— (7R)-6-N-(2,4-dimethylphenyl)-5-methyl-7-(4-methylphenyl)-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C30H29N5O2
(7R)-6-N-(2,4-dimethylphenyl)-5-methyl-7-(4-methylphenyl)-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide