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—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H25N5O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C20H26N6O3S
7-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2R)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H27FN4O2
7-(cyclopropylmethyl)-2-[(2R)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H25FN6O2
7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O2
7-[2-(4-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(6-methylpyridine-3-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C26H33N5O2
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(6-methylpyridine-3-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H23FN6O2
7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-(pyrazine-2-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— [7-(1,5-dimethylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-3-hydroxy-3-(4-methylphenyl)pyrrolidin-1-yl]methanone —— C23H24N6O2
[7-(1,5-dimethylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-3-hydroxy-3-(4-methylphenyl)pyrrolidin-1-yl]methanone
—— [7-(1,5-dimethylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-hydroxy-3-(4-methylphenyl)pyrrolidin-1-yl]methanone —— C23H24N6O2
[7-(1,5-dimethylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-hydroxy-3-(4-methylphenyl)pyrrolidin-1-yl]methanone
—— (7-amino-2-methylpyrazolo[1,5-a]pyrimidin-6-yl)-[(2S)-2-(4-ethoxyphenyl)pyrrolidin-1-yl]methanone —— C20H23N5O2
(7-amino-2-methylpyrazolo[1,5-a]pyrimidin-6-yl)-[(2S)-2-(4-ethoxyphenyl)pyrrolidin-1-yl]methanone
—— 7-(difluoromethyl)-5-methyl-N-[(1S)-1-(1-propan-2-ylbenzimidazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H22F2N6O
7-(difluoromethyl)-5-methyl-N-[(1S)-1-(1-propan-2-ylbenzimidazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-methoxy-2-methyl-N-[(1S)-1-(4-morpholin-4-ylphenyl)ethyl]quinoline-3-carboxamide —— C24H27N3O3
7-methoxy-2-methyl-N-[(1S)-1-(4-morpholin-4-ylphenyl)ethyl]quinoline-3-carboxamide
—— 7-(4-fluorophenyl)-N-[(2R)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H23FN6O
7-(4-fluorophenyl)-N-[(2R)-1-(1,3,5-trimethylpyrazol-4-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 7-(difluoromethyl)-N-[(4R)-2,2-dimethyl-3,4-dihydrochromen-4-yl]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H20F2N4O2
7-(difluoromethyl)-N-[(4R)-2,2-dimethyl-3,4-dihydrochromen-4-yl]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-amino-2-methyl-N-[(1S)-1-phenyl-3-piperidin-1-ylpropyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H28N6O
7-amino-2-methyl-N-[(1S)-1-phenyl-3-piperidin-1-ylpropyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-methoxy-N-[(3R)-1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-methylquinoline-3-carboxamide —— C23H23N3O4
7-methoxy-N-[(3R)-1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-methylquinoline-3-carboxamide
—— 7-ethyl-1-methyl-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C18H25N5O4
7-ethyl-1-methyl-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-ethyl-1-methyl-N-[(2S)-1-morpholin-4-ylpropan-2-yl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C18H25N5O4
7-ethyl-1-methyl-N-[(2S)-1-morpholin-4-ylpropan-2-yl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-ethyl-5-[(3S)-3-hydroxy-3-(4-methylphenyl)pyrrolidine-1-carbonyl]-1-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H24N4O4
7-ethyl-5-[(3S)-3-hydroxy-3-(4-methylphenyl)pyrrolidine-1-carbonyl]-1-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-(benzenesulfonyl)-N-methyl-2-(1-methylpiperidin-4-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C20H27N5O2S
7-(benzenesulfonyl)-N-methyl-2-(1-methylpiperidin-4-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-(4-fluoro-3-methylphenyl)sulfonyl-3-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C18H24FN5O2S
7-(4-fluoro-3-methylphenyl)sulfonyl-3-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(4-fluoro-3-methylphenyl)sulfonyl-N-methyl-2-(1-methylpiperidin-4-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C21H28FN5O2S
7-(4-fluoro-3-methylphenyl)sulfonyl-N-methyl-2-(1-methylpiperidin-4-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-(3,4-dimethylphenyl)sulfonyl-N-methyl-2-[(3S)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C22H31N5O2S
7-(3,4-dimethylphenyl)sulfonyl-N-methyl-2-[(3S)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-methyl-2-[(3S)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C19H28N6O3S
7-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-methyl-2-[(3S)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-(4-methoxyphenyl)sulfonyl-N-methyl-2-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C21H29N5O3S
7-(4-methoxyphenyl)sulfonyl-N-methyl-2-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-[(3-cyclopentyloxyphenyl)methyl]-N-methyl-2-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C24H33N5O
7-[(3-cyclopentyloxyphenyl)methyl]-N-methyl-2-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-(3,4-dimethylphenyl)sulfonyl-N-methyl-2-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C22H31N5O2S
7-(3,4-dimethylphenyl)sulfonyl-N-methyl-2-[(3R)-1-methylpiperidin-3-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-(2-Fluoro-5-methylphenyl)sulfonyl-3-piperidin-4-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C18H24FN5O2S
7-(2-Fluoro-5-methylphenyl)sulfonyl-3-piperidin-4-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-[[3-(4-fluorophenyl)phenyl]methyl]-3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C23H26FN5
7-[[3-(4-fluorophenyl)phenyl]methyl]-3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-(4-fluoro-2-methylphenyl)sulfonyl-3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C18H24FN5O2S
7-(4-fluoro-2-methylphenyl)sulfonyl-3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— (7R)-5-(isoquinoline-1-carbonyl)-N,N,2-trimethyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C20H21N5O2
(7R)-5-(isoquinoline-1-carbonyl)-N,N,2-trimethyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— 7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C22H31N5O
7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— (7R)-N-[(4-methoxyphenyl)methyl]-5-[(E)-3-(2-methoxyphenyl)prop-2-enyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C26H30N4O3
(7R)-N-[(4-methoxyphenyl)methyl]-5-[(E)-3-(2-methoxyphenyl)prop-2-enyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— 7-(2-chlorophenyl)-1,3,4,5-tetrahydroimidazo[4,5-e][2,1,3]benzoxadiazol-6-ium 6-oxide —— C13H10ClN4O2+
7-(2-chlorophenyl)-1,3,4,5-tetrahydroimidazo[4,5-e][2,1,3]benzoxadiazol-6-ium 6-oxide
—— 7-(2-chlorophenyl)sulfonyl-3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C17H22ClN5O2S
7-(2-chlorophenyl)sulfonyl-3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— (7S)-N-[2-(4-fluorophenyl)ethyl]-2-methyl-5-(quinolin-6-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C26H26FN5O
(7S)-N-[2-(4-fluorophenyl)ethyl]-2-methyl-5-(quinolin-6-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-N-benzyl-N-ethyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C16H20N4O
(7R)-N-benzyl-N-ethyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— [(7R)-5-benzoyl-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-7-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone —— C25H26FN5O2
[(7R)-5-benzoyl-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-7-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone
—— 7-Hydroxy-2-methyl-3-phenyl-8-(piperidin-1-ium-1-ylmethyl)chromen-4-one —— C22H24NO3+
7-Hydroxy-2-methyl-3-phenyl-8-(piperidin-1-ium-1-ylmethyl)chromen-4-one
—— (7R)-5-[2-(2-fluorophenyl)acetyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C22H22FN5O2
(7R)-5-[2-(2-fluorophenyl)acetyl]-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-(4-methoxyphenyl)sulfonyl-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C21H23N5O4S
(7R)-5-(4-methoxyphenyl)sulfonyl-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-2-methyl-N,N-dipropyl-4,5,6,7-tetrahydropyrazolo[4,3-c]pyridine-7-carboxamide —— C14H24N4O
(7S)-2-methyl-N,N-dipropyl-4,5,6,7-tetrahydropyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-5-(2-methoxy-3-methylbenzoyl)-N-[(4-methoxyphenyl)methyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C25H28N4O4
(7S)-5-(2-methoxy-3-methylbenzoyl)-N-[(4-methoxyphenyl)methyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-N-(2,3-dihydro-1H-inden-2-yl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C16H18N4O
(7R)-N-(2,3-dihydro-1H-inden-2-yl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-5-acetyl-2-methyl-N-(3-methylbutyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C15H24N4O2
(7S)-5-acetyl-2-methyl-N-(3-methylbutyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-N-[2-(4-fluorophenyl)ethyl]-2-methyl-5-[(4-propan-2-ylphenyl)methyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C26H31FN4O
(7R)-N-[2-(4-fluorophenyl)ethyl]-2-methyl-5-[(4-propan-2-ylphenyl)methyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-[2-[3-(dimethylamino)phenoxy]acetyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C18H23N5O3
(7R)-5-[2-[3-(dimethylamino)phenoxy]acetyl]-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-5-(4-methoxyphenyl)sulfonyl-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C21H23N5O4S
(7S)-5-(4-methoxyphenyl)sulfonyl-2-methyl-N-(pyridin-2-ylmethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7R)-5-acetyl-N-(2,2-dimethylpropyl)-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C15H24N4O2
(7R)-5-acetyl-N-(2,2-dimethylpropyl)-2-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide
—— (7S)-N-[2-(4-fluorophenyl)ethyl]-2-methyl-5-[2-(2-oxopyrrolidin-1-yl)acetyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide —— C22H26FN5O3
(7S)-N-[2-(4-fluorophenyl)ethyl]-2-methyl-5-[2-(2-oxopyrrolidin-1-yl)acetyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-7-carboxamide