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—— 7-oxo-N'-[(Z)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]-2-(trifluoromethyl)-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbohydrazide —— C14H9F3N6O3
7-oxo-N'-[(Z)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]-2-(trifluoromethyl)-1H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbohydrazide
—— (7S)-7-(2,4-dimorpholin-4-yl-5-nitrophenyl)-2,4-dimethyl-8-oxa-2,4-diazabicyclo[4.2.0]oct-1(6)-ene-3,5-dione —— C21H25N5O7
(7S)-7-(2,4-dimorpholin-4-yl-5-nitrophenyl)-2,4-dimethyl-8-oxa-2,4-diazabicyclo[4.2.0]oct-1(6)-ene-3,5-dione
—— (7Z)-7-[(4-bromo-1-ethyl-1H-pyrazol-5-yl)methylidene]-3-(difluoromethyl)-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C17H13BrF2N6S
(7Z)-7-[(4-bromo-1-ethyl-1H-pyrazol-5-yl)methylidene]-3-(difluoromethyl)-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7R)-7-[2,4-bis(4-methylpiperidin-1-yl)-5-nitrophenyl]-8-oxa-2,4-diazabicyclo[4.2.0]oct-1(6)-ene-3,5-dione —— C23H29N5O5
(7R)-7-[2,4-bis(4-methylpiperidin-1-yl)-5-nitrophenyl]-8-oxa-2,4-diazabicyclo[4.2.0]oct-1(6)-ene-3,5-dione
—— (7S)-4-imino-2,7-dimethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-3-amine —— C12H16N4S
(7S)-4-imino-2,7-dimethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-3-amine
—— (7S)-2-amino-N-(2-fluorophenyl)-7-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-b]pyridine-3-carboxamide —— C20H17F4N3OS
(7S)-2-amino-N-(2-fluorophenyl)-7-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-b]pyridine-3-carboxamide
—— (7R)-2-amino-N-(2-fluorophenyl)-7-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-b]pyridine-3-carboxamide —— C20H17F4N3OS
(7R)-2-amino-N-(2-fluorophenyl)-7-methyl-4-(trifluoromethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-b]pyridine-3-carboxamide
—— (7Z)-7-(3-bromo-5-methoxy-4-propoxybenzylidene)-3-methyl-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C22H21BrN4O2S
(7Z)-7-(3-bromo-5-methoxy-4-propoxybenzylidene)-3-methyl-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-(difluoromethyl)-7-[(1,5-dimethyl-1H-pyrazol-4-yl)methylidene]-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C17H14F2N6S
(7Z)-3-(difluoromethyl)-7-[(1,5-dimethyl-1H-pyrazol-4-yl)methylidene]-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-7-{[5-(2-chlorophenyl)furan-2-yl]methylidene}-6-(2,4-difluorophenyl)-3-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C22H13ClF2N4OS
(7Z)-7-{[5-(2-chlorophenyl)furan-2-yl]methylidene}-6-(2,4-difluorophenyl)-3-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-[chloro(difluoro)methyl]-6-(2,4-dichlorophenyl)-7-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methylidene]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C18H13Cl3F2N6S
(7Z)-3-[chloro(difluoro)methyl]-6-(2,4-dichlorophenyl)-7-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methylidene]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-(difluoromethyl)-7-{3-methoxy-4-[2-(morpholin-4-yl)ethoxy]benzylidene}-6-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C20H23F2N5O3S
(7Z)-3-(difluoromethyl)-7-{3-methoxy-4-[2-(morpholin-4-yl)ethoxy]benzylidene}-6-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-6-(2,4-difluorophenyl)-7-[(1,3-dimethyl-1H-pyrazol-4-yl)methylidene]-3-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C17H14F2N6S
(7Z)-6-(2,4-difluorophenyl)-7-[(1,3-dimethyl-1H-pyrazol-4-yl)methylidene]-3-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-[chloro(difluoro)methyl]-6-methyl-7-{[5-(4-nitrophenyl)furan-2-yl]methylidene}-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C17H10ClF2N5O3S
(7Z)-3-[chloro(difluoro)methyl]-6-methyl-7-{[5-(4-nitrophenyl)furan-2-yl]methylidene}-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-(difluoromethyl)-7-[(5-methylthiophen-2-yl)methylidene]-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C17H12F2N4S2
(7Z)-3-(difluoromethyl)-7-[(5-methylthiophen-2-yl)methylidene]-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-(difluoromethyl)-6-methyl-7-(pyridin-2-ylmethylidene)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C12H9F2N5S
(7Z)-3-(difluoromethyl)-6-methyl-7-(pyridin-2-ylmethylidene)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-7-[[5-[(3-bromophenoxy)methyl]furan-2-yl]methylidene]-3-(difluoromethyl)-6-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C18H13BrF2N4O2S
(7Z)-7-[[5-[(3-bromophenoxy)methyl]furan-2-yl]methylidene]-3-(difluoromethyl)-6-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7E)-3-(difluoromethyl)-6-methyl-7-[(1-methyl-1H-pyrazol-3-yl)methylidene]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C11H10F2N6S
(7E)-3-(difluoromethyl)-6-methyl-7-[(1-methyl-1H-pyrazol-3-yl)methylidene]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— 7-[(2-chlorophenyl)methyl]-8-[3-[(E)-hydroxyiminomethyl]phenoxy]-1,3-dimethylpurine-2,6-dione —— C21H18ClN5O4
7-[(2-chlorophenyl)methyl]-8-[3-[(E)-hydroxyiminomethyl]phenoxy]-1,3-dimethylpurine-2,6-dione
—— (7Z)-3-(difluoromethyl)-7-{[1-(3-nitrophenyl)-1H-pyrrol-2-yl]methylidene}-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C22H14F2N6O2S
(7Z)-3-(difluoromethyl)-7-{[1-(3-nitrophenyl)-1H-pyrrol-2-yl]methylidene}-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-7-[(4-bromothiophen-2-yl)methylidene]-3-(difluoromethyl)-6-(2,4-difluorophenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C16H7BrF4N4S2
(7Z)-7-[(4-bromothiophen-2-yl)methylidene]-3-(difluoromethyl)-6-(2,4-difluorophenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-(difluoromethyl)-7-(2,4-dimethoxybenzylidene)-6-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C15H14F2N4O2S
(7Z)-3-(difluoromethyl)-7-(2,4-dimethoxybenzylidene)-6-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— 7H-[1,2,4]Triazolo[3,4-b][1,3,4]thiadiazine, 3-difluoromethyl-6-phenyl-7-thiophen-2-ylmethylene- —— C16H10F2N4S2
7H-[1,2,4]Triazolo[3,4-b][1,3,4]thiadiazine, 3-difluoromethyl-6-phenyl-7-thiophen-2-ylmethylene-
—— (7Z)-7-{[5-(2-chloro-4-nitrophenyl)furan-2-yl]methylidene}-3-(difluoromethyl)-6-(2,4-difluorophenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C22H10ClF4N5O3S
(7Z)-7-{[5-(2-chloro-4-nitrophenyl)furan-2-yl]methylidene}-3-(difluoromethyl)-6-(2,4-difluorophenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-[chloro(difluoro)methyl]-6-methyl-7-[(5-methylthiophen-2-yl)methylidene]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C12H9ClF2N4S2
(7Z)-3-[chloro(difluoro)methyl]-6-methyl-7-[(5-methylthiophen-2-yl)methylidene]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-(difluoromethyl)-6-(2,4-difluorophenyl)-7-(thiophen-2-ylmethylidene)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C16H8F4N4S2
(7Z)-3-(difluoromethyl)-6-(2,4-difluorophenyl)-7-(thiophen-2-ylmethylidene)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-[chloro(difluoro)methyl]-6-phenyl-7-(thiophen-2-ylmethylidene)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C16H9ClF2N4S2
(7Z)-3-[chloro(difluoro)methyl]-6-phenyl-7-(thiophen-2-ylmethylidene)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-6-(2,4-difluorophenyl)-3-methyl-7-[(5-methylthiophen-2-yl)methylidene]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C17H12F2N4S2
(7Z)-6-(2,4-difluorophenyl)-3-methyl-7-[(5-methylthiophen-2-yl)methylidene]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-7-[(6-bromo-1,3-benzodioxol-5-yl)methylidene]-3-(difluoromethyl)-6-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C14H9BrF2N4O2S
(7Z)-7-[(6-bromo-1,3-benzodioxol-5-yl)methylidene]-3-(difluoromethyl)-6-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7Z)-3-(difluoromethyl)-7-[(1-methyl-1H-pyrazol-3-yl)methylidene]-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C16H12F2N6S
(7Z)-3-(difluoromethyl)-7-[(1-methyl-1H-pyrazol-3-yl)methylidene]-6-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— 7-methoxy-N-[(2S)-4-phenylbutan-2-yl]-1-benzofuran-2-carboxamide —— C20H21NO3
7-methoxy-N-[(2S)-4-phenylbutan-2-yl]-1-benzofuran-2-carboxamide
—— 7-methoxy-N-[2-[[(1R)-1-phenylethyl]carbamoyl]phenyl]-1-benzofuran-2-carboxamide —— C25H22N2O4
7-methoxy-N-[2-[[(1R)-1-phenylethyl]carbamoyl]phenyl]-1-benzofuran-2-carboxamide
—— 7-methoxy-N-[2-(piperidine-1-carbonyl)phenyl]-1-benzofuran-2-carboxamide —— C22H22N2O4
7-methoxy-N-[2-(piperidine-1-carbonyl)phenyl]-1-benzofuran-2-carboxamide
—— 7-methoxy-N-[2-[[(1S)-1-phenylethyl]carbamoyl]phenyl]-1-benzofuran-2-carboxamide —— C25H22N2O4
7-methoxy-N-[2-[[(1S)-1-phenylethyl]carbamoyl]phenyl]-1-benzofuran-2-carboxamide
—— 7-[(2S)-2-hydroxy-3-(4-methoxyphenoxy)propyl]-3-methyl-8-[(2Z)-2-[1-(3-nitrophenyl)ethylidene]hydrazinyl]purine-2,6-dione —— C24H25N7O7
7-[(2S)-2-hydroxy-3-(4-methoxyphenoxy)propyl]-3-methyl-8-[(2Z)-2-[1-(3-nitrophenyl)ethylidene]hydrazinyl]purine-2,6-dione
—— 7-methoxy-N-[4-(phenylsulfanylmethyl)phenyl]-1-benzofuran-2-carboxamide —— C23H19NO3S
7-methoxy-N-[4-(phenylsulfanylmethyl)phenyl]-1-benzofuran-2-carboxamide
—— (7R)-5-(3,4-difluorophenyl)-7-[2-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H11F5N4
(7R)-5-(3,4-difluorophenyl)-7-[2-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-methoxy-N-[2-[(2-methylphenyl)methylsulfanyl]ethyl]-1-benzofuran-2-carboxamide —— C20H21NO3S
7-methoxy-N-[2-[(2-methylphenyl)methylsulfanyl]ethyl]-1-benzofuran-2-carboxamide
—— (7aS)-7a-morpholin-4-yl-4,5,6,7-tetrahydro-1-benzofuran-2-one —— C12H17NO3
(7aS)-7a-morpholin-4-yl-4,5,6,7-tetrahydro-1-benzofuran-2-one
—— 7-benzyl-4-methyl-2-[(3R)-1-(4-methylthiadiazole-5-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H24N6O2S
7-benzyl-4-methyl-2-[(3R)-1-(4-methylthiadiazole-5-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(3R)-1-(2-morpholin-4-ylacetyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H31N5O3
7-benzyl-4-methyl-2-[(3R)-1-(2-morpholin-4-ylacetyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(3S)-1-(2-morpholin-4-ylacetyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H31N5O3
7-benzyl-4-methyl-2-[(3S)-1-(2-morpholin-4-ylacetyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(3-methylbutanoyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(3-methylbutanoyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[1-(2-Cyclopentylacetyl)piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H32N4O4
7-[1-(2-Cyclopentylacetyl)piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-benzyl-4-methyl-2-[(3R)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H24N6O3
7-benzyl-4-methyl-2-[(3R)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H29FN4O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-2-[(2R)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H27N5O3
7-benzyl-2-[(2R)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(2-methylpropanoyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(2-methylpropanoyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one