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—— (7S)-2-[(1R)-1-[3-[(2S)-1-methoxypropan-2-yl]-4-oxoquinazolin-2-yl]sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H28N4O3S2
(7S)-2-[(1R)-1-[3-[(2S)-1-methoxypropan-2-yl]-4-oxoquinazolin-2-yl]sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-3-(2-methylpropyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H28N4O2S2
(7R)-7-methyl-2-[(8-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methylsulfanyl]-3-(2-methylpropyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H27N5O2S2
(7R)-2-[(1S)-1-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H27N5O2S2
(7S)-2-[(1R)-1-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1R)-1-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H27N5O2S2
(7R)-2-[(1R)-1-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-Hydroxy-8-[(4-methylpiperidin-1-ium-1-yl)methyl]-4-phenylchromen-2-one —— C22H24NO3+
7-Hydroxy-8-[(4-methylpiperidin-1-ium-1-yl)methyl]-4-phenylchromen-2-one
—— 7-(4-ethoxyphenyl)-10-[2-methyl-4-(1-pyrrolidinyl)benzylidene]-5,7-dihydro-6H-benzo[h][1,3]thiazolo[2,3-b]quinazolin-9(10H)-one —— C34H33N3O2S
7-(4-ethoxyphenyl)-10-[2-methyl-4-(1-pyrrolidinyl)benzylidene]-5,7-dihydro-6H-benzo[h][1,3]thiazolo[2,3-b]quinazolin-9(10H)-one
—— (7R)-7-tert-butyl-3-(4-methoxyphenyl)-2-[(5-methyl-1,3,4-oxadiazol-2-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C25H28N4O3S2
(7R)-7-tert-butyl-3-(4-methoxyphenyl)-2-[(5-methyl-1,3,4-oxadiazol-2-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1S)-1-(1-oxidopyridin-1-ium-2-yl)sulfanylethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H19N3O2S2
(7S)-7-methyl-2-[(1S)-1-(1-oxidopyridin-1-ium-2-yl)sulfanylethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-(1-oxidopyridin-1-ium-2-yl)sulfanylethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H19N3O2S2
(7R)-7-methyl-2-[(1R)-1-(1-oxidopyridin-1-ium-2-yl)sulfanylethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfanyl]-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H23N3O3S2
(7R)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfanyl]-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-[(5-ethyl-[1,2,4]triazino[5,6-b]indol-3-yl)sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H24N6OS2
(7S)-2-[(1S)-1-[(5-ethyl-[1,2,4]triazino[5,6-b]indol-3-yl)sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[(2,4-dichlorophenyl)methyl]-8-[2-methoxy-4-[(E)-[3-(4-methylphenyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]phenoxy]-1,3-dimethylpurine-2,6-dione —— C32H25Cl2N5O5S2
7-[(2,4-dichlorophenyl)methyl]-8-[2-methoxy-4-[(E)-[3-(4-methylphenyl)-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]methyl]phenoxy]-1,3-dimethylpurine-2,6-dione
—— 7-methyl-N-[(2R)-4-phenylbutan-2-yl]-3-(4-propan-2-ylphenyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H30N4O
7-methyl-N-[(2R)-4-phenylbutan-2-yl]-3-(4-propan-2-ylphenyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidine —— C23H24N6
7-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-Tert-butyl-2-[4-(2,5-dimethoxyphenyl)sulfonylpiperazin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C21H28N6O4S
7-Tert-butyl-2-[4-(2,5-dimethoxyphenyl)sulfonylpiperazin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-decyl-3-methyl-8-[2-[1-(4-oxocyclohexa-2,5-dien-1-ylidene)ethyl]hydrazinyl]purine-2,6-dione —— C24H34N6O3
7-decyl-3-methyl-8-[2-[1-(4-oxocyclohexa-2,5-dien-1-ylidene)ethyl]hydrazinyl]purine-2,6-dione
—— (7S)-3-[(2-chlorophenyl)methyl]-7-[4-(2-methoxyethyl)piperazin-1-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H29ClN4O2S
(7S)-3-[(2-chlorophenyl)methyl]-7-[4-(2-methoxyethyl)piperazin-1-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-(4-ethylpiperazin-1-yl)-3-(3-methylbutyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H32N4OS
(7R)-7-(4-ethylpiperazin-1-yl)-3-(3-methylbutyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-3-[2-(2-chlorophenyl)ethyl]-7-(4-ethylpiperazin-1-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H29ClN4OS
(7R)-3-[2-(2-chlorophenyl)ethyl]-7-(4-ethylpiperazin-1-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-[4-(2-methoxyethyl)piperazin-1-yl]-3-(3-phenylpropyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C26H34N4O2S
(7R)-7-[4-(2-methoxyethyl)piperazin-1-yl]-3-(3-phenylpropyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-methyl-N-[(2R)-4-methylpentan-2-yl]-3-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H23F3N4O
7-methyl-N-[(2R)-4-methylpentan-2-yl]-3-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-methyl-N-[(2S)-4-methylpentan-2-yl]-3-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H23F3N4O
7-methyl-N-[(2S)-4-methylpentan-2-yl]-3-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R,11bR)-N-(2,4-dibromo-6-fluorophenyl)-7-methyl-4-oxo-3,6,7,11b-tetrahydro-1H-pyrazino[2,1-a]isoquinoline-2-carboxamide —— C20H18Br2FN3O2
(7R,11bR)-N-(2,4-dibromo-6-fluorophenyl)-7-methyl-4-oxo-3,6,7,11b-tetrahydro-1H-pyrazino[2,1-a]isoquinoline-2-carboxamide
—— (7R,11bS)-N-(2,4-dibromo-6-fluorophenyl)-7-methyl-4-oxo-3,6,7,11b-tetrahydro-1H-pyrazino[2,1-a]isoquinoline-2-carboxamide —— C20H18Br2FN3O2
(7R,11bS)-N-(2,4-dibromo-6-fluorophenyl)-7-methyl-4-oxo-3,6,7,11b-tetrahydro-1H-pyrazino[2,1-a]isoquinoline-2-carboxamide
—— (7S,11bS)-N-(2,4-dibromo-6-fluorophenyl)-7-methyl-4-oxo-3,6,7,11b-tetrahydro-1H-pyrazino[2,1-a]isoquinoline-2-carboxamide —— C20H18Br2FN3O2
(7S,11bS)-N-(2,4-dibromo-6-fluorophenyl)-7-methyl-4-oxo-3,6,7,11b-tetrahydro-1H-pyrazino[2,1-a]isoquinoline-2-carboxamide
—— 7-[4-[(3S)-3-methylpiperidin-1-yl]piperidin-1-yl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidine —— C22H28N6
7-[4-[(3S)-3-methylpiperidin-1-yl]piperidin-1-yl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7E)-4-(3-chlorophenyl)-7-[(2-chlorophenyl)methylidene]-2-ethoxy-5,6-dihydrocyclopenta[b]pyridine-3-carbonitrile —— C24H18Cl2N2O
(7E)-4-(3-chlorophenyl)-7-[(2-chlorophenyl)methylidene]-2-ethoxy-5,6-dihydrocyclopenta[b]pyridine-3-carbonitrile
—— 7-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C14H18N4OS
7-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (7-ethyl-2-oxochromen-4-yl)methyl 2-[3-chloro-2-oxo-5-(trifluoromethyl)pyridin-1-yl]acetate —— C20H15ClF3NO5
(7-ethyl-2-oxochromen-4-yl)methyl 2-[3-chloro-2-oxo-5-(trifluoromethyl)pyridin-1-yl]acetate
—— 7-hydroxy-8-methyl-6-[(4-methylpiperidin-1-yl)methyl]-4-phenyl-2H-chromen-2-one —— C23H25NO3
7-hydroxy-8-methyl-6-[(4-methylpiperidin-1-yl)methyl]-4-phenyl-2H-chromen-2-one
—— 7-[[4-[(3S)-1-(4-butylphenyl)-5-oxopyrrolidine-3-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C26H31N5O3S
7-[[4-[(3S)-1-(4-butylphenyl)-5-oxopyrrolidine-3-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-benzyl-3-methyl-8-[2-[(E)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]hydrazinyl]purine-2,6-dione —— C20H18N6O3
7-benzyl-3-methyl-8-[2-[(E)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]hydrazinyl]purine-2,6-dione
—— (7R)-3-cyclopentyl-7-[[1-(4-methylpiperazin-1-yl)cyclohexyl]methylamino]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C27H41N5OS
(7R)-3-cyclopentyl-7-[[1-(4-methylpiperazin-1-yl)cyclohexyl]methylamino]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7-methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl (E)-3-(3-fluorophenyl)prop-2-enoate —— C23H21FO4
(7-methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl (E)-3-(3-fluorophenyl)prop-2-enoate
—— (7S)-3-[2-(2-acetylphenoxy)ethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H22N2O3S
(7S)-3-[2-(2-acetylphenoxy)ethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-3-[2-(2,2-dimethyl-3-oxo-4H-quinoxalin-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24N4O3S
(7S)-3-[2-(2,2-dimethyl-3-oxo-4H-quinoxalin-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-3-[2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H25FN4O2S
(7S)-3-[2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— [(7E)-3-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-[1-(4-chlorophenyl)sulfonylpyrrolidin-2-yl]methanone —— C31H28Cl3N3O3S
[(7E)-3-(4-chlorophenyl)-7-[(4-chlorophenyl)methylidene]-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-[1-(4-chlorophenyl)sulfonylpyrrolidin-2-yl]methanone
—— (7R)-3-[2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H25FN4O2S
(7R)-3-[2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-3-[(6-chloro-7-methyl-2-oxochromen-4-yl)methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H19ClN2O3S
(7S)-3-[(6-chloro-7-methyl-2-oxochromen-4-yl)methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3S)-3-acetamido-3-(4-methylphenyl)propanoate —— C22H23N3O4
(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3S)-3-acetamido-3-(4-methylphenyl)propanoate
—— 7,7-dimethyl-9-[[(2R)-oxolan-2-yl]methyl]-6,9-diazaspiro[4.5]decane —— C15H28N2O
7,7-dimethyl-9-[[(2R)-oxolan-2-yl]methyl]-6,9-diazaspiro[4.5]decane
—— 7-[[4-[2-[(2R)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolidin-1-yl]-2-oxoethyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C25H29N5O4S
7-[[4-[2-[(2R)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrrolidin-1-yl]-2-oxoethyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3R)-3-acetamido-3-(4-methylphenyl)propanoate —— C22H23N3O4
(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3R)-3-acetamido-3-(4-methylphenyl)propanoate
—— (7R)-7-methyl-N-[2-(4-methylpiperazin-1-yl)ethyl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide —— C19H28N6O
(7R)-7-methyl-N-[2-(4-methylpiperazin-1-yl)ethyl]-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline-3-carboxamide
—— 7-[2-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one —— C17H19N5O4
7-[2-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one
—— 7-Hydroxy-3-(3-methoxyphenoxy)-2-methyl-8-[(3-methylpiperidin-1-yl)methyl]chromen-4-one —— C24H27NO5
7-Hydroxy-3-(3-methoxyphenoxy)-2-methyl-8-[(3-methylpiperidin-1-yl)methyl]chromen-4-one
—— 7-chloro-N-[(Z)-(1-methyl-2-phenylindol-3-yl)methylideneamino]quinolin-4-amine —— C25H19ClN4
7-chloro-N-[(Z)-(1-methyl-2-phenylindol-3-yl)methylideneamino]quinolin-4-amine
—— 7-[[4-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C23H27N5O2S2
7-[[4-[2-[(2R)-2-methyl-3,4-dihydro-2H-1,5-benzothiazepin-5-yl]-2-oxoethyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one