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—— (R)-Spiro[2.5]oct-5-ylamine —— C8H15N
(R)-Spiro[2.5]oct-5-ylamine
—— (R)-[6-(2,4-dichlorophenyl)-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-3-yl]-phenylmethanamine —— C17H13Cl2N5S
(R)-[6-(2,4-dichlorophenyl)-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-3-yl]-phenylmethanamine
—— (R)-1,3,3-trimethyl-butylamine trifluoroacetate —— (x)C2HF3O2*C7H17N
(R)-1,3,3-trimethyl-butylamine trifluoroacetate
—— ((R)-2,2-dichloro-cyclopropyl)-methylamine —— C4H7Cl2N
((R)-2,2-dichloro-cyclopropyl)-methylamine
—— ((R)-1,3,3-trimethyl-butyl)-carbamic acid tert-butyl ester —— C12H25NO2
((R)-1,3,3-trimethyl-butyl)-carbamic acid tert-butyl ester
—— (R)-4-[(R)-5-(1-methanesulfonyl-1,2,3,6-tetrahydro-pyridin-4-yl )-2-methyl-2,3-dihydrofuro[2,3-c]pyridin-2-yl]-piperidine-1-carboxylic acid 2,2,2-trifluoro-1-methyl-ethyl ester —— C23H30F3N3O5S
(R)-4-[(R)-5-(1-methanesulfonyl-1,2,3,6-tetrahydro-pyridin-4-yl )-2-methyl-2,3-dihydrofuro[2,3-c]pyridin-2-yl]-piperidine-1-carboxylic acid 2,2,2-trifluoro-1-methyl-ethyl ester
—— (R)-4-[(R)-5-(4-methanesulfonyl-phenyl)-2-methyl-2.3-dihydro-furo[2.3-c]pyridin-2-yl]piperidine-1-carboxylic acid 2,2,2-trifluoro-1-methyl-ethyl ester —— C24H27F3N2O5S
(R)-4-[(R)-5-(4-methanesulfonyl-phenyl)-2-methyl-2.3-dihydro-furo[2.3-c]pyridin-2-yl]piperidine-1-carboxylic acid 2,2,2-trifluoro-1-methyl-ethyl ester
—— (R)-3-phenyl-cyclopentylamine —— C11H15N
(R)-3-phenyl-cyclopentylamine
—— (R)-1-(2-phenoxyethyl)piperidine carboxylic acid hydrochloride —— C14H20ClNO3
(R)-1-(2-phenoxyethyl)piperidine carboxylic acid hydrochloride
—— [(R)-1-((R)-2,2-dichloro-cyclopropyl)-2-hydroxy-ethyl]-carbamic acid tert-butyl ester —— C10H17Cl2NO3
[(R)-1-((R)-2,2-dichloro-cyclopropyl)-2-hydroxy-ethyl]-carbamic acid tert-butyl ester
—— (R)-4-[(R)-5-(1-methanesulfonyl-1,2,3,6-tetrahydro-pyridin-4-yl )-2,3-dihydro-furo[2.3-c]pyridin-2-yl]-piperidine-1-carboxylic acid 2,2,2-trifluoro-1-methyl-ethyl ester —— C22H28F3N3O5S
(R)-4-[(R)-5-(1-methanesulfonyl-1,2,3,6-tetrahydro-pyridin-4-yl )-2,3-dihydro-furo[2.3-c]pyridin-2-yl]-piperidine-1-carboxylic acid 2,2,2-trifluoro-1-methyl-ethyl ester
—— rac-(1R,2S)-2-(3-chloro-2-fluorophenyl)cyclopropan-1-amine —— C9H9ClFN
rac-(1R,2S)-2-(3-chloro-2-fluorophenyl)cyclopropan-1-amine
—— [(R)-[(2S,4S,5R)-5-ethenyl-1-azabicyclo[2.2.2]octan-2-yl]-(6-methoxyquinolin-4-yl)methyl] 2,2,2-trifluoroacetate —— C22H23F3N2O3
[(R)-[(2S,4S,5R)-5-ethenyl-1-azabicyclo[2.2.2]octan-2-yl]-(6-methoxyquinolin-4-yl)methyl] 2,2,2-trifluoroacetate
—— (R)-(3-hydroxypiperidin-1-yl)(4-(6-((1-(3,3,3-trifluoro-2,2-dimethylpropyl)piperidin-4-yl)methoxy)pyridin-3-yl)phenyl)methanone —— C28H36F3N3O3
(R)-(3-hydroxypiperidin-1-yl)(4-(6-((1-(3,3,3-trifluoro-2,2-dimethylpropyl)piperidin-4-yl)methoxy)pyridin-3-yl)phenyl)methanone
—— (R)-(5-(3-fluoro-4-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)phenyl)pyridin-2-yl)(3-hydroxypiperidin-1-yl)methanone —— C29H35F4N3O3
(R)-(5-(3-fluoro-4-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)phenyl)pyridin-2-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(4′-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methylamino)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C28H38FN3O2
(R)-(4′-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methylamino)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(2-(hydroxymethyl)pyrrolidin-1-yl)(4-(6-((1-((1-(trifluoromethyl)cyclopentyl)methyl)piperidin-4-yl)methoxy)pyridin-3-yl)phenyl)methanone —— C30H38F3N3O3
(R)-(2-(hydroxymethyl)pyrrolidin-1-yl)(4-(6-((1-((1-(trifluoromethyl)cyclopentyl)methyl)piperidin-4-yl)methoxy)pyridin-3-yl)phenyl)methanone
—— (R)-1-(4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenylcarbonyl)pyrrolidine-2-carboxamide —— C28H36FN3O3
(R)-1-(4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenylcarbonyl)pyrrolidine-2-carboxamide
—— (R)-(3'-fluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C28H36F2N2O3
(R)-(3'-fluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(4-(6-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-3-yl)phenyl)(3-hydroxypyrrolidine-1-yl)methanone —— C26H34FN3O3
(R)-(4-(6-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-3-yl)phenyl)(3-hydroxypyrrolidine-1-yl)methanone
—— (R)-(2',3-difluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(2-(hydroxymethyl)pyrrolidine-1-yl)methanone —— C28H35F3N2O3
(R)-(2',3-difluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(2-(hydroxymethyl)pyrrolidine-1-yl)methanone
—— (R)-(4'-((1-((1-fluorocyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(2-(hydroxymethyl)pyrrolidin-1-yl)methanone —— C29H37FN2O3
(R)-(4'-((1-((1-fluorocyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(2-(hydroxymethyl)pyrrolidin-1-yl)methanone
—— (R)-1-(2-fluoro-4-(6-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-3-yl)benzoyl)piperidin-2-carboxamide —— C28H36F2N4O3
(R)-1-(2-fluoro-4-(6-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-3-yl)benzoyl)piperidin-2-carboxamide
—— (R)-(4'-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)-2,3'-difluorobiphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C30H39F3N2O3
(R)-(4'-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)-2,3'-difluorobiphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(3-hydroxypiperidin-1-yl)(4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)methanone —— C30H37F3N2O3
(R)-(3-hydroxypiperidin-1-yl)(4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)methanone
—— (R)-(2-fluoro-4-(6-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)pyridin-3-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone —— C29H35F4N3O3
(R)-(2-fluoro-4-(6-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)pyridin-3-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(2,3'-difluoro-4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C30H35F5N2O3
(R)-(2,3'-difluoro-4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-1-(4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyrazine-2-yl)benzoyl)piperidin-2-carboxamide —— C27H36FN5O3
(R)-1-(4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyrazine-2-yl)benzoyl)piperidin-2-carboxamide
—— (R)-2-(3-Benzyl-3-methyl-ureido)-3-phenyl-propionic acid methyl ester —— C19H22N2O3
(R)-2-(3-Benzyl-3-methyl-ureido)-3-phenyl-propionic acid methyl ester
—— ((R)-1-{5-[(E)-2-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)-vinyl]-1-methyl-1H-[1,2,4]triazol-3-yl}-pyrrolidin-3-yl)-carbamic acid tert-butyl ester —— C21H29N9O2
((R)-1-{5-[(E)-2-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)-vinyl]-1-methyl-1H-[1,2,4]triazol-3-yl}-pyrrolidin-3-yl)-carbamic acid tert-butyl ester
—— (R)-3'-fluoro-4-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)-4'-(3-hydroxypiperidin-1-carbonyl)biphenyl-2-carbonitrile —— C29H35F2N3O3
(R)-3'-fluoro-4-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)-4'-(3-hydroxypiperidin-1-carbonyl)biphenyl-2-carbonitrile
—— ((R)-1-{5-[2-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)-ethyl]-1-methyl-1H-[1,2,4]triazol-3-yl}-pyrrolidin-3-yl)-carbamic acid tert-butyl ester —— C21H31N9O2
((R)-1-{5-[2-(5,8-dimethyl-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)-ethyl]-1-methyl-1H-[1,2,4]triazol-3-yl}-pyrrolidin-3-yl)-carbamic acid tert-butyl ester
—— (R)-(3-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone —— C27H35F2N3O3
(R)-(3-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(2,3'-difluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(2-(hydroxymethyl)pyrrolidine-1-yl)methanone —— C28H35F3N2O3
(R)-(2,3'-difluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(2-(hydroxymethyl)pyrrolidine-1-yl)methanone
—— (R)-(4'-(((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methyl)(methyl)amino)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C29H40FN3O2
(R)-(4'-(((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methyl)(methyl)amino)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(3-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-2-yl)phenyl)(2-(hydroxymethyl)pyrrolidine-1-yl)methanone —— C27H35F2N3O3
(R)-(3-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-2-yl)phenyl)(2-(hydroxymethyl)pyrrolidine-1-yl)methanone
—— (R)-(2-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone —— C27H35F2N3O3
(R)-(2-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(3-hydroxypiperidin-1-yl)(4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methylamino)biphenyl-4-yl)methanone —— C30H38F3N3O2
(R)-(3-hydroxypiperidin-1-yl)(4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methylamino)biphenyl-4-yl)methanone
—— (R)-(2-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyrimidin-2-yl)phenyl)(3-hydroxypyrrolidin-1-yl)methanone —— C25H32F2N4O3
(R)-(2-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyrimidin-2-yl)phenyl)(3-hydroxypyrrolidin-1-yl)methanone
—— (R)-(2-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyrazin-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone —— C26H34F2N4O3
(R)-(2-fluoro-4-(5-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyrazin-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(4'-(ethyl((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methyl)amino)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C30H42FN3O2
(R)-(4'-(ethyl((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methyl)amino)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(4-(5-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)pyridin-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone —— C29H40FN3O3
(R)-(4-(5-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)pyridin-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(4-(5-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)pyridin-2-yl)-2-fluorophenyl)(3-hydroxypiperidin-1-yl)methanone —— C29H39F2N3O3
(R)-(4-(5-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)pyridin-2-yl)-2-fluorophenyl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(4'-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)-3-fluorobiphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C30H40F2N2O3
(R)-(4'-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)-3-fluorobiphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(2-fluoro-4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C30H36F4N2O3
(R)-(2-fluoro-4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(3,3'-difluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C28H35F3N2O3
(R)-(3,3'-difluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(4-(5-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)pyrimidin-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone —— C28H39FN4O3
(R)-(4-(5-((1-(2-ethyl-2-fluorobutyl)piperidin-4-yl)methoxy)pyrimidin-2-yl)phenyl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(2',3-difluoro-4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone —— C30H35F5N2O3
(R)-(2',3-difluoro-4'-((1-((1-(trifluoromethyl)cyclobutyl)methyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypiperidin-1-yl)methanone
—— (R)-(2-fluoro-4-(6-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-3-yl)phenyl)(3-hydroxypyrrolidine-1-yl)methanone —— C26H33F2N3O3
(R)-(2-fluoro-4-(6-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)pyridine-3-yl)phenyl)(3-hydroxypyrrolidine-1-yl)methanone
—— (R)-(3-fluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypyrrolidine-1-yl)methanone —— C27H34F2N2O3
(R)-(3-fluoro-4'-((1-(2-fluoro-2-methylpropyl)piperidin-4-yl)methoxy)biphenyl-4-yl)(3-hydroxypyrrolidine-1-yl)methanone