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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R5)-7-ethyl-4-hydroxy-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carbonyl chloride —— C13H13ClN2O2S
(R5)-7-ethyl-4-hydroxy-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carbonyl chloride
—— (R)-N-(4-((tert-butyldimethylsilyl)oxy)-1-cyclobutylbutyl)-2-chloro-7-(4-(trifluoromethyl)benzyl)-7H-purin-6-amine —— C27H37ClF3N5OSi
(R)-N-(4-((tert-butyldimethylsilyl)oxy)-1-cyclobutylbutyl)-2-chloro-7-(4-(trifluoromethyl)benzyl)-7H-purin-6-amine
—— (R)-7-(4-chlorobenzyl)-6-((1-cyclobutyl-4-hydroxybutyl)amino)-8-(3-methylphenyl)-7H-purine-2-carbonitrile —— C28H29ClN6O
(R)-7-(4-chlorobenzyl)-6-((1-cyclobutyl-4-hydroxybutyl)amino)-8-(3-methylphenyl)-7H-purine-2-carbonitrile
—— (R5)-4-chloro-7-ethyl-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carbonyl chloride —— C13H12Cl2N2OS
(R5)-4-chloro-7-ethyl-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidine-7-carbonyl chloride
—— (R)-6-((4-((tert-butyldimethylsilyl)oxy)-1-cyclobutylbutyl)amino)-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile —— C35H43F3N6OSi
(R)-6-((4-((tert-butyldimethylsilyl)oxy)-1-cyclobutylbutyl)amino)-8-(3-methylphenyl)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile
—— (R)-[(1S)-4-[(Z)-amino-(5-amino-2,3-dihydro-1H-pyridin-6-ylidene)methyl]-5-fluorocyclohexa-2,4-dien-1-yl]-[[4-(trifluoromethyl)pyridin-2-yl]amino]methanol —— C19H21F4N5O
(R)-[(1S)-4-[(Z)-amino-(5-amino-2,3-dihydro-1H-pyridin-6-ylidene)methyl]-5-fluorocyclohexa-2,4-dien-1-yl]-[[4-(trifluoromethyl)pyridin-2-yl]amino]methanol
—— (R)-[4-[(Z)-amino-(3-amino-1H-pyridin-2-ylidene)methyl]-2-methylphenyl]-[[(Z,3S)-5-amino-3-cyclopropylpent-4-enyl]amino]methanol —— C22H31N5O
(R)-[4-[(Z)-amino-(3-amino-1H-pyridin-2-ylidene)methyl]-2-methylphenyl]-[[(Z,3S)-5-amino-3-cyclopropylpent-4-enyl]amino]methanol
—— (R)-[(1S)-4-[(Z)-amino-(5-amino-2,3-dihydro-1H-pyrazin-6-ylidene)methyl]cyclohexa-2,4-dien-1-yl]-[[4-(trifluoromethyl)-2,3-dihydropyridin-6-yl]amino]methanol —— C18H23F3N6O
(R)-[(1S)-4-[(Z)-amino-(5-amino-2,3-dihydro-1H-pyrazin-6-ylidene)methyl]cyclohexa-2,4-dien-1-yl]-[[4-(trifluoromethyl)-2,3-dihydropyridin-6-yl]amino]methanol
—— (R)-tert-butyl 4-((2-bromophenyl)sulfonyl)-3-methylpiperazine-1-carboxylate —— C16H23BrN2O4S
(R)-tert-butyl 4-((2-bromophenyl)sulfonyl)-3-methylpiperazine-1-carboxylate
—— (R)-1-(1-benzylpyrrolidin-3-yl)-N-(3-(3,4-dichlorophenyl)propyl)-4-hydroxy-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429292-26-1 C25H27Cl2N3O3
(R)-1-(1-benzylpyrrolidin-3-yl)-N-(3-(3,4-dichlorophenyl)propyl)-4-hydroxy-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(3-(3,4-dichlorophenyl)propyl)-4-hydroxy-1-(2-hydroxy-2-phenylethyl)-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429293-00-4 C22H22Cl2N2O4
(R)-N-(3-(3,4-dichlorophenyl)propyl)-4-hydroxy-1-(2-hydroxy-2-phenylethyl)-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(chroman-2-ylmethyl)-1-ethyl-4-hydroxy-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429292-92-1 C17H20N2O4
(R)-N-(chroman-2-ylmethyl)-1-ethyl-4-hydroxy-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— racemic 5-({[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfanyl}methyl)-1,3-oxazolidin-2-one —— C20H17FN4O2S
racemic 5-({[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfanyl}methyl)-1,3-oxazolidin-2-one
—— (R)-4-hydroxy-N-(1-(naphthalen-2-yl)ethyl)-5-oxo-1-(2,2,2-trifluoroethyl)-2,5-dihydro-1H-pyrrole-3-carboxamide 1429292-95-4 C19H17F3N2O3
(R)-4-hydroxy-N-(1-(naphthalen-2-yl)ethyl)-5-oxo-1-(2,2,2-trifluoroethyl)-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-methyl-N-piperidin-3-ylbiphenyl-2-sulfonamide —— C22H24FN5O2S
(R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-methyl-N-piperidin-3-ylbiphenyl-2-sulfonamide
—— racemic 5-(3-fluoro-2'-{[2-(trifluoromethyl)morpholin-4-yl]carbonyl}biphenyl-4-yl)pyrazin-2-amine —— C22H18F4N4O2
racemic 5-(3-fluoro-2'-{[2-(trifluoromethyl)morpholin-4-yl]carbonyl}biphenyl-4-yl)pyrazin-2-amine
—— (R)-4''-(5-Aminopyrazin-2-yl)-3''-fluoro-N-[(1R)-2-hydroxy-1-methylethyl]biphenyl-2-sulfonamide —— C19H19FN4O3S
(R)-4''-(5-Aminopyrazin-2-yl)-3''-fluoro-N-[(1R)-2-hydroxy-1-methylethyl]biphenyl-2-sulfonamide
—— racemic-1-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-4-morpholin-4-ylpyrrolidin-3-ol trifluoroacetic acid salt —— (x)C2HF3O2*C24H26FN5O4S
racemic-1-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-4-morpholin-4-ylpyrrolidin-3-ol trifluoroacetic acid salt
—— racemic 1-((2-bromophenyl)sulfonyl)-4-morpholinopyrrolidin-3-ol —— C14H19BrN2O4S
racemic 1-((2-bromophenyl)sulfonyl)-4-morpholinopyrrolidin-3-ol
—— (racemic)-1-((4'-(6-amino-5-fluoropyridin-3-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)piperidin-3-ol —— C22H21F2N3O3S
(racemic)-1-((4'-(6-amino-5-fluoropyridin-3-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)piperidin-3-ol
—— racemic (trans)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-[2-(hydroxymethyl)cyclohexyl]biphenyl-2-sulfonamide —— C23H25FN4O3S
racemic (trans)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-[2-(hydroxymethyl)cyclohexyl]biphenyl-2-sulfonamide
—— racemic 2-bromo-N-[(1,2-cis)-2-(hydroxymethyl)cyclohexyl]benzenesulfonamide —— C13H18BrNO3S
racemic 2-bromo-N-[(1,2-cis)-2-(hydroxymethyl)cyclohexyl]benzenesulfonamide
—— racemic 1-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-3-phenylpyrrolidin-3-ol —— C26H23FN4O3S
racemic 1-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-3-phenylpyrrolidin-3-ol
—— (R)-2-bromo-N-(1-hydroxybutan-2-yl)benzenesulfonamide —— C10H14BrNO3S
(R)-2-bromo-N-(1-hydroxybutan-2-yl)benzenesulfonamide
—— (R)-4'-(5-amino-1,3,4-thiadiazol-2-yl)-3'-fluoro-N-(1-hydroxypropan-2-yl)-[1,1'-biphenyl]-2-sulfonamide —— C17H17FN4O3S2
(R)-4'-(5-amino-1,3,4-thiadiazol-2-yl)-3'-fluoro-N-(1-hydroxypropan-2-yl)-[1,1'-biphenyl]-2-sulfonamide
—— (R)-4'-(5-aminopyrazin-2-yl)-N-(2,3-dihydroxypropyl)-3'-fluoro-[1,1'-biphenyl]-2-sulfonamide —— C19H19FN4O4S
(R)-4'-(5-aminopyrazin-2-yl)-N-(2,3-dihydroxypropyl)-3'-fluoro-[1,1'-biphenyl]-2-sulfonamide
—— (R)-5-(2'-((3-aminopyrrolidin-1-yl)sulfonyl)-3-fluoro-[1,1'-biphenyl]-4-yl)pyrazin-2-amine —— C20H20FN5O2S
(R)-5-(2'-((3-aminopyrrolidin-1-yl)sulfonyl)-3-fluoro-[1,1'-biphenyl]-4-yl)pyrazin-2-amine
—— (R)-(1-((4'-(5-aminopyrazin-2-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)pyrrolidin-2-yl)methanol —— C21H21FN4O3S
(R)-(1-((4'-(5-aminopyrazin-2-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)pyrrolidin-2-yl)methanol
—— racemic 5-[3-fluoro-2'-(methylsulfinyl)biphenyl-4-yl]pyrazin-2-amine —— C17H14FN3OS
racemic 5-[3-fluoro-2'-(methylsulfinyl)biphenyl-4-yl]pyrazin-2-amine
—— racemic 1-((2-bromophenyl)sulfonyl)piperidin-3-amine hydrochloride salt —— C11H15BrN2O2S*ClH
racemic 1-((2-bromophenyl)sulfonyl)piperidin-3-amine hydrochloride salt
—— (racemic)-1'-((2-bromophenyl)sulfonyl)-[1,3'-bipyrrolidin]-4'-ol —— C14H19BrN2O3S
(racemic)-1'-((2-bromophenyl)sulfonyl)-[1,3'-bipyrrolidin]-4'-ol
—— racemic-1-((2-bromophenyl)sulfonyl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol —— C15H22BrN3O3S
racemic-1-((2-bromophenyl)sulfonyl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
—— (R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-(1-hydroxy-3,3-dimethylbutan-2-yl)-[1,1'-biphenyl]-2-sulfonamide —— C22H25FN4O3S
(R)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-(1-hydroxy-3,3-dimethylbutan-2-yl)-[1,1'-biphenyl]-2-sulfonamide
—— racemic-1'-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-1,3'-bipyrrolidin-4'-ol —— C24H26FN5O3S
racemic-1'-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-1,3'-bipyrrolidin-4'-ol
—— (R)-tert-butyl 3-(2-bromo-N-methylphenylsulfonamido)piperidine-1-carboxylate —— C17H25BrN2O4S
(R)-tert-butyl 3-(2-bromo-N-methylphenylsulfonamido)piperidine-1-carboxylate
—— racemic (4-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}morpholin-2-yl)methanol —— C21H21FN4O4S
racemic (4-{[4'-(2-aminopyrimidin-5-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}morpholin-2-yl)methanol
—— racemic-1-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-4-(4-methylpiperazin-1-yl)-pyrrolidin-3-ol trifluoroacetic acid salt —— (x)C2HF3O2*C25H29FN6O3S
racemic-1-{[4'-(5-aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-4-(4-methylpiperazin-1-yl)-pyrrolidin-3-ol trifluoroacetic acid salt
—— (R)-(1,1-dichloro-2-phenylethyl)-[(1R)-1-phenylethyl]-(trichloromethyl)phosphane —— C17H16Cl5P
(R)-(1,1-dichloro-2-phenylethyl)-[(1R)-1-phenylethyl]-(trichloromethyl)phosphane
—— (R)-4'-(6-aminopyridin-3-yl)-3'-fluoro-N-(1-hydroxypropan-2-yl)-[1,1'-biphenyl]-2-sulfonamide —— C20H20FN3O3S
(R)-4'-(6-aminopyridin-3-yl)-3'-fluoro-N-(1-hydroxypropan-2-yl)-[1,1'-biphenyl]-2-sulfonamide
—— racemic 2-bromo-N-[(1,2-trans)-2-(hydroxymethyl)cyclohexyl]benzenesulfonamide —— C13H18BrNO3S
racemic 2-bromo-N-[(1,2-trans)-2-(hydroxymethyl)cyclohexyl]benzenesulfonamide
—— (R)-tert-butyl 4-((4'-(2-aminopyrimidin-5-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)-3-(hydroxymethyl)piperazine-1-carboxylate —— C26H30FN5O5S
(R)-tert-butyl 4-((4'-(2-aminopyrimidin-5-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)-3-(hydroxymethyl)piperazine-1-carboxylate
—— racemic (cis)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-[2-(hydroxymethyl)cyclohexyl]biphenyl-2-sulfonamide —— C23H25FN4O3S
racemic (cis)-4'-(5-aminopyrazin-2-yl)-3'-fluoro-N-[2-(hydroxymethyl)cyclohexyl]biphenyl-2-sulfonamide
—— (R)-(1,1-dichloro-2-phenylethyl)-[(1S)-1-phenylethyl]-(trichloromethyl)phosphane —— C17H16Cl5P
(R)-(1,1-dichloro-2-phenylethyl)-[(1S)-1-phenylethyl]-(trichloromethyl)phosphane
—— (R)-(1-((4'-(5-aminopyrazin-2-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)pyrrolidin-3-yl)methanol —— C21H21FN4O3S
(R)-(1-((4'-(5-aminopyrazin-2-yl)-3'-fluoro-[1,1'-biphenyl]-2-yl)sulfonyl)pyrrolidin-3-yl)methanol
—— (R)-4'-(5-aminopyrazin-2-yl)-N-(1-cyanopropan-2-yl)-3'-fluoro-[1,1'-biphenyl]-2-sulfonamide —— C20H18FN5O2S
(R)-4'-(5-aminopyrazin-2-yl)-N-(1-cyanopropan-2-yl)-3'-fluoro-[1,1'-biphenyl]-2-sulfonamide
—— Racemic-1'-{[4'-(5-Aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-1,3'-bipyrrolidin-4'-ol —— C24H26FN5O3S
Racemic-1'-{[4'-(5-Aminopyrazin-2-yl)-3'-fluorobiphenyl-2-yl]sulfonyl}-1,3'-bipyrrolidin-4'-ol
—— (R)-4-(8-amino-3-(4-(2-hydroxyethyl)morpholin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide —— C25H24F3N7O3
(R)-4-(8-amino-3-(4-(2-hydroxyethyl)morpholin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— (R)-4-(8-amino-3-(4-(2-methoxyethyl)morpholin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide —— C26H26F3N7O3
(R)-4-(8-amino-3-(4-(2-methoxyethyl)morpholin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)benzamide
—— (R)-tert-butyl 4,4-difluoro-2-(3-(5-(pyridin-2-ylethynyl)pyridin-2-yl)-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxylate 1415144-37-4 C23H21F2N5O3
(R)-tert-butyl 4,4-difluoro-2-(3-(5-(pyridin-2-ylethynyl)pyridin-2-yl)-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxylate
—— (R)-4-(8-amino-3-(piperidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-methylpyridin-2-yl)benzamide —— C24H25N7O
(R)-4-(8-amino-3-(piperidin-3-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-methylpyridin-2-yl)benzamide