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—— Rel-{4-[2-(4-chlorophenoxy)ethyl]-1-piperazinyl}(4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}phenyl)methanone —— C24H27ClN4O4S2
Rel-{4-[2-(4-chlorophenoxy)ethyl]-1-piperazinyl}(4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}phenyl)methanone
—— Rel-(4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}phenyl)[4-(2-fluorophenyl)-1-piperazinyl]methanone —— C22H23FN4O3S2
Rel-(4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}phenyl)[4-(2-fluorophenyl)-1-piperazinyl]methanone
—— Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-phenylglycinamide —— C21H23N3O3S2
Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-phenylglycinamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethylphenyl)-N-(2-methoxyphenyl)glycinamide —— C22H25N3O4S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethylphenyl)-N-(2-methoxyphenyl)glycinamide
—— Rel-(3AR,6AR)-N-(2-chloro-4-fluorobenzyl)-N-(2-fluorophenyl)-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-amine 5,5-dioxide —— C18H15ClF2N2O2S2
Rel-(3AR,6AR)-N-(2-chloro-4-fluorobenzyl)-N-(2-fluorophenyl)-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-amine 5,5-dioxide
—— Rel-N,N~2~-bis(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]glycinamide —— C23H27N3O3S2
Rel-N,N~2~-bis(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]glycinamide
—— Rel-N~2~-(3-chlorophenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-fluorophenyl)glycinamide —— C19H17ClFN3O3S2
Rel-N~2~-(3-chlorophenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-fluorophenyl)glycinamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(2-fluorophenyl)-N-(3-methylphenyl)glycinamide —— C20H20FN3O3S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(2-fluorophenyl)-N-(3-methylphenyl)glycinamide
—— Rel-N-(5-chloro-2-methoxyphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethylphenyl)glycinamide —— C22H24ClN3O4S2
Rel-N-(5-chloro-2-methoxyphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethylphenyl)glycinamide
—— Rel-(3AR,6AR)-N-(4-chlorobenzyl)-N-(4-ethylphenyl)-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-amine 5,5-dioxide —— C20H21ClN2O2S2
Rel-(3AR,6AR)-N-(4-chlorobenzyl)-N-(4-ethylphenyl)-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-amine 5,5-dioxide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethylphenyl)-N-(4-fluorophenyl)glycinamide —— C21H22FN3O3S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethylphenyl)-N-(4-fluorophenyl)glycinamide
—— rac-N-[2-(4-chlorophenyl)-2-hydroxyethyl]-2,6-dimethyl-8-[4,4,4-trifluoro-3-(trifluoromethyl)butoxy]imidazo[1,2-a]pyridine-3-carboxamide 1609165-34-5 C23H22ClF6N3O3
rac-N-[2-(4-chlorophenyl)-2-hydroxyethyl]-2,6-dimethyl-8-[4,4,4-trifluoro-3-(trifluoromethyl)butoxy]imidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-hydroxybutyl)-2,6-dimethyl-8-[4,4,4-trifluoro-3-(trifluoromethyl)butoxy]imidazo[1,2-a]pyridine-3-carboxamide 1609165-33-4 C19H23F6N3O3
rac-N-(2-hydroxybutyl)-2,6-dimethyl-8-[4,4,4-trifluoro-3-(trifluoromethyl)butoxy]imidazo[1,2-a]pyridine-3-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-N-(1-ethoxy-3-hydroxypropan-2-yl)-2-methylimidazo[1,2-a]-pyridine-3-carboxamide 1609165-20-9 C21H23F2N3O4
rac-8-[(2,6-difluorobenzyl)oxy]-N-(1-ethoxy-3-hydroxypropan-2-yl)-2-methylimidazo[1,2-a]-pyridine-3-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(1,1,1-trifluoro-4-hydroxy-4-methylpentan-3-yl)-imidazo[1,2-a]pyridine-3-carboxamide 1609165-11-8 C22H22F5N3O3
rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(1,1,1-trifluoro-4-hydroxy-4-methylpentan-3-yl)-imidazo[1,2-a]pyridine-3-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-N-{2-hydroxy-1-[4-(methylsulphonyl)phenyl]ethyl}-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609164-85-3 C25H23F2N3O5S
rac-8-[(2,6-difluorobenzyl)oxy]-N-{2-hydroxy-1-[4-(methylsulphonyl)phenyl]ethyl}-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— Rac-6,6,6-trifluoro-5-hydroxynorleucine —— C6H10F3NO3
Rac-6,6,6-trifluoro-5-hydroxynorleucine
—— rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(7,7,7-trifluoro-2-hydroxy-2-methylheptan-3-yl)imidazo[1,2-a]pyridine-3-carboxamide 1609165-13-0 C24H26F5N3O3
rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(7,7,7-trifluoro-2-hydroxy-2-methylheptan-3-yl)imidazo[1,2-a]pyridine-3-carboxamide
—— rac-Methyl N-[(benzyloxy)carbonyl]-5,5,6,6,6-pentafluoronorleucinate —— C15H16F5NO4
rac-Methyl N-[(benzyloxy)carbonyl]-5,5,6,6,6-pentafluoronorleucinate
—— rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(6,6,6-trifluoro-1-hydroxyhexan-2-yl)imidazo[1,2-a]-pyridine-3-carboxamide 1609164-71-7 C22H22F5N3O3
rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(6,6,6-trifluoro-1-hydroxyhexan-2-yl)imidazo[1,2-a]-pyridine-3-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-N-[1-(4-fluorophenyl)-2-hydroxy-2-methylpropyl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609165-15-2 C26H24F3N3O3
rac-8-[(2,6-difluorobenzyl)oxy]-N-[1-(4-fluorophenyl)-2-hydroxy-2-methylpropyl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-methyl 2-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}-carbonyl)amino]-4,4,4-trifluorobutanoate 1609081-96-0 C21H18F5N3O4
rac-methyl 2-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}-carbonyl)amino]-4,4,4-trifluorobutanoate
—— (R)-2-((R)-1-hydroxy-19-((1S,2R)-2-((2S,18S,19S)-18-methoxy-19-methylheptatriacontan-2-yl)cyclopropyl)nonadecyl)hexacosanoic acid —— C87H172O4
(R)-2-((R)-1-hydroxy-19-((1S,2R)-2-((2S,18S,19S)-18-methoxy-19-methylheptatriacontan-2-yl)cyclopropyl)nonadecyl)hexacosanoic acid
—— rac-Methyl N-[(benzyloxy)carbonyl]-6,6,6-trifluoronorleucinate —— C15H18F3NO4
rac-Methyl N-[(benzyloxy)carbonyl]-6,6,6-trifluoronorleucinate
—— rac-N-[1-(4-chlorophenyl)-2-hydroxy-2-methylpropyl]-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609165-14-1 C26H24ClF2N3O3
rac-N-[1-(4-chlorophenyl)-2-hydroxy-2-methylpropyl]-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— (rac)-8-(cyclohexylmethoxy)-N-(1-hydroxypent-4-en-2-yl)-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609164-45-5 C21H29N3O3
(rac)-8-(cyclohexylmethoxy)-N-(1-hydroxypent-4-en-2-yl)-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-[1-(4-chlorophenyl)-2-hydroxyethyl]-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide trifluoroacetate 1609164-77-3 C2HF3O2*C24H20ClF2N3O3
rac-N-[1-(4-chlorophenyl)-2-hydroxyethyl]-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide trifluoroacetate
—— rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(6,6,6-trifluoro-2-hydroxy-2-methylhexan-3-yl)imidazo[1,2-a]pyridine-3-carboxamide 1609165-12-9 C23H24F5N3O3
rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-(6,6,6-trifluoro-2-hydroxy-2-methylhexan-3-yl)imidazo[1,2-a]pyridine-3-carboxamide
—— (R)-1-Butylpyrrolidine-2-carboxamide —— C9H18N2O
(R)-1-Butylpyrrolidine-2-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-N-(2,3-dihydro-1H-indol-3-yl)-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609340-40-0 C24H20F2N4O2
rac-8-[(2,6-difluorobenzyl)oxy]-N-(2,3-dihydro-1H-indol-3-yl)-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-Methyl 5,5,6,6,6-pentafluoronorleucinate hydrochloride —— C7H11ClF5NO2
rac-Methyl 5,5,6,6,6-pentafluoronorleucinate hydrochloride
—— rac-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethyl-N-[2-(morpholin-4-yl)propyl]imidazo[1,2-a]pyridine-3-carboxamide 1609341-52-7 C24H28F2N4O3
rac-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethyl-N-[2-(morpholin-4-yl)propyl]imidazo[1,2-a]pyridine-3-carboxamide
—— rac-tert-Butyl 2-{[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}-carbonyl)amino]methyl}-3,4-dihydroquinoline-1(2H)-carboxylate —— C32H34F2N4O4
rac-tert-Butyl 2-{[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}-carbonyl)amino]methyl}-3,4-dihydroquinoline-1(2H)-carboxylate
—— rac-tert-butyl 4-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)-amino]-3,4-dihydroquinoline-1(2H)-carboxylate 1609345-18-7 C30H30F2N4O4
rac-tert-butyl 4-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)-amino]-3,4-dihydroquinoline-1(2H)-carboxylate
—— rac-N-(2-Amino-2,4-dimethylpentyl)-2,6-dimethyl-8-[4,4,4-trifluoro-3-(trifluoromethyl)butoxy]-imidazo[1,2-a]pyridine-3-carboxamide —— C22H30F6N4O2
rac-N-(2-Amino-2,4-dimethylpentyl)-2,6-dimethyl-8-[4,4,4-trifluoro-3-(trifluoromethyl)butoxy]-imidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-aminopropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide 1609340-37-5 C20H22F2N4O2
rac-N-(2-aminopropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-Amino-1-phenylethyl)-8-(cyclohexylmethoxy)-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609340-56-8 C24H30N4O2
rac-N-(2-Amino-1-phenylethyl)-8-(cyclohexylmethoxy)-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-[2-amino-3-(benzyloxy)-2-methylpropyl]-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C27H28F2N4O3
rac-N-[2-amino-3-(benzyloxy)-2-methylpropyl]-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-Amino-2-methylpentyl)-8-[(2,6-difluorobenzyl)oxy]-7-fluoro-2-methylimidazo[1,2-a]-pyridine-3-carboxamide —— C22H25F3N4O2
rac-N-(2-Amino-2-methylpentyl)-8-[(2,6-difluorobenzyl)oxy]-7-fluoro-2-methylimidazo[1,2-a]-pyridine-3-carboxamide
—— rac-N-[2-Amino-1-(4-chlorophenyl)ethyl]-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide dihydrochloride —— C24H23Cl3F2N4O2
rac-N-[2-Amino-1-(4-chlorophenyl)ethyl]-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide dihydrochloride
—— rac-8-[(2,6-difluorobenzyl)oxy]-N-[2-(isopropylamino)ethyl]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide 1609341-49-2 C22H26F2N4O2
rac-8-[(2,6-difluorobenzyl)oxy]-N-[2-(isopropylamino)ethyl]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(3-azabicyclo[4.1.0]hept-1-yl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide 1609341-36-7 C22H22F2N4O2
rac-N-(3-azabicyclo[4.1.0]hept-1-yl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide
—— rac-N-(2-Amino-3-methoxy-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide —— C21H24F2N4O3
rac-N-(2-Amino-3-methoxy-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide
—— rac-N-[2-amino-1-(3,4-difluorophenyl)ethyl]-8-(cyclohexylmethoxy)-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609340-58-0 C24H28F2N4O2
rac-N-[2-amino-1-(3,4-difluorophenyl)ethyl]-8-(cyclohexylmethoxy)-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-Amino-4-hydroxy-2-methylbutyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C22H26F2N4O3
rac-N-(2-Amino-4-hydroxy-2-methylbutyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-amino-4,4,4-trifluorobutyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609341-62-9 C20H18ClF5N4O2
rac-N-(2-amino-4,4,4-trifluorobutyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— Rel-N-(5-chloro-2-methoxyphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)glycinamide —— C21H22ClN3O5S2
Rel-N-(5-chloro-2-methoxyphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)glycinamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethoxyphenyl)-N-(4-methylphenyl)glycinamide —— C22H25N3O4S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethoxyphenyl)-N-(4-methylphenyl)glycinamide
—— rac-N-(2-Amino-3,3,3-trifluoro-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethyl-imidazo[1,2-a]pyridine-3-carboxamide —— C21H21F5N4O2
rac-N-(2-Amino-3,3,3-trifluoro-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethyl-imidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-amino-3-methoxy-2-methylpropyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609341-75-4 C21H23ClF2N4O3
rac-N-(2-amino-3-methoxy-2-methylpropyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide