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—— (R)-N-((S)-1-(2-fluoro-4-(1H-pyrazol-4-yl)phenyl)ethyl)-2-methylpropane-2-sulfinamide —— C15H20FN3OS
(R)-N-((S)-1-(2-fluoro-4-(1H-pyrazol-4-yl)phenyl)ethyl)-2-methylpropane-2-sulfinamide
—— (R)-N-((S)-1-(5-chloro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)ethyl)-2-methylpropane-2-sulfinamide —— C13H18ClF3N2O2S
(R)-N-((S)-1-(5-chloro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)ethyl)-2-methylpropane-2-sulfinamide
—— (R)-N-(4-acetylphenyl)-3-(1-(4-fluorophenyl)ethoxy)benzamide 1616243-43-6 C23H20FNO3
(R)-N-(4-acetylphenyl)-3-(1-(4-fluorophenyl)ethoxy)benzamide
—— (R)-3-hydroxy-1-methyl-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-4-carboxamide 1429216-39-6 C17H18N2O3
(R)-3-hydroxy-1-methyl-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-4-carboxamide
—— (R)-2-methyl-N-[(Z)-(3-methylpyrazol-4-ylidene)methyl]propane-2-sulfinamide —— C9H15N3OS
(R)-2-methyl-N-[(Z)-(3-methylpyrazol-4-ylidene)methyl]propane-2-sulfinamide
—— (R)-3-hydroxy-1-methyl-N-(1-(naphthalen-2-yl)ethyl)-2-oxo-1,2-dihydropyridine-4-carboxamide 1429204-34-1 C19H18N2O3
(R)-3-hydroxy-1-methyl-N-(1-(naphthalen-2-yl)ethyl)-2-oxo-1,2-dihydropyridine-4-carboxamide
—— (R)-3-hydroxy-1-methyl-2-oxo-N-(6-(trifluoromethyl)-2,3-dihydro-1H-inden-1-yl)-1,2-dihydropyridine-4-carboxamide 1429216-41-0 C17H15F3N2O3
(R)-3-hydroxy-1-methyl-2-oxo-N-(6-(trifluoromethyl)-2,3-dihydro-1H-inden-1-yl)-1,2-dihydropyridine-4-carboxamide
—— (R)-N-(4-(2,6-dichlorophenoxy)butan-2-yl)-3-hydroxy-1-isobutyl-2-oxo-1,2-dihydropyridine-4-carboxamide 1429203-94-0 C20H24Cl2N2O4
(R)-N-(4-(2,6-dichlorophenoxy)butan-2-yl)-3-hydroxy-1-isobutyl-2-oxo-1,2-dihydropyridine-4-carboxamide
—— (R)-methyl 3-((4-((2-acrylamidophenyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)pyrrolidine-1-carboxylate 1621999-48-1 C20H21F3N6O3
(R)-methyl 3-((4-((2-acrylamidophenyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)pyrrolidine-1-carboxylate
—— (R)-tert-butyl 4-(4-((4-(2-ethoxy-2-oxoethyl)phenyl)amino)-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)-2-methylpiperazine-1-carboxylate —— C28H38N4O4
(R)-tert-butyl 4-(4-((4-(2-ethoxy-2-oxoethyl)phenyl)amino)-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)-2-methylpiperazine-1-carboxylate
—— (R)-methyl 2-(4-((2-(3-methylpiperazin-1-yl)-6,7-dihydro-5H-cyclopenta[b]pyridin-4-yl)amino)phenyl)acetate —— C22H28N4O2
(R)-methyl 2-(4-((2-(3-methylpiperazin-1-yl)-6,7-dihydro-5H-cyclopenta[b]pyridin-4-yl)amino)phenyl)acetate
—— (R)-1-(4-((2-(3-chlorophenyl)-6,7-dihydro-5H-cyclopenta[b]pyridin-4-yl)amino)phenyl)propan-2-ol 1606973-98-1 C23H23ClN2O
(R)-1-(4-((2-(3-chlorophenyl)-6,7-dihydro-5H-cyclopenta[b]pyridin-4-yl)amino)phenyl)propan-2-ol
—— (R)-1-(4-((2-(3-chlorophenyl)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino)phenyl)propan-2-ol 1606974-64-4 C22H22ClN3O
(R)-1-(4-((2-(3-chlorophenyl)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino)phenyl)propan-2-ol
—— (R)-2-(Methylsulfinyl)ethanol —— C3H8O2S
(R)-2-(Methylsulfinyl)ethanol
—— (R)-ethyl 4-(5'-fluoro-2'-methoxy-[1,1'-biphenyl]-4-yl)-3-(5-oxo-4,5-dihydro-1,3,4-oxadiazole-2-carboxamido)butanoate —— C22H22FN3O6
(R)-ethyl 4-(5'-fluoro-2'-methoxy-[1,1'-biphenyl]-4-yl)-3-(5-oxo-4,5-dihydro-1,3,4-oxadiazole-2-carboxamido)butanoate
—— (R)-6-((1-cyclopropylethyl)amino)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile —— C19H17F3N6
(R)-6-((1-cyclopropylethyl)amino)-7-(4-(trifluoromethyl)benzyl)-7H-purine-2-carbonitrile
—— (R)-(5-ethenyl-1-azabicyclo[2.2.2]octan-2-yl)-naphthalen-1-ylmethanol —— C20H23NO
(R)-(5-ethenyl-1-azabicyclo[2.2.2]octan-2-yl)-naphthalen-1-ylmethanol
—— (R)-2-methyl-N-[(1R)-6-methyl-2,3-dihydro-1H-inden-1-yl]propane-2-sulfinamide —— C14H21NOS
(R)-2-methyl-N-[(1R)-6-methyl-2,3-dihydro-1H-inden-1-yl]propane-2-sulfinamide
—— (R)-(3-((1-(5'-chloro-2'-fluoro-[1,1'-biphenyl]-4-yl)-4-((5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy)-4-oxobutan-2-yl)amino)-3-oxopropyl)phosphonic acid 1621527-41-0 C24H24ClFNO9P
(R)-(3-((1-(5'-chloro-2'-fluoro-[1,1'-biphenyl]-4-yl)-4-((5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy)-4-oxobutan-2-yl)amino)-3-oxopropyl)phosphonic acid
—— (R)-1H-benzimidazol-2-yl(furan-2-yl)methanol —— C12H10N2O2
(R)-1H-benzimidazol-2-yl(furan-2-yl)methanol
—— (R)-3-chloro-N-[4-(2-chlorophenyl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfinamide —— C22H26Cl2N2O2S
(R)-3-chloro-N-[4-(2-chlorophenyl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfinamide
—— (R)-3-Amino-3-(4-(difluoromethoxy)phenyl)propanoic acid —— C10H11F2NO3
(R)-3-Amino-3-(4-(difluoromethoxy)phenyl)propanoic acid
—— (R)-(3-((1-(5'-chloro-2'-fluoro-[1,1'-biphenyl]-4-yl)-4-oxo-4-((pivaloyloxy)methoxy)butan-2-yl)amino)-3-oxopropyl)phosphonic acid 1621527-40-9 C25H30ClFNO8P
(R)-(3-((1-(5'-chloro-2'-fluoro-[1,1'-biphenyl]-4-yl)-4-oxo-4-((pivaloyloxy)methoxy)butan-2-yl)amino)-3-oxopropyl)phosphonic acid
—— (R)-1-(4-((4-((2-acrylamidophenyl)amino)-5-chloropyrimidin-2-yl)amino)-3-cyanophenyl)pyrrolidine-2-carboxamide 1622000-88-7 C25H23ClN8O2
(R)-1-(4-((4-((2-acrylamidophenyl)amino)-5-chloropyrimidin-2-yl)amino)-3-cyanophenyl)pyrrolidine-2-carboxamide
—— rel-N-[(4aR,6R,8aS)-8a-(2,4-difluorophenyl)-6-(6-methylpyridin-3-yl)-4,4a,5,6,8,8a-hexahydropyrano[3,4-d][1,3]thiazin-2-yl]benzamide —— C26H23F2N3O2S
rel-N-[(4aR,6R,8aS)-8a-(2,4-difluorophenyl)-6-(6-methylpyridin-3-yl)-4,4a,5,6,8,8a-hexahydropyrano[3,4-d][1,3]thiazin-2-yl]benzamide
—— (R)-4-(2-acrylamido-4-methoxyphenoxy)-2-((4-(2-carbamoylpyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide 1622001-72-2 C27H29N7O6
(R)-4-(2-acrylamido-4-methoxyphenoxy)-2-((4-(2-carbamoylpyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide
—— rel-{(2R,4R,5S)-5-amino-5-(2,4-difluorophenyl)-2-(5-methylpyrazin-2-yl)tetrahydro-2H-pyran-4-yl}methanol —— C17H19F2N3O2
rel-{(2R,4R,5S)-5-amino-5-(2,4-difluorophenyl)-2-(5-methylpyrazin-2-yl)tetrahydro-2H-pyran-4-yl}methanol
—— rac-trans-4-((2-acrylamidocyclohexyl)oxy)-2-((5-(methoxycarbamoyl)-2-methylphenyl)amino)pyrimidine-5-carboxamide —— C23H28N6O5
rac-trans-4-((2-acrylamidocyclohexyl)oxy)-2-((5-(methoxycarbamoyl)-2-methylphenyl)amino)pyrimidine-5-carboxamide
—— rac-trans-4-((2-acrylamidocyclohexyl)oxy)-2-((5-carbamoyl-2-methylphenyl)amino)pyrimidine-5-carboxamide —— C22H26N6O4
rac-trans-4-((2-acrylamidocyclohexyl)oxy)-2-((5-carbamoyl-2-methylphenyl)amino)pyrimidine-5-carboxamide
—— (R)-(3-((1-(5'-chloro-2'-fluoro-[1,1'-biphenyl]-4-yl)-4-((2,3-dihydro-1H-inden-5-yl)oxy)-4-oxobutan-2-yl)amino)-3-oxopropyl)phosphonic acid 1621527-48-7 C28H28ClFNO6P
(R)-(3-((1-(5'-chloro-2'-fluoro-[1,1'-biphenyl]-4-yl)-4-((2,3-dihydro-1H-inden-5-yl)oxy)-4-oxobutan-2-yl)amino)-3-oxopropyl)phosphonic acid
—— rac-trans-4-((2-acrylamidocyclohexyl)amino)-2-((5-((2-hydroxyethoxy) carbamoyl)-2-methylphenyl)amino)pyrimidine-5-carboxamide —— C24H31N7O5
rac-trans-4-((2-acrylamidocyclohexyl)amino)-2-((5-((2-hydroxyethoxy) carbamoyl)-2-methylphenyl)amino)pyrimidine-5-carboxamide
—— (R)-N-(2-((2-((1-acetylpiperidin-3-yl)amino)-5-chloropyrimidin-4-yl)amino)phenyl)acrylamide 1622000-36-5 C20H23ClN6O2
(R)-N-(2-((2-((1-acetylpiperidin-3-yl)amino)-5-chloropyrimidin-4-yl)amino)phenyl)acrylamide
—— (R)-N-(2-((5-chloro-2-((2-cyano-4-(2-(hydroxymethyl)pyrrolidin-1-yl)phenyl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide 1622000-82-1 C25H24ClN7O2
(R)-N-(2-((5-chloro-2-((2-cyano-4-(2-(hydroxymethyl)pyrrolidin-1-yl)phenyl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide
—— (R)-N-(2-((5-chloro-2-((2-cyano-4-(2-(hydroxymethyl)pyrrolidin-1-yl)phenyl)amino)pyrimidin-4-yl)amino)-5-methoxyphenyl)acrylamide 1622000-90-1 C26H26ClN7O3
(R)-N-(2-((5-chloro-2-((2-cyano-4-(2-(hydroxymethyl)pyrrolidin-1-yl)phenyl)amino)pyrimidin-4-yl)amino)-5-methoxyphenyl)acrylamide
—— rac-trans-4-((2-acrylamidocyclohexyl)amino)-2-((5-(methoxycarbamoyl)-2-methylphenyl)amino)pyrimidine-5-carboxamide —— C23H29N7O4
rac-trans-4-((2-acrylamidocyclohexyl)amino)-2-((5-(methoxycarbamoyl)-2-methylphenyl)amino)pyrimidine-5-carboxamide
—— rac-cis-N-(2-((5-chloro-2-((3-(hydroxymethyl)cyclohexyl)amino) pyrimidin-4-yl)amino)phenyl)acrylamide —— C20H24ClN5O2
rac-cis-N-(2-((5-chloro-2-((3-(hydroxymethyl)cyclohexyl)amino) pyrimidin-4-yl)amino)phenyl)acrylamide
—— (R)-N-(5-methyl-2-((5-(trifluoromethyl)-2-((1-(vinylsulfonyl)pyrrolidin-3-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide 1621999-55-0 C21H23F3N6O3S
(R)-N-(5-methyl-2-((5-(trifluoromethyl)-2-((1-(vinylsulfonyl)pyrrolidin-3-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide
—— (R)-4-hydroxy-1-methyl-5-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-95-5 C16H18N2O3
(R)-4-hydroxy-1-methyl-5-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-4-(2-acrylamido-4-methoxyphenoxy)-2-((4-(2-(hydroxymethyl)pyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide 1622001-74-4 C27H30N6O6
(R)-4-(2-acrylamido-4-methoxyphenoxy)-2-((4-(2-(hydroxymethyl)pyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide
—— (R)-N-(2-((2-((1-acetylpyrrolidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)acrylamide 1621999-47-0 C20H21F3N6O2
(R)-N-(2-((2-((1-acetylpyrrolidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)acrylamide
—— (R)-1-(4-((4-((2-acrylamido-4-methoxyphenyl)amino)-5-chloropyrimidin-2-yl)amino)-3-cyanophenyl)pyrrolidine-2-carboxamide 1622000-89-8 C26H25ClN8O3
(R)-1-(4-((4-((2-acrylamido-4-methoxyphenyl)amino)-5-chloropyrimidin-2-yl)amino)-3-cyanophenyl)pyrrolidine-2-carboxamide
—— (R)-4-hydroxy-1-methyl-N-(1-(4’-(methylsulfonyl)biphenyl-3-yl)ethyl)-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-42-2 C21H22N2O5S
(R)-4-hydroxy-1-methyl-N-(1-(4’-(methylsulfonyl)biphenyl-3-yl)ethyl)-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(1-(3'-carbamoylbiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-46-6 C21H21N3O4
(R)-N-(1-(3'-carbamoylbiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(1-(3',5'-dichlorobiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-33-1 C20H18Cl2N2O3
(R)-N-(1-(3',5'-dichlorobiphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— rac-trans-4-((2-acrylamidocyclohexyl)amino)-2-((5-carbamoyl-2-methylphenyl)amino)pyrimidine-5-carboxamide —— C22H27N7O3
rac-trans-4-((2-acrylamidocyclohexyl)amino)-2-((5-carbamoyl-2-methylphenyl)amino)pyrimidine-5-carboxamide
—— (R)-N-(5-bromo-2,3-dihydro-1H-inden-1-yl)-1-ethyl-4-hydroxy-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-83-1 C16H17BrN2O3
(R)-N-(5-bromo-2,3-dihydro-1H-inden-1-yl)-1-ethyl-4-hydroxy-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(2-((2-((1-(2-hydroxyacetyl)pyrrolidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)acrylamide 1621999-49-2 C20H21F3N6O3
(R)-N-(2-((2-((1-(2-hydroxyacetyl)pyrrolidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)acrylamide
—— [(R)-[5-chloro-2-[(3,4,5-trimethoxybenzoyl)amino]phenyl]-phenylmethyl]-(2-hydrazinyl-2-oxoethyl)azanium —— C25H28ClN4O5+
[(R)-[5-chloro-2-[(3,4,5-trimethoxybenzoyl)amino]phenyl]-phenylmethyl]-(2-hydrazinyl-2-oxoethyl)azanium
—— (R)-N-( 1-(4’-(dimethylcarbamoyl)biphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-45-5 C23H25N3O4
(R)-N-( 1-(4’-(dimethylcarbamoyl)biphenyl-3-yl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide
—— (R)-N-(1-(3-(3-chloropyridin-4-yl)phenyl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide 1429344-51-3 C19H18ClN3O3
(R)-N-(1-(3-(3-chloropyridin-4-yl)phenyl)ethyl)-4-hydroxy-1-methyl-5-oxo-2,5-dihydro-1H-pyrrole-3-carboxamide