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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-5-methoxy-2-(2-((pyridin-3-yloxy)methyl)piperazin-1-yl)benzo[d]oxazole hydrochloride —— C18H20N4O3*ClH
(R)-5-methoxy-2-(2-((pyridin-3-yloxy)methyl)piperazin-1-yl)benzo[d]oxazole hydrochloride
—— rel-(3R,3aR,5R,7aS)-5-cyclopropyl-7a-(2,4-difluorophenyl)-3-(fluoromethyl)hexahydro-1H-pyrano[3,4-c][1,2]oxazole —— C16H18F3NO2
rel-(3R,3aR,5R,7aS)-5-cyclopropyl-7a-(2,4-difluorophenyl)-3-(fluoromethyl)hexahydro-1H-pyrano[3,4-c][1,2]oxazole
—— rel-N-({(3S,4R,6R)-6-cyclopropyl-3-(2,4-difluorophenyl)-4-[(1R)-2-fluoro-1-hydroxyethyl]tetrahydro-2H-pyran-3-yl}carbamothioyl)benzamide —— C24H25F3N2O3S
rel-N-({(3S,4R,6R)-6-cyclopropyl-3-(2,4-difluorophenyl)-4-[(1R)-2-fluoro-1-hydroxyethyl]tetrahydro-2H-pyran-3-yl}carbamothioyl)benzamide
—— rel-(3aR,5S,7aS)-5-(Cyclopropylmethyl)-7a-(2,4-difluorophenyl) hexahydro-1H-pyrano[3,4-c][1,2]oxazole —— C16H19F2NO2
rel-(3aR,5S,7aS)-5-(Cyclopropylmethyl)-7a-(2,4-difluorophenyl) hexahydro-1H-pyrano[3,4-c][1,2]oxazole
—— rel-(3R,3aR,5R)-5-cyclopropyl-3-(methoxymethyl)-3,3a,4,5-tetrahydro-7H-pyrano[3,4-c][1,2]oxazole —— C11H17NO3
rel-(3R,3aR,5R)-5-cyclopropyl-3-(methoxymethyl)-3,3a,4,5-tetrahydro-7H-pyrano[3,4-c][1,2]oxazole
—— (R)-N-[(E,2S)-2-(2,4-difluorophenyl)-5-methyl-4-oxohept-5-en-2-yl]-2-methylpropane-2-sulfinamide —— C18H25F2NO2S
(R)-N-[(E,2S)-2-(2,4-difluorophenyl)-5-methyl-4-oxohept-5-en-2-yl]-2-methylpropane-2-sulfinamide
—— rel-N-[(4aR,6R,8aS)-6-cyclopropyl-8a-(2,4-difluorophenyl)-4,4a,5,6,8,8a-hexahydropyrano[3,4-d][1,3]thiazin-2-yl]benzamide —— C23H22F2N2O2S
rel-N-[(4aR,6R,8aS)-6-cyclopropyl-8a-(2,4-difluorophenyl)-4,4a,5,6,8,8a-hexahydropyrano[3,4-d][1,3]thiazin-2-yl]benzamide
—— rel-(1R)-1-[(2R,4R,5S)-5-amino-2-cyclopropyl-5-(2,4-difluorophenyl)tetrahydro-2H-pyran-4-yl]-2-methoxyethanol —— C17H23F2NO3
rel-(1R)-1-[(2R,4R,5S)-5-amino-2-cyclopropyl-5-(2,4-difluorophenyl)tetrahydro-2H-pyran-4-yl]-2-methoxyethanol
—— (R)-N-(4-cyanophenyl)-5-(1-(4-fluorophenyl)ethoxy)nicotinamide 1616242-54-6 C21H16FN3O2
(R)-N-(4-cyanophenyl)-5-(1-(4-fluorophenyl)ethoxy)nicotinamide
—— (R)-1-(2-(2-((6-(azetidine-1-carbonyl)pyridin-3-yl)oxy)-5-nitrophenyl)pyrrolidin-1-yl)ethanone 1616280-94-4 C21H22N4O5
(R)-1-(2-(2-((6-(azetidine-1-carbonyl)pyridin-3-yl)oxy)-5-nitrophenyl)pyrrolidin-1-yl)ethanone
—— (R)-5-(1-(4-acetylphenyl)ethoxy)-N-(4-cyanophenyl)nicotinamide 1616242-97-7 C23H19N3O3
(R)-5-(1-(4-acetylphenyl)ethoxy)-N-(4-cyanophenyl)nicotinamide
—— (R)-5-(1-(4-acetylphenyl)ethoxy)-N-(4-bromophenyl)nicotinamide 1616243-42-5 C22H19BrN2O3
(R)-5-(1-(4-acetylphenyl)ethoxy)-N-(4-bromophenyl)nicotinamide
—— (R)-N-(4-cyanophenyl)-3-(1-(4-fluorophenyl)ethoxy)benzamide 1616242-42-2 C22H17FN2O2
(R)-N-(4-cyanophenyl)-3-(1-(4-fluorophenyl)ethoxy)benzamide
—— rac-2-[(Diphenylmethylene)amino]-4-fluoro-2-methylbutanonitrile —— C18H17FN2
rac-2-[(Diphenylmethylene)amino]-4-fluoro-2-methylbutanonitrile
—— (R,R,S,R,S)-N,N'-((ethane-1,2-diylbis(oxy))bis(ethane-2,1-diyl))bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide) 1616111-58-0 C32H44N2O14
(R,R,S,R,S)-N,N'-((ethane-1,2-diylbis(oxy))bis(ethane-2,1-diyl))bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide)
—— (R,R,S,R,S)-N,N'-(hexane-1,6-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide) 1616111-55-7 C32H44N2O12
(R,R,S,R,S)-N,N'-(hexane-1,6-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide)
—— (R,R,S,R,S)-N,N'-(octane-1,8-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide) 1616111-57-9 C34H48N2O12
(R,R,S,R,S)-N,N'-(octane-1,8-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide)
—— (R,R,S,R,S)-N,N'-(ethane-1,2-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide) 1616111-51-3 C28H36N2O12
(R,R,S,R,S)-N,N'-(ethane-1,2-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide)
—— (R,R,S,R,S)-N,N'-(propane-1,3-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide) 1616111-52-4 C29H38N2O12
(R,R,S,R,S)-N,N'-(propane-1,3-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide)
—— (R,R,S,R,S)-N,N'-(heptane-1,7-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide) 1616111-56-8 C33H46N2O12
(R,R,S,R,S)-N,N'-(heptane-1,7-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide)
—— (R,R,S,R,S)-N,N'-(pentane-1,5-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide) 1616111-54-6 C31H42N2O12
(R,R,S,R,S)-N,N'-(pentane-1,5-diyl)bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide)
—— (R,R,S,R,S)-N,N'-(methylenebis(4,1-phenylene))bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide) 1616111-59-1 C39H42N2O12
(R,R,S,R,S)-N,N'-(methylenebis(4,1-phenylene))bis(3-((2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)benzamide)
—— (R)-bis(2-methylpropoxy)phosphoryl-(2-fluorophenyl)methanol —— C15H24FO4P
(R)-bis(2-methylpropoxy)phosphoryl-(2-fluorophenyl)methanol
—— (R)-2,6-difluoro-N-(6-(4-(4-fluorophenyl)-1-(1-(3,3,3-trifluoro-2-hydroxypropyI)piperidin-4-yl)-1H-imidazol-5-yl)imidazo[1,2-b]pyridazin-2-yl)isonicotinamide 1615721-63-5 C29H24F6N8O2
(R)-2,6-difluoro-N-(6-(4-(4-fluorophenyl)-1-(1-(3,3,3-trifluoro-2-hydroxypropyI)piperidin-4-yl)-1H-imidazol-5-yl)imidazo[1,2-b]pyridazin-2-yl)isonicotinamide
—— ((R)-2-Benzyloxycarbonylamino-3-methyl-butyrylamino)-acetic acid tert-butyl ester 65443-45-0 C19H28N2O5
((R)-2-Benzyloxycarbonylamino-3-methyl-butyrylamino)-acetic acid tert-butyl ester
—— (R)-4-[2-(2,3-dihydro-pyrrolo[2,3-b]pyridin-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester 1403899-91-1 C19H28N4O3
(R)-4-[2-(2,3-dihydro-pyrrolo[2,3-b]pyridin-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester
—— (R)-2-fluoro-N-(6-(3-(4-fluorophenyl)-1-methyl-5-(1-(3,3,3-trifluoro-2-hydroxypropyl)piperidin-4-yl)-1H-pyrazol-4-yl)imidazo[1,2-b]pyridazin-2-yl)isonicotinamide 1616234-84-4 C30H27F5N8O2
(R)-2-fluoro-N-(6-(3-(4-fluorophenyl)-1-methyl-5-(1-(3,3,3-trifluoro-2-hydroxypropyl)piperidin-4-yl)-1H-pyrazol-4-yl)imidazo[1,2-b]pyridazin-2-yl)isonicotinamide
—— (R)-2-hydroxy-2-((R)-3-oxo-4-(6-(trifluoromethyl)pyridin-2-yl)morpholin-2-yl)propanoic anhydride —— C26H24F6N4O9
(R)-2-hydroxy-2-((R)-3-oxo-4-(6-(trifluoromethyl)pyridin-2-yl)morpholin-2-yl)propanoic anhydride
—— (R)-4-((1-cyclobutylethyl)amino)-7-methyl-6-(m-tolyl)-5-(4-(trifluoromethyl)benzyl)-5H-pyrrolo[3,2-d]pyrimidine-2-carbonitrile —— C29H28F3N5
(R)-4-((1-cyclobutylethyl)amino)-7-methyl-6-(m-tolyl)-5-(4-(trifluoromethyl)benzyl)-5H-pyrrolo[3,2-d]pyrimidine-2-carbonitrile
—— racemic 2-bromo-4-(5-chloropyridin-3-yl)-3-[1-(trans-4-methylcyclohexyl)ethyl]-3H-imidazo[4,5-c]pyridine-6-carbonitrile —— C21H21BrClN5
racemic 2-bromo-4-(5-chloropyridin-3-yl)-3-[1-(trans-4-methylcyclohexyl)ethyl]-3H-imidazo[4,5-c]pyridine-6-carbonitrile
—— rac-(3aR,4S,9bS)-6,8-dichloro-3H,3aH,4H,5H,9bH-cyclopenta[c]quinoline-4-carboxylic acid —— C13H11Cl2NO2
rac-(3aR,4S,9bS)-6,8-dichloro-3H,3aH,4H,5H,9bH-cyclopenta[c]quinoline-4-carboxylic acid
—— racemic 4-(5-chloropyridin-3-yl)-2-(ethoxy(phenyl)methyl)-3-((trans-4-methylcyclohexyl)methyl)-3H-imidazo[4,5-c]pyridine-6-carbonitrile —— C29H30ClN5O
racemic 4-(5-chloropyridin-3-yl)-2-(ethoxy(phenyl)methyl)-3-((trans-4-methylcyclohexyl)methyl)-3H-imidazo[4,5-c]pyridine-6-carbonitrile
—— racemic 4-(5-chloropyridin-3-yl)-3-[1-(trans-4-methylcyclohexyl)ethyl]-3H-imidazo[4,5-c]pyridine-6-carbonitrile —— C21H22ClN5
racemic 4-(5-chloropyridin-3-yl)-3-[1-(trans-4-methylcyclohexyl)ethyl]-3H-imidazo[4,5-c]pyridine-6-carbonitrile
—— racemic 4-(5-chloropyridin-3-yl)-2-(cyclopentyl(ethoxy)methyl)-3-((trans-4-methylcyclohexyl)methyl)-3H-imidazo[4,5-c]pyridine-6-carbonitrile —— C28H34ClN5O
racemic 4-(5-chloropyridin-3-yl)-2-(cyclopentyl(ethoxy)methyl)-3-((trans-4-methylcyclohexyl)methyl)-3H-imidazo[4,5-c]pyridine-6-carbonitrile
—— [(R)-(4-chlorophenyl)-phenylmethyl]-[(2R)-4-methyl-4-(5-methylfuran-2-yl)pentan-2-yl]azanium —— C24H29ClNO+
[(R)-(4-chlorophenyl)-phenylmethyl]-[(2R)-4-methyl-4-(5-methylfuran-2-yl)pentan-2-yl]azanium
—— [(R)-(4-chlorophenyl)-phenylmethyl]-[(2S)-4-methyl-4-(5-methylfuran-2-yl)pentan-2-yl]azanium —— C24H29ClNO+
[(R)-(4-chlorophenyl)-phenylmethyl]-[(2S)-4-methyl-4-(5-methylfuran-2-yl)pentan-2-yl]azanium
—— rac-(4aR,7aS)-hexahydro-2H-furo[3,4-b]morpholine —— C6H11NO2
rac-(4aR,7aS)-hexahydro-2H-furo[3,4-b]morpholine
—— (R)-2-fluoro-5-(1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamido)pyridine 1-oxide 1616084-98-0 C23H27FN8O2
(R)-2-fluoro-5-(1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamido)pyridine 1-oxide
—— (R)-5-(3,5-dimethylisoxazol-4-yl)-1-(1-(4-fluorophenyl)ethyl)pyridin-2(1H)-one 1616401-08-1 C18H17FN2O2
(R)-5-(3,5-dimethylisoxazol-4-yl)-1-(1-(4-fluorophenyl)ethyl)pyridin-2(1H)-one
—— (R)-2,4-diamino-6-((1-(5-chloro-3-(3,5-difluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-2-methoxyethyl)amino)pyrimidine-5-carbonitrile 1615253-01-4 C22H17ClF2N8O2
(R)-2,4-diamino-6-((1-(5-chloro-3-(3,5-difluorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-2-methoxyethyl)amino)pyrimidine-5-carbonitrile
—— (R)-6-(3,5-dimethylisoxazol-4-yl)-2-(1-phenylethyl)pyridazin-3(2H)-one 1616401-05-8 C17H17N3O2
(R)-6-(3,5-dimethylisoxazol-4-yl)-2-(1-phenylethyl)pyridazin-3(2H)-one
—— (R)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((R)-pyrrolidin-3-yl)pyrrolidine-2-carboxamide 1616083-96-5 C22H32N8O
(R)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((R)-pyrrolidin-3-yl)pyrrolidine-2-carboxamide
—— (R)-(3-aminoazetidin-1-yl)(1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidin-2-yl)methanone 1616084-00-4 C21H30N8O
(R)-(3-aminoazetidin-1-yl)(1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidin-2-yl)methanone
—— (R)-5-(3,5-Dimethylisoxazol-4-yl)-1-(1-phenylethyl)pyridin-2(1H)-one 1616401-31-0 C18H18N2O2
(R)-5-(3,5-Dimethylisoxazol-4-yl)-1-(1-phenylethyl)pyridin-2(1H)-one
—— (R)-N-(6-fluoropyridin-3-yl)-1-(4-(3-isopropyl-1H-pyrazol-5-ylamino)-6,6-dimethyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide 1616084-74-2 C25H31FN8O
(R)-N-(6-fluoropyridin-3-yl)-1-(4-(3-isopropyl-1H-pyrazol-5-ylamino)-6,6-dimethyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide
—— (R)-N-(6-fluoropyridin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-4-oxopyrrolidine-2-carboxamide 1616085-48-3 C23H25FN8O2
(R)-N-(6-fluoropyridin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-4-oxopyrrolidine-2-carboxamide
—— (R)-N-(6-fluoropyridin-3-yl)-1-(4-(1-hydroxy-5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide 1616085-42-7 C23H27FN8O2
(R)-N-(6-fluoropyridin-3-yl)-1-(4-(1-hydroxy-5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide
—— (R)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((R)-piperidin-3-yl)pyrrolidine-2-carboxamide 1616084-06-0 C23H34N8O
(R)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((R)-piperidin-3-yl)pyrrolidine-2-carboxamide
—— (R)-N-(6-fluoropyridin-3-yl)-1-(4-(5-(2-hydroxypropan-2-yl)-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide 1616085-38-1 C23H27FN8O2
(R)-N-(6-fluoropyridin-3-yl)-1-(4-(5-(2-hydroxypropan-2-yl)-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide
—— (R)-N-(6-aminopyridin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide 1616085-32-5 C23H29N9O
(R)-N-(6-aminopyridin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide