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—— (R)-N-((S)-1-(1-(4-chlorophenyl)-2-methyl-1H-imidazol-4-yl)ethyl)-2-methylpropane-2-sulfinamide —— C16H22ClN3OS
(R)-N-((S)-1-(1-(4-chlorophenyl)-2-methyl-1H-imidazol-4-yl)ethyl)-2-methylpropane-2-sulfinamide
—— (R)-3-(2-{1-[3-(2,4-dichlorophenyl)isoxazol-5-yl]ethylamino}-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C20H18Cl2FN5O4
(R)-3-(2-{1-[3-(2,4-dichlorophenyl)isoxazol-5-yl]ethylamino}-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R,E)-2-methyl-N-((5-phenylthiophen-2-yl)methylene)propane-2-sulfinamide —— C15H17NOS2
(R,E)-2-methyl-N-((5-phenylthiophen-2-yl)methylene)propane-2-sulfinamide
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(6-chloro-2-((S)-1-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C25H30ClFN6O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(6-chloro-2-((S)-1-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C25H30F2N6O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-(4-fluorophenyl)isoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C24H27ClFN5O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-(4-fluorophenyl)isoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(4-chlorophenyl)isoxazol-5-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C24H27ClFN5O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(4-chlorophenyl)isoxazol-5-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-(1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C24H28F2N6O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-(1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-((1-(4-(4-chlorophenyl)-5-methylthiazol-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C21H22ClN5O3S
(R)-3-(2-((1-(4-(4-chlorophenyl)-5-methylthiazol-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(5-(3-methyl-4-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C23H23F3N6O3
(R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(5-(3-methyl-4-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-(1-methylcyclopropyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C25H33FN4O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-(1-methylcyclopropyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-((1-(5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C19H19FN6O4
(R)-3-(2-((1-(5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(5-fluoro-2-(((S)-1-(2-fluoro-4-(2-hydroxypropan-2-yl)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C24H32F2N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(5-fluoro-2-(((S)-1-(2-fluoro-4-(2-hydroxypropan-2-yl)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(5-(4-chlorophenyl)isoxazol-3-yl)ethyl)amino)-6-(fluoromethyl)pyrimidin-4-yl)oxazolidin-2-one —— C25H29ClFN5O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(5-(4-chlorophenyl)isoxazol-3-yl)ethyl)amino)-6-(fluoromethyl)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-{2-[1-(5-benzyl-[1,2,4]-oxadiazol-3-yl)ethylamino]-5-fluoropyrimidin-4-yl}-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C20H21FN6O4
(R)-3-{2-[1-(5-benzyl-[1,2,4]-oxadiazol-3-yl)ethylamino]-5-fluoropyrimidin-4-yl}-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(5-(4-chlorophenyl)isoxazol-3-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one —— C25H30ClN5O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(5-(4-chlorophenyl)isoxazol-3-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-{1-[3-(3,4-dichlorophenyl)isoxazol-5-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C20H19Cl2N5O4
(R)-3-(2-{1-[3-(3,4-dichlorophenyl)isoxazol-5-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(2,5-difluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C25H29ClF2N6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(2,5-difluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-isopropylphenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C24H33FN4O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-isopropylphenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2,5-difluoro-4-(2,2,2-trifluoroethoxy)phenyl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one —— C24H29F5N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2,5-difluoro-4-(2,2,2-trifluoroethoxy)phenyl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(6-chloro-2-((S)-1-(2-fluoro-4-(trifluoromethyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C22H25ClF4N4O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(6-chloro-2-((S)-1-(2-fluoro-4-(trifluoromethyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R,E)-N-((1-(4-chlorophenyl)-2-methyl-1H-imidazol-4-yl)methylene)-2-methylpropane-2-sulfinamide —— C15H18ClN3OS
(R,E)-N-((1-(4-chlorophenyl)-2-methyl-1H-imidazol-4-yl)methylene)-2-methylpropane-2-sulfinamide
—— (R)-3-(2-((1-(3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C19H19FN6O4
(R)-3-(2-((1-(3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-3-(2-((1-(5-(2-fluoro-3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C22H20F4N6O3
(R)-3-(2-((1-(5-(2-fluoro-3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(5-(m-tolyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C20H22N6O4
(R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(5-(m-tolyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(5-(4-chlorophenyl)isoxazol-3-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C24H27ClFN5O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(5-(4-chlorophenyl)isoxazol-3-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-2-methyl-N-((S)-1-(1-(6-(trifluoromethyl)pyridin-3-yl)-1H-pyrazol-3-yl)ethyl)propane-2-sulfinamide —— C15H19F3N4OS
(R)-2-methyl-N-((S)-1-(1-(6-(trifluoromethyl)pyridin-3-yl)-1H-pyrazol-3-yl)ethyl)propane-2-sulfinamide
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-2-methyl-1H-imidazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C25H31ClN6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-2-methyl-1H-imidazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl)ethylamino)-6-(trifluoromethyl)pyrimidin-4-yl)oxazolidin-2-one —— C24H26ClF3N6O4
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl)ethylamino)-6-(trifluoromethyl)pyrimidin-4-yl)oxazolidin-2-one
—— (R,E)-2-methyl-N-((2-(pyridin-2-yl)thiazol-5-yl)methylene)propane-2-sulfinamide —— C13H15N3OS2
(R,E)-2-methyl-N-((2-(pyridin-2-yl)thiazol-5-yl)methylene)propane-2-sulfinamide
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C25H31FN6O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C23H28ClN7O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(5-fluoro-2-((1-(5-(3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C22H20F4N6O3
(R)-3-(5-fluoro-2-((1-(5-(3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-3-(2-((1-(5-(3,4-dichlorophenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C21H20Cl2N6O3
(R)-3-(2-((1-(5-(3,4-dichlorophenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-3-(2-((1-(5-(3,4-dichlorophenyl)pyrimidin-2-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C21H19Cl2FN6O3
(R)-3-(2-((1-(5-(3,4-dichlorophenyl)pyrimidin-2-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(2-(4-chlorophenyl)thiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C24H27Cl2N5O3S
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(2-(4-chlorophenyl)thiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R,E)-2-methyl-N-((2-(pyridin-4-yl)thiazol-5-yl)methylene)propane-2-sulfinamide —— C13H15N3OS2
(R,E)-2-methyl-N-((2-(pyridin-4-yl)thiazol-5-yl)methylene)propane-2-sulfinamide
—— (R)-3-(2-{1-[3-(2,4-dichlorophenyl)isoxazol-5-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C20H19Cl2N5O4
(R)-3-(2-{1-[3-(2,4-dichlorophenyl)isoxazol-5-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C24H29ClN6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-((1-(5-(4-chloro-3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C22H20ClF3N6O3
(R)-3-(2-((1-(5-(4-chloro-3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-3-(2-{1-[5-(3-fluorophenyl)-[1,3,4]-oxadiazol-2-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C19H19FN6O4
(R)-3-(2-{1-[5-(3-fluorophenyl)-[1,3,4]-oxadiazol-2-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-2-methyl-N-((S)-1-(2-(6-methylpyridin-3-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide —— C15H21N3OS2
(R)-2-methyl-N-((S)-1-(2-(6-methylpyridin-3-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide
—— (R)-2-methyl-N-((R)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethyl)propane-2-sulfinamide —— C14H25N3O3S
(R)-2-methyl-N-((R)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethyl)propane-2-sulfinamide
—— (R,E)-2-methyl-N-((2-morpholinothiazol-5-yl)methylene)propane-2-sulfinamide —— C12H19N3O2S2
(R,E)-2-methyl-N-((2-morpholinothiazol-5-yl)methylene)propane-2-sulfinamide
—— (R)-2-methyl-N-((S)-1-(2-morpholinothiazol-5-yl)ethyl)propane-2-sulfinamide —— C13H23N3O2S2
(R)-2-methyl-N-((S)-1-(2-morpholinothiazol-5-yl)ethyl)propane-2-sulfinamide
—— (R)-N-((S)-1-(1-(4-fluorophenyl)-1H-pyrazol-4-yl)ethyl)-2-methylpropane-2-sulfinamide —— C15H20FN3OS
(R)-N-((S)-1-(1-(4-fluorophenyl)-1H-pyrazol-4-yl)ethyl)-2-methylpropane-2-sulfinamide
—— (R,E)-2-methyl-N-((2-(2-(trifluoromethyl)pyridin-4-yl)thiazol-5-yl)methylene)propane-2-sulfinamide —— C14H14F3N3OS2
(R,E)-2-methyl-N-((2-(2-(trifluoromethyl)pyridin-4-yl)thiazol-5-yl)methylene)propane-2-sulfinamide
—— (R)-methyl 2-(4-((2-formyl-5-oxopyrrolidin-1-yl)methyl)phenyl)acetate —— C15H17NO4
(R)-methyl 2-(4-((2-formyl-5-oxopyrrolidin-1-yl)methyl)phenyl)acetate
—— (R,E)-2-methyl-N-((2-(pyridin-3-yl)thiazol-5-yl)methylene)propane-2-sulfinamide —— C13H15N3OS2
(R,E)-2-methyl-N-((2-(pyridin-3-yl)thiazol-5-yl)methylene)propane-2-sulfinamide
—— (R)-2-methyl-N-((S)-1-(5-(pyridin-2-yl)thiophen-2-yl)ethyl)propane-2-sulfinamide —— C15H20N2OS2
(R)-2-methyl-N-((S)-1-(5-(pyridin-2-yl)thiophen-2-yl)ethyl)propane-2-sulfinamide