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—— (R)-N-(6-hydroxypyridin-3-yl)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide 1616085-04-1 C23H28N8O2
(R)-N-(6-hydroxypyridin-3-yl)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide
—— (R)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((S)-piperidin-3-yl)pyrrolidine-2-carboxamide 1616084-08-2 C23H34N8O
(R)-1-(4-((5-isopropyl-1H-pyrazol-3-yl)amino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((S)-piperidin-3-yl)pyrrolidine-2-carboxamide
—— (R,R)-N-(1-acetylpyrrolidin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide 1616085-50-7 C24H34N8O2
(R,R)-N-(1-acetylpyrrolidin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide
—— (R)-N-(1-phenylethyl)-(R)-2-(2,4-dichlorophenoxy)propionamide —— C17H17Cl2NO2
(R)-N-(1-phenylethyl)-(R)-2-(2,4-dichlorophenoxy)propionamide
—— (R)-4-(4-amino-6-chloropyrimidin-5-yl)but-3-yn-2-ol 1615681-07-6 C8H8ClN3O
(R)-4-(4-amino-6-chloropyrimidin-5-yl)but-3-yn-2-ol
—— Rac-1,2-dimethylcyclobutane-1,2-diamine dihydrochloride —— C6H16Cl2N2
Rac-1,2-dimethylcyclobutane-1,2-diamine dihydrochloride
—— rac-N-[2-amino-3-(4-fluorophenyl)-2-methylpropyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C27H27F3N4O2
rac-N-[2-amino-3-(4-fluorophenyl)-2-methylpropyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-amino-2-cyanoethyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C20H19F2N5O2
rac-N-(2-amino-2-cyanoethyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-8-[(2,6-Difluorobenzyl)oxy]-2,6-dimethyl-N-(morpholin-2-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide —— C22H24F2N4O3
rac-8-[(2,6-Difluorobenzyl)oxy]-2,6-dimethyl-N-(morpholin-2-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
—— Rac-tert-butyl 3-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbon-yl)amino]azepane-1-carboxylate trifluoroacetate —— C30H35F5N4O6
Rac-tert-butyl 3-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbon-yl)amino]azepane-1-carboxylate trifluoroacetate
—— rac-N-(2-amino-2-methylpentyl)-2,6-dimethyl-8-[(2,3,5,6-tetrafluorobenzyl)oxy]imidazo[1,2-a]pyridine-3-carboxamide —— C23H26F4N4O2
rac-N-(2-amino-2-methylpentyl)-2,6-dimethyl-8-[(2,3,5,6-tetrafluorobenzyl)oxy]imidazo[1,2-a]pyridine-3-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-N-(5,5-difluoropiperidin-3-yl)-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C22H22F4N4O2
rac-8-[(2,6-difluorobenzyl)oxy]-N-(5,5-difluoropiperidin-3-yl)-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— (R)-2-(1-amino-2-methoxyethyl)-5-chloro-3-(3,5-difluorophenyl)quinazolin-4(3H)-one 1615256-14-8 C17H14ClF2N3O2
(R)-2-(1-amino-2-methoxyethyl)-5-chloro-3-(3,5-difluorophenyl)quinazolin-4(3H)-one
—— rac-N-(2-amino-3-fluoro-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide Formate —— C22H25F3N4O4
rac-N-(2-amino-3-fluoro-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide Formate
—— rac-tert-Butyl 4-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-3,3-difluoropiperidine-1-carboxylate —— C27H30F4N4O4
rac-tert-Butyl 4-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-3,3-difluoropiperidine-1-carboxylate
—— rac-N-[(4-benzylmorpholin-2-yl)methyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C29H30F2N4O3
rac-N-[(4-benzylmorpholin-2-yl)methyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-tert-Butyl 3-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-4-fluoropyrrolidine-1-carboxylate Trifluoroacetate —— C28H30F6N4O6
rac-tert-Butyl 3-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-4-fluoropyrrolidine-1-carboxylate Trifluoroacetate
—— rac-N-(2-amino-2-methylpentyl)-8-[(2,3-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C23H28F2N4O2
rac-N-(2-amino-2-methylpentyl)-8-[(2,3-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-amino-2-methylpentyl)-8-[(2-chlorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C23H29ClN4O2
rac-N-(2-amino-2-methylpentyl)-8-[(2-chlorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-2-Methyl-3-[1-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]propane-1,2-diamine —— C10H16N6O
rac-2-Methyl-3-[1-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]propane-1,2-diamine
—— rac-N-(3-amino-2,2-dimethylcyclopropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C22H24F2N4O2
rac-N-(3-amino-2,2-dimethylcyclopropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethyl-N-[2-(trifluoromethyl)piperidin-4-yl]imidazo[1,2-a]pyridine-3-carboxamide —— C23H23F5N4O2
rac-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethyl-N-[2-(trifluoromethyl)piperidin-4-yl]imidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-amino-2-methylpentyl)-8-(benzyloxy)-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C23H30N4O2
rac-N-(2-amino-2-methylpentyl)-8-(benzyloxy)-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-tert-Butyl 5-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-3,3-difluoropiperidine-1-carboxylate —— C27H30F4N4O4
rac-tert-Butyl 5-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-3,3-difluoropiperidine-1-carboxylate
—— rac-N-(2-amino-2-methylpentyl)-2,6-dimethyl-8-[(2,3,6-trifluorobenzyl)oxy]imidazo[1,2-a]pyridine-3-carboxamide —— C23H27F3N4O2
rac-N-(2-amino-2-methylpentyl)-2,6-dimethyl-8-[(2,3,6-trifluorobenzyl)oxy]imidazo[1,2-a]pyridine-3-carboxamide
—— rac-2-Amino-2-methyl-3-[1-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]propanonitrile —— C10H12N6O
rac-2-Amino-2-methyl-3-[1-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]propanonitrile
—— Rac-tert-butyl 3-{[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]methyl}thiomorpholine-4-carboxylate —— C27H32F2N4O4S
Rac-tert-butyl 3-{[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]methyl}thiomorpholine-4-carboxylate
—— rac-3-(1,3-Benzothiazol-2-yl)-2-methylpropane-1,2-diamine —— C11H15N3S
rac-3-(1,3-Benzothiazol-2-yl)-2-methylpropane-1,2-diamine
—— rac-N-(azepan-3-yl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C23H26F2N4O2
rac-N-(azepan-3-yl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-{2-amino-2-methyl-3-[1-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]propyl}-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C27H28F2N8O3
rac-N-{2-amino-2-methyl-3-[1-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]propyl}-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-amino-2-methylpentyl)-8-[(2-fluoro-6-methoxybenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C24H31FN4O3
rac-N-(2-amino-2-methylpentyl)-8-[(2-fluoro-6-methoxybenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-N-(3,3-difluoropiperidin-4-yl)-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C22H22F4N4O2
rac-8-[(2,6-difluorobenzyl)oxy]-N-(3,3-difluoropiperidin-4-yl)-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-aminocyclopropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C20H20F2N4O2
rac-N-(2-aminocyclopropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— (R)-2-methyl-4-[2-(6-methylsulfamoyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-piperazine-1-carboxylic acid tert-butyl ester 1403900-56-0 C21H32N4O5S
(R)-2-methyl-4-[2-(6-methylsulfamoyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-piperazine-1-carboxylic acid tert-butyl ester
—— rac-tert-Butyl 1-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-3-azabicyclo[3.2.0]heptane-3-carboxylate —— C28H32F2N4O4
rac-tert-Butyl 1-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]-3-azabicyclo[3.2.0]heptane-3-carboxylate
—— rac-N-(2-amino-1,2-dimethylcyclopropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C22H24F2N4O2
rac-N-(2-amino-1,2-dimethylcyclopropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— (R)-4-[2-(5-bromo-6-dimethylsulfamoyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester 1403899-85-3 C22H33BrN4O5S
(R)-4-[2-(5-bromo-6-dimethylsulfamoyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester
—— rac-N-[1-(3-acetamidophenyl)-2-aminoethyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C27H27F2N5O3
rac-N-[1-(3-acetamidophenyl)-2-aminoethyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-amino-2-methylpentyl)-8-[(3-fluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C23H29FN4O2
rac-N-(2-amino-2-methylpentyl)-8-[(3-fluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— Rac-tert-butyl 3-{[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]methyl}thiomorpholine-4-carboxylate 1,1-dioxide trifluoroacetate —— C29H33F5N4O8S
Rac-tert-butyl 3-{[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}carbonyl)amino]methyl}thiomorpholine-4-carboxylate 1,1-dioxide trifluoroacetate
—— rac-N-[2-amino-3-(3,4-difluorophenoxy)-2-methylpropyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C27H26F4N4O3
rac-N-[2-amino-3-(3,4-difluorophenoxy)-2-methylpropyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— (R)-4-[2-(4-chloro-3,3-dimethyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester 1403899-79-5 C22H32ClN3O3
(R)-4-[2-(4-chloro-3,3-dimethyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester
—— (R)-4-{2-[5-bromo-6-(pyrrolidine-1-sulfonyl)-2,3-dihydro-indol-1-yl]2-oxo-ethyl}-2-methyl-piperazine-1-carboxylic acid tert-butyl ester 1403899-69-3 C24H35BrN4O5S
(R)-4-{2-[5-bromo-6-(pyrrolidine-1-sulfonyl)-2,3-dihydro-indol-1-yl]2-oxo-ethyl}-2-methyl-piperazine-1-carboxylic acid tert-butyl ester
—— rac-3-(4-Fluorophenyl)-2-methylpropane-1,2-diamine —— C10H15FN2
rac-3-(4-Fluorophenyl)-2-methylpropane-1,2-diamine
—— (R)-4-[2-(5-fluoro-6-phenyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester 1403899-83-1 C26H32FN3O3
(R)-4-[2-(5-fluoro-6-phenyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester
—— (R)-4-[2-(5-bromo-6-methylsulfamoyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester 1403899-84-2 C21H31BrN4O5S
(R)-4-[2-(5-bromo-6-methylsulfamoyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-2-methyl-piperazine-1-carboxylic acid tert-butyl ester
—— (R)-7-(2-fluorophenyl)-4-methyl-6-((R)-1-methylpyrrolidin-3-yl)-2,10-dihydro-9-oxa-1,2,4a-triazaphenanthren-3-one —— C22H23FN4O2
(R)-7-(2-fluorophenyl)-4-methyl-6-((R)-1-methylpyrrolidin-3-yl)-2,10-dihydro-9-oxa-1,2,4a-triazaphenanthren-3-one
—— Racemic 3-methyl-3-(1-methyl-2-oxo-1,2,3,5,8,9-hexahydro-6-oxa-3,4,10,11b-tetraaza-cyclopenta[b]phenanthren-10-yl)-azetidine-1-carboxylic acid tert-butyl ester —— C22H29N5O4
Racemic 3-methyl-3-(1-methyl-2-oxo-1,2,3,5,8,9-hexahydro-6-oxa-3,4,10,11b-tetraaza-cyclopenta[b]phenanthren-10-yl)-azetidine-1-carboxylic acid tert-butyl ester
—— Rhodanine, 1-11 —— C16H12ClNO2S2
Rhodanine, 1-11
—— (R)-2-{2-[4-(4-methoxy-1-methyl-1H-benzimidazol-2-yl)-piperazin-1-yl]-5-oxo-6,7-dihydro-5H-5λ<sup>4</sup>-thieno[3,2-d]pyrimidin-4-ylamino}-3-methylbutan-1-ol trifluoroacetate —— (x)C2HF3O2*C24H33N7O3S
(R)-2-{2-[4-(4-methoxy-1-methyl-1H-benzimidazol-2-yl)-piperazin-1-yl]-5-oxo-6,7-dihydro-5H-5λ<sup>4</sup>-thieno[3,2-d]pyrimidin-4-ylamino}-3-methylbutan-1-ol trifluoroacetate