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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-(4-methylphenyl)-(5-phenyl-1,3,4-oxadiazol-2-yl)methanol —— C16H14N2O2
(R)-(4-methylphenyl)-(5-phenyl-1,3,4-oxadiazol-2-yl)methanol
—— rac-(6S,7R,8R)-5-acetyl-6-cyclopropyl-7-methyl-8-(phenylamino)-5,6,7,8-tetrahydro-1,5-naphthyridin-2-yl trifluoromethanesulfonate —— C21H22F3N3O4S
rac-(6S,7R,8R)-5-acetyl-6-cyclopropyl-7-methyl-8-(phenylamino)-5,6,7,8-tetrahydro-1,5-naphthyridin-2-yl trifluoromethanesulfonate
—— rac-6-(((2S,3R,4R)-1-acetyl-2-cyclopropyl-6-(3,6-dihydro-2H-pyran-4-yl)-3-methyl-1,2,3,4-tetrahydroquinolin-4-yl)amino)nicotinonitrile —— C26H28N4O2
rac-6-(((2S,3R,4R)-1-acetyl-2-cyclopropyl-6-(3,6-dihydro-2H-pyran-4-yl)-3-methyl-1,2,3,4-tetrahydroquinolin-4-yl)amino)nicotinonitrile
—— rac-5-((6S,7R,8R)-5-acetyl-6-cyclopropyl-7-methyl-8-(phenylamino)-5,6,7,8-tetrahydro-1,5-naphthyridin-2-yl)-N-methylpicolinamide —— C27H29N5O2
rac-5-((6S,7R,8R)-5-acetyl-6-cyclopropyl-7-methyl-8-(phenylamino)-5,6,7,8-tetrahydro-1,5-naphthyridin-2-yl)-N-methylpicolinamide
—— rac-1-((2S,3R,4R)-2-cyclopropyl-6-fluoro-4-((6-methoxypyridin-2-yl)amino)-3-methyl-3,4-dihydroquinolin-1(2H)-yl)ethanone —— C21H24FN3O2
rac-1-((2S,3R,4R)-2-cyclopropyl-6-fluoro-4-((6-methoxypyridin-2-yl)amino)-3-methyl-3,4-dihydroquinolin-1(2H)-yl)ethanone
—— rac-(2S,3S,4R)-ethyl 4-(((benzyloxy)carbonyl)amino)-2,3-dimethyl-1,2,3,4-tetrahydroquinoline-6-carboxylate —— C22H26N2O4
rac-(2S,3S,4R)-ethyl 4-(((benzyloxy)carbonyl)amino)-2,3-dimethyl-1,2,3,4-tetrahydroquinoline-6-carboxylate
—— rac-1-((2S,3R,4R)-4-amino-2,3-diethyl-3,4-dihydroquinolin-1(2H)-yl)ethanone —— C15H22N2O
rac-1-((2S,3R,4R)-4-amino-2,3-diethyl-3,4-dihydroquinolin-1(2H)-yl)ethanone
—— rac-tert-butyl 3-((2S,3R,4R)-1-acetyl-4-amino-2,3-dimethyl-1,2,3,4-tetrahydroquinolin-6-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxylate —— C24H36N4O3
rac-tert-butyl 3-((2S,3R,4R)-1-acetyl-4-amino-2,3-dimethyl-1,2,3,4-tetrahydroquinolin-6-yl)-3,8-diazabicyclo[3.2.1]octane-8-carboxylate
—— rac-1-((2S,3R,4R)-4-Amino-3-methyl-2-propyl-3,4-dihydro-1,7-naphthyridin-1(2H)-yl)ethanone —— C14H21N3O
rac-1-((2S,3R,4R)-4-Amino-3-methyl-2-propyl-3,4-dihydro-1,7-naphthyridin-1(2H)-yl)ethanone
—— rac-(2S,3R,4R)-1-acetyl-2-cyclopropyl-7-methoxy-3-methyl-4-((4-methylpyrimidin-2-yl)amino)-1,2,3,4-tetrahydroquinoline-6-carboxylic acid —— C22H26N4O4
rac-(2S,3R,4R)-1-acetyl-2-cyclopropyl-7-methoxy-3-methyl-4-((4-methylpyrimidin-2-yl)amino)-1,2,3,4-tetrahydroquinoline-6-carboxylic acid
—— rac-(2S,3R,4R)-ethyl 1-acetyl-4-(((benzyloxy)carbonyl)amino)-2-cyclopropyl-3-methyl-8-(((trifluoromethyl)sulfonyl)oxy)-1,2,3,4-tetrahydro-1,7-naphthyridine-6-carboxylate —— C26H28F3N3O8S
rac-(2S,3R,4R)-ethyl 1-acetyl-4-(((benzyloxy)carbonyl)amino)-2-cyclopropyl-3-methyl-8-(((trifluoromethyl)sulfonyl)oxy)-1,2,3,4-tetrahydro-1,7-naphthyridine-6-carboxylate
—— rac-1-((2S,3R,4R)-2-cyclopropyl-6-fluoro-3-methyl-4-((6-methylpyridin-2-yl)amino)-3,4-dihydroquinolin-1(2H)-yl)ethanone —— C21H24FN3O
rac-1-((2S,3R,4R)-2-cyclopropyl-6-fluoro-3-methyl-4-((6-methylpyridin-2-yl)amino)-3,4-dihydroquinolin-1(2H)-yl)ethanone
—— rac-(6S,7R,8R)-5-acetyl-6-cyclopropyl-7-methyl-8-((6-methylpyridin-2-yl)amino)-5,6,7,8-tetrahydro-1,5-naphthyridin-2-yl trifluoromethanesulfonate —— C21H23F3N4O4S
rac-(6S,7R,8R)-5-acetyl-6-cyclopropyl-7-methyl-8-((6-methylpyridin-2-yl)amino)-5,6,7,8-tetrahydro-1,5-naphthyridin-2-yl trifluoromethanesulfonate
—— rac-5-(((2S,3R,4R)-1-acetyl-2-ethyl-3-methyl-6-(piperazin-1-yl)-1,2,3,4-tetrahydroquinolin-4-yl)amino)pyrazine-2-carbonitrile —— C23H29N7O
rac-5-(((2S,3R,4R)-1-acetyl-2-ethyl-3-methyl-6-(piperazin-1-yl)-1,2,3,4-tetrahydroquinolin-4-yl)amino)pyrazine-2-carbonitrile
—— rac-1-((2S,3R,4R)-2-cyclopropyl-6-fluoro-3-methyl-4-((5-methylpyrazin-2-yl)amino)-3,4-dihydroquinolin-1(2H)-yl)ethanone —— C20H23FN4O
rac-1-((2S,3R,4R)-2-cyclopropyl-6-fluoro-3-methyl-4-((5-methylpyrazin-2-yl)amino)-3,4-dihydroquinolin-1(2H)-yl)ethanone
—— rac-(2S,3R,4R)-ethyl 1-acetyl-4-amino-2-ethyl-3-methyl-1,2,3,4-tetrahydroquinoline-6-carboxylate —— C17H24N2O3
rac-(2S,3R,4R)-ethyl 1-acetyl-4-amino-2-ethyl-3-methyl-1,2,3,4-tetrahydroquinoline-6-carboxylate
—— rac-(2S,3R,4R)-1-acetyl-4-amino-N,2,3-trimethyl-1,2,3,4-tetrahydroquinoline-6-carboxamide —— C15H21N3O2
rac-(2S,3R,4R)-1-acetyl-4-amino-N,2,3-trimethyl-1,2,3,4-tetrahydroquinoline-6-carboxamide
—— rac-1-((2S,3R,4R)-2-cyclopropyl-4-((6-hydroxypyridin-2-yl)amino)-3-methyl-6-(1,2,3,6-tetrahydropyridin-4-yl)-3,4-dihydroquinolin-1(2H)-yl)ethanone —— C25H30N4O2
rac-1-((2S,3R,4R)-2-cyclopropyl-4-((6-hydroxypyridin-2-yl)amino)-3-methyl-6-(1,2,3,6-tetrahydropyridin-4-yl)-3,4-dihydroquinolin-1(2H)-yl)ethanone
—— rac-(2S,3R,4R)-ethyl 1-acetyl-4-(((benzyloxy)carbonyl)amino)-2-cyclopropyl-8-methoxy-3-methyl-1,2,3,4-tetrahydro-1,7-naphthyridine-6-carboxylate —— C26H31N3O6
rac-(2S,3R,4R)-ethyl 1-acetyl-4-(((benzyloxy)carbonyl)amino)-2-cyclopropyl-8-methoxy-3-methyl-1,2,3,4-tetrahydro-1,7-naphthyridine-6-carboxylate
—— rac-(2S,3R,4R)-ethyl 1-acetyl-4-(((benzyloxy)carbonyl)amino)-2-cyclopropyl-8-hydroxy-3-methyl-1,2,3,4-tetrahydro-1,7-naphthyridine-6-carboxylate —— C25H29N3O6
rac-(2S,3R,4R)-ethyl 1-acetyl-4-(((benzyloxy)carbonyl)amino)-2-cyclopropyl-8-hydroxy-3-methyl-1,2,3,4-tetrahydro-1,7-naphthyridine-6-carboxylate
—— rac-(2S,3R,4R)-1-acetyl-N-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)-2-ethyl-3-methyl-4-((6-methylpyridin2-yl)amino)-1,2,3,4-tetrahydroquinoline-6-carboxamide —— C26H34N4O4S
rac-(2S,3R,4R)-1-acetyl-N-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)-2-ethyl-3-methyl-4-((6-methylpyridin2-yl)amino)-1,2,3,4-tetrahydroquinoline-6-carboxamide
—— rac-(2S,3R,4R)-1-acetyl-2-cyclopropyl-3-methyl-4-(pyrimidin-2-ylamino)-1,2,3,4-tetrahydroquinoline-6-carboxylic acid —— C20H22N4O3
rac-(2S,3R,4R)-1-acetyl-2-cyclopropyl-3-methyl-4-(pyrimidin-2-ylamino)-1,2,3,4-tetrahydroquinoline-6-carboxylic acid
—— rac-(2S,3R,4R)-ethyl 1-acetyl-4-(((benzyloxy)carbonyl)amino)-2-ethyl-3-methyl-1,2,3,4-tetrahydroquinoline-6-carboxylate —— C25H30N2O5
rac-(2S,3R,4R)-ethyl 1-acetyl-4-(((benzyloxy)carbonyl)amino)-2-ethyl-3-methyl-1,2,3,4-tetrahydroquinoline-6-carboxylate
—— (R)-1-(phenyl)ethyl N-[5-(4-Bromo-phenyl)-1,3-dimethyl-1H-pyrazole-4-yl]-carbamate —— C20H20BrN3O2
(R)-1-(phenyl)ethyl N-[5-(4-Bromo-phenyl)-1,3-dimethyl-1H-pyrazole-4-yl]-carbamate
—— (R)-[(2S,4S,5R)-5-ethenyl-1-azabicyclo[2.2.2]octan-2-yl]-(6-methoxyquinolin-4-yl)methanol;propan-2-yl tetradecanoate —— C37H58N2O4
(R)-[(2S,4S,5R)-5-ethenyl-1-azabicyclo[2.2.2]octan-2-yl]-(6-methoxyquinolin-4-yl)methanol;propan-2-yl tetradecanoate
—— rac-(2S,3R,4R)-ethyl 1-acetyl-4-amino-2,3-dimethyl-1,2,3,4-tetrahydroquinoline-6-carboxylate —— C16H22N2O3
rac-(2S,3R,4R)-ethyl 1-acetyl-4-amino-2,3-dimethyl-1,2,3,4-tetrahydroquinoline-6-carboxylate
—— rac-tert-butyl 4-((2S,3R,4R)-1-acetyl-2,3-dimethyl-4-(phenylamino)-1,2,3,4-tetrahydroquinolin-6-yl)piperazine-1-carboxylate —— C28H38N4O3
rac-tert-butyl 4-((2S,3R,4R)-1-acetyl-2,3-dimethyl-4-(phenylamino)-1,2,3,4-tetrahydroquinolin-6-yl)piperazine-1-carboxylate
—— rac-1-((2S,3R,4R)-4-amino-2-cyclopropyl-3-methyl-6-morpholino-3,4-dihydroquinolin-1 (2H)-yl)ethanone —— C19H27N3O2
rac-1-((2S,3R,4R)-4-amino-2-cyclopropyl-3-methyl-6-morpholino-3,4-dihydroquinolin-1 (2H)-yl)ethanone
—— rac-tert-butyl 4-(((2S,3R,4R)-1-acetyl-2,3-dimethyl-4-(phenylamino)-1,2,3,4-tetrahydroquinolin-6-yl)amino)piperidine-1-carboxylate —— C29H40N4O3
rac-tert-butyl 4-(((2S,3R,4R)-1-acetyl-2,3-dimethyl-4-(phenylamino)-1,2,3,4-tetrahydroquinolin-6-yl)amino)piperidine-1-carboxylate
—— rac-1-((2S,3R,4R)-4-amino-2-ethyl-3-methyl-3,4-dihydroquinolin-1(2H)-yl)ethanone hydrobromide —— C14H21BrN2O
rac-1-((2S,3R,4R)-4-amino-2-ethyl-3-methyl-3,4-dihydroquinolin-1(2H)-yl)ethanone hydrobromide
—— (RS)-3-(4-chlorophenyl)-2-{4-[3-methyl-4-((R)-1-phenylethoxycarbonyloxy)isoxazol-5-yl]benzyloxy}propionic acid methyl ester —— C30H28ClNO7
(RS)-3-(4-chlorophenyl)-2-{4-[3-methyl-4-((R)-1-phenylethoxycarbonyloxy)isoxazol-5-yl]benzyloxy}propionic acid methyl ester
—— rac-1-((2S.3R.4R)-6-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-2,3-dimethyl-4-(phenylamino)-3.4-dihydroquinolin-1(2H)-yl)ethanone —— C25H31N3O2
rac-1-((2S.3R.4R)-6-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-2,3-dimethyl-4-(phenylamino)-3.4-dihydroquinolin-1(2H)-yl)ethanone
—— rac-1-((2S,3R,4R)-4-amino-2-ethyl-3-methyl-3,4-dihydroquinolin-1(2H)-yl)ethanone —— C14H20N2O
rac-1-((2S,3R,4R)-4-amino-2-ethyl-3-methyl-3,4-dihydroquinolin-1(2H)-yl)ethanone
—— rac-(2S,3R,4R)-ethyl 1-acetyl-2-cyclopropyl-3-methyl-4-(pyrimidin-2-ylamino)-1,2,3,4-tetrahydro-1,7-naphthyridine-6-carboxylate —— C21H25N5O3
rac-(2S,3R,4R)-ethyl 1-acetyl-2-cyclopropyl-3-methyl-4-(pyrimidin-2-ylamino)-1,2,3,4-tetrahydro-1,7-naphthyridine-6-carboxylate
—— (R)-2-(2-mercaptoethyl)-5-(diethylamino)pentanol —— C11H25NOS
(R)-2-(2-mercaptoethyl)-5-(diethylamino)pentanol
—— rac-(2S,3S,4R)-ethyl 4-(((benzyloxy)carbonyl)amino)-2-ethyl-3-methyl-1,2,3,4-tetrahydroquinoline-6-carboxylate —— C23H28N2O4
rac-(2S,3S,4R)-ethyl 4-(((benzyloxy)carbonyl)amino)-2-ethyl-3-methyl-1,2,3,4-tetrahydroquinoline-6-carboxylate
—— (R)-(2-(tert-butyl-dimethylsilanyloxy)-3-{4-chloro-3-[4-(2,3-dimethyl-2,6-dihydro-4H-pyrrolo[3,4-c]pyrazol-5-yl)-6-(3,5-dimethyl-isoxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy}propyl)methylcarbamic acid tert-butyl ester —— C38H54ClN7O5Si
(R)-(2-(tert-butyl-dimethylsilanyloxy)-3-{4-chloro-3-[4-(2,3-dimethyl-2,6-dihydro-4H-pyrrolo[3,4-c]pyrazol-5-yl)-6-(3,5-dimethyl-isoxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy}propyl)methylcarbamic acid tert-butyl ester
—— (R)-2-(4-{4-[1-((R)-2-chlorophenyl)ethoxycarbonylamino]-3-methylisoxazol-5-yl}benzoylamino)-3-cyclopropyl-propionic acid —— C26H26ClN3O6
(R)-2-(4-{4-[1-((R)-2-chlorophenyl)ethoxycarbonylamino]-3-methylisoxazol-5-yl}benzoylamino)-3-cyclopropyl-propionic acid
—— rac-1-((2S,3R,4R)-4-amino-3-methyl-2-(2,2,2-trifluoroethyl)-3,4-dihydroquinolin-1(2H)-yl)ethanone —— C14H17F3N2O
rac-1-((2S,3R,4R)-4-amino-3-methyl-2-(2,2,2-trifluoroethyl)-3,4-dihydroquinolin-1(2H)-yl)ethanone
—— (R)-1-(tetrahydrofuran-3-yl)imidazolidin-2-one —— C7H12N2O2
(R)-1-(tetrahydrofuran-3-yl)imidazolidin-2-one
—— (RS)-3-(4-chlorophenyl)-2-{4-[3-methyl-4-((R)-1-phenylethoxycarbonyloxy)isoxazol-5-yl]benzyloxy}propionic acid —— C29H26ClNO7
(RS)-3-(4-chlorophenyl)-2-{4-[3-methyl-4-((R)-1-phenylethoxycarbonyloxy)isoxazol-5-yl]benzyloxy}propionic acid
—— (R)-(2-(tert-butyl-dimethylsilanyloxy)-3-{4-chloro-3-[4-(3,5-dimethylisoxazol-4-yl)-5-methyl-6-(3-methyl-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazol-5-yl)pyrimidin-2-yl]phenoxy}propyl)methylcarbamic acid tert-butyl ester —— C37H52ClN7O5Si
(R)-(2-(tert-butyl-dimethylsilanyloxy)-3-{4-chloro-3-[4-(3,5-dimethylisoxazol-4-yl)-5-methyl-6-(3-methyl-4,6-dihydro-1H-pyrrolo[3,4-c]pyrazol-5-yl)pyrimidin-2-yl]phenoxy}propyl)methylcarbamic acid tert-butyl ester
—— (R)-2-(4-{4-[(R)-1-(2-chlorophenyl)ethoxycarbonylamino]-3-methylisoxazol-5-yl}benzylamino)-3-phenylpropionic acid methyl ester —— C30H30ClN3O5
(R)-2-(4-{4-[(R)-1-(2-chlorophenyl)ethoxycarbonylamino]-3-methylisoxazol-5-yl}benzylamino)-3-phenylpropionic acid methyl ester
—— (R)-2-[2-{5-[3-(tert-butoxycarbonyl-methyl-amino)-2-(tert-butyl-dimethyl-silanyloxy)propoxy]-2-chloro-phenyl}-6-(3,5-dimethyl-isoxazol-4-yl)-5-methyl-pyrimidin-4-yl]-2,7-diaza-spiro[3.5]nonane-7-carboxylic acid methyl ester —— C40H59ClN6O7Si
(R)-2-[2-{5-[3-(tert-butoxycarbonyl-methyl-amino)-2-(tert-butyl-dimethyl-silanyloxy)propoxy]-2-chloro-phenyl}-6-(3,5-dimethyl-isoxazol-4-yl)-5-methyl-pyrimidin-4-yl]-2,7-diaza-spiro[3.5]nonane-7-carboxylic acid methyl ester
—— (R)-(2-(tert-butyl-dimethylsilanyloxy)-3-{4-chloro-3-[4-(7-cyclopropyl-2,7-diazaspiro[3.5]non-2-yl)-6-(3,5-dimethylisoxazol-4-yl)-5-methylpyrimidin-2-yl]-phenoxy}propyl)methylcarbamic acid tert-butyl ester —— C41H61ClN6O5Si
(R)-(2-(tert-butyl-dimethylsilanyloxy)-3-{4-chloro-3-[4-(7-cyclopropyl-2,7-diazaspiro[3.5]non-2-yl)-6-(3,5-dimethylisoxazol-4-yl)-5-methylpyrimidin-2-yl]-phenoxy}propyl)methylcarbamic acid tert-butyl ester
—— (R)-1-(3-bromo-4-fluorophenoxy)-3-(methyl-amino)propan-2-ol —— C10H13BrFNO2
(R)-1-(3-bromo-4-fluorophenoxy)-3-(methyl-amino)propan-2-ol
—— (R)-1-(1-methoxypropan-2-yl)imidazolidin-2-one —— C7H14N2O2
(R)-1-(1-methoxypropan-2-yl)imidazolidin-2-one
—— (R)-tert-butyl 3-(3-bromo-4-fluoro phenoxy)-2-hydroxypropyl(methyl)carbamate —— C15H21BrFNO4
(R)-tert-butyl 3-(3-bromo-4-fluoro phenoxy)-2-hydroxypropyl(methyl)carbamate
—— (R)-methyl 3-((5-fluoro-2-(1-(2-fluorobenzyl)-5-(isoxazol-3-yl)-1H-pyrazol-3-yl)pyrimidin-4-yl)amino)-4-methylpentanoate —— C24H24F2N6O3
(R)-methyl 3-((5-fluoro-2-(1-(2-fluorobenzyl)-5-(isoxazol-3-yl)-1H-pyrazol-3-yl)pyrimidin-4-yl)amino)-4-methylpentanoate
—— Racemic cis-3-[4-(4-fluoro-3-methyl-phenyl)-2-(3-fluoro-piperidin-4-yl)-imidazol-1-ylmethyl]-azetidine-1-carboxylic acid tert-butyl ester —— C24H32F2N4O2
Racemic cis-3-[4-(4-fluoro-3-methyl-phenyl)-2-(3-fluoro-piperidin-4-yl)-imidazol-1-ylmethyl]-azetidine-1-carboxylic acid tert-butyl ester