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—— (R)-N-[(2R)-2-(5-bromo-2-fluorophenyl)-1-(1-cyanocyclobutyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide —— C18H24BrFN2O3S2
(R)-N-[(2R)-2-(5-bromo-2-fluorophenyl)-1-(1-cyanocyclobutyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2S)-2-(5-bromo-3-chlorothiophen-2-yl)-1-(1-cyanocyclobutyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide —— C16H22BrClN2O3S3
(R)-N-[(2S)-2-(5-bromo-3-chlorothiophen-2-yl)-1-(1-cyanocyclobutyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2R)-2-(5-bromo-2-fluorophenyl)-1-(1-cyanocyclopentyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide —— C19H26BrFN2O3S2
(R)-N-[(2R)-2-(5-bromo-2-fluorophenyl)-1-(1-cyanocyclopentyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2S)-2-(5-bromo-3-chlorothiophen-2-yl)-1-(1-cyanocyclohexyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide —— C18H26BrClN2O3S3
(R)-N-[(2S)-2-(5-bromo-3-chlorothiophen-2-yl)-1-(1-cyanocyclohexyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2R)-1-(3-cyanooxetan-3-yl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide —— C17H22FN3O6S2
(R)-N-[(2R)-1-(3-cyanooxetan-3-yl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2R)-1-(1-cyanocyclopentyl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide —— C19H26FN3O5S2
(R)-N-[(2R)-1-(1-cyanocyclopentyl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2S)-1-(1-cyanocyclohexyl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide —— C20H28FN3O5S2
(R)-N-[(2S)-1-(1-cyanocyclohexyl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2S)-2-(5-bromo-3-chlorothiophen-2-yl)-1-(1-cyanocyclopentyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide —— C17H24BrClN2O3S3
(R)-N-[(2S)-2-(5-bromo-3-chlorothiophen-2-yl)-1-(1-cyanocyclopentyl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2S)-2-(5-bromo-3-chlorothiophen-2-yl)-1-(4-cyanooxan-4-yl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide —— C17H24BrClN2O4S3
(R)-N-[(2S)-2-(5-bromo-3-chlorothiophen-2-yl)-1-(4-cyanooxan-4-yl)sulfonylpropan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2S)-1-(1-cyanocyclobutyl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide —— C18H24FN3O5S2
(R)-N-[(2S)-1-(1-cyanocyclobutyl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2R)-1-[(3R)-3-cyanooxolan-3-yl]sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide —— C18H24FN3O6S2
(R)-N-[(2R)-1-[(3R)-3-cyanooxolan-3-yl]sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2R)-1-(1-cyanocyclopropyl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide —— C17H22FN3O5S2
(R)-N-[(2R)-1-(1-cyanocyclopropyl)sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2R)-1-[(3S)-3-cyanooxolan-3-yl]sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide —— C18H24FN3O6S2
(R)-N-[(2R)-1-[(3S)-3-cyanooxolan-3-yl]sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-4-(6-chloro-1,5-naphthyridin-3-yl)-3-methylmorpholine —— C13H14ClN3O
(R)-4-(6-chloro-1,5-naphthyridin-3-yl)-3-methylmorpholine
—— [(R)-anilino(methylsulfanyl)methyl]-(3-hydroxy-3,3-diphosphonatopropyl)azanium —— C11H17N2O7P2S-3
[(R)-anilino(methylsulfanyl)methyl]-(3-hydroxy-3,3-diphosphonatopropyl)azanium
—— (R)-N-[(1S)-6-bromo-1-(1-ethoxyethenyl)-4'-methoxyspiro[3H-indene-2,1'-cyclohexane]-1-yl]-2-methylpropane-2-sulfinamide —— C23H34BrNO3S
(R)-N-[(1S)-6-bromo-1-(1-ethoxyethenyl)-4'-methoxyspiro[3H-indene-2,1'-cyclohexane]-1-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2R)-1-[1-cyano-3-[(4-methoxyphenyl)methoxy]cyclopentyl]sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide —— C27H34FN3O7S2
(R)-N-[(2R)-1-[1-cyano-3-[(4-methoxyphenyl)methoxy]cyclopentyl]sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-[(2R)-1-[1-cyano-3-[(4-methoxyphenyl)methoxy]cyclobutyl]sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide —— C26H32FN3O7S2
(R)-N-[(2R)-1-[1-cyano-3-[(4-methoxyphenyl)methoxy]cyclobutyl]sulfonyl-2-(2-fluoro-5-nitrophenyl)propan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-methyl 1-(3-amino-4-(phenylthio)butyl)-3-methylazetidine-3-carboxylate 1619923-65-7 C16H24N2O2S
(R)-methyl 1-(3-amino-4-(phenylthio)butyl)-3-methylazetidine-3-carboxylate
—— (R)-(+)-1-Methoxy-1,2,2,2-tetrafuoropropionamide —— C4H5F4NO2
(R)-(+)-1-Methoxy-1,2,2,2-tetrafuoropropionamide
—— (R)-1-((R)-3-methoxy-tetrahydro-pyran-4-yl)-3-[(3S,3aR,6S,6aS)-6-(2-methyl-pyridin-3-yloxy)-hexahydro-furo[3,2-b]furan-3-yl]-urea —— C19H27N3O6
(R)-1-((R)-3-methoxy-tetrahydro-pyran-4-yl)-3-[(3S,3aR,6S,6aS)-6-(2-methyl-pyridin-3-yloxy)-hexahydro-furo[3,2-b]furan-3-yl]-urea
—— (R)-2-amino-N-(4-methoxybenzyl)-3-phenylpropionamide hydrochloride —— C17H20N2O2*ClH
(R)-2-amino-N-(4-methoxybenzyl)-3-phenylpropionamide hydrochloride
—— (R)-N-cyclohexylmethyl-2-{N'-[2-(3,4-dimethoxyphenyl)acetyl]guanidino}-3-phenylpropionamide trifluoroacetate —— C2HF3O2*C27H36N4O4
(R)-N-cyclohexylmethyl-2-{N'-[2-(3,4-dimethoxyphenyl)acetyl]guanidino}-3-phenylpropionamide trifluoroacetate
—— (R)-3-Cyclohexyl-2-{N'-[2-(3,4-dimethoxyphenyl)acetyl]-guanidino}-N-(1-ethylpropyl)propionamide —— C25H40N4O4
(R)-3-Cyclohexyl-2-{N'-[2-(3,4-dimethoxyphenyl)acetyl]-guanidino}-N-(1-ethylpropyl)propionamide
—— (R)-methyl 3-methyl-2-(2-((4-methyl-2-oxo-2H-chromen-7-yl)oxy)acetamido)butanoate —— C18H21NO6
(R)-methyl 3-methyl-2-(2-((4-methyl-2-oxo-2H-chromen-7-yl)oxy)acetamido)butanoate
—— (R)-3-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-yl)-4-(1-methyl-1H-1,2,4-triazol-5-yl)oxazolidin-2-one —— C16H13F2N5O5
(R)-3-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-yl)-4-(1-methyl-1H-1,2,4-triazol-5-yl)oxazolidin-2-one
—— (R)-6,7-difluoro-3-(4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-oxooxazolidin-3-yl)benzo[d]isoxazole-5-carbaldehyde —— C14H9F2N5O4
(R)-6,7-difluoro-3-(4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-oxooxazolidin-3-yl)benzo[d]isoxazole-5-carbaldehyde
—— (R)-3-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-yl)-4-(difluoromethyl)oxazolidin-2-one —— C14H10F4N2O5
(R)-3-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-yl)-4-(difluoromethyl)oxazolidin-2-one
—— (R)-2-Acetyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid 1842525-43-2 C12H13NO3
(R)-2-Acetyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
—— (R)-8-cyclopropyl-6-(4-(furan-2-carbonyl)-3-methylpiperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C25H29N3O3
(R)-8-cyclopropyl-6-(4-(furan-2-carbonyl)-3-methylpiperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-8-cyclohexyl-6-(4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416269-59-4 C24H32N4O2
(R)-8-cyclohexyl-6-(4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(2-methylindolizine-3-carbonyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile —— C31H37N5O2
(R)-8-cyclopropyl-6-(3-isopropyl-4-(2-methylindolizine-3-carbonyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-ethyl-6-(3-isopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416269-97-0 C24H36N4O3
(R)-8-ethyl-6-(3-isopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-isopropyl-6-(3-isopropyl-4-(4-methyloxazole-5-carbonyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-63-4 C26H35N5O3
(R)-8-isopropyl-6-(3-isopropyl-4-(4-methyloxazole-5-carbonyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-2-isopropyl-N-(4-methoxyphenyl)piperazine-1-carboxamide 1416269-00-5 C29H37N5O3
(R)-4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-2-isopropyl-N-(4-methoxyphenyl)piperazine-1-carboxamide
—— (R)-8-cyclopropyl-6-(4-(2-cyclopropylacetyl)-3-isopropylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416269-66-3 C26H36N4O2
(R)-8-cyclopropyl-6-(4-(2-cyclopropylacetyl)-3-isopropylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-isopropyl-3,3-dimethyl-6-(3-methyl-4-(2-oxo-2-phenylacetyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416266-35-7 C27H32N4O3
(R)-8-isopropyl-3,3-dimethyl-6-(3-methyl-4-(2-oxo-2-phenylacetyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(2-(2-methoxyphenyl)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C31H39N3O3
(R)-8-cyclopropyl-6-(3-isopropyl-4-(2-(2-methoxyphenyl)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-4-(5-cyano-8-cyclopropyl-3,3-dimethylisochroman-6-yl)-N,2-diisopropylpiperazine-1-carboxamide —— C26H38N4O2
(R)-4-(5-cyano-8-cyclopropyl-3,3-dimethylisochroman-6-yl)-N,2-diisopropylpiperazine-1-carboxamide
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(2-(prop-2-ynylamino)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416269-57-2 C26H35N5O2
(R)-8-cyclopropyl-6-(3-isopropyl-4-(2-(prop-2-ynylamino)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-isopropyl-6-(3-isopropyl-4-(2-(thiophen-2-yl)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-28-1 C27H36N4O2S
(R)-8-isopropyl-6-(3-isopropyl-4-(2-(thiophen-2-yl)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-ethyl-4-(3-methoxypropanoyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-81-9 C24H34N4O3
(R)-8-cyclopropyl-6-(3-ethyl-4-(3-methoxypropanoyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-propionylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416269-38-9 C24H34N4O2
(R)-8-cyclopropyl-6-(3-isopropyl-4-propionylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-6-(4-(5-chlorothiophen-2-ylsulfonyl)-3-isopropylpiperazin-1-yl)-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-69-3 C25H31ClN4O3S2
(R)-6-(4-(5-chlorothiophen-2-ylsulfonyl)-3-isopropylpiperazin-1-yl)-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-4-(5-cyano-8-cyclohexyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-2-methyl-N-(prop-2-ynyl)piperazine-1-carboxamide 1416269-45-8 C24H31N5O2
(R)-4-(5-cyano-8-cyclohexyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-2-methyl-N-(prop-2-ynyl)piperazine-1-carboxamide
—— (R)-8-isopropyl-6-(3-isopropyl-4-(2-(pyridin-2-yl)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-64-5 C28H37N5O2
(R)-8-isopropyl-6-(3-isopropyl-4-(2-(pyridin-2-yl)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(4-methyloxazole-5-carbonyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C27H34N4O3
(R)-8-cyclopropyl-6-(3-isopropyl-4-(4-methyloxazole-5-carbonyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-8-cyclohexyl-6-(3-methyl-4-(2-methylfuran-3-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-06-5 C26H32N4O3
(R)-8-cyclohexyl-6-(3-methyl-4-(2-methylfuran-3-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-isopropyl-6-(3-isopropyl-4-(2-(pyridin-3-yl)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-30-8 C28H37N5O2
(R)-8-isopropyl-6-(3-isopropyl-4-(2-(pyridin-3-yl)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-isopropyl-6-(3-isopropyl-4-(2-(3-methoxyphenyl)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-99-6 C30H40N4O3
(R)-8-isopropyl-6-(3-isopropyl-4-(2-(3-methoxyphenyl)acetyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile