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—— rac-tert-Butyl 2-{[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)-amino]methyl}-3,4-dihydroquinoline-1(2H)-carboxylate —— C31H32F2N4O4
rac-tert-Butyl 2-{[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)-amino]methyl}-3,4-dihydroquinoline-1(2H)-carboxylate
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)-N-(3-methylphenyl)glycinamide —— C21H23N3O4S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)-N-(3-methylphenyl)glycinamide
—— rac-N-(2-Amino-2,4-dimethylpentyl)-2,6-dimethyl-8-(3-methylbutoxy)imidazo[1,2-a]pyridine-3-carboxamide —— C22H36N4O2
rac-N-(2-Amino-2,4-dimethylpentyl)-2,6-dimethyl-8-(3-methylbutoxy)imidazo[1,2-a]pyridine-3-carboxamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-[2-(morpholin-4-yl)-1-phenylethyl]imidazo[1,2-a]pyridine-3-carboxamide 1609341-48-1 C28H28F2N4O3
rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-[2-(morpholin-4-yl)-1-phenylethyl]imidazo[1,2-a]pyridine-3-carboxamide
—— Rel-N-(5-chloro-2-methoxyphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethoxyphenyl)glycinamide —— C22H24ClN3O5S2
Rel-N-(5-chloro-2-methoxyphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethoxyphenyl)glycinamide
—— rac-3-Isopropoxypropane-1,2-diamine dihydrochloride —— C6H18Cl2N2O
rac-3-Isopropoxypropane-1,2-diamine dihydrochloride
—— rac-tert-butyl 3-[({6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridin-3-yl}carbonyl)amino]indolin-1-carboxylate 1609345-17-6 C29H27ClF2N4O4
rac-tert-butyl 3-[({6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridin-3-yl}carbonyl)amino]indolin-1-carboxylate
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethoxyphenyl)-N-(2-fluorophenyl)glycinamide —— C21H22FN3O4S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethoxyphenyl)-N-(2-fluorophenyl)glycinamide
—— rac-N-(2-Amino-2,4-dimethylpentyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C23H28F2N4O2
rac-N-(2-Amino-2,4-dimethylpentyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-[2-amino-4-(benzyloxy)-2-methylbutyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C29H32F2N4O3
rac-N-[2-amino-4-(benzyloxy)-2-methylbutyl]-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-Amino-1-phenylethyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide dihydrochloride —— C24H24Cl2F2N4O2
rac-N-(2-Amino-1-phenylethyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide dihydrochloride
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-isopropylphenyl)-N-(3-methyl-1H-pyrazol-5-YL)glycinamide —— C20H25N5O3S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-isopropylphenyl)-N-(3-methyl-1H-pyrazol-5-YL)glycinamide
—— Rel-(3AR,6AR)-N-(2-chloro-4-fluorobenzyl)-N-(3-methoxyphenyl)-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-amine 5,5-dioxide —— C19H18ClFN2O3S2
Rel-(3AR,6AR)-N-(2-chloro-4-fluorobenzyl)-N-(3-methoxyphenyl)-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-amine 5,5-dioxide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-isopropylphenyl)-N-(4-methylphenyl)glycinamide —— C23H27N3O3S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-isopropylphenyl)-N-(4-methylphenyl)glycinamide
—— Rel-N-(3-chloro-4-fluorophenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)glycinamide —— C20H19ClFN3O4S2
Rel-N-(3-chloro-4-fluorophenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)glycinamide
—— rac-N-(1-amino-3-isopropoxypropan-2-yl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609340-73-9 C22H26F2N4O3
rac-N-(1-amino-3-isopropoxypropan-2-yl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-amino-3-methoxy-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide 1609341-83-4 C22H26F2N4O3
rac-N-(2-amino-3-methoxy-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethoxyphenyl)-N-(3-methyl-1H-pyrazol-5-YL)glycinamide —— C19H23N5O4S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-ethoxyphenyl)-N-(3-methyl-1H-pyrazol-5-YL)glycinamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-[2-(morpholin-4-yl)propyl]imidazo[1,2-a]pyridine-3-carboxamide 1609341-46-9 C23H26F2N4O3
rac-8-[(2,6-difluorobenzyl)oxy]-2-methyl-N-[2-(morpholin-4-yl)propyl]imidazo[1,2-a]pyridine-3-carboxamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(3-fluoro-4-methylphenyl)-N~2~-(4-methoxyphenyl)glycinamide —— C21H22FN3O4S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(3-fluoro-4-methylphenyl)-N~2~-(4-methoxyphenyl)glycinamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(2-methoxyphenyl)-N~2~-(4-methoxyphenyl)glycinamide —— C21H23N3O5S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(2-methoxyphenyl)-N~2~-(4-methoxyphenyl)glycinamide
—— rac-N-(2-Amino-2,4-dimethylpentyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C23H27ClF2N4O2
rac-N-(2-Amino-2,4-dimethylpentyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-Amino-2-methylpentyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide —— C23H28F2N4O2
rac-N-(2-Amino-2-methylpentyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
—— rac-N-(2-Amino-3-hydroxy-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide —— C20H22F2N4O3
rac-N-(2-Amino-3-hydroxy-2-methylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-ethoxyphenyl)-N~2~-(4-isopropylphenyl)glycinamide —— C24H29N3O4S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-ethoxyphenyl)-N~2~-(4-isopropylphenyl)glycinamide
—— rac-N-(2-aminopropyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609340-35-3 C19H19ClF2N4O2
rac-N-(2-aminopropyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— Rel-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}-N-[2-(2-furyl)ethyl]benzamide —— C18H19N3O4S2
Rel-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}-N-[2-(2-furyl)ethyl]benzamide
—— rac-8-[(2,6-difluorobenzyl)oxy]-N-[2-(dimethylamino)-3-methylbutyl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609341-57-2 C23H28F2N4O2
rac-8-[(2,6-difluorobenzyl)oxy]-N-[2-(dimethylamino)-3-methylbutyl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— Rel-(3AR,6AR)-N-(4-ethoxyphenyl)-N-(2-fluorobenzyl)-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-amine 5,5-dioxide —— C20H21FN2O3S2
Rel-(3AR,6AR)-N-(4-ethoxyphenyl)-N-(2-fluorobenzyl)-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-amine 5,5-dioxide
—— rac-N-(2-Amino-2-cyclopropylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]-pyridine-3-carboxamide —— C23H26F2N4O2
rac-N-(2-Amino-2-cyclopropylpropyl)-8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]-pyridine-3-carboxamide
—— rac-N-(2-Amino-2-methylpentyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide —— C22H25ClF2N4O2
rac-N-(2-Amino-2-methylpentyl)-6-chloro-8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]-pyridine-3-carboxamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)-N-(2-methylphenyl)glycinamide —— C21H23N3O4S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)-N-(2-methylphenyl)glycinamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)-N-[3-(trifluoromethyl)phenyl]glycinamide —— C21H20F3N3O4S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N~2~-(4-methoxyphenyl)-N-[3-(trifluoromethyl)phenyl]glycinamide
—— rac-6-chloro-8-[(2,6-difluorobenzyl)oxy]-N-(2,3-dihydro-1H-indol-3-yl)-2-methylimidazo[1,2-a]pyridine-3-carboxamide 1609340-60-4 C24H19ClF2N4O2
rac-6-chloro-8-[(2,6-difluorobenzyl)oxy]-N-(2,3-dihydro-1H-indol-3-yl)-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-methylphenyl)-N~2~-phenylglycinamide —— C20H21N3O3S2
Rel-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-methylphenyl)-N~2~-phenylglycinamide
—— rac-3-(Benzyloxy)-2-methylpropane-1,2-diamine —— C11H18N2O
rac-3-(Benzyloxy)-2-methylpropane-1,2-diamine
—— rac-tert-butyl 3-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)-amino]indolin-1-carboxylate 1609345-16-5 C29H28F2N4O4
rac-tert-butyl 3-[({8-[(2,6-difluorobenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-yl}carbonyl)-amino]indolin-1-carboxylate
—— Rel-N-[2-(2,5-dimethoxyphenyl)ethyl]-2-(4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}phenyl)acetamide —— C23H27N3O5S2
Rel-N-[2-(2,5-dimethoxyphenyl)ethyl]-2-(4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}phenyl)acetamide
—— Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(3-methyl-1H-pyrazol-5-YL)glycinamide —— C19H23N5O3S2
Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(3-methyl-1H-pyrazol-5-YL)glycinamide
—— Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-mesitylglycinamide —— C24H29N3O3S2
Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-mesitylglycinamide
—— Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(3-methoxyphenyl)glycinamide —— C22H25N3O4S2
Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(3-methoxyphenyl)glycinamide
—— Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-fluorophenyl)glycinamide —— C21H22FN3O3S2
Rel-N~2~-(3,5-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-fluorophenyl)glycinamide
—— Rel-N~2~-(3,4-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-ethylphenyl)glycinamide —— C23H27N3O3S2
Rel-N~2~-(3,4-dimethylphenyl)-N~2~-[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]-N-(4-ethylphenyl)glycinamide
—— Rel-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}-N-[2-(4-sulfamoylphenyl)ethyl]benzamide —— C20H22N4O5S3
Rel-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}-N-[2-(4-sulfamoylphenyl)ethyl]benzamide
—— Rel-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}-N-[2-(4-ethoxyphenyl)ethyl]benzamide —— C22H25N3O4S2
Rel-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}-N-[2-(4-ethoxyphenyl)ethyl]benzamide
—— rac-(3R,6S,7S,8aS)-2,3,7-trimethyl-1,4-dioxo-6-(1-(phenylsulfonyl)-1H-indol-3-yl)octahydropyrrolo[1,2-a]pyrazine-7-carbonitrile —— C25H24N4O4S
rac-(3R,6S,7S,8aS)-2,3,7-trimethyl-1,4-dioxo-6-(1-(phenylsulfonyl)-1H-indol-3-yl)octahydropyrrolo[1,2-a]pyrazine-7-carbonitrile
—— Rel-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}-N-{2-[3-(trifluoromethyl)phenoxy]ethyl}benzamide —— C21H20F3N3O4S2
Rel-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}-N-{2-[3-(trifluoromethyl)phenoxy]ethyl}benzamide
—— rac-4-(3-(6-cyano-5-(trifluoromethyl)pyridin-3-yl)-7,7-dimethyl-4-oxo-2-thioxo-1,3-diazaspiro[4.5]decan-1-yl)-2-fluoro-N-methylbenzamide 1607853-89-3 C25H23F4N5O2S
rac-4-(3-(6-cyano-5-(trifluoromethyl)pyridin-3-yl)-7,7-dimethyl-4-oxo-2-thioxo-1,3-diazaspiro[4.5]decan-1-yl)-2-fluoro-N-methylbenzamide
—— Rel-N-[2-(2,4-dimethoxyphenyl)ethyl]-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}benzamide —— C22H25N3O5S2
Rel-N-[2-(2,4-dimethoxyphenyl)ethyl]-4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}benzamide
—— Rel-1-(1-azepanyl)-2-(4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}phenyl)ethanone —— C19H25N3O3S2
Rel-1-(1-azepanyl)-2-(4-{[(3AR,6AR)-5,5-dioxido-3A,4,6,6A-tetrahydrothieno[3,4-D][1,3]thiazol-2-YL]amino}phenyl)ethanone