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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-N-(1-(4-(4-chlorophenyl)isoxazol-3-yl)-2-(3,5-difluorophenyl)ethyl)-2-(5-hydroxy-1H-indol-3-yl)acetamide 1620231-86-8 C27H20ClF2N3O3
(R)-N-(1-(4-(4-chlorophenyl)isoxazol-3-yl)-2-(3,5-difluorophenyl)ethyl)-2-(5-hydroxy-1H-indol-3-yl)acetamide
—— (R)-N-(2-(3,5-difluorophenyl)-1-(1-(4-methoxyphenyl)-1H-imidazol-2-yl)ethyl)-2-(5-hydroxy-1H-indol-3-yl)acetamide 1620231-43-7 C28H24F2N4O3
(R)-N-(2-(3,5-difluorophenyl)-1-(1-(4-methoxyphenyl)-1H-imidazol-2-yl)ethyl)-2-(5-hydroxy-1H-indol-3-yl)acetamide
—— (R)-N-(2-(3,5-difluorophenyl)-1-(1-(4-methoxyphenyl)-1H-imidazol-2-yl)ethyl)-2-(3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl)acetamide 1620231-41-5 C28H26F5N5O2
(R)-N-(2-(3,5-difluorophenyl)-1-(1-(4-methoxyphenyl)-1H-imidazol-2-yl)ethyl)-2-(3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl)acetamide
—— (R)-1-(3-(4-(N-(4-(4-(3-(2-(4-chlorophenyl)-1-isopropyl-5-methyl-4-(methylsulfonyl)-1H-pyrrol-3-yl)-5-fluorophenyl)piperazin-1-yl)phenyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)-3-methylazetidine-3-carboxylic acid 1619923-49-7 C53H57ClF4N6O8S4
(R)-1-(3-(4-(N-(4-(4-(3-(2-(4-chlorophenyl)-1-isopropyl-5-methyl-4-(methylsulfonyl)-1H-pyrrol-3-yl)-5-fluorophenyl)piperazin-1-yl)phenyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)-3-methylazetidine-3-carboxylic acid
—— (R)-3-(1-(3-(4-(N-(4-(4-(3-(2-(4-chlorophenyl)-1-isopropyl-5-methyl-4-(methylsulfonyl)-1H-pyrrol-3-yl)-5-fluorophenyl)piperazin-1-yl)phenyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)-3-methylazetidine-3-carbonyloxy)propylphosphonic acid 1619923-51-1 C56H64ClF4N6O11PS4
(R)-3-(1-(3-(4-(N-(4-(4-(3-(2-(4-chlorophenyl)-1-isopropyl-5-methyl-4-(methylsulfonyl)-1H-pyrrol-3-yl)-5-fluorophenyl)piperazin-1-yl)phenyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)-3-methylazetidine-3-carbonyloxy)propylphosphonic acid
—— (R)-2-(1-(3-(4-(N-(4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex-1-enyl)methyl) piperazin-1-yl)benzoyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)piperidine-4-carbonyloxy)ethylphosphonic acid 1619923-45-3 C51H62ClF3N5O10PS3
(R)-2-(1-(3-(4-(N-(4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex-1-enyl)methyl) piperazin-1-yl)benzoyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)piperidine-4-carbonyloxy)ethylphosphonic acid
—— (R)-(1-(3-(4-(N-(4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex-1-enyl)methyl)piperazin-1-yl)benzoyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)piperidine-4-carbonyloxy)methylphosphonic acid 1619923-44-2 C50H60ClF3N5O10PS3
(R)-(1-(3-(4-(N-(4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex-1-enyl)methyl)piperazin-1-yl)benzoyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)piperidine-4-carbonyloxy)methylphosphonic acid
—— (R)-2-(1-(3-(4-(N-(4-(4-(3-(2-(4-chlorophenyl)-1-isopropyl-5-methyl-4-(methylsulfonylcarbamoyl)-1H-pyrrol-3-yl)phenyl)piperazin-1-yl)phenyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)piperidine-4-carbonyloxy)ethylphosphonic acid 1619923-48-6 C57H66ClF3N7O12PS4
(R)-2-(1-(3-(4-(N-(4-(4-(3-(2-(4-chlorophenyl)-1-isopropyl-5-methyl-4-(methylsulfonylcarbamoyl)-1H-pyrrol-3-yl)phenyl)piperazin-1-yl)phenyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)piperidine-4-carbonyloxy)ethylphosphonic acid
—— (R)-1-(3-(4-(N-(4-(4-(3-(2-(4-chlorophenyl)-1-isopropyl-5-methyl-4-(methylsulfonylcarbamoyl)-1H-pyrrol-3-yl)phenyl)piperazin-1-yl)phenyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)piperidine-4-carboxylic acid 1619923-47-5 C55H61ClF3N7O9S4
(R)-1-(3-(4-(N-(4-(4-(3-(2-(4-chlorophenyl)-1-isopropyl-5-methyl-4-(methylsulfonylcarbamoyl)-1H-pyrrol-3-yl)phenyl)piperazin-1-yl)phenyl)sulfamoyl)-2-(trifluoromethylsulfonyl)phenylamino)-4-(phenylthio)butyl)piperidine-4-carboxylic acid
—— (R)-4-((5-(4-chlorophenyl)-1-ethyl-4-(3-(4-(4-(4-((4-(4-hydroxypiperidin-1-yl)-1-(phenylthio)butan-2-yl)amino)-3-((trifluoromethyl)sulfonyl)phenylsulfonamido)phenyl)piperazin-1-yl)phenyl)-2-methyl-1H-pyrrole-3-carbonyl)oxy)cyclohexane carboxylic acid —— C59H66ClF3N6O9S3
(R)-4-((5-(4-chlorophenyl)-1-ethyl-4-(3-(4-(4-(4-((4-(4-hydroxypiperidin-1-yl)-1-(phenylthio)butan-2-yl)amino)-3-((trifluoromethyl)sulfonyl)phenylsulfonamido)phenyl)piperazin-1-yl)phenyl)-2-methyl-1H-pyrrole-3-carbonyl)oxy)cyclohexane carboxylic acid
—— (R)-(7-(trifluoromethyl)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl 4-bromobenzenesulfonate —— C16H12BrF3O5S
(R)-(7-(trifluoromethyl)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl 4-bromobenzenesulfonate
—— (R)-4-((3-fluorophenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazidin-2-one —— C17H23FN2O3
(R)-4-((3-fluorophenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazidin-2-one
—— (R)-tert-butyl 4-(2-(4-(((tert-butyldimethylsilyl)oxy)methyl)-5,5-dimethyl-2-oxooxazolidin-3-yl)ethyl)piperidine-1-carboxylate —— C24H46N2O5Si
(R)-tert-butyl 4-(2-(4-(((tert-butyldimethylsilyl)oxy)methyl)-5,5-dimethyl-2-oxooxazolidin-3-yl)ethyl)piperidine-1-carboxylate
—— (R)-(7-fluoro-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl 4-bromobenzenesulfonate —— C15H12BrFO5S
(R)-(7-fluoro-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl 4-bromobenzenesulfonate
—— (R)-3-(2-(1-(((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperidin-4-yl)ethyl)-4-((3-fluorophenoxy)methyl)oxazolidin-2-one —— C26H31FN2O5
(R)-3-(2-(1-(((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperidin-4-yl)ethyl)-4-((3-fluorophenoxy)methyl)oxazolidin-2-one
—— (R)-4-((3-(benzyloxy)phenoxy)methyl)-3-(2-(1-(((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperidin-4-yl)ethyl)oxazolidin-2-one —— C33H38N2O6
(R)-4-((3-(benzyloxy)phenoxy)methyl)-3-(2-(1-(((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperidin-4-yl)ethyl)oxazolidin-2-one
—— (R)-4-((4-(benzyloxy)phenoxy)methyl)-3-(2-(1-(((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperidin-4-yl)ethyl)oxazolidin-2-one —— C33H38N2O6
(R)-4-((4-(benzyloxy)phenoxy)methyl)-3-(2-(1-(((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperidin-4-yl)ethyl)oxazolidin-2-one
—— (R)-4-((4-fluorophenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one —— C17H23FN2O3
(R)-4-((4-fluorophenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one
—— (R)-7-bromo-2-(bromomethyl)-2,3-dihydrobenzo[b][1,4]dioxine —— C9H8Br2O2
(R)-7-bromo-2-(bromomethyl)-2,3-dihydrobenzo[b][1,4]dioxine
—— (R)-4-((3,4-dimethoxyphenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one —— C19H28N2O5
(R)-4-((3,4-dimethoxyphenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one
—— (R)-3-(2-(1-(((S)-6-(benzyloxy)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperidin-4-yl)ethyl)-4-(phenoxymethyl)oxazolidin-2-one —— C33H38N2O6
(R)-3-(2-(1-(((S)-6-(benzyloxy)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)piperidin-4-yl)ethyl)-4-(phenoxymethyl)oxazolidin-2-one
—— (R)-4-phenyl-3-(3-(piperidin-4-yl)propyl)-oxazolidin-2-one —— C17H24N2O2
(R)-4-phenyl-3-(3-(piperidin-4-yl)propyl)-oxazolidin-2-one
—— (R)-4-(hydroxymethyl)-5,5-dimethyl-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one —— C13H24N2O3
(R)-4-(hydroxymethyl)-5,5-dimethyl-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one
—— (R)-4-phenyl-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one —— C16H22N2O2
(R)-4-phenyl-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one
—— (R)-6-phenyl-4-(2-(piperidin-4-yl)ethyl)morpholin-3-one —— C17H24N2O2
(R)-6-phenyl-4-(2-(piperidin-4-yl)ethyl)morpholin-3-one
—— (R)-4-((2,6-dimethylphenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one —— C19H28N2O3
(R)-4-((2,6-dimethylphenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one
—— (R)-4-((4-(benzyloxy)phenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one —— C24H30N2O4
(R)-4-((4-(benzyloxy)phenoxy)methyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one
—— (R)-4-(phenoxymethyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one —— C17H24N2O3
(R)-4-(phenoxymethyl)-3-(2-(piperidin-4-yl)ethyl)oxazolidin-2-one
—— (R)-tert-butyl 4-(2-(2-oxo-4-(phenoxymethyl)oxazolidin-3-yl)ethyl)piperidine-1-carboxylate —— C22H32N2O5
(R)-tert-butyl 4-(2-(2-oxo-4-(phenoxymethyl)oxazolidin-3-yl)ethyl)piperidine-1-carboxylate
—— racemic (1R,2S)-2-phenylcyclopentanecarboxamidine hydrochloride —— C12H16N2*ClH
racemic (1R,2S)-2-phenylcyclopentanecarboxamidine hydrochloride
—— (R)-2-hydroxy-3-[(1H-pyrrolo[2,3-b]pyridine-5-carbonyl)-amino]-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-66-8 C17H14BN3O5
(R)-2-hydroxy-3-[(1H-pyrrolo[2,3-b]pyridine-5-carbonyl)-amino]-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-3-(2-(6-(2-aminoethylamino)pyridin-3-yl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-91-9 C18H21BN4O5
(R)-3-(2-(6-(2-aminoethylamino)pyridin-3-yl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-3-(2-(4-(2-aminoethoxy)-3-hydroxyphenyl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-90-8 C19H21BN2O7
(R)-3-(2-(4-(2-aminoethoxy)-3-hydroxyphenyl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-2-hydroxy-3-[4-(1H-imidazol-2-yl)-benzoylamino]-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-78-2 C19H16BN3O5
(R)-2-hydroxy-3-[4-(1H-imidazol-2-yl)-benzoylamino]-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-3-(2-(4-(2-aminoethylamino)phenyl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-88-4 C19H22BN3O5
(R)-3-(2-(4-(2-aminoethylamino)phenyl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-3-(5,6-bis(aminomethyl)nicotinamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-93-1 C17H19BN4O5
(R)-3-(5,6-bis(aminomethyl)nicotinamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-3-(3,5-bis(aminomethyl)benzamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-75-9 C18H20BN3O5
(R)-3-(3,5-bis(aminomethyl)benzamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-3-(2-(2-aminoethylcarbamoyl)benzamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-85-1 C19H20BN3O6
(R)-3-(2-(2-aminoethylcarbamoyl)benzamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-3-(3,4-bis((isopropylamino)methyl)benzamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-87-3 C24H32BN3O5
(R)-3-(3,4-bis((isopropylamino)methyl)benzamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-3-(2-(3,4-bis(2-aminoethoxy)phenyl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid 1618082-89-5 C21H26BN3O7
(R)-3-(2-(3,4-bis(2-aminoethoxy)phenyl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid
—— (R)-N-(3,4-difluorophenyl)-2-fluoro-5-(N-(1-(tetrahydro-2H-pyran-4-yl)ethyl)sulfamoyl)benzamide 1616807-92-1 C20H21F3N2O4S
(R)-N-(3,4-difluorophenyl)-2-fluoro-5-(N-(1-(tetrahydro-2H-pyran-4-yl)ethyl)sulfamoyl)benzamide
—— (R)-N-(3,4-difluorophenyl)-2-methoxy-5-(N-(3-methylbutan-2-yl)sulfamoyl)benzamide 1616807-84-1 C19H22F2N2O4S
(R)-N-(3,4-difluorophenyl)-2-methoxy-5-(N-(3-methylbutan-2-yl)sulfamoyl)benzamide
—— (R)-5-(N-(1-cyclohexylethyl)sulfamoyl)-N-(3,4-difluorophenyl)-2-fluorobenzamide 1616807-81-8 C21H23F3N2O3S
(R)-5-(N-(1-cyclohexylethyl)sulfamoyl)-N-(3,4-difluorophenyl)-2-fluorobenzamide
—— (R)-N-(3,4-difluorophenyl)-2-fluoro-5-(N-(1-phenylethyl)sulfamoyl)benzamide 1616807-56-7 C21H17F3N2O3S
(R)-N-(3,4-difluorophenyl)-2-fluoro-5-(N-(1-phenylethyl)sulfamoyl)benzamide
—— (R)-5-(N-(1-cyclopentylethyl)sulfamoyl)-N-(3,4-difluorophenyl)-2-fluorobenzamide 1616807-85-2 C20H21F3N2O3S
(R)-5-(N-(1-cyclopentylethyl)sulfamoyl)-N-(3,4-difluorophenyl)-2-fluorobenzamide
—— (R)-5-(N-(1-cyclobutylethyl)sulfamoyl)-N-(3,4-difluorophenyl)-2-fluorobenzamide 1616807-83-0 C19H19F3N2O3S
(R)-5-(N-(1-cyclobutylethyl)sulfamoyl)-N-(3,4-difluorophenyl)-2-fluorobenzamide
—— (R)-N-(3,4-difluorophenyl)-2,4-difluoro-5-(N-(3-methylbutan-2-yl)sulfamoyl)benzamide 1616807-86-3 C18H18F4N2O3S
(R)-N-(3,4-difluorophenyl)-2,4-difluoro-5-(N-(3-methylbutan-2-yl)sulfamoyl)benzamide
—— (R)-N-(3,4-difluorophenyl)-2-fluoro-5-(N-(1-(pyridin-4-yl)ethyl)sulfamoyl)benzamide 1616808-00-4 C20H16F3N3O3S
(R)-N-(3,4-difluorophenyl)-2-fluoro-5-(N-(1-(pyridin-4-yl)ethyl)sulfamoyl)benzamide
—— (R)-N-(3,4-difluorophenyl)-2-fluoro-5-(N-(1-hydroxypropan-2-yl)sulfamoyl)benzamide 1616807-60-3 C16H15F3N2O4S
(R)-N-(3,4-difluorophenyl)-2-fluoro-5-(N-(1-hydroxypropan-2-yl)sulfamoyl)benzamide
—— (R)-2-(1-Methoxyethyl)thiophene —— C7H10OS
(R)-2-(1-Methoxyethyl)thiophene