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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-4-(fluoromethyl)-3-(2-fluoropyrimidin-4-yl)oxazolidin-2-one —— C8H7F2N3O2
(R)-4-(fluoromethyl)-3-(2-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-(((S)-1-(5-chloro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C18H18ClF4N5O4
(R)-3-(2-(((S)-1-(5-chloro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— racemic cis-3-{1-[2-fluoro-4-(6-methoxypyridin-3-yl)benzyl]-5-(quinolin-2-ylmethoxy)-1H-benzimidazol-2-yl}-2,2-dimethylcyclopropanecarboxylic acid —— C36H31FN4O4
racemic cis-3-{1-[2-fluoro-4-(6-methoxypyridin-3-yl)benzyl]-5-(quinolin-2-ylmethoxy)-1H-benzimidazol-2-yl}-2,2-dimethylcyclopropanecarboxylic acid
—— racemic cis-3-{1-[(3,4'-difluorobiphenyl-4-yl)methyl]-5-(quinolin-2-ylmethoxy)-1H-benzimidazol-2-yl}-2,2-dimethylcyclopropanecarboxylic acid —— C36H29F2N3O3
racemic cis-3-{1-[(3,4'-difluorobiphenyl-4-yl)methyl]-5-(quinolin-2-ylmethoxy)-1H-benzimidazol-2-yl}-2,2-dimethylcyclopropanecarboxylic acid
—— (R)-4-((R)-1-hydroxyethyl)-3-(2-(((S)-1-(3-(isoquinolin-8-yl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C22H21N7O4
(R)-4-((R)-1-hydroxyethyl)-3-(2-(((S)-1-(3-(isoquinolin-8-yl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-(difluoromethoxy)-3-fluorophenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C22H27F3N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-(difluoromethoxy)-3-fluorophenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-(((S)-1-(3-(4-ethylphenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C21H24N6O4
(R)-3-(2-(((S)-1-(3-(4-ethylphenyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((S)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chloro-3-(trifluoromethoxy)phenyl)piperidin-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C27H35ClF3N5O4
(R)-4-((S)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chloro-3-(trifluoromethoxy)phenyl)piperidin-4-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— racemic cis-2-(5-((6-fluoroquinolin-2-yl)methoxy)-1-((4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl)methyl)-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid —— C38H31F4N3O3
racemic cis-2-(5-((6-fluoroquinolin-2-yl)methoxy)-1-((4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl)methyl)-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-(difluoromethoxy)-2-fluorophenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C22H27F3N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-(difluoromethoxy)-2-fluorophenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(3-((S)-tetrahydrofuran-3-yloxy)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C25H34N4O5
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(3-((S)-tetrahydrofuran-3-yloxy)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-(((S)-1-(1-(4-(difluoromethyl)-3-fluorophenyl)-1H-imidazol-4-yl)ethyl)amino)pyrimidin-4-yl)-4-(fluoromethyl)oxazolidin-2-one —— C20H18F4N6O2
(R)-3-(2-(((S)-1-(1-(4-(difluoromethyl)-3-fluorophenyl)-1H-imidazol-4-yl)ethyl)amino)pyrimidin-4-yl)-4-(fluoromethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(difluoromethoxy)phenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C22H27F3N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3-(difluoromethoxy)phenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-(((S)-1-(1-(2,4-difluorophenyl)-1H-imidazol-4-yl)ethyl)amino)pyrimidin-4-yl)-4-((S)-1-fluoroethyl)oxazolidin-2-one —— C20H19F3N6O2
(R)-3-(2-(((S)-1-(1-(2,4-difluorophenyl)-1H-imidazol-4-yl)ethyl)amino)pyrimidin-4-yl)-4-((S)-1-fluoroethyl)oxazolidin-2-one
—— racemic cis-2-{1-(4-bromobenzyl)-5-[(6-chloroquinolin-2-yl)methoxy]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid —— C31H27BrClN3O3
racemic cis-2-{1-(4-bromobenzyl)-5-[(6-chloroquinolin-2-yl)methoxy]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid
—— (R)-4-((S)-1-(tert-butoxy)ethyl)-3-(2-chloropyrimidin-4-yl)oxazolidin-2-one —— C13H18ClN3O3
(R)-4-((S)-1-(tert-butoxy)ethyl)-3-(2-chloropyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(5-fluoro-2-(((R)-1-(5-(3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C22H20F4N6O3
(R)-3-(5-fluoro-2-(((R)-1-(5-(3-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((S)-1-hydroxyethyl)-3-(2-(((R)-1-(2-phenylthiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C20H21N5O3S
(R)-4-((S)-1-hydroxyethyl)-3-(2-(((R)-1-(2-phenylthiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— racemic cis-2,2-dimethyl-3-{5-(quinolin-2-ylmethoxy)-1-[3-(1,3-thiazol-4-yl)benzyl]-1H-benzimidazol-2-yl}cyclopropanecarboxylic acid —— C33H28N4O3S
racemic cis-2,2-dimethyl-3-{5-(quinolin-2-ylmethoxy)-1-[3-(1,3-thiazol-4-yl)benzyl]-1H-benzimidazol-2-yl}cyclopropanecarboxylic acid
—— racemic cis-2-(1-(4-bromobenzyl)-5-((6-fluoroquinolin-2-yl)methoxy)-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid —— C31H27BrFN3O3
racemic cis-2-(1-(4-bromobenzyl)-5-((6-fluoroquinolin-2-yl)methoxy)-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid
—— (R)-3-(2-{(S)-1-[5-(3-fluorophenyl)-[1,3,4]-oxadiazol-2-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C19H19FN6O4
(R)-3-(2-{(S)-1-[5-(3-fluorophenyl)-[1,3,4]-oxadiazol-2-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-chloro-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C13H17ClFN3O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-chloro-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-(((R)-1-(5-(4-chloro-3-methylphenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C22H23ClN6O3
(R)-3-(2-(((R)-1-(5-(4-chloro-3-methylphenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-hydroxyethyl)-3-(2-(((S)-1-phenylethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C17H20N4O3
(R)-4-((R)-1-hydroxyethyl)-3-(2-(((S)-1-phenylethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-(4-chlorophenyl)isoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C24H27Cl2N5O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(6-chloro-2-(((S)-1-(5-(4-chlorophenyl)isoxazol-3-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— racemic cis-3-[1-(2,4-dichlorobenzyl)-5-(quinolin-2-ylmethoxy)-1H-benzimidazol-2-yl]-2,2-dimethylcyclopropanecarboxylic acid —— C30H25Cl2N3O3
racemic cis-3-[1-(2,4-dichlorobenzyl)-5-(quinolin-2-ylmethoxy)-1H-benzimidazol-2-yl]-2,2-dimethylcyclopropanecarboxylic acid
—— (R)-4-((R)-1-hydroxyethyl)-3-(2-(((R)-1-(5-(3-methyl-4-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C23H23F3N6O3
(R)-4-((R)-1-hydroxyethyl)-3-(2-(((R)-1-(5-(3-methyl-4-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— racemic trans-2-{1-(4-bromobenzyl)-5-[(8-fluoroquinolin-2-yl)methoxy]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid —— C31H27BrFN3O3
racemic trans-2-{1-(4-bromobenzyl)-5-[(8-fluoroquinolin-2-yl)methoxy]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid
—— racemic cis-2-(5-(benzo[d]thiazol-2-ylmethoxy)-1-(4-(piperidin-1-yl)benzyl)-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid —— C34H36N4O3S
racemic cis-2-(5-(benzo[d]thiazol-2-ylmethoxy)-1-(4-(piperidin-1-yl)benzyl)-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-(difluoromethoxy)-3-fluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C22H26F4N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-(difluoromethoxy)-3-fluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— racemic cis-2-(5-(benzo[d]thiazol-2-ylmethoxy)-1-(4-(pyrimidin-2-yl)benzyl)-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid —— C33H29N5O3S
racemic cis-2-(5-(benzo[d]thiazol-2-ylmethoxy)-1-(4-(pyrimidin-2-yl)benzyl)-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid
—— (R)-3-(2-(((S)-1-(1-(4-chloro-3-(trifluoromethoxy)phenyl)piperidin-4-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-4-((S)-1-hydroxyethyl)oxazolidin-2-one —— C23H26ClF4N5O4
(R)-3-(2-(((S)-1-(1-(4-chloro-3-(trifluoromethoxy)phenyl)piperidin-4-yl)ethyl)amino)-5-fluoropyrimidin-4-yl)-4-((S)-1-hydroxyethyl)oxazolidin-2-one
—— racemic cis-2-(1-(4-Bromobenzyl)-5-hydroxy-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid —— C21H21BrN2O3
racemic cis-2-(1-(4-Bromobenzyl)-5-hydroxy-1H-benzo[d]imidazol-2-yl)cyclohexanecarboxylic acid
—— (R)-5-bromo-4-fluoro-N-(1-(3-fluorophenyl)ethyl)-2-nitroaniline —— C14H11BrF2N2O2
(R)-5-bromo-4-fluoro-N-(1-(3-fluorophenyl)ethyl)-2-nitroaniline
—— (R)-1-(1-(4-chlorophenyl)-1H-pyrazol-3-yl)ethanamine —— C11H12ClN3
(R)-1-(1-(4-chlorophenyl)-1H-pyrazol-3-yl)ethanamine
—— (R)-tert-butyl 3-(5-chloro-4-(1H-pyrrolo[3,2-b]pyridin-6-yl)pyridin-2-ylcarbamoyl)piperidine-1-carboxylate —— C23H26ClN5O3
(R)-tert-butyl 3-(5-chloro-4-(1H-pyrrolo[3,2-b]pyridin-6-yl)pyridin-2-ylcarbamoyl)piperidine-1-carboxylate
—— (R)-6-bromo-5-fluoro-1-(1-(3-fluorophenyl)ethyl)-1H-benzo[d][1,2,3]triazole —— C14H10BrF2N3
(R)-6-bromo-5-fluoro-1-(1-(3-fluorophenyl)ethyl)-1H-benzo[d][1,2,3]triazole
—— (R)-tert-butyl 4,4-difluoro-2-formylpyrrolidine-1-carboxylate —— C10H15F2NO3
(R)-tert-butyl 4,4-difluoro-2-formylpyrrolidine-1-carboxylate
—— (R)-tert-butyl 3-(5-chloro-4-(1-(2-oxo-2-(tetrahydro-2H-pyran-4-yl)ethyl)-1H-pyrrolo[3,2-b]pyridin-6-yl)pyridin-2-ylcarbamoyl)piperidine-1-carboxylate —— C30H36ClN5O5
(R)-tert-butyl 3-(5-chloro-4-(1-(2-oxo-2-(tetrahydro-2H-pyran-4-yl)ethyl)-1H-pyrrolo[3,2-b]pyridin-6-yl)pyridin-2-ylcarbamoyl)piperidine-1-carboxylate
—— (R)-tert-butyl 3-(5-chloro-4-(1-((1-methyl-1H-benzo[d][1,2,3]triazol-6-yl)methyl)-1H-pyrrolo[3,2-b]pyridin-6-yl)pyridin-2-ylcarbamoyl)piperidine-1-carboxylate —— C31H33ClN8O3
(R)-tert-butyl 3-(5-chloro-4-(1-((1-methyl-1H-benzo[d][1,2,3]triazol-6-yl)methyl)-1H-pyrrolo[3,2-b]pyridin-6-yl)pyridin-2-ylcarbamoyl)piperidine-1-carboxylate
—— (R)-tert-butyl 2-(((6-bromo-5-chloropyridin-2-yl)amino)methyl)-4,4-difluoropyrrolidine-1-carboxylate —— C15H19BrClF2N3O2
(R)-tert-butyl 2-(((6-bromo-5-chloropyridin-2-yl)amino)methyl)-4,4-difluoropyrrolidine-1-carboxylate
—— (R)-tert-butyl 3-(5-chloro-4-(3-formyl-1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-pyrrolo[3,2-b]pyridin-6-yl)pyridin-2-ylcarbamoyl)piperidine-1-carboxylate —— C30H36ClN5O5
(R)-tert-butyl 3-(5-chloro-4-(3-formyl-1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-pyrrolo[3,2-b]pyridin-6-yl)pyridin-2-ylcarbamoyl)piperidine-1-carboxylate
—— (R)-tert-butyl 3-(4-bromopyridin-2-ylcarbamoyl)piperidine-1-carboxylate —— C16H22BrN3O3
(R)-tert-butyl 3-(4-bromopyridin-2-ylcarbamoyl)piperidine-1-carboxylate
—— (R)-tert-butyl 4-(4-(6-(((1-(tert-butoxycarbonyl)-4,4-difluoropyrrolidin-2-yl)methyl)amino)-3-chloropyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl)piperidine-1-carboxylate —— C32H41ClF2N6O4
(R)-tert-butyl 4-(4-(6-(((1-(tert-butoxycarbonyl)-4,4-difluoropyrrolidin-2-yl)methyl)amino)-3-chloropyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl)piperidine-1-carboxylate
—— (R)-1-(4-(1-(4-(trifluoromethoxy)phenyl)-1H-1,2,4-triazol-3-yl)phenyl)propan-2-amine —— C18H17F3N4O
(R)-1-(4-(1-(4-(trifluoromethoxy)phenyl)-1H-1,2,4-triazol-3-yl)phenyl)propan-2-amine
—— racemic cis-2-{1-[3-Fluoro-4-(trifluoromethoxy)benzyl]-6-[(5-methylpyridin-2-yl)methoxy]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid —— C29H27F4N3O4
racemic cis-2-{1-[3-Fluoro-4-(trifluoromethoxy)benzyl]-6-[(5-methylpyridin-2-yl)methoxy]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid
—— racemic cis-2-{6-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methoxy]-1-(4-piperidin-1-ylbenzyl)-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid —— C31H36ClN5O3
racemic cis-2-{6-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methoxy]-1-(4-piperidin-1-ylbenzyl)-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid
—— racemic cis-2-{1-[4-(3,3-difluoroazetidin-1-yl)benzyl]-4-fluoro-6-[(1-methyl-1H-pyrazol-3-yl)methoxy]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid —— C29H30F3N5O3
racemic cis-2-{1-[4-(3,3-difluoroazetidin-1-yl)benzyl]-4-fluoro-6-[(1-methyl-1H-pyrazol-3-yl)methoxy]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid
—— racemic cis-3-{1-(4-bromobenzyl)-4-chloro-6-[(5-methylpyridin-2-yl)methoxy]-1H-benzimidazol-2-yl}-2,2-dimethylcyclopropanecarboxylic acid —— C27H25BrClN3O3
racemic cis-3-{1-(4-bromobenzyl)-4-chloro-6-[(5-methylpyridin-2-yl)methoxy]-1H-benzimidazol-2-yl}-2,2-dimethylcyclopropanecarboxylic acid
—— racemic cis-2-{4-fluoro-6-[(5-methylpyridin-2-yl)methoxy]-1-[4-(trifluoromethoxy)benzyl]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid —— C29H27F4N3O4
racemic cis-2-{4-fluoro-6-[(5-methylpyridin-2-yl)methoxy]-1-[4-(trifluoromethoxy)benzyl]-1H-benzimidazol-2-yl}cyclohexanecarboxylic acid