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—— (R)-6-(4-(2,5-dimethylfuran-3-carbonyl)-3-methylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-29-2 C26H34N4O3
(R)-6-(4-(2,5-dimethylfuran-3-carbonyl)-3-methylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-50-2 C25H36N4O3
(R)-8-cyclopropyl-6-(3-isopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(thiophene-3-carbonyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C27H33N3O2S
(R)-8-cyclopropyl-6-(3-isopropyl-4-(thiophene-3-carbonyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-N-benzyl-4-(5-cyano-8-cyclopropyl-3,3-dimethylisochroman-6-yl)-2-isopropylpiperazine-1-carboxamide —— C30H38N4O2
(R)-N-benzyl-4-(5-cyano-8-cyclopropyl-3,3-dimethylisochroman-6-yl)-2-isopropylpiperazine-1-carboxamide
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(oxazole-4-carbonyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C26H32N4O3
(R)-8-cyclopropyl-6-(3-isopropyl-4-(oxazole-4-carbonyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-8-isopropyl-6-(4-(2-(3-methoxyphenyl)acetyl)-3-methylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-77-0 C28H36N4O3
(R)-8-isopropyl-6-(4-(2-(3-methoxyphenyl)acetyl)-3-methylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-1-((4-(benzo[d]thiazol-5-ylamino)-6-(tert-butylsulfonyl)quinazolin-7-yl)oxy)propan-2-ol —— C22H24N4O4S2
(R)-1-((4-(benzo[d]thiazol-5-ylamino)-6-(tert-butylsulfonyl)quinazolin-7-yl)oxy)propan-2-ol
—— (R)-6-(4-(2-(4-bromo-1H-pyrazol-1-yl)acetyl)-3-isopropylpiperazin-1-yl)-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416269-99-2 C26H33BrN6O2
(R)-6-(4-(2-(4-bromo-1H-pyrazol-1-yl)acetyl)-3-isopropylpiperazin-1-yl)-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-6-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416266-01-7 C24H30N4O3
(R)-6-(4-(furan-3-carbonyl)-3-methylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-6-(4-(furan-2-carbonyl)-3-methylpiperazin-1-yl)-8-isopropyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416265-91-2 C22H26N4O3
(R)-6-(4-(furan-2-carbonyl)-3-methylpiperazin-1-yl)-8-isopropyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-4-(5-cyano-8-cyclohexyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-N-(2-fluorophenyl)-2-methylpiperazine-1-carboxamide 1416268-84-2 C27H32FN5O2
(R)-4-(5-cyano-8-cyclohexyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-N-(2-fluorophenyl)-2-methylpiperazine-1-carboxamide
—— (R)-6-(4-(benzo[b]thiophene-3-carbonyl)-3-methylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-25-1 C28H32N4O2S
(R)-6-(4-(benzo[b]thiophene-3-carbonyl)-3-methylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-6-(4-(2-(3-fluorophenyl)acetyl)-3-isopropylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-01-3 C29H37FN4O2
(R)-6-(4-(2-(3-fluorophenyl)acetyl)-3-isopropylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(2-(methoxy(methyl)amino)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C26H38N4O3
(R)-8-cyclopropyl-6-(3-isopropyl-4-(2-(methoxy(methyl)amino)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-4-methoxyphenyl 4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]-pyridine-6-yl)-2-isopropylpiperazine-1-carboxylate 1416269-21-0 C29H36N4O4
(R)-4-methoxyphenyl 4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]-pyridine-6-yl)-2-isopropylpiperazine-1-carboxylate
—— (R)-1-cyclopropyl-3-(3-cyclopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-6-propioloyl-5,6,7,8-tetrahydro-2,6-naphthyridine-4-carbonitrile 1416270-69-3 C26H31N5O3
(R)-1-cyclopropyl-3-(3-cyclopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-6-propioloyl-5,6,7,8-tetrahydro-2,6-naphthyridine-4-carbonitrile
—— (R)-4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-2-isopropyl-N-p-tolylpiperazine-1-carboxamide 1416268-85-3 C29H37N5O2
(R)-4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-2-isopropyl-N-p-tolylpiperazine-1-carboxamide
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(2-(pyridin-3-yl)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C29H36N4O2
(R)-8-cyclopropyl-6-(3-isopropyl-4-(2-(pyridin-3-yl)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-8-cyclopropyl-6-(4-(2-(2-hydroxyethoxy)acetyl)-3-isopropylpiperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C26H37N3O4
(R)-8-cyclopropyl-6-(4-(2-(2-hydroxyethoxy)acetyl)-3-isopropylpiperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-6-(4-(furan-3-carbonyl)-3-phenylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-36-4 C29H32N4O3
(R)-6-(4-(furan-3-carbonyl)-3-phenylpiperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-4-(5-cyano-8-cyclohexyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-2-methyl-N-o-tolylpiperazine-1-carboxamide 1416268-63-7 C28H35N5O2
(R)-4-(5-cyano-8-cyclohexyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-2-methyl-N-o-tolylpiperazine-1-carboxamide
—— (R)-8-cyclobutyl-6-(3-isopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416269-79-8 C26H38N4O3
(R)-8-cyclobutyl-6-(3-isopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-6-(4-acetyl-3-isopropylpiperazin-1-yl)-8-cyclopropyl-3,3-dimethylisochroman-5-carbonitrile —— C24H33N3O2
(R)-6-(4-acetyl-3-isopropylpiperazin-1-yl)-8-cyclopropyl-3,3-dimethylisochroman-5-carbonitrile
—— (R)-(4-(5-(2-chloro-4-(1H-pyrazol-4-yl)phenyl)-1,3,4-thiadiazol-2-yl)piperazin-2-yl)methanol Hydrochloride Salt 1620515-72-1 C16H17ClN6OS*ClH
(R)-(4-(5-(2-chloro-4-(1H-pyrazol-4-yl)phenyl)-1,3,4-thiadiazol-2-yl)piperazin-2-yl)methanol Hydrochloride Salt
—— (R)-6-(4-(2-chloroacetyl)-3-methylpiperazin-1-yl)-8-cyclohexyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416269-24-3 C22H29ClN4O2
(R)-6-(4-(2-chloroacetyl)-3-methylpiperazin-1-yl)-8-cyclohexyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-cyclopropylmethyl 4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]-pyridine-6-yl)-2-isopropylpiperazine-1-carboxylate 1416269-54-9 C26H36N4O3
(R)-cyclopropylmethyl 4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]-pyridine-6-yl)-2-isopropylpiperazine-1-carboxylate
—— (R)-8-cyclopropyl-6-(4-(2,5-dimethylfuran-3-carbonyl)-3-methylpiperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C27H33N3O3
(R)-8-cyclopropyl-6-(4-(2,5-dimethylfuran-3-carbonyl)-3-methylpiperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-8-cyclopropyl-6-(4-(furan-2-carbonyl)-2-methylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-45-2 C24H28N4O3
(R)-8-cyclopropyl-6-(4-(furan-2-carbonyl)-2-methylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-ethyl-4-(2-methylfuran-3-carbonyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-07-9 C26H32N4O3
(R)-8-cyclopropyl-6-(3-ethyl-4-(2-methylfuran-3-carbonyl)piperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(4-(2-(furan-2-ylmethoxy)acetyl)-3-isopropylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416269-88-9 C28H36N4O4
(R)-8-cyclopropyl-6-(4-(2-(furan-2-ylmethoxy)acetyl)-3-isopropylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclohexyl-6-(3-methyl-4-(thiazole-4-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-11-5 C24H29N5O2S
(R)-8-cyclohexyl-6-(3-methyl-4-(thiazole-4-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-ethyl-4-(2-(thiophen-2-yl)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C27H33N3O2S
(R)-8-cyclopropyl-6-(3-ethyl-4-(2-(thiophen-2-yl)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-8-isopropyl-3,3-dimethyl-6-(3-methyl-4-(3-methylfuran-2-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416266-83-5 C25H32N4O3
(R)-8-isopropyl-3,3-dimethyl-6-(3-methyl-4-(3-methylfuran-2-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclohexyl-6-(3-methyl-4-(4-methyloxazol-5-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-84-9 C25H31N5O3
(R)-8-cyclohexyl-6-(3-methyl-4-(4-methyloxazol-5-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-ethyl-4-(2-(2-methoxyphenyl)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C30H37N3O3
(R)-8-cyclopropyl-6-(3-ethyl-4-(2-(2-methoxyphenyl)acetyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile
—— (R)-6-(4-(2-(3,5-difluorophenyl)acetyl)-3-methylpiperazin-1-yl)-8isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416266-42-6 C27H32F2N4O2
(R)-6-(4-(2-(3,5-difluorophenyl)acetyl)-3-methylpiperazin-1-yl)-8isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-N-cyclopropyl-2-isopropylpiperazine-1-carboxamide 1416269-82-3 C25H35N5O2
(R)-4-(5-cyano-8-cyclopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-N-cyclopropyl-2-isopropylpiperazine-1-carboxamide
—— (R)-1-cyclopropyl-3-(3-cyclopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-7-(2-hydroxyethyl)-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile 1416270-67-1 C25H35N5O3
(R)-1-cyclopropyl-3-(3-cyclopropyl-4-(3-methoxypropanoyl)piperazin-1-yl)-7-(2-hydroxyethyl)-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
—— (R)-N-(4-((3-chloro-4-fluorophenyl)amino)-7-((tetrahydrofuran-3-yl)oxy)quinazolin-6-yl)-4-(dimethylamino)-2-fluorobut-2-enamide —— C24H24ClF2N5O3
(R)-N-(4-((3-chloro-4-fluorophenyl)amino)-7-((tetrahydrofuran-3-yl)oxy)quinazolin-6-yl)-4-(dimethylamino)-2-fluorobut-2-enamide
—— (R)-N-{4-(3-chloro-4-fluorophenylamino)-7-[2-(1-methylpiperidin-2-yl)ethoxy]quinazolin-6-yl}-2-fluoroacrylamide 1420406-73-0 C25H26ClF2N5O2
(R)-N-{4-(3-chloro-4-fluorophenylamino)-7-[2-(1-methylpiperidin-2-yl)ethoxy]quinazolin-6-yl}-2-fluoroacrylamide
—— (R)-8-cyclobutyl-6-(4-(furan-3-carbonyl)-3-isopropylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-72-8 C27H34N4O3
(R)-8-cyclobutyl-6-(4-(furan-3-carbonyl)-3-isopropylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-6-(3-ethyl-4-(2-(thiophen-2-yl)acetyl)piperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416267-48-5 C26H34N4O2S
(R)-6-(3-ethyl-4-(2-(thiophen-2-yl)acetyl)piperazin-1-yl)-8-isopropyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclohexyl-3,3-dimethyl-6-(3-methyl-4-(2-phenylacetyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416266-18-6 C30H38N4O2
(R)-8-cyclohexyl-3,3-dimethyl-6-(3-methyl-4-(2-phenylacetyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-isopropyl-3,3-dimethyl-6-(3-methyl-4-(thiophene-3-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-31-9 C24H30N4O2S
(R)-8-isopropyl-3,3-dimethyl-6-(3-methyl-4-(thiophene-3-carbonyl)piperazin-1-yl)-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-N-[4-(3-chloro-2,4-difluorophenylamino)-7-(tetrahydrofuran-3-ylmethoxy)quinazolin-6-yl]-2-fluoroacrylamide —— C22H18ClF3N4O3
(R)-N-[4-(3-chloro-2,4-difluorophenylamino)-7-(tetrahydrofuran-3-ylmethoxy)quinazolin-6-yl]-2-fluoroacrylamide
—— (R)-6-(4-butyryl-3-isopropylpiperazin-1-yl)-8-cyclopropyl-3,3-dimethylisochroman-5-carbonitrile —— C26H37N3O2
(R)-6-(4-butyryl-3-isopropylpiperazin-1-yl)-8-cyclopropyl-3,3-dimethylisochroman-5-carbonitrile
—— (R)-8-cyclohexyl-6-(4-(furan-2-carbonyl)-3-methylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416266-16-4 C27H34N4O3
(R)-8-cyclohexyl-6-(4-(furan-2-carbonyl)-3-methylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-6-(4-(furan-3-carbonyl)-3-isopropylpiperazin-1-yl)-3,3-dimethyl-8-(1-methylcyclopropyl)isochroman-5-carbonitrile —— C28H35N3O3
(R)-6-(4-(furan-3-carbonyl)-3-isopropylpiperazin-1-yl)-3,3-dimethyl-8-(1-methylcyclopropyl)isochroman-5-carbonitrile
—— (R)-8-cyclohexyl-6-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile 1416268-96-6 C26H38N4O3
(R)-8-cyclohexyl-6-(4-(3-methoxypropanoyl)-3-methylpiperazin-1-yl)-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— (R)-8-cyclopropyl-6-(3-isopropyl-4-(2-methylfuran-3-carbonyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile —— C28H35N3O3
(R)-8-cyclopropyl-6-(3-isopropyl-4-(2-methylfuran-3-carbonyl)piperazin-1-yl)-3,3-dimethylisochroman-5-carbonitrile