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—— (R)-tert-butyl 3-(5-bromo-4-chloro-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidine-1-carboxylate —— C16H20BrClN4O2
(R)-tert-butyl 3-(5-bromo-4-chloro-7H-pyrrolo[2,3-d]pyrimidin-7-yl)piperidine-1-carboxylate
—— (R)-2-(1-bromo-8-chloroimidazolo[1,5-a]pyrazin-3-yl)morpholine-4-carboxylic acid tert-butyl ester —— C15H18BrClN4O3
(R)-2-(1-bromo-8-chloroimidazolo[1,5-a]pyrazin-3-yl)morpholine-4-carboxylic acid tert-butyl ester
—— (R)-6-(2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-2,3,4,5,6,7-hexahydro-1H-cyclopenta[d]pyrimidin-4-yl)nicotinonitrile 1621270-83-4 C20H13F3N4O2
(R)-6-(2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-2,3,4,5,6,7-hexahydro-1H-cyclopenta[d]pyrimidin-4-yl)nicotinonitrile
—— (R)-5-(4,4-difluoro-1-methylpyrrolidin-2-yl)-3-(5-(pyridin-2-ylethynyl)pyridin-2-yl)-1,2,4-oxadiazole 1415143-46-2 C19H15F2N5O
(R)-5-(4,4-difluoro-1-methylpyrrolidin-2-yl)-3-(5-(pyridin-2-ylethynyl)pyridin-2-yl)-1,2,4-oxadiazole
—— (R)-4-(2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-2,3,4,5,6,7-hexahydro-1H-cyclopenta[d]pyrimidin-4-yl)-3-(ethylsulfonyl)benzonitrile 1621270-73-2 C23H18F3N3O4S
(R)-4-(2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-2,3,4,5,6,7-hexahydro-1H-cyclopenta[d]pyrimidin-4-yl)-3-(ethylsulfonyl)benzonitrile
—— (R)-4-(1-(3-(difluoromethyl)phenyl)-2,5-dioxo-2,3,4,5,6,7-hexahydro-1H-cyclopenta [d]pyrimidin-4-yl)-3-(methylsulfonyl)benzonitrile 1621270-85-6 C22H17F2N3O4S
(R)-4-(1-(3-(difluoromethyl)phenyl)-2,5-dioxo-2,3,4,5,6,7-hexahydro-1H-cyclopenta [d]pyrimidin-4-yl)-3-(methylsulfonyl)benzonitrile
—— racemic-4-(4-cyanophenyl)-N-(2-hydroxyethyl)-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidine-3(2H)-carboxamide 1621270-47-0 C24H19F3N4O4
racemic-4-(4-cyanophenyl)-N-(2-hydroxyethyl)-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidine-3(2H)-carboxamide
—— [(R)-(4-methylphenyl)sulfonyl-(1-nitronaphthalen-2-yl)methyl] N,N-diethylcarbamodithioate —— C23H24N2O4S3
[(R)-(4-methylphenyl)sulfonyl-(1-nitronaphthalen-2-yl)methyl] N,N-diethylcarbamodithioate
—— racemic-6-(2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-2,3,4,5,6,7-hexahydro-1H-cyclopenta[d]pyrimidin-4-yl)nicotinonitrile 1621270-77-6 C20H13F3N4O2
racemic-6-(2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-2,3,4,5,6,7-hexahydro-1H-cyclopenta[d]pyrimidin-4-yl)nicotinonitrile
—— rac-2-(2,6-difluorophenyl)-N-(4-((trans)-2,5-dimethyl-1-piperazinyl)-3-pyridinyl)imidazo[1,5-b]pyridazin-7-amine —— C23H23F2N7
rac-2-(2,6-difluorophenyl)-N-(4-((trans)-2,5-dimethyl-1-piperazinyl)-3-pyridinyl)imidazo[1,5-b]pyridazin-7-amine
—— (R)-4-(4-cyanophenyl)-N-methyl-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidine-3(2H)-carboxamide 1621270-57-2 C23H17F3N4O3
(R)-4-(4-cyanophenyl)-N-methyl-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidine-3(2H)-carboxamide
—— (R)-4-(4-cyanophenyl)-N-(2-hydroxyethyl)-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidine-3(2H)-carboxamide 1621270-59-4 C24H19F3N4O4
(R)-4-(4-cyanophenyl)-N-(2-hydroxyethyl)-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidine-3(2H)-carboxamide
—— (R)-4-(4-cyanophenyl)-1-(3-(difluoromethyl)phenyl)-N-(3-hydroxypropyl)-2,5-dioxo-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidine-3(2H)-carboxamide 1621272-60-3 C25H22F2N4O4
(R)-4-(4-cyanophenyl)-1-(3-(difluoromethyl)phenyl)-N-(3-hydroxypropyl)-2,5-dioxo-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidine-3(2H)-carboxamide
—— (R)-4-(3-methyl-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-2,3,4,5,6,7-hexahydro-1H-cyclopenta[d]pyrimidin-4-yl)benzonitrile 1621269-93-9 C22H16F3N3O2
(R)-4-(3-methyl-2,5-dioxo-1-(3-(trifluoromethyl)phenyl)-2,3,4,5,6,7-hexahydro-1H-cyclopenta[d]pyrimidin-4-yl)benzonitrile
—— (R)-N,2-dimethyl-N-(6-methylhept-5-en-2-yl)propane-2-sulfinamide —— C13H27NOS
(R)-N,2-dimethyl-N-(6-methylhept-5-en-2-yl)propane-2-sulfinamide
—— (R)-2-methyl-N-(6-methylhept-5-en-2-yl)propane-2-sulfinamide —— C12H25NOS
(R)-2-methyl-N-(6-methylhept-5-en-2-yl)propane-2-sulfinamide
—— (R)-(4-amino-3,5-dichlorophenyl)-[2-(pyridin-3-ylmethylidene)hydrazinyl]methanol —— C13H12Cl2N4O
(R)-(4-amino-3,5-dichlorophenyl)-[2-(pyridin-3-ylmethylidene)hydrazinyl]methanol
—— (R)-1,2-dimethyl-8-((2,4,5-trifluorobenzyl)oxy)-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620678-96-7 C16H16F3N3O2
(R)-1,2-dimethyl-8-((2,4,5-trifluorobenzyl)oxy)-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((4-fluorobenzyl)oxy)-2-methyl-3,4-dmydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-01-7 C15H16FN3O2
(R)-8-((4-fluorobenzyl)oxy)-2-methyl-3,4-dmydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((3,4-difluorobenzyl)oxy)-2-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-02-8 C15H15F2N3O2
(R)-8-((3,4-difluorobenzyl)oxy)-2-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-2-methyl-8-((3,4,5-trifluorobenzyl)oxy)-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-03-9 C15H14F3N3O2
(R)-2-methyl-8-((3,4,5-trifluorobenzyl)oxy)-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((3,5-difluoro-4-isopropoxybenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-56-2 C19H23F2N3O3
(R)-8-((3,5-difluoro-4-isopropoxybenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((2,3-difluorobenzyl)oxy)-2-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-04-0 C15H15F2N3O2
(R)-8-((2,3-difluorobenzyl)oxy)-2-methyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— [(R)-(4-fluorophenyl)-[[(1S)-1-phenylethyl]amino]methyl]phosphonic acid —— C15H17FNO3P
[(R)-(4-fluorophenyl)-[[(1S)-1-phenylethyl]amino]methyl]phosphonic acid
—— [(R)-(4-fluorophenyl)-phosphonatomethyl]-[(1R)-1-phenylethyl]azanium —— C15H16FNO3P-
[(R)-(4-fluorophenyl)-phosphonatomethyl]-[(1R)-1-phenylethyl]azanium
—— [(R)-(4-fluorophenyl)-phosphonatomethyl]-[(1S)-1-phenylethyl]azanium —— C15H16FNO3P-
[(R)-(4-fluorophenyl)-phosphonatomethyl]-[(1S)-1-phenylethyl]azanium
—— (R)-2-(4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl)-6-cyclopropyl-5-(2-methyl-1-oxoisoindolin-4-yl)nicotinonitrile 1416147-38-0 C26H27N5O2
(R)-2-(4-(cyclopropanecarbonyl)-3-methylpiperazin-1-yl)-6-cyclopropyl-5-(2-methyl-1-oxoisoindolin-4-yl)nicotinonitrile
—— [(R)-[(2S,4R)-5-ethyl-1-azabicyclo[2.2.2]octan-2-yl]-(6-methylquinolin-4-yl)methyl] 4-chlorobenzoate —— C27H29ClN2O2
[(R)-[(2S,4R)-5-ethyl-1-azabicyclo[2.2.2]octan-2-yl]-(6-methylquinolin-4-yl)methyl] 4-chlorobenzoate
—— [(R)-(benzylamino)-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)methyl]phosphonic acid —— C22H21N4O3P
[(R)-(benzylamino)-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)methyl]phosphonic acid
—— (R)-8-((3-fluoro-4-((5-(trifluoromethyl)pyridin-3-yl)oxy)benzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620680-23-0 C22H20F4N4O3
(R)-8-((3-fluoro-4-((5-(trifluoromethyl)pyridin-3-yl)oxy)benzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— [(R)-(benzylamino)-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]methyl]phosphonic acid —— C26H22N3O5P
[(R)-(benzylamino)-[3-(2-oxochromen-3-yl)-1-phenylpyrazol-4-yl]methyl]phosphonic acid
—— (R)-4-(((1,2-dimethyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidin-8-yl)oxy)methyl)benzonitrile 1620678-95-6 C17H18N4O2
(R)-4-(((1,2-dimethyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidin-8-yl)oxy)methyl)benzonitrile
—— (R)-8-((3,5-difluorophenyl)dideuteromethoxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-24-4 C16H17F2N3O2
(R)-8-((3,5-difluorophenyl)dideuteromethoxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((4-(4-chloro-3-fluorophenoxy)-3,5-difluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-37-9 C22H19ClF3N3O3
(R)-8-((4-(4-chloro-3-fluorophenoxy)-3,5-difluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-4-(((2-methyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidin-8-yl)oxy)methyl)benzonitrile 1620679-05-1 C16H16N4O2
(R)-4-(((2-methyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidin-8-yl)oxy)methyl)benzonitrile
—— (R)-1,2-dimethyl-8-((3,4,5-trifluorobenzyl)oxy)-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620678-90-1 C16H16F3N3O2
(R)-1,2-dimethyl-8-((3,4,5-trifluorobenzyl)oxy)-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((2,3-difluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620678-92-3 C16H17F2N3O2
(R)-8-((2,3-difluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-8-((4-(cyclohexyloxy)-3,5-difluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1620679-57-3 C22H27F2N3O3
(R)-8-((4-(cyclohexyloxy)-3,5-difluorobenzyl)oxy)-1,2-dimethyl-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— (R)-2-(3-chloro-4-fluorophenoxy)-5-(((1,2-dimethyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidin-8-yl)oxy)methyl)benzonitrile 1620679-53-9 C23H20ClFN4O3
(R)-2-(3-chloro-4-fluorophenoxy)-5-(((1,2-dimethyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidin-8-yl)oxy)methyl)benzonitrile
—— (R)-tert-butyl 8-chloro-2-methyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidine-1-carboxylate 1620680-37-6 C13H18ClN3O3
(R)-tert-butyl 8-chloro-2-methyl-6-oxo-2,3,4,6-tetrahydro-1H-pyrimido[1,6-a]pyrimidine-1-carboxylate
—— (R)-2-methyl-N-((2R,3R,4S)-5,5,5-trifluoro-2-(2-fluorophenyl)-4-hydroxy-3-(2,2,2-trifluoroethoxy)pentan-2-yl)propane-2-sulfinamide 1620829-28-8 C17H22F7NO3S
(R)-2-methyl-N-((2R,3R,4S)-5,5,5-trifluoro-2-(2-fluorophenyl)-4-hydroxy-3-(2,2,2-trifluoroethoxy)pentan-2-yl)propane-2-sulfinamide
—— (R)-N-[(2R,3R)-3-(2,2-dimethylpropoxy)-2-(2-fluorophenyl)-4-oxobutan-2-yl]-2-methylpropane-2-sulfinamide —— C19H30FNO3S
(R)-N-[(2R,3R)-3-(2,2-dimethylpropoxy)-2-(2-fluorophenyl)-4-oxobutan-2-yl]-2-methylpropane-2-sulfinamide
—— (R)-N-((2S,4S)-2-(5-bromo-2-fluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide 1620828-11-6 C15H20BrF4NO2S
(R)-N-((2S,4S)-2-(5-bromo-2-fluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-2-methyl-N-((2R,3R,4S)-3,5,5,5-tetrafluoro-2-(2-fluorophenyl)-4-hydroxy-3-methylpentan-2-yl)propane-2-sulfinamide 1620828-07-0 C16H22F5NO2S
(R)-2-methyl-N-((2R,3R,4S)-3,5,5,5-tetrafluoro-2-(2-fluorophenyl)-4-hydroxy-3-methylpentan-2-yl)propane-2-sulfinamide
—— (R)-N-((2S,4R)-2-(4-bromothiophen-2-yl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide 1620828-19-4 C13H19BrF3NO2S2
(R)-N-((2S,4R)-2-(4-bromothiophen-2-yl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-((2R,3R)-3-fluoro-2-(2-fluorophenyl)-3-methyl-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide 1620828-01-4 C15H21F2NO2S
(R)-N-((2R,3R)-3-fluoro-2-(2-fluorophenyl)-3-methyl-4-oxobutan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-((2S,4R)-2-(5-bromo-2,4-difluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide 1620828-17-2 C15H19BrF5NO2S
(R)-N-((2S,4R)-2-(5-bromo-2,4-difluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-((2S,4R)-2-(5-bromo-2-fluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide 1620828-13-8 C15H20BrF4NO2S
(R)-N-((2S,4R)-2-(5-bromo-2-fluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-N-((2S,4S)-2-(5-bromo-2,4-difluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide 1620828-15-0 C15H19BrF5NO2S
(R)-N-((2S,4S)-2-(5-bromo-2,4-difluorophenyl)-5,5,5-trifluoro-4-hydroxypentan-2-yl)-2-methylpropane-2-sulfinamide
—— (R)-2-methyl-N-((2R,3R,4R)-3,5,5,5-tetrafluoro-2-(2-fluorophenyl)-4-hydroxy-3-methylpentan-2-yl)propane-2-sulfinamide 1620828-09-2 C16H22F5NO2S
(R)-2-methyl-N-((2R,3R,4R)-3,5,5,5-tetrafluoro-2-(2-fluorophenyl)-4-hydroxy-3-methylpentan-2-yl)propane-2-sulfinamide