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—— (R,E)-N-((2-(4-chlorophenyl)thiazol-5-yl)methylene)-2-methyl propane-2-sulfinamide —— C14H15ClN2OS2
(R,E)-N-((2-(4-chlorophenyl)thiazol-5-yl)methylene)-2-methyl propane-2-sulfinamide
—— (R)-2-methyl-N-((S)-1-(2-(6-(trifluoromethyl)pyridin-3-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide —— C15H18F3N3OS2
(R)-2-methyl-N-((S)-1-(2-(6-(trifluoromethyl)pyridin-3-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide
—— (R,E)-N-((2-(4-(difluoromethyl)phenyl)thiazol-5-yl)methylene)-2-methylpropane-2-sulfinamide —— C15H16F2N2OS2
(R,E)-N-((2-(4-(difluoromethyl)phenyl)thiazol-5-yl)methylene)-2-methylpropane-2-sulfinamide
—— (R)-2-methyl-N-((S)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethyl)propane-2-sulfinamide —— C14H25N3O3S
(R)-2-methyl-N-((S)-1-(5-(morpholinomethyl)isoxazol-3-yl)ethyl)propane-2-sulfinamide
—— (R)-2-methyl-N-((S)-1-(2-(pyridin-2-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide —— C14H19N3OS2
(R)-2-methyl-N-((S)-1-(2-(pyridin-2-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide
—— (R,E)-N-((1-(4-chlorophenyl)-1H-pyrazol-4-yl)methylene)-2-methyl propane-2-sulfinamide —— C14H16ClN3OS
(R,E)-N-((1-(4-chlorophenyl)-1H-pyrazol-4-yl)methylene)-2-methyl propane-2-sulfinamide
—— (R)-2-methyl-N-((S)-1-(2-(pyridin-3-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide —— C14H19N3OS2
(R)-2-methyl-N-((S)-1-(2-(pyridin-3-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide
—— (R,E)-N-((1-(4-fluorophenyl)-1H-pyrazol-4-yl)methylene)-2-methyl propane-2-sulfinamide —— C14H16FN3OS
(R,E)-N-((1-(4-fluorophenyl)-1H-pyrazol-4-yl)methylene)-2-methyl propane-2-sulfinamide
—— (R,E)-2-methyl-N-((5-(morpholinomethyl)isoxazol-3-yl)methylene)propane-2-sulfinamide —— C13H21N3O3S
(R,E)-2-methyl-N-((5-(morpholinomethyl)isoxazol-3-yl)methylene)propane-2-sulfinamide
—— (R)-N-((S)-1-(2-(4-(difluoromethyl)phenyl)thiazol-5-yl)ethyl)-2-methylpropane-2-sulfinamide —— C16H20F2N2OS2
(R)-N-((S)-1-(2-(4-(difluoromethyl)phenyl)thiazol-5-yl)ethyl)-2-methylpropane-2-sulfinamide
—— (R)-methyl 2-(4-((2-(hydroxymethyl)-5-oxopyrrolidin-1-yl)methyl)phenyl)acetate —— C15H19NO4
(R)-methyl 2-(4-((2-(hydroxymethyl)-5-oxopyrrolidin-1-yl)methyl)phenyl)acetate
—— (R)-2-methyl-N-((S)-1-(2-(2-(trifluoromethyl)pyridin-4-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide —— C15H18F3N3OS2
(R)-2-methyl-N-((S)-1-(2-(2-(trifluoromethyl)pyridin-4-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide
—— (R,E)-2-methyl-N-((2-(6-methylpyridin-3-yl)thiazol-5-yl) methylene)propane-2-sulfinamide —— C14H17N3OS2
(R,E)-2-methyl-N-((2-(6-methylpyridin-3-yl)thiazol-5-yl) methylene)propane-2-sulfinamide
—— (R)-N-((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)-2-methylpropane-2-sulfinamide —— C15H20ClN3OS
(R)-N-((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)-2-methylpropane-2-sulfinamide
—— (R)-2-methyl-N-((S)-1-(2-(pyridin-4-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide —— C14H19N3OS2
(R)-2-methyl-N-((S)-1-(2-(pyridin-4-yl)thiazol-5-yl)ethyl)propane-2-sulfinamide
—— (R,E)-2-methyl-N-((5-phenylisoxazol-3-yl)methylene)propane-2-sulfinamide —— C14H16N2O2S
(R,E)-2-methyl-N-((5-phenylisoxazol-3-yl)methylene)propane-2-sulfinamide
—— (R)-methyl 5-(3-(2-formyl-5-oxopyrrolidin-1-yl)prop-1-yn-1-yl)thiophene-2-carboxylate —— C14H13NO4S
(R)-methyl 5-(3-(2-formyl-5-oxopyrrolidin-1-yl)prop-1-yn-1-yl)thiophene-2-carboxylate
—— (R,E)-N-((5-(4-fluorophenyl)isoxazol-3-yl)methylene)-2-methyl propane-2-sulfinamide —— C14H15FN2O2S
(R,E)-N-((5-(4-fluorophenyl)isoxazol-3-yl)methylene)-2-methyl propane-2-sulfinamide
—— (R)-tert-butyl 1-(3-(5-(methoxycarbonyl)-thiophen-2-yl)prop-2-yn-1-yl)-5-oxopyrrolidine-2-carboxylate —— C18H21NO5S
(R)-tert-butyl 1-(3-(5-(methoxycarbonyl)-thiophen-2-yl)prop-2-yn-1-yl)-5-oxopyrrolidine-2-carboxylate
—— (R,Z)-1-(3-(5-(methoxycarbonyl)thiophen-2-yl)allyl)-5-oxopyrrolidine-2-carboxylic acid —— C14H15NO5S
(R,Z)-1-(3-(5-(methoxycarbonyl)thiophen-2-yl)allyl)-5-oxopyrrolidine-2-carboxylic acid
—— (R)-4-(N-benzyl-1'-(methoxycarbonyl)-1-((5-methoxythiazolo[5,4-b]pyridin-2-yl)carbamoyl)spiro[indoline-3,3'-pyrrolidin]-5-ylsulfonamido)butyric acid —— C32H34N6O8S2
(R)-4-(N-benzyl-1'-(methoxycarbonyl)-1-((5-methoxythiazolo[5,4-b]pyridin-2-yl)carbamoyl)spiro[indoline-3,3'-pyrrolidin]-5-ylsulfonamido)butyric acid
—— (R)-5-cyano-N1-(5-fluorothiazol-2-yl)-N1'-methylspiro[indoline-3,3’-pyrrolidine]-1,1'-dicarboxamide —— C18H17FN6O2S
(R)-5-cyano-N1-(5-fluorothiazol-2-yl)-N1'-methylspiro[indoline-3,3’-pyrrolidine]-1,1'-dicarboxamide
—— (R)-5-chloro-N-(5-chlorothiazol-2-yl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide —— C15H14Cl2N4OS
(R)-5-chloro-N-(5-chlorothiazol-2-yl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide
—— (R)-2-((2-(5-bromo-1'-(methoxycarbonyl)spiro[indoline-3,3'-pyrrolidin]-1-ylcarboxamido)thiazol-5-yl)thio)acetic acid —— C19H19BrN4O5S2
(R)-2-((2-(5-bromo-1'-(methoxycarbonyl)spiro[indoline-3,3'-pyrrolidin]-1-ylcarboxamido)thiazol-5-yl)thio)acetic acid
—— (R)-N1-(5-methoxythiazol-2-yl)-N1'-methyl-5-(trifluoromethyl)spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide —— C19H20F3N5O3S
(R)-N1-(5-methoxythiazol-2-yl)-N1'-methyl-5-(trifluoromethyl)spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide
—— (R)-5-chloro-N1-(5-chlorothiazol-2-yl)-N1'-methyl spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide —— C17H17Cl2N5O2S
(R)-5-chloro-N1-(5-chlorothiazol-2-yl)-N1'-methyl spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide
—— (R)-N1-(5-chlorothiazol-2-yl)-5-cyano-N1'-methylspiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide —— C18H17ClN6O2S
(R)-N1-(5-chlorothiazol-2-yl)-5-cyano-N1'-methylspiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide
—— (R)-5-chloro-N1-(5-methoxythiazol-2-yl)-N1'-methylspiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide —— C18H20ClN5O3S
(R)-5-chloro-N1-(5-methoxythiazol-2-yl)-N1'-methylspiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide
—— (R)-3-((2-(1'-acetyl-5-chlorospiro[indoline-3,3'-pyrrolidin]-1-ylcarboxamido)thiazol-5-yl)thio)propionic acid —— C20H21ClN4O4S2
(R)-3-((2-(1'-acetyl-5-chlorospiro[indoline-3,3'-pyrrolidin]-1-ylcarboxamido)thiazol-5-yl)thio)propionic acid
—— (R)-N1'-methyl-N1-(5-methylpyrazin-2-yl)-5-(trifluoromethyl)spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide —— C20H21F3N6O2
(R)-N1'-methyl-N1-(5-methylpyrazin-2-yl)-5-(trifluoromethyl)spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide
—— (R)-3-(N-benzyl-1'-(methoxycarbonyl)-1-((5-methoxythiazolo[5,4-b]pyridin-2-yl)carbamoyl)spiro[indoline-3,3'-pyrrolidin]-5-ylsulfonamido)propionic acid —— C31H32N6O8S2
(R)-3-(N-benzyl-1'-(methoxycarbonyl)-1-((5-methoxythiazolo[5,4-b]pyridin-2-yl)carbamoyl)spiro[indoline-3,3'-pyrrolidin]-5-ylsulfonamido)propionic acid
—— (R)-5-chloro-N-(5-chlorothiazol-2-yl)-1'-(2-hydroxyacetyl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide —— C17H16Cl2N4O3S
(R)-5-chloro-N-(5-chlorothiazol-2-yl)-1'-(2-hydroxyacetyl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide
—— (R)-5-chloro-N1-(5-fluorothiazol-2-yl)-N1'-methyl spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide —— C17H17ClFN5O2S
(R)-5-chloro-N1-(5-fluorothiazol-2-yl)-N1'-methyl spiro[indoline-3,3'-pyrrolidine]-1,1'-dicarboxamide
—— (R)-1'-acetyl-N-(5-methoxythiazol-2-yl)-5-(trifluoromethyl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide —— C19H19F3N4O3S
(R)-1'-acetyl-N-(5-methoxythiazol-2-yl)-5-(trifluoromethyl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide
—— (R)-2-methoxy-N-(3-(2,2,2-trifluoro-1-(6-(oxazol-5-yl) pyridin-3-yl)ethoxy)quinoxalin-2-yl)ethanesulfonamide —— C21H18F3N5O5S
(R)-2-methoxy-N-(3-(2,2,2-trifluoro-1-(6-(oxazol-5-yl) pyridin-3-yl)ethoxy)quinoxalin-2-yl)ethanesulfonamide
—— (R)-1'-acetyl-5-chloro-N-(5-fluorothiazol-2-yl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide —— C17H16ClFN4O2S
(R)-1'-acetyl-5-chloro-N-(5-fluorothiazol-2-yl)spiro[indoline-3,3'-pyrrolidine]-1-carboxamide
—— (R)-2-((2-(1'-acetyl-5-bromospiro[indoline-3,3'-pyrrolidin]-1-ylcarboxamido)thiazol-5-yl)thio)acetic acid —— C19H19BrN4O4S2
(R)-2-((2-(1'-acetyl-5-bromospiro[indoline-3,3'-pyrrolidin]-1-ylcarboxamido)thiazol-5-yl)thio)acetic acid
—— (R)-3-(tert-butoxy)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)-2-methylpropanamide —— C19H25F3N4O2
(R)-3-(tert-butoxy)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)-2-methylpropanamide
—— (R)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)-3-phenylbutanamide —— C21H21F3N4O
(R)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)-3-phenylbutanamide
—— (R)-N-(5-chloro-3-(4-fluorophenyl)-3H-imidazo[4,5-b]pyridin-2-yl)-2-(6,6-dimethyltetrahydro-2H-pyran-2-yl)acetamide —— C21H22ClFN4O2
(R)-N-(5-chloro-3-(4-fluorophenyl)-3H-imidazo[4,5-b]pyridin-2-yl)-2-(6,6-dimethyltetrahydro-2H-pyran-2-yl)acetamide
—— (R)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)-2-(6,6-dimethyltetrahydro2H-pyran-2-yl)acetamide —— C20H25F3N4O2
(R)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)-2-(6,6-dimethyltetrahydro2H-pyran-2-yl)acetamide
—— (R)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)-2-(5,5-dimethyltetrahydrofuran-2-yl)acetamide —— C19H23F3N4O2
(R)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)-2-(5,5-dimethyltetrahydrofuran-2-yl)acetamide
—— (R)-N-(3-(tert-butyl)-5-chloro-3H-imidazo[4,5-b]pyridin-2-yl)-2-(6,6-dimethyltetrahydro2H-pyran-2-yl)acetamide —— C19H27ClN4O2
(R)-N-(3-(tert-butyl)-5-chloro-3H-imidazo[4,5-b]pyridin-2-yl)-2-(6,6-dimethyltetrahydro2H-pyran-2-yl)acetamide
—— (R)-3-(tert-butoxy)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)butanamide —— C19H25F3N4O2
(R)-3-(tert-butoxy)-N-(3-cyclobutyl-5-(trifluoromethyl)-3H-imidazo[4,5-b]pyridin-2-yl)butanamide
—— (R)-N-(5-chloro-3-cyclobutyl-3H-imidazo[4,5-b]pyridin-2-yl)-2-(5,5-dimethyltetrahydrofuran-2-yl)acetamide —— C18H23ClN4O2
(R)-N-(5-chloro-3-cyclobutyl-3H-imidazo[4,5-b]pyridin-2-yl)-2-(5,5-dimethyltetrahydrofuran-2-yl)acetamide
—— (R)-2-oxo-3-(tetrahydrofuran-3-yl)imidazolidine-1-carbonyl chloride —— C8H11ClN2O3
(R)-2-oxo-3-(tetrahydrofuran-3-yl)imidazolidine-1-carbonyl chloride
—— (R/S)-Benzyl 7-azabicyclo[2.2.1]hept-5-ene-7-carboxylate —— C14H15NO2
(R/S)-Benzyl 7-azabicyclo[2.2.1]hept-5-ene-7-carboxylate
—— (R)-[(3S)-1-(7-morpholin-4-yl-1,2,3-benzotriazin-4-yl)piperidin-3-yl]-(1-propan-2-ylpyrazol-4-yl)methanol —— C23H31N7O2
(R)-[(3S)-1-(7-morpholin-4-yl-1,2,3-benzotriazin-4-yl)piperidin-3-yl]-(1-propan-2-ylpyrazol-4-yl)methanol
—— (R)-[4-(difluoromethyl)-1,3-thiazol-2-yl]-[(3S)-1-(7-morpholin-4-yl-1,2,3-benzotriazin-4-yl)piperidin-3-yl]methanol —— C21H24F2N6O2S
(R)-[4-(difluoromethyl)-1,3-thiazol-2-yl]-[(3S)-1-(7-morpholin-4-yl-1,2,3-benzotriazin-4-yl)piperidin-3-yl]methanol
—— (R)-[3-[(1-benzylbenzimidazol-2-yl)amino]-5-methyl-2-phenyl-1H-pyrazol-2-ium-4-yl]-pyridin-4-ylmethanol —— C30H27N6O+
(R)-[3-[(1-benzylbenzimidazol-2-yl)amino]-5-methyl-2-phenyl-1H-pyrazol-2-ium-4-yl]-pyridin-4-ylmethanol