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中文名称 英文名称 CAS号 化学式 结构式图片
—— rac-(3aR,8S,8aR)-8-hydroxy-3a-methyl-3,3a,8,8a-tetrahydro-2H-indeno[1,2-d][1,3]oxazol-2-one —— C11H11NO3
rac-(3aR,8S,8aR)-8-hydroxy-3a-methyl-3,3a,8,8a-tetrahydro-2H-indeno[1,2-d][1,3]oxazol-2-one
—— rac-8-[(2,6-difluorobenzyl)oxy]-N-[(1R,2S)-2-hydroxy-1-(hydroxymethyl)-2,3-dihydro-1H-indan-1-yl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C26H23F2N3O4
rac-8-[(2,6-difluorobenzyl)oxy]-N-[(1R,2S)-2-hydroxy-1-(hydroxymethyl)-2,3-dihydro-1H-indan-1-yl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— Racemic-3-amino-5-(3-fluorophenyl)-9-methyl-1H-benzo[e][1,4]diazepin-2(3H)-one —— C16H14FN3O
Racemic-3-amino-5-(3-fluorophenyl)-9-methyl-1H-benzo[e][1,4]diazepin-2(3H)-one
—— rac-methyl (1R,2R)-1-amino-2,3-dihydro-1H-indene-2-carboxylate —— C11H13NO2
rac-methyl (1R,2R)-1-amino-2,3-dihydro-1H-indene-2-carboxylate
—— Rel-methyl (1S,2S)-1-amino-1,2,3,4-tetrahydronaphthalene-2-carboxylate hydrochloride —— C12H16ClNO2
Rel-methyl (1S,2S)-1-amino-1,2,3,4-tetrahydronaphthalene-2-carboxylate hydrochloride
—— [(R)-(4-chlorophenyl)-phenylmethyl] 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-oxobutanoate —— C25H21ClO5
[(R)-(4-chlorophenyl)-phenylmethyl] 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-oxobutanoate
—— (R)-(2-(((4-amino-2,2-dioxido-1H-benzo[c][1,2,6]thiadiazin-5-yl)oxy)methyl)piperidin-1-yl)(pyridin-4-yl)methanone 1554633-35-0 C19H21N5O4S
(R)-(2-(((4-amino-2,2-dioxido-1H-benzo[c][1,2,6]thiadiazin-5-yl)oxy)methyl)piperidin-1-yl)(pyridin-4-yl)methanone
—— (R)-1-(3-(((4-amino-2,2-dioxido-1H-benzo[c][1,2,6]thiadiazin-5-yl)oxy)methyl)piperidin-1-yl)-3-methylbutan-1-one 1554633-18-9 C18H26N4O4S
(R)-1-(3-(((4-amino-2,2-dioxido-1H-benzo[c][1,2,6]thiadiazin-5-yl)oxy)methyl)piperidin-1-yl)-3-methylbutan-1-one
—— (R)-2-sulfamoylamino-6-((1-(3-methylbutanoyl)piperidin-3-yl)methoxy)benzonitrile 1554633-20-3 C18H26N4O4S
(R)-2-sulfamoylamino-6-((1-(3-methylbutanoyl)piperidin-3-yl)methoxy)benzonitrile
—— (R)-2-((2-cyano-3-(sulfamoylamino)phenoxy)methyl)-N-(pyridin-4-ylmethyl)piperidine-1-carboxamide 1554632-85-7 C20H24N6O4S
(R)-2-((2-cyano-3-(sulfamoylamino)phenoxy)methyl)-N-(pyridin-4-ylmethyl)piperidine-1-carboxamide
—— (R)-7-chloro-N-(2,6-difluorophenyl)-2-((S)-3-methyl-2-((S)-2-(methylamino)propanamido)butanoyl)-1,2,3,4-tetrahydroisoquinoline-1-carboxamide 1567382-11-9 C25H29ClF2N4O3
(R)-7-chloro-N-(2,6-difluorophenyl)-2-((S)-3-methyl-2-((S)-2-(methylamino)propanamido)butanoyl)-1,2,3,4-tetrahydroisoquinoline-1-carboxamide
—— rac-(4aR,8aR)-6-[3-(4,6-dimethyl-1H-benzimidazol-2-yl)-5-(3,5-dimethylphenyl)-4-pyridinyl]octahydro-1H-pyrido[3,4-b][1,4]oxazine —— C29H33N5O
rac-(4aR,8aR)-6-[3-(4,6-dimethyl-1H-benzimidazol-2-yl)-5-(3,5-dimethylphenyl)-4-pyridinyl]octahydro-1H-pyrido[3,4-b][1,4]oxazine
—— rac-(3R, 4S)-1-[3-(3,5-dimethylphenyl)-5-(6-methyl-1H-benzimidazol-2-yl)-4-pyridinyl]-3-fluoro-4-piperidinamine —— C26H28FN5
rac-(3R, 4S)-1-[3-(3,5-dimethylphenyl)-5-(6-methyl-1H-benzimidazol-2-yl)-4-pyridinyl]-3-fluoro-4-piperidinamine
—— (R)-6-chloro-N-(2,6-difluorophenyl)-2-((S)-3-methyl-2-((S)-2-(methylamino)propanamido)butanoyl)-1,2,3,4-tetrahydroisoquinoline-1-carboxamide 1567382-46-0 C25H29ClF2N4O3
(R)-6-chloro-N-(2,6-difluorophenyl)-2-((S)-3-methyl-2-((S)-2-(methylamino)propanamido)butanoyl)-1,2,3,4-tetrahydroisoquinoline-1-carboxamide
—— (R)-N-(2,6-difluorophenyl)-7-fluoro-2-((S)-3-methyl-2-((S)-2-(methylamino) propanamido)butanoyl)-1,2,3,4-tetrahydroisoquinoline-1-carboxamide 1567382-10-8 C25H29F3N4O3
(R)-N-(2,6-difluorophenyl)-7-fluoro-2-((S)-3-methyl-2-((S)-2-(methylamino) propanamido)butanoyl)-1,2,3,4-tetrahydroisoquinoline-1-carboxamide
—— rac-(3R,4S)-4-amino-1-[3-(3,5-dimethoxyphenyl)-5-(4,6-dimethyl-1H-benzimidazol-2-yl)-4-pyridinyl]-3-piperidinol —— C27H31N5O3
rac-(3R,4S)-4-amino-1-[3-(3,5-dimethoxyphenyl)-5-(4,6-dimethyl-1H-benzimidazol-2-yl)-4-pyridinyl]-3-piperidinol
—— (R)-2-((4-(1-(oxetan-3-yl)piperidin-4-yl)-6-(2-(trifluoromethyl)pyrrolidin-1-yl)pyridin-2-yl)amino)isonicotinonitrile —— C24H27F3N6O
(R)-2-((4-(1-(oxetan-3-yl)piperidin-4-yl)-6-(2-(trifluoromethyl)pyrrolidin-1-yl)pyridin-2-yl)amino)isonicotinonitrile
—— (R)-2-(4-(1-acetylpiperidin-4-yl)-6-(2-(methylpyrrolidin-1-yl)pyridin-2-yl)amino)isonicotinonitrile —— C23H28N6O
(R)-2-(4-(1-acetylpiperidin-4-yl)-6-(2-(methylpyrrolidin-1-yl)pyridin-2-yl)amino)isonicotinonitrile
—— (R)-2-((4-(4-cyanotetrahydro-2H-pyran-4-yl)-6-(2-methylpyrrolidin-1-yl)pyridin-2-yl)amino)isonicotinonitrile —— C22H24N6O
(R)-2-((4-(4-cyanotetrahydro-2H-pyran-4-yl)-6-(2-methylpyrrolidin-1-yl)pyridin-2-yl)amino)isonicotinonitrile
—— (R)-6-(2-methylpyrrolidin-1-yl)-4-(1-(methylsulfonyl)piperidin-4-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)pyridin-2-amine —— C22H28F3N5O2S
(R)-6-(2-methylpyrrolidin-1-yl)-4-(1-(methylsulfonyl)piperidin-4-yl)-N-(4-(trifluoromethyl)pyridin-2-yl)pyridin-2-amine
—— (R)-1-Methanesulfonyl-pyrrolidine-2-carboxylic acid —— C6H11NO4S
(R)-1-Methanesulfonyl-pyrrolidine-2-carboxylic acid
—— (R)-N-((4-difluoromethyl)pyridin-2-yl)-6-(2-methylpyrrolidin-1-yl)-4-(1-(oxetan-3-yl)piperidin-4-yl)pyridin-2-amine —— C24H31F2N5O
(R)-N-((4-difluoromethyl)pyridin-2-yl)-6-(2-methylpyrrolidin-1-yl)-4-(1-(oxetan-3-yl)piperidin-4-yl)pyridin-2-amine
—— (R)-2-(6-(2-(methylpyrrolidin-1-yl)-4-(1-(oxetan-3-yl)piperidin-4-yl)pyridin-2-yl)amino)isonicotinonitrile —— C24H30N6O
(R)-2-(6-(2-(methylpyrrolidin-1-yl)-4-(1-(oxetan-3-yl)piperidin-4-yl)pyridin-2-yl)amino)isonicotinonitrile
—— (R)-1-(4-(2-(2-methylpyrrolidin-1-yl)-6-((4-(trifluoromethyl)pyridin-2-yl)amino)pyridin-4-yl)piperidin-1-yl)ethanone —— C23H28F3N5O
(R)-1-(4-(2-(2-methylpyrrolidin-1-yl)-6-((4-(trifluoromethyl)pyridin-2-yl)amino)pyridin-4-yl)piperidin-1-yl)ethanone
—— (R)-N-(4-methylpyridin-2-yl)-6-(2-methylpyrrolidin-1-yl)-4-(1-(oxetan-3-yl)piperidin-4-yl)pyridin-2-amine —— C24H33N5O
(R)-N-(4-methylpyridin-2-yl)-6-(2-methylpyrrolidin-1-yl)-4-(1-(oxetan-3-yl)piperidin-4-yl)pyridin-2-amine
—— (R)-1-(4-(2-((4-cyclopropylpyridin-2-yl)amino)-6-(2-methylpyrrolidin-1-yl)pyridin-4-yl)piperidin-1-yl)ethanone —— C25H33N5O
(R)-1-(4-(2-((4-cyclopropylpyridin-2-yl)amino)-6-(2-methylpyrrolidin-1-yl)pyridin-4-yl)piperidin-1-yl)ethanone
—— (R)-2-(4-(2-(2-methylpyrrolidin-1-yl)-6-((4-(trifluoromethyl)pyridin-2-yl)amino)pyridin-4-yl)piperidin-1-yl)ethanol —— C23H30F3N5O
(R)-2-(4-(2-(2-methylpyrrolidin-1-yl)-6-((4-(trifluoromethyl)pyridin-2-yl)amino)pyridin-4-yl)piperidin-1-yl)ethanol
—— (R)-2-amino-3-(3-ethylbenzamido)propanoic acid —— C12H16N2O3
(R)-2-amino-3-(3-ethylbenzamido)propanoic acid
—— (R)-5-(5-bromo-2-fluoro-phenyl)-2,2,5-trimethyl-1,1-dioxo-1λ6-thiomorpholin-3-thione —— C13H15BrFNO2S2
(R)-5-(5-bromo-2-fluoro-phenyl)-2,2,5-trimethyl-1,1-dioxo-1λ6-thiomorpholin-3-thione
—— (R)-4-(1-(4-(3-methoxypyrrolidin-1-yl)-2-methyl-5-(5-methyl-4H-1,2,4-triazol-3-yl)benzoyl)piperidin-4-yl)benzonitrile 1533437-29-4 C28H32N6O2
(R)-4-(1-(4-(3-methoxypyrrolidin-1-yl)-2-methyl-5-(5-methyl-4H-1,2,4-triazol-3-yl)benzoyl)piperidin-4-yl)benzonitrile
—— (R)-4-(1-(2-methyl-5-(5-methyl-4H-1,2,4-triazol-3-yl)-4-(2-methylpyrrolidin-1-yl)benzoyl)piperidin-4-yl)benzonitrile 1533437-30-7 C28H32N6O
(R)-4-(1-(2-methyl-5-(5-methyl-4H-1,2,4-triazol-3-yl)-4-(2-methylpyrrolidin-1-yl)benzoyl)piperidin-4-yl)benzonitrile
—— (R)-1-(5-((4-((1R,4R,5R)-5-Amino-2-azabicyclo[2.2.1]heptan-2-yl)-6-fluoro-8-(methylamino)-9H-pyrimido[4,5-b]indol-2-yl)oxy)pyrimidin-2-yl)ethyl ethyl hydrogen phosphate —— C25H30FN8O5P
(R)-1-(5-((4-((1R,4R,5R)-5-Amino-2-azabicyclo[2.2.1]heptan-2-yl)-6-fluoro-8-(methylamino)-9H-pyrimido[4,5-b]indol-2-yl)oxy)pyrimidin-2-yl)ethyl ethyl hydrogen phosphate
—— (R)-1-(5-((4-((1R,4R,5R)-5-amino-2-azabicyclo[2.2.1]heptan-2-yl)-5,6-difluoro-8-(methylamino)-9H-pyrimido[4,5-b]indol-2-yl)oxy)pyrimidin-2-yl)ethyl dihydrogen phosphate —— C23H25F2N8O5P
(R)-1-(5-((4-((1R,4R,5R)-5-amino-2-azabicyclo[2.2.1]heptan-2-yl)-5,6-difluoro-8-(methylamino)-9H-pyrimido[4,5-b]indol-2-yl)oxy)pyrimidin-2-yl)ethyl dihydrogen phosphate
—— rac-(2R,3S)-2-ethylpyrrolidin-3-amine —— C6H14N2
rac-(2R,3S)-2-ethylpyrrolidin-3-amine
—— rel-((1R,8S,9s)-Bicyclo[6.1.0]non-4-yn-9-yl)methanamine —— C10H15N
rel-((1R,8S,9s)-Bicyclo[6.1.0]non-4-yn-9-yl)methanamine
—— (R)-1-((3-(trifluoromethyl)phenyl)sulfonyl)piperidine-3-carboxylic acid —— C13H14F3NO4S
(R)-1-((3-(trifluoromethyl)phenyl)sulfonyl)piperidine-3-carboxylic acid
—— (R)-2-(2-Oxo-ethyl)-azetidine-1-carboxylic acid tert-butyl ester —— C10H17NO3
(R)-2-(2-Oxo-ethyl)-azetidine-1-carboxylic acid tert-butyl ester
—— (R)-2-Amino-7-methyloctanoic acid —— C9H19NO2
(R)-2-Amino-7-methyloctanoic acid
—— (R,S)-2-bromo-5-(3-chloro-4-fluoro-phenyl)-6-(4-chloro-phenyl)-1-((R)-2-methoxy-1-methyl-ethyl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C22H18BrCl2FN2O2
(R,S)-2-bromo-5-(3-chloro-4-fluoro-phenyl)-6-(4-chloro-phenyl)-1-((R)-2-methoxy-1-methyl-ethyl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— (R)-1-(1-(2-chloro-6-(trifluoromethyl)benzoyl)-6-(3-methoxypyrrolidine-1-carbonyl)-1H-indazol-3-yl)piperidine-4-carboxylic acid 1561771-55-8 C27H26ClF3N4O5
(R)-1-(1-(2-chloro-6-(trifluoromethyl)benzoyl)-6-(3-methoxypyrrolidine-1-carbonyl)-1H-indazol-3-yl)piperidine-4-carboxylic acid
—— (R,S)-5-(5-chloro-1-methyl-6-oxo-1,6-dihydro-pyridin-3-yl)-6-(4-chloro-phenyl)-2-(2,4-dimethoxy-pyrimidin-5-yl)-1-((R)-2-methoxy-1-methyl-ethyl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C28H27Cl2N5O5
(R,S)-5-(5-chloro-1-methyl-6-oxo-1,6-dihydro-pyridin-3-yl)-6-(4-chloro-phenyl)-2-(2,4-dimethoxy-pyrimidin-5-yl)-1-((R)-2-methoxy-1-methyl-ethyl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— (R,S)-2-(2-amino-4-methoxy-pyrimidin-5-yl)-5-(3-chloro-4-fluoro-phenyl)-6-(4-chloro-phenyl)-1-((R)-2-methoxy-1-methyl-ethyl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C27H24Cl2FN5O3
(R,S)-2-(2-amino-4-methoxy-pyrimidin-5-yl)-5-(3-chloro-4-fluoro-phenyl)-6-(4-chloro-phenyl)-1-((R)-2-methoxy-1-methyl-ethyl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— (R,S)-4-[2-bromo-5-(5-chloro-1-methyl-6-oxo-1,6-dihydro-pyridin-3-yl)-1-((R)-2-methoxy-1-methyl-ethyl)-4-oxo-1,4,5,6-tetrahydro-pyrrolo[3,4-b]pyrrol-6-yl]-benzonitrile —— C23H20BrClN4O3
(R,S)-4-[2-bromo-5-(5-chloro-1-methyl-6-oxo-1,6-dihydro-pyridin-3-yl)-1-((R)-2-methoxy-1-methyl-ethyl)-4-oxo-1,4,5,6-tetrahydro-pyrrolo[3,4-b]pyrrol-6-yl]-benzonitrile
—— (R,S)-2-bromo-5-(5-chloro-1-methyl-6-oxo-1,6-dihydro-pyridin-3-yl)-6-(4-chloro-phenyl)-1-((R)-2-methoxy-1-methyl-ethyl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one —— C22H20BrCl2N3O3
(R,S)-2-bromo-5-(5-chloro-1-methyl-6-oxo-1,6-dihydro-pyridin-3-yl)-6-(4-chloro-phenyl)-1-((R)-2-methoxy-1-methyl-ethyl)-5,6-dihydro-1H-pyrrolo[3,4-b]pyrrol-4-one
—— (R)-2-[[7-(3-aminopiperidin-1-yl)-3,5-dimethyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl]methyl]naphthonitrile trifluoroacetate —— C2HF3O2*C25H26N6O
(R)-2-[[7-(3-aminopiperidin-1-yl)-3,5-dimethyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl]methyl]naphthonitrile trifluoroacetate
—— (R)-2-[[7-(3-aminopyrrolidin-1-yl)-3,5-dimethyl-2-oxo-2,3.dihydro-1H-imidazo[4, 5-b]pyridin-1-yl]methyl]benzonitrile trifluoroacetate 1314944-21-2 C2HF3O2*C20H22N6O
(R)-2-[[7-(3-aminopyrrolidin-1-yl)-3,5-dimethyl-2-oxo-2,3.dihydro-1H-imidazo[4, 5-b]pyridin-1-yl]methyl]benzonitrile trifluoroacetate
—— (R)-(-)-ethyl 2-methyl-5-phenylpentanoate 1263428-82-5 C14H20O2
(R)-(-)-ethyl 2-methyl-5-phenylpentanoate
—— (R)-methyl 4-(2-(3,3-difluoro-5-formyl-2-oxopyrrolidin-1-yl)ethyl)benzoate 1544279-30-2 C15H15F2NO4
(R)-methyl 4-(2-(3,3-difluoro-5-formyl-2-oxopyrrolidin-1-yl)ethyl)benzoate
—— (R,Z)-methyl 5-(3-(3,3-difluoro-5-formyl-2-oxopyrrolidin-1-yl)prop-1-en-1-yl)thiophene-2-carboxylate 1544279-42-6 C14H13F2NO4S
(R,Z)-methyl 5-(3-(3,3-difluoro-5-formyl-2-oxopyrrolidin-1-yl)prop-1-en-1-yl)thiophene-2-carboxylate
—— (R)-methyl 5-(3-(3,3-difluoro-5-formyl-2-oxopyrrolidin-1-yl)prop-1-yn-1-yl)thiophene-2-carboxylate 1544279-37-9 C14H11F2NO4S
(R)-methyl 5-(3-(3,3-difluoro-5-formyl-2-oxopyrrolidin-1-yl)prop-1-yn-1-yl)thiophene-2-carboxylate