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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-N-(2-(3-methyl-5-oxo-2,3,4,5-tetrahydro-1H-benzo[4,5]thieno[3,2-e][1,4]diazepin-9-yl)benzo[d]oxazol-5-yl)acrylamide —— C22H18N4O3S
(R)-N-(2-(3-methyl-5-oxo-2,3,4,5-tetrahydro-1H-benzo[4,5]thieno[3,2-e][1,4]diazepin-9-yl)benzo[d]oxazol-5-yl)acrylamide
—— (R)-5-bromo-2-(trifluoromethyl)-2,3-dihydro-1H-inden-2-ol —— C10H8BrF3O
(R)-5-bromo-2-(trifluoromethyl)-2,3-dihydro-1H-inden-2-ol
—— (R)-N-(2-acrylamidophenyl)-3-methyl-5-oxo-2,3,4,5-tetrahydro-1H-benzo[4,5]thieno[3,2-e][1,4]diazepine-9-carboxamide —— C22H20N4O3S
(R)-N-(2-acrylamidophenyl)-3-methyl-5-oxo-2,3,4,5-tetrahydro-1H-benzo[4,5]thieno[3,2-e][1,4]diazepine-9-carboxamide
—— (R)-1-(1-((1H-benzo[d]imidazol-6-yl)methyl)piperidin-4-yl)-2-(pyrrolidin-3-yl)-1H-benzo[d]imidazole —— C24H28N6
(R)-1-(1-((1H-benzo[d]imidazol-6-yl)methyl)piperidin-4-yl)-2-(pyrrolidin-3-yl)-1H-benzo[d]imidazole
—— (R)-N-(1-acryloylpiperidin-3-yl)-1-oxo-1,2,3,4-tetrahydropyrazino[1,2-a]indole-7-carboxamide —— C20H22N4O3
(R)-N-(1-acryloylpiperidin-3-yl)-1-oxo-1,2,3,4-tetrahydropyrazino[1,2-a]indole-7-carboxamide
—— (R)-N-(4-acryloyl-2,2-dimethyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-3-methyl-5-oxo-2,3,4,5-tetrahydro-1H-benzo[4,5]thieno[3,2-e][1,4]diazepine-9-carboxamide —— C26H26N4O4S
(R)-N-(4-acryloyl-2,2-dimethyl-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-3-methyl-5-oxo-2,3,4,5-tetrahydro-1H-benzo[4,5]thieno[3,2-e][1,4]diazepine-9-carboxamide
—— (R)-3-(oxiran-2-yl)-6-(1H-tetrazol-1-yl)pyridazine —— C7H6N6O
(R)-3-(oxiran-2-yl)-6-(1H-tetrazol-1-yl)pyridazine
—— (R)-5-((1-amino-1-oxopropan-2-yl)amino)-3-((4,6-dimethylpyridin-2-yl)amino)picolinamide —— C16H20N6O2
(R)-5-((1-amino-1-oxopropan-2-yl)amino)-3-((4,6-dimethylpyridin-2-yl)amino)picolinamide
—— (R)-1-(2-bromo-5-ethylphenylcarbamoyl)pyrrolidine-2-carboxylic acid —— C14H17BrN2O3
(R)-1-(2-bromo-5-ethylphenylcarbamoyl)pyrrolidine-2-carboxylic acid
—— racemic N-(4,4,4-trifluoro-2-methylbutyl)cyclohexanamine —— C11H20F3N
racemic N-(4,4,4-trifluoro-2-methylbutyl)cyclohexanamine
—— (R)-N-((S)-1-(3-bromophenyl)-2,2,2-trifluoroethyl)-2-methylpropane-2-sulfinamide —— C12H15BrF3NOS
(R)-N-((S)-1-(3-bromophenyl)-2,2,2-trifluoroethyl)-2-methylpropane-2-sulfinamide
—— (R)-3-(4-(diisobutylamino)-3-(3-(5-methylisoxazol-3-yl)ureido)phenyl)butanoic acid —— C23H34N4O4
(R)-3-(4-(diisobutylamino)-3-(3-(5-methylisoxazol-3-yl)ureido)phenyl)butanoic acid
—— racemic (1S,2R)-2-(4-(diisobutylamino)-2-fluoro-5-(3-(6-methylpyridin-3-yl)ureido)phenyl)cyclopropanecarboxylic acid —— C25H33FN4O3
racemic (1S,2R)-2-(4-(diisobutylamino)-2-fluoro-5-(3-(6-methylpyridin-3-yl)ureido)phenyl)cyclopropanecarboxylic acid
—— (R)-3-(4-(diisobutylamino)-3-(3-(2-methylpyrimidin-5-yl)ureido)phenyl)butanoic acid —— C24H35N5O3
(R)-3-(4-(diisobutylamino)-3-(3-(2-methylpyrimidin-5-yl)ureido)phenyl)butanoic acid
—— (R)-3-(2-Hydroxy-1-(methylamino)ethyl)phenol —— C9H13NO2
(R)-3-(2-Hydroxy-1-(methylamino)ethyl)phenol
—— (R)-tert-butyl 3-((S)-2-((R)-(1-benzyl-4-(2,5-difluorophenyl)-1H-imidazol-2-yl)(tetrahydro-2H-pyran-4-yl)methyl)-14-(2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)-5-methyl-3,8-dioxo-7,12-dioxa-2,4,9-triazatetradecyl)pyrrolidine-1-carboxylate —— C45H57F2N7O9
(R)-tert-butyl 3-((S)-2-((R)-(1-benzyl-4-(2,5-difluorophenyl)-1H-imidazol-2-yl)(tetrahydro-2H-pyran-4-yl)methyl)-14-(2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)-5-methyl-3,8-dioxo-7,12-dioxa-2,4,9-triazatetradecyl)pyrrolidine-1-carboxylate
—— (R)-2-((tert-butoxycarbonyl)amino)-2-(4-methyltetrahydro-2H-pyran-4-yl)acetic acid —— C13H23NO5
(R)-2-((tert-butoxycarbonyl)amino)-2-(4-methyltetrahydro-2H-pyran-4-yl)acetic acid
—— (R)-2-(azetidin-3-yloxy)-N-(1-(1-benzyl-4-(2,5-difluorophenyl)-1H-imidazol-2-yl)-4-((2-(2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)ethyl)amino)-2,2-dimethyl-4-oxobutyl)benzamide —— C38H38F2N6O5
(R)-2-(azetidin-3-yloxy)-N-(1-(1-benzyl-4-(2,5-difluorophenyl)-1H-imidazol-2-yl)-4-((2-(2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)ethyl)amino)-2,2-dimethyl-4-oxobutyl)benzamide
—— racemic (1S,2R)-2-(4-(cyclohexyl(isobutyl)amino)-3-(3-(p-tolyl)ureido)phenyl)cyclopropanecarboxylic acid —— C28H37N3O3
racemic (1S,2R)-2-(4-(cyclohexyl(isobutyl)amino)-3-(3-(p-tolyl)ureido)phenyl)cyclopropanecarboxylic acid
—— (R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(4-methyloxan-4-yl)methanamine —— C23H25F2N3O
(R)-[1-benzyl-4-(2,5-difluorophenyl)imidazol-2-yl]-(4-methyloxan-4-yl)methanamine
—— (R)-1-((4-chloro-6-morpholinopyrimidin-2-yl)amino) propan-2-ol —— C11H17ClN4O2
(R)-1-((4-chloro-6-morpholinopyrimidin-2-yl)amino) propan-2-ol
—— (R)-N-(3-(2-((2-hydroxypropyl)amino)-6-morpholinopyridin-4-yl)-4-methylphenyl)-2-(trifluoromethyl)isonicotinamide —— C26H28F3N5O3
(R)-N-(3-(2-((2-hydroxypropyl)amino)-6-morpholinopyridin-4-yl)-4-methylphenyl)-2-(trifluoromethyl)isonicotinamide
—— (R)-N-(6'-(2-hydroxypropoxy)-2-methyl-5'-morpholino-[3,3'-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide —— C26H27F3N4O4
(R)-N-(6'-(2-hydroxypropoxy)-2-methyl-5'-morpholino-[3,3'-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide
—— (R)-N-(6'-((1-aminopropan-2-yl)oxy)-2-methyl-5'-morpholino-[3,3'-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide —— C26H28F3N5O3
(R)-N-(6'-((1-aminopropan-2-yl)oxy)-2-methyl-5'-morpholino-[3,3'-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide
—— (R)-2-(2-naphthylsulfonyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxylic acid 140645-46-1 C20H17NO4S
(R)-2-(2-naphthylsulfonyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxylic acid
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3,4-difluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C21H25F3N4O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(3,4-difluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(5-fluoro-2-(((S)-1-(2-fluoro-4-methoxyphenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C22H28F2N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(5-fluoro-2-(((S)-1-(2-fluoro-4-methoxyphenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-N-[tert-butyl(dimethyl)silyl]-2-(4-methylphenyl)propane-2-sulfinamide —— C16H29NOSSi
(R)-N-[tert-butyl(dimethyl)silyl]-2-(4-methylphenyl)propane-2-sulfinamide
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-isobutoxyphenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C25H36N4O4
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(4-isobutoxyphenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-N-[(1S)-1-[2,5-difluoro-4-[2-(fluoromethyl)pyridin-4-yl]phenyl]ethyl]-2-methylpropane-2-sulfinamide —— C18H21F3N2OS
(R)-N-[(1S)-1-[2,5-difluoro-4-[2-(fluoromethyl)pyridin-4-yl]phenyl]ethyl]-2-methylpropane-2-sulfinamide
—— (R)-3-(6-chloro-2-(((S)-1-(2,5-difluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-methoxyethyl)oxazolidin-2-one —— C22H23ClF2N6O3
(R)-3-(6-chloro-2-(((S)-1-(2,5-difluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-methoxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2 ,3-difluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C21H25F3N4O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2 ,3-difluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2,3-difluorophenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C21H26F2N4O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2,3-difluorophenyl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-(2-(tert-butyl-dimethyl-silanyloxy)-3-{4-chloro-3-[4-(7-cyclopropyl-2,7-diaza-spiro[4.4]non-2-yl)-6-(3,5-dimethylisoxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy}propyl)methylcarbamic acid tert-butyl ester —— C42H62ClN5O5Si
(R)-(2-(tert-butyl-dimethyl-silanyloxy)-3-{4-chloro-3-[4-(7-cyclopropyl-2,7-diaza-spiro[4.4]non-2-yl)-6-(3,5-dimethylisoxazol-4-yl)-5-methylpyrimidin-2-yl]phenoxy}propyl)methylcarbamic acid tert-butyl ester
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2,4-difluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C21H25F3N4O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2,4-difluorophenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(5-(p-tolyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C20H22N6O4
(R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(5-(p-tolyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-{1-[3-(3,4-difluorophenyl)-[1,2,4]-oxadiazol-5-yl]ethylamino}-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C19H17F3N6O4
(R)-3-(2-{1-[3-(3,4-difluorophenyl)-[1,2,4]-oxadiazol-5-yl]ethylamino}-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C25H32N6O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(2-((S)-1-(4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-((1-(3-(2,3-dihydro-1H-inden-5-yl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C22H24N6O4
(R)-3-(2-((1-(3-(2,3-dihydro-1H-inden-5-yl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-(trifluoromethyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C22H25F5N4O3
(R)-4-((R)-1-tert-butoxyethyl)-3-(5-fluoro-2-((S)-1-(2-fluoro-4-(trifluoromethyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-((1-(5-(3-chloro-5-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C22H20ClF3N6O3
(R)-3-(2-((1-(5-(3-chloro-5-(trifluoromethyl)phenyl)pyrimidin-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-3-(2-{1-[3-(3,4-dichlorophenyl)isoxazol-5-yl]ethylamino}-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C20H18Cl2FN5O4
(R)-3-(2-{1-[3-(3,4-dichlorophenyl)isoxazol-5-yl]ethylamino}-5-fluoropyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-3-(5-fluoro-2-{1-[3-(3-fluoro-4-methylphenyl)-[1,2,4]-oxadiazol-5-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C20H20F2N6O4
(R)-3-(5-fluoro-2-{1-[3-(3-fluoro-4-methylphenyl)-[1,2,4]-oxadiazol-5-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one —— C25H31ClN6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(1-(4-chlorophenyl)-1H-pyrazol-4-yl)ethyl)amino)-6-methylpyrimidin-4-yl)oxazolidin-2-one
—— (R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(3-(2-phenoxyethyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C21H24N6O5
(R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(3-(2-phenoxyethyl)-1,2,4-oxadiazol-5-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-{1-[4-(3-chloro-4-fluorophenyl)thiazol-2-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C20H19ClFN5O3S
(R)-3-(2-{1-[4-(3-chloro-4-fluorophenyl)thiazol-2-yl]ethylamino}pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(4-methyl-5-(2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl)thiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one —— C24H27F3N6O3S
(R)-4-((R)-1-hydroxyethyl)-3-(2-((1-(4-methyl-5-(2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl)thiazol-2-yl)ethyl)amino)pyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-(2-((1-(5-(2-fluorophenyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C19H19FN6O4
(R)-3-(2-((1-(5-(2-fluorophenyl)-1,3,4-oxadiazol-2-yl)ethyl)amino)pyrimidin-4-yl)-4-((R)-1-hydroxyethyl)oxazolidin-2-one
—— (R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2,5-difluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C25H29F3N6O3
(R)-4-((R)-1-(tert-butoxy)ethyl)-3-(2-(((S)-1-(2,5-difluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)ethyl)amino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— (R)-3-{2-[1-(5-benzyl-[1,2,4]-oxadiazol-3-yl)ethylamino]pyrimidin-4-yl}-4-((R)-1-hydroxyethyl)oxazolidin-2-one —— C20H22N6O4
(R)-3-{2-[1-(5-benzyl-[1,2,4]-oxadiazol-3-yl)ethylamino]pyrimidin-4-yl}-4-((R)-1-hydroxyethyl)oxazolidin-2-one