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—— 7-[4-[(1S)-1-(2,4-difluorophenyl)ethyl]piperazin-1-yl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H20F2N6
7-[4-[(1S)-1-(2,4-difluorophenyl)ethyl]piperazin-1-yl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7,8-Dimethyl-2-oxochromen-4-yl)methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate —— C18H17NO4S
(7,8-Dimethyl-2-oxochromen-4-yl)methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate
—— (7-Bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate —— C15H12BrN3O3S
(7-Bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate —— C17H15NO5S
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate
—— (7S)-7-methyl-2-[(1R)-1-(2-methylsulfonylethylsulfanyl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C16H22N2O3S3
(7S)-7-methyl-2-[(1R)-1-(2-methylsulfonylethylsulfanyl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[2-(1,3-Benzodioxol-5-yl)-2-oxoethoxy]-6-chloro-4-methylchromen-2-one —— C19H13ClO6
7-[2-(1,3-Benzodioxol-5-yl)-2-oxoethoxy]-6-chloro-4-methylchromen-2-one
—— 7-cyclopropyl-N-[[4-[[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C28H35N5O3
7-cyclopropyl-N-[[4-[[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-1-ethyl-N-[[2-[[(3R)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C27H33N5O3
7-cyclopropyl-1-ethyl-N-[[2-[[(3R)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-N-[[4-[[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C28H35N5O3
7-cyclopropyl-N-[[4-[[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C28H35N5O3
7-cyclopropyl-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-1-ethyl-N-[[2-[[(3S)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C27H33N5O3
7-cyclopropyl-1-ethyl-N-[[2-[[(3S)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-1-ethyl-N-[[4-[[(3R)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C27H33N5O3
7-cyclopropyl-1-ethyl-N-[[4-[[(3R)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-N-[(1S)-1-[3-(difluoromethoxy)phenyl]ethyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C22H22F2N4O4
7-cyclopropyl-N-[(1S)-1-[3-(difluoromethoxy)phenyl]ethyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-1-ethyl-N-[[4-[[(3S)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C27H33N5O3
7-cyclopropyl-1-ethyl-N-[[4-[[(3S)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-N-[(1R)-1-[3-(difluoromethoxy)phenyl]ethyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide —— C22H22F2N4O4
7-cyclopropyl-N-[(1R)-1-[3-(difluoromethoxy)phenyl]ethyl]-1-ethyl-2,4-dioxopyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-1-ethyl-2,4-dioxo-N-[(2S)-2-(4-phenylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidine-5-carboxamide —— C26H32N6O3
7-cyclopropyl-1-ethyl-2,4-dioxo-N-[(2S)-2-(4-phenylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidine-5-carboxamide
—— 7-cyclopropyl-1-ethyl-2,4-dioxo-N-[(2R)-2-(4-phenylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidine-5-carboxamide —— C26H32N6O3
7-cyclopropyl-1-ethyl-2,4-dioxo-N-[(2R)-2-(4-phenylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidine-5-carboxamide
—— (7-Ethyl-2-oxochromen-4-yl)methyl 2,4-difluorobenzoate —— C19H14F2O4
(7-Ethyl-2-oxochromen-4-yl)methyl 2,4-difluorobenzoate
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 4-(4-fluorophenyl)-4-oxobutanoate —— C21H17FO6
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 4-(4-fluorophenyl)-4-oxobutanoate
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 2,4-difluorobenzoate —— C17H10F2O5
(7-Hydroxy-2-oxochromen-4-yl)methyl 2,4-difluorobenzoate
—— (7-Ethyl-2-oxochromen-4-yl)methyl 2-(1,3-dioxoisoindol-2-yl)acetate —— C22H17NO6
(7-Ethyl-2-oxochromen-4-yl)methyl 2-(1,3-dioxoisoindol-2-yl)acetate
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2-(2,4-dichlorophenyl)acetate —— C19H14Cl2O5
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2-(2,4-dichlorophenyl)acetate
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2,4-difluorobenzoate —— C18H12F2O5
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2,4-difluorobenzoate
—— 7-methyl-N-[(2S)-2-(4-methylpiperidin-1-yl)-2-phenylethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide —— C24H28N4O2
7-methyl-N-[(2S)-2-(4-methylpiperidin-1-yl)-2-phenylethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 2-(4-chlorophenoxy)-2-methylpropanoate —— C20H17ClO6
(7-Hydroxy-2-oxochromen-4-yl)methyl 2-(4-chlorophenoxy)-2-methylpropanoate
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 3,3-dimethylbutanoate —— C16H18O5
(7-Hydroxy-2-oxochromen-4-yl)methyl 3,3-dimethylbutanoate
—— (7-Bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3,3-dimethylbutanoate —— C15H17BrN2O3
(7-Bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3,3-dimethylbutanoate
—— (7-Methoxy-2-oxochromen-4-yl)methyl 3,3-dimethylbutanoate —— C17H20O5
(7-Methoxy-2-oxochromen-4-yl)methyl 3,3-dimethylbutanoate
—— 7-methyl-N-[(2R)-2-(4-methylpiperidin-1-yl)-2-phenylethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide —— C24H28N4O2
7-methyl-N-[(2R)-2-(4-methylpiperidin-1-yl)-2-phenylethyl]-4-oxopyrido[1,2-a]pyrimidine-3-carboxamide
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 5-methylpyrazine-2-carboxylate —— C16H12N2O5
(7-Hydroxy-2-oxochromen-4-yl)methyl 5-methylpyrazine-2-carboxylate
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 4-acetamidobenzoate —— C19H15NO6
(7-Hydroxy-2-oxochromen-4-yl)methyl 4-acetamidobenzoate
—— (7-Ethyl-2-oxochromen-4-yl)methyl 5-methylpyrazine-2-carboxylate —— C18H16N2O4
(7-Ethyl-2-oxochromen-4-yl)methyl 5-methylpyrazine-2-carboxylate
—— (7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 4-acetamidobenzoate —— C23H23NO5
(7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 4-acetamidobenzoate
—— (7-methoxy-2-oxochromen-4-yl)methyl (E)-3-(2,5-dimethoxyphenyl)prop-2-enoate —— C22H20O7
(7-methoxy-2-oxochromen-4-yl)methyl (E)-3-(2,5-dimethoxyphenyl)prop-2-enoate
—— (7-ethyl-2-oxochromen-4-yl)methyl (E)-3-(2,5-dimethoxyphenyl)prop-2-enoate —— C23H22O6
(7-ethyl-2-oxochromen-4-yl)methyl (E)-3-(2,5-dimethoxyphenyl)prop-2-enoate
—— (7-hydroxy-8-methyl-2-oxochromen-4-yl)methyl (E)-3-(2,5-dimethoxyphenyl)prop-2-enoate —— C22H20O7
(7-hydroxy-8-methyl-2-oxochromen-4-yl)methyl (E)-3-(2,5-dimethoxyphenyl)prop-2-enoate
—— (7-hydroxy-2-oxochromen-4-yl)methyl (E)-3-(2,5-dimethoxyphenyl)prop-2-enoate —— C21H18O7
(7-hydroxy-2-oxochromen-4-yl)methyl (E)-3-(2,5-dimethoxyphenyl)prop-2-enoate
—— 7-chloro-3-(3-ethoxypropyl)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one —— C19H23ClN4O3S
7-chloro-3-(3-ethoxypropyl)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one
—— (7S)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H24N4O3S2
(7S)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H24N4O3S2
(7R)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-chloro-3-(3-ethoxypropyl)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one —— C19H23ClN4O3S
7-chloro-3-(3-ethoxypropyl)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanylquinazolin-4-one
—— (7S)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H24N4O3S2
(7S)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[[4-[(2S)-1-butanoylpiperidine-2-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C21H29N5O3S
7-[[4-[(2S)-1-butanoylpiperidine-2-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (7R)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-7-methyl-3-[[(2S)-oxolan-2-yl]methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H28N4O3S2
(7R)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-7-methyl-3-[[(2S)-oxolan-2-yl]methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-7-methyl-3-[[(2S)-oxolan-2-yl]methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H28N4O3S2
(7S)-2-[(1R)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-7-methyl-3-[[(2S)-oxolan-2-yl]methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H24N4O3S2
(7R)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-3-(furan-2-ylmethyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-7-methyl-3-[[(2S)-oxolan-2-yl]methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H28N4O3S2
(7S)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-7-methyl-3-[[(2S)-oxolan-2-yl]methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-7-methyl-3-[[(2S)-oxolan-2-yl]methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H28N4O3S2
(7R)-2-[(1S)-1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl-7-methyl-3-[[(2S)-oxolan-2-yl]methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-chloro-3-methyl-N-(2-methylphenyl)-1-benzofuran-2-carboxamide —— C17H14ClNO2
7-chloro-3-methyl-N-(2-methylphenyl)-1-benzofuran-2-carboxamide
—— 7-bromo-N-[(2R)-2-methoxy-2-phenylethyl]-1-benzofuran-2-carboxamide —— C18H16BrNO3
7-bromo-N-[(2R)-2-methoxy-2-phenylethyl]-1-benzofuran-2-carboxamide