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—— (7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O3
(7S)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O4
(7R)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-methylsulfanyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23N5O3S
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-methylsulfanyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-phenyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24N6O3
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-phenyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C20H14ClN3O3S
(7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— (7R)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H19ClF3N5O3
(7R)-N-(4-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-phenyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H20F3N5O3
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-phenyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(furan-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H23N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(furan-2-yl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-(3-methoxypyrazin-2-yl)-2-methyl-N-[(3R)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine —— C18H24N6O2
7-(3-methoxypyrazin-2-yl)-2-methyl-N-[(3R)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine
—— 7-[(3S)-3-methoxypiperidin-1-yl]-5-pyridin-4-ylpyrazolo[1,5-a]pyrimidine —— C17H19N5O
7-[(3S)-3-methoxypiperidin-1-yl]-5-pyridin-4-ylpyrazolo[1,5-a]pyrimidine
—— 7-(3-methoxypyrazin-2-yl)-2-methyl-N-[(3S)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine —— C18H24N6O2
7-(3-methoxypyrazin-2-yl)-2-methyl-N-[(3S)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine
—— 7-Hydroxy-8-methyl-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one —— C14H13N3O3S2
7-Hydroxy-8-methyl-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one
—— 7-Methyl-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-6-propan-2-ylchromen-2-one —— C17H19N3O2S2
7-Methyl-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-6-propan-2-ylchromen-2-one
—— 7-Methoxy-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one —— C14H13N3O3S2
7-Methoxy-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one
—— 7-Hydroxy-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one —— C13H11N3O3S2
7-Hydroxy-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one
—— 7-[[5-(Methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C10H9N5OS3
7-[[5-(Methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-Ethyl-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one —— C15H15N3O2S2
7-Ethyl-4-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]chromen-2-one
—— 7-[(4-Tert-butylphenyl)methylsulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H20N2OS2
7-[(4-Tert-butylphenyl)methylsulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-Bromo-2-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C12H10BrN5OS2
7-Bromo-2-[[5-(methylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-[(2-Fluorophenyl)methylsulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C14H11FN2OS2
7-[(2-Fluorophenyl)methylsulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-[(3S)-piperidin-3-yl]-N-(2-thiophen-2-ylethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine —— C19H27N5S
7-[(3S)-piperidin-3-yl]-N-(2-thiophen-2-ylethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine
—— 7-[(3R)-piperidin-3-yl]-N-(2-thiophen-2-ylethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine —— C19H27N5S
7-[(3R)-piperidin-3-yl]-N-(2-thiophen-2-ylethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine
—— (7-Bromo-2,3-dioxoindol-1-yl)methyl-[(2-chloro-6-fluorophenyl)methyl]-methylazanium —— C17H14BrClFN2O2+
(7-Bromo-2,3-dioxoindol-1-yl)methyl-[(2-chloro-6-fluorophenyl)methyl]-methylazanium
—— 7-(2-aminoethyl)-2-(ethoxymethyl)-N-[[(2R)-oxolan-2-yl]methyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine —— C18H31N5O2
7-(2-aminoethyl)-2-(ethoxymethyl)-N-[[(2R)-oxolan-2-yl]methyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine
—— 7-Bromo-1-[[methyl-[(4-prop-2-enoxyphenyl)methyl]amino]methyl]indole-2,3-dione —— C20H19BrN2O3
7-Bromo-1-[[methyl-[(4-prop-2-enoxyphenyl)methyl]amino]methyl]indole-2,3-dione
—— 7-Methoxy-1-[[methyl-[(4-prop-2-enoxyphenyl)methyl]amino]methyl]naphthalen-2-ol —— C23H25NO3
7-Methoxy-1-[[methyl-[(4-prop-2-enoxyphenyl)methyl]amino]methyl]naphthalen-2-ol
—— (7-Bromo-2,3-dioxoindol-1-yl)methyl-methyl-[(4-prop-2-enoxyphenyl)methyl]azanium —— C20H20BrN2O3+
(7-Bromo-2,3-dioxoindol-1-yl)methyl-methyl-[(4-prop-2-enoxyphenyl)methyl]azanium
—— 7-(2-aminoethyl)-2-(ethoxymethyl)-N-[[(2S)-oxolan-2-yl]methyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine —— C18H31N5O2
7-(2-aminoethyl)-2-(ethoxymethyl)-N-[[(2S)-oxolan-2-yl]methyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine
—— 7-[[(3R)-oxolan-3-yl]methyl]-4-N-(thiophen-2-ylmethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-2,4-diamine —— C18H25N5OS
7-[[(3R)-oxolan-3-yl]methyl]-4-N-(thiophen-2-ylmethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-2,4-diamine
—— 7-[[(3S)-oxolan-3-yl]methyl]-4-N-(thiophen-2-ylmethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-2,4-diamine —— C18H25N5OS
7-[[(3S)-oxolan-3-yl]methyl]-4-N-(thiophen-2-ylmethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-2,4-diamine
—— 7-[2-[4-(2-Methoxyphenyl)piperazin-1-yl]-2-oxoethoxy]-4,8-dimethylchromen-2-one —— C24H26N2O5
7-[2-[4-(2-Methoxyphenyl)piperazin-1-yl]-2-oxoethoxy]-4,8-dimethylchromen-2-one
—— 7-(furan-2-yl)-4-methyl-3-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine —— C22H18N8O
7-(furan-2-yl)-4-methyl-3-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine
—— 7-[2-[4-(2-Fluorophenyl)piperazin-1-yl]-2-oxoethoxy]-4,8-dimethylchromen-2-one —— C23H23FN2O4
7-[2-[4-(2-Fluorophenyl)piperazin-1-yl]-2-oxoethoxy]-4,8-dimethylchromen-2-one
—— 7-(furan-2-yl)-4-methyl-3-[2-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine —— C19H20N8O
7-(furan-2-yl)-4-methyl-3-[2-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine
—— 7-ethyl-4-methyl-3-[2-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine —— C17H22N8
7-ethyl-4-methyl-3-[2-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine
—— 7-ethyl-4-methyl-3-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine —— C20H20N8
7-ethyl-4-methyl-3-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine
—— 7-ethyl-4-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine —— C20H20N8
7-ethyl-4-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine
—— 7-methyl-N-(2-methylphenyl)-2,4-dioxo-1-[[(2S)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidine-6-carboxamide —— C21H22N4O4
7-methyl-N-(2-methylphenyl)-2,4-dioxo-1-[[(2S)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidine-6-carboxamide
—— 7-(furan-2-yl)-4-methyl-3-[2-[(3R)-3-methylpiperidin-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine —— C19H20N8O
7-(furan-2-yl)-4-methyl-3-[2-[(3R)-3-methylpiperidin-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine
—— 7-methyl-2,4-dioxo-1-[[(2R)-oxolan-2-yl]methyl]-N-[3-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidine-6-carboxamide —— C21H19F3N4O4
7-methyl-2,4-dioxo-1-[[(2R)-oxolan-2-yl]methyl]-N-[3-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidine-6-carboxamide
—— 7-(furan-2-yl)-4-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine —— C22H18N8O
7-(furan-2-yl)-4-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine
—— 7-methyl-2,4-dioxo-1-[[(2S)-oxolan-2-yl]methyl]-N-[3-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidine-6-carboxamide —— C21H19F3N4O4
7-methyl-2,4-dioxo-1-[[(2S)-oxolan-2-yl]methyl]-N-[3-(trifluoromethyl)phenyl]pyrido[2,3-d]pyrimidine-6-carboxamide
—— (7S)-3-(4-chlorophenyl)-2-ethyl-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline —— C19H20ClN3
(7S)-3-(4-chlorophenyl)-2-ethyl-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
—— (7S)-3-(3-chlorophenyl)-2-ethyl-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline —— C19H20ClN3
(7S)-3-(3-chlorophenyl)-2-ethyl-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
—— (7S)-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline —— C11H13N3
(7S)-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
—— (7S)-3-(4-chlorophenyl)-2,7-dimethyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline —— C18H18ClN3
(7S)-3-(4-chlorophenyl)-2,7-dimethyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
—— (7R)-3-(4-chlorophenyl)-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline —— C17H16ClN3
(7R)-3-(4-chlorophenyl)-7-methyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline
—— (7R)-7-methyl-2-pyridin-4-yl-6,7,8,9-tetrahydro-[1,2,4]triazolo[1,5-a]quinazoline —— C15H15N5
(7R)-7-methyl-2-pyridin-4-yl-6,7,8,9-tetrahydro-[1,2,4]triazolo[1,5-a]quinazoline
—— 7-(methoxymethyl)-4-methyl-3-[2-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine —— C17H22N8O
7-(methoxymethyl)-4-methyl-3-[2-[(3S)-3-methylpiperidin-1-yl]pyrimidin-4-yl]-[1,2,4]triazolo[5,1-c][1,2,4]triazine
—— (7R)-2,7-dimethyl-3-phenyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline —— C18H19N3
(7R)-2,7-dimethyl-3-phenyl-6,7,8,9-tetrahydropyrazolo[1,5-a]quinazoline