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—— 7-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-3-piperidin-4-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C22H31N5O2
7-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methyl]-3-piperidin-4-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N6O2
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[[3-(4-fluorophenyl)phenyl]methyl]-3-piperidin-4-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C23H26FN5
7-[[3-(4-fluorophenyl)phenyl]methyl]-3-piperidin-4-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(4-fluorophenyl)methyl]-2-[(2S)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O3
7-[(4-fluorophenyl)methyl]-2-[(2S)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(2R)-1-(4-methylthiadiazole-5-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H24N6O2S
7-benzyl-4-methyl-2-[(2R)-1-(4-methylthiadiazole-5-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-2-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O3
7-[2-(4-fluorophenyl)ethyl]-2-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C19H26N4O3
7-(cyclopropylmethyl)-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O3
7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-2-[(2S)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O4
7-[(4-methoxyphenyl)methyl]-2-[(2S)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-2-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O3
7-[2-(4-fluorophenyl)ethyl]-2-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-2-[(2S)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O4
7-[(4-methoxyphenyl)methyl]-2-[(2S)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O2
7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O3
7-[(3-fluorophenyl)methyl]-2-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-2-[(2S)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O3
7-[2-(4-fluorophenyl)ethyl]-2-[(2S)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2S)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N6O2
7-(cyclopropylmethyl)-2-[(2S)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(2S)-1-(4-methylthiadiazole-5-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H24N6O2S
7-benzyl-4-methyl-2-[(2S)-1-(4-methylthiadiazole-5-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C19H26N4O3
7-(cyclopropylmethyl)-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H34N4O2
7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H32N4O2
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N6O2
7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O2
7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O3
7-[(4-fluorophenyl)methyl]-2-[(2S)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-2-[(2S)-1-[2-(diethylamino)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H33N5O2
7-benzyl-2-[(2S)-1-[2-(diethylamino)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(2-fluorophenyl)ethyl]-2-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O3
7-[2-(2-fluorophenyl)ethyl]-2-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H26N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H30N4O3
7-(cyclopropylmethyl)-2-[(2R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H26N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O3
7-[(4-fluorophenyl)methyl]-2-[(2R)-1-(2-methoxyacetyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H25FN6O2
7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-(1-methylpyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-(1-propanoylpiperidin-4-yl)-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-(1-propanoylpiperidin-4-yl)-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-2-[1-(3-methoxypropanoyl)piperidin-4-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O4
7-[(4-methoxyphenyl)methyl]-2-[1-(3-methoxypropanoyl)piperidin-4-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O3
7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(2R)-1-[3-(2-methylimidazol-1-yl)propanoyl]pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H28N6O2
7-benzyl-4-methyl-2-[(2R)-1-[3-(2-methylimidazol-1-yl)propanoyl]pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-2-[(2R)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O3
7-[2-(4-fluorophenyl)ethyl]-2-[(2R)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-2-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O4
7-[(4-methoxyphenyl)methyl]-2-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(2-fluorophenyl)ethyl]-2-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H29FN4O3
7-[2-(2-fluorophenyl)ethyl]-2-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H32N4O2
7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-2-[(2S)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H34N4O3
7-(cyclohexylmethyl)-2-[(2S)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O3
7-[(4-fluorophenyl)methyl]-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(3S)-1-propan-2-ylpiperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H29FN4O
7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(3S)-1-propan-2-ylpiperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O2
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2S)-1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H30N4O3
7-(cyclopropylmethyl)-2-[(2S)-1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-2-[(2R)-1-[2-(diethylamino)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H33N5O2
7-benzyl-2-[(2R)-1-[2-(diethylamino)acetyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-(1-propan-2-ylpiperidin-4-yl)-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H30N4O2
7-[(4-methoxyphenyl)methyl]-4-methyl-2-(1-propan-2-ylpiperidin-4-yl)-5H-pyrrolo[2,3-d]pyrimidin-6-one