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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7,7-dimethyl-2-(3-pyridin-2-yl-2H-1,2,4-oxadiazol-5-ylidene)-6,8-dihydro-5H-imidazo[4,5-c]azepin-4-one —— C16H16N6O2
7,7-dimethyl-2-(3-pyridin-2-yl-2H-1,2,4-oxadiazol-5-ylidene)-6,8-dihydro-5H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-phenyl-2-(3-pyridin-2-yl-2H-1,2,4-oxadiazol-5-ylidene)-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one —— C20H16N6O2
(7R)-7-phenyl-2-(3-pyridin-2-yl-2H-1,2,4-oxadiazol-5-ylidene)-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one
—— (7S)-7-phenyl-2-(3-pyridin-2-yl-2H-1,2,4-oxadiazol-5-ylidene)-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one —— C20H16N6O2
(7S)-7-phenyl-2-(3-pyridin-2-yl-2H-1,2,4-oxadiazol-5-ylidene)-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one
—— [7-(Ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 5-chlorothiophene-2-carboxylate —— C18H14ClNO6S
[7-(Ethoxycarbonylamino)-2-oxochromen-4-yl]methyl 5-chlorothiophene-2-carboxylate
—— (7S)-7-(4-chlorophenyl)-2-(ethylsulfanylmethyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C16H18ClN3OS
(7S)-7-(4-chlorophenyl)-2-(ethylsulfanylmethyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(4-chlorophenyl)-2-(ethylsulfanylmethyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C16H18ClN3OS
(7R)-7-(4-chlorophenyl)-2-(ethylsulfanylmethyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-3-(2-fluorophenyl)-7-methyl-2-(2-methylsulfanylethylsulfanyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H21FN2OS3
(7R)-3-(2-fluorophenyl)-7-methyl-2-(2-methylsulfanylethylsulfanyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-Methyl-4-[(2-methylquinazolin-4-yl)sulfanylmethyl]chromen-2-one —— C20H16N2O2S
7-Methyl-4-[(2-methylquinazolin-4-yl)sulfanylmethyl]chromen-2-one
—— 7-[4-[(1R)-1-morpholin-4-ylethyl]phenyl]-2H-isoquinolin-1-one —— C21H22N2O2
7-[4-[(1R)-1-morpholin-4-ylethyl]phenyl]-2H-isoquinolin-1-one
—— (7S)-7-(4-fluorophenyl)-2-[1-(2-methoxyethyl)piperidin-4-yl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C21H27FN4O2
(7S)-7-(4-fluorophenyl)-2-[1-(2-methoxyethyl)piperidin-4-yl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(4-fluorophenyl)-2-[1-(2-methoxyethyl)piperidin-4-yl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C21H27FN4O2
(7R)-7-(4-fluorophenyl)-2-[1-(2-methoxyethyl)piperidin-4-yl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— 7-Methyl-4-[(2-methylquinazolin-4-yl)sulfanylmethyl]-6-propan-2-ylchromen-2-one —— C23H22N2O2S
7-Methyl-4-[(2-methylquinazolin-4-yl)sulfanylmethyl]-6-propan-2-ylchromen-2-one
—— (7S)-7-methyl-6-[(E)-2-methyl-3-phenylprop-2-enyl]-4-pyridin-4-yl-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine —— C22H23N5
(7S)-7-methyl-6-[(E)-2-methyl-3-phenylprop-2-enyl]-4-pyridin-4-yl-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine
—— 7-[4-[(1S)-1-morpholin-4-ylethyl]phenyl]-2H-isoquinolin-1-one —— C21H22N2O2
7-[4-[(1S)-1-morpholin-4-ylethyl]phenyl]-2H-isoquinolin-1-one
—— (7-methyl-2-oxochromen-4-yl)methyl (2S)-2-(4-chlorophenyl)-3-methylbutanoate —— C22H21ClO4
(7-methyl-2-oxochromen-4-yl)methyl (2S)-2-(4-chlorophenyl)-3-methylbutanoate
—— (7R)-7-methyl-6-[(E)-2-methyl-3-phenylprop-2-enyl]-4-pyridin-4-yl-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine —— C22H23N5
(7R)-7-methyl-6-[(E)-2-methyl-3-phenylprop-2-enyl]-4-pyridin-4-yl-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine
—— 7,7-dimethyl-2-[(2S)-2-pyrrolidin-1-ylpropyl]-1,5,6,8-tetrahydroimidazo[4,5-c]azepin-4-one —— C16H26N4O
7,7-dimethyl-2-[(2S)-2-pyrrolidin-1-ylpropyl]-1,5,6,8-tetrahydroimidazo[4,5-c]azepin-4-one
—— (7R)-7-(4-chlorophenyl)-2-(3,5-dimethyl-1,2-oxazol-4-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C18H17ClN4O2
(7R)-7-(4-chlorophenyl)-2-(3,5-dimethyl-1,2-oxazol-4-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7S)-2-(ethylsulfanylmethyl)-7-(3-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C17H21N3O2S
(7S)-2-(ethylsulfanylmethyl)-7-(3-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-2-[2-(2-ethylimidazol-1-yl)ethyl]-7-(4-fluorophenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C20H22FN5O
(7R)-2-[2-(2-ethylimidazol-1-yl)ethyl]-7-(4-fluorophenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— 7-[(4R)-2,2-dimethyloxane-4-carbonyl]-2,3-dimethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-one —— C18H27N3O3
7-[(4R)-2,2-dimethyloxane-4-carbonyl]-2,3-dimethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-one
—— (7S)-7-(4-chlorophenyl)-2-(3,5-dimethyl-1,2-oxazol-4-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C18H17ClN4O2
(7S)-7-(4-chlorophenyl)-2-(3,5-dimethyl-1,2-oxazol-4-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-2-(ethylsulfanylmethyl)-7-(3-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C17H21N3O2S
(7R)-2-(ethylsulfanylmethyl)-7-(3-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— 7,7-dimethyl-2-[(2R)-2-pyrrolidin-1-ylpropyl]-1,5,6,8-tetrahydroimidazo[4,5-c]azepin-4-one —— C16H26N4O
7,7-dimethyl-2-[(2R)-2-pyrrolidin-1-ylpropyl]-1,5,6,8-tetrahydroimidazo[4,5-c]azepin-4-one
—— (7S)-2-[2-(2-ethylimidazol-1-yl)ethyl]-7-(4-fluorophenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C20H22FN5O
(7S)-2-[2-(2-ethylimidazol-1-yl)ethyl]-7-(4-fluorophenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— 7-methyl-2-[[(6R)-2,2,6-trimethylmorpholin-4-yl]methyl]pyrido[1,2-a]pyrimidin-4-one —— C17H23N3O2
7-methyl-2-[[(6R)-2,2,6-trimethylmorpholin-4-yl]methyl]pyrido[1,2-a]pyrimidin-4-one
—— (7S)-7-methyl-4-pyridin-4-yl-6-(quinolin-4-ylmethyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine —— C22H20N6
(7S)-7-methyl-4-pyridin-4-yl-6-(quinolin-4-ylmethyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine
—— (7S)-2-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-7-(2-methoxyphenyl)-1,3,5,6,7,8-hexahydroimidazo[4,5-c]azepin-4-one —— C21H21N3O4
(7S)-2-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-7-(2-methoxyphenyl)-1,3,5,6,7,8-hexahydroimidazo[4,5-c]azepin-4-one
—— (7R)-2-(3-ethylimidazol-4-yl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C19H21N5O2
(7R)-2-(3-ethylimidazol-4-yl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-methyl-4-pyridin-4-yl-6-(quinolin-4-ylmethyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine —— C22H20N6
(7R)-7-methyl-4-pyridin-4-yl-6-(quinolin-4-ylmethyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine
—— 7-[(4S)-2,2-dimethyloxane-4-carbonyl]-2,3-dimethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-one —— C18H27N3O3
7-[(4S)-2,2-dimethyloxane-4-carbonyl]-2,3-dimethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-one
—— (7S)-7-(2-methoxyphenyl)-4-oxo-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepine-2-carboxamide —— C15H16N4O3
(7S)-7-(2-methoxyphenyl)-4-oxo-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepine-2-carboxamide
—— (7S)-2-(4-hydroxyhepta-1,6-dien-4-yl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C21H25N3O3
(7S)-2-(4-hydroxyhepta-1,6-dien-4-yl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C18H15ClN4O
(7R)-7-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(2-methoxyphenyl)-2-(propoxymethyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C18H23N3O3
(7R)-7-(2-methoxyphenyl)-2-(propoxymethyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7S)-2-(3-ethylimidazol-4-yl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C19H21N5O2
(7S)-2-(3-ethylimidazol-4-yl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-2-(4-hydroxyhepta-1,6-dien-4-yl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C21H25N3O3
(7R)-2-(4-hydroxyhepta-1,6-dien-4-yl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-2-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-7-(2-methoxyphenyl)-1,3,5,6,7,8-hexahydroimidazo[4,5-c]azepin-4-one —— C21H21N3O4
(7R)-2-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-7-(2-methoxyphenyl)-1,3,5,6,7,8-hexahydroimidazo[4,5-c]azepin-4-one
—— (7S)-7-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C18H15ClN4O
(7S)-7-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7S)-7-(2-methoxyphenyl)-2-(propoxymethyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C18H23N3O3
(7S)-7-(2-methoxyphenyl)-2-(propoxymethyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(3-methoxyphenyl)-2-(3-pyrrolidin-1-ylpropyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C21H28N4O2
(7R)-7-(3-methoxyphenyl)-2-(3-pyrrolidin-1-ylpropyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-2-[4-(hydroxymethyl)phenyl]-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C21H21N3O3
(7R)-2-[4-(hydroxymethyl)phenyl]-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(3-methoxyphenyl)-2-(1-propylpyrazol-4-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C20H23N5O2
(7R)-7-(3-methoxyphenyl)-2-(1-propylpyrazol-4-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7S)-7-(4-chlorophenyl)-2-[3-(methoxymethyl)-2H-1,2,4-oxadiazol-5-ylidene]-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one —— C17H16ClN5O3
(7S)-7-(4-chlorophenyl)-2-[3-(methoxymethyl)-2H-1,2,4-oxadiazol-5-ylidene]-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one
—— (7S)-2-[4-(hydroxymethyl)phenyl]-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C21H21N3O3
(7S)-2-[4-(hydroxymethyl)phenyl]-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7S)-7-(3-methoxyphenyl)-2-(1-propylpyrazol-4-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C20H23N5O2
(7S)-7-(3-methoxyphenyl)-2-(1-propylpyrazol-4-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(4-chlorophenyl)-2-[2-(diethylamino)ethyl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C19H25ClN4O
(7R)-7-(4-chlorophenyl)-2-[2-(diethylamino)ethyl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(2-methoxyphenyl)-2-(3-pyridin-2-ylpropyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C22H24N4O2
(7R)-7-(2-methoxyphenyl)-2-(3-pyridin-2-ylpropyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(4-fluorophenyl)-2-[2-(1,2,4-triazol-1-yl)pyridin-3-yl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C20H16FN7O
(7R)-7-(4-fluorophenyl)-2-[2-(1,2,4-triazol-1-yl)pyridin-3-yl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7S)-7-(4-chlorophenyl)-2-(4-methylpyridin-2-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C19H17ClN4O
(7S)-7-(4-chlorophenyl)-2-(4-methylpyridin-2-yl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one