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—— (7R)-7-methyl-2-[(1S)-1-[[5-(propylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H23N5OS3
(7R)-7-methyl-2-[(1S)-1-[[5-(propylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-[[5-(propylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H23N5OS3
(7R)-7-methyl-2-[(1R)-1-[[5-(propylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-N-(4-methylphenyl)-5-oxo-2-phenyl-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C20H18N4O2
(7S)-N-(4-methylphenyl)-5-oxo-2-phenyl-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(4-bromophenyl)-2-(4-methylphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C20H17BrN4O2
(7S)-N-(4-bromophenyl)-2-(4-methylphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(4-methoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C15H16N4O3
(7S)-N-(4-methoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(5-chloro-2-methoxyphenyl)-3-(4-chlorophenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C20H16Cl2N4O3
(7R)-N-(5-chloro-2-methoxyphenyl)-3-(4-chlorophenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S,11S)-7,11-bis(4-fluorophenyl)-3-sulfanylidene-2,4,8,10-tetrazaspiro[5.5]undecane-1,5,9-trione —— C19H14F2N4O3S
(7S,11S)-7,11-bis(4-fluorophenyl)-3-sulfanylidene-2,4,8,10-tetrazaspiro[5.5]undecane-1,5,9-trione
—— 7-[[(1S,2S,4aR,6S,8aS)-1,6-dihydroxy-1,5,5,8a-tetramethyl-3,4,4a,6,7,8-hexahydro-2H-naphthalen-2-yl]methoxy]chromen-2-one —— C24H32O5
7-[[(1S,2S,4aR,6S,8aS)-1,6-dihydroxy-1,5,5,8a-tetramethyl-3,4,4a,6,7,8-hexahydro-2H-naphthalen-2-yl]methoxy]chromen-2-one
—— (7R,11R)-7,11-bis(4-fluorophenyl)-3-sulfanylidene-2,4,8,10-tetrazaspiro[5.5]undecane-1,5,9-trione —— C19H14F2N4O3S
(7R,11R)-7,11-bis(4-fluorophenyl)-3-sulfanylidene-2,4,8,10-tetrazaspiro[5.5]undecane-1,5,9-trione
—— (7R)-2-methyl-N-(4-methylphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C15H16N4O2
(7R)-2-methyl-N-(4-methylphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-7-(3-ethoxy-4-hydroxyphenyl)-6-N-(4-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C24H25N5O5
(7S)-7-(3-ethoxy-4-hydroxyphenyl)-6-N-(4-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-6-(3,4-difluorophenyl)-7-methyl-3-(2-methylfuran-3-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C16H12F2N4OS
(7S)-6-(3,4-difluorophenyl)-7-methyl-3-(2-methylfuran-3-yl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— (7R)-N-(5-chloro-2-methoxyphenyl)-2-(4-chlorophenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C20H16Cl2N4O3
(7R)-N-(5-chloro-2-methoxyphenyl)-2-(4-chlorophenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R,11S)-7,11-bis(4-fluorophenyl)-3-sulfanylidene-2,4,8,10-tetrazaspiro[5.5]undecane-1,5,9-trione —— C19H14F2N4O3S
(7R,11S)-7,11-bis(4-fluorophenyl)-3-sulfanylidene-2,4,8,10-tetrazaspiro[5.5]undecane-1,5,9-trione
—— (7S)-3-cyano-N-(2,4-dimethylphenyl)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H23N5O3
(7S)-3-cyano-N-(2,4-dimethylphenyl)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,5-dimethoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C16H18N4O4
(7S)-N-(2,5-dimethoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-2-(4-chlorophenyl)-5-methyl-N-phenyl-7-pyridin-3-yl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H20ClN5O
(7S)-2-(4-chlorophenyl)-5-methyl-N-phenyl-7-pyridin-3-yl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-ethoxy-4-hydroxyphenyl)-6-N-(4-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C24H25N5O5
(7R)-7-(3-ethoxy-4-hydroxyphenyl)-6-N-(4-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C21H18ClN5O2
(7R)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(4-chlorophenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClN4O2
(7S)-7-(4-chlorophenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-3-cyano-5-methyl-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H16ClN5O
(7S)-N-(4-chlorophenyl)-3-cyano-5-methyl-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-hydroxy-3-methoxyphenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26N4O4
(7S)-7-(4-hydroxy-3-methoxyphenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-phenyl-2-(trifluoromethyl)-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one —— C12H9F3N4O
(7R)-7-phenyl-2-(trifluoromethyl)-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one
—— (7S)-N-(4-chlorophenyl)-5-methyl-7-(4-nitrophenyl)-2-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H20ClN5O3
(7S)-N-(4-chlorophenyl)-5-methyl-7-(4-nitrophenyl)-2-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C29H27ClN4O3
(7R)-2-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3-cyano-7-(3-hydroxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H17N5O2
(7R)-3-cyano-7-(3-hydroxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-5-methyl-7-(4-nitrophenyl)-2-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H20ClN5O3
(7R)-N-(4-chlorophenyl)-5-methyl-7-(4-nitrophenyl)-2-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C29H27ClN4O3
(7S)-2-(4-chlorophenyl)-N-(2,4-dimethylphenyl)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-2,5-dimethyl-7-(4-nitrophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H18ClN5O3
(7R)-N-(4-chlorophenyl)-2,5-dimethyl-7-(4-nitrophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-3-cyano-5-methyl-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H16ClN5O
(7R)-N-(4-chlorophenyl)-3-cyano-5-methyl-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2,5-dimethyl-7-(4-nitrophenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H19N5O3
(7S)-2,5-dimethyl-7-(4-nitrophenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-cyanophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C23H20N6O3
(7R)-7-(4-cyanophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-N-(4-chlorophenyl)-7-(4-methoxyphenyl)-2,5-dioxo-1,6,7,8-tetrahydroquinoline-3-carboxamide —— C23H19ClN2O4
(7S)-N-(4-chlorophenyl)-7-(4-methoxyphenyl)-2,5-dioxo-1,6,7,8-tetrahydroquinoline-3-carboxamide
—— (7R)-2-(4-chlorophenyl)-5-methyl-N-phenyl-7-pyridin-3-yl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C25H20ClN5O
(7R)-2-(4-chlorophenyl)-5-methyl-N-phenyl-7-pyridin-3-yl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-cyanophenyl)-2,5-dimethyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H19N5O
(7R)-7-(4-cyanophenyl)-2,5-dimethyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C21H18ClN5O2
(7S)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(4-bromophenyl)-2,5-dimethyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H19BrN4O
(7S)-7-(4-bromophenyl)-2,5-dimethyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-(4-chlorophenyl)-5-methyl-7-(4-nitrophenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C26H20ClN5O3
(7R)-2-(4-chlorophenyl)-5-methyl-7-(4-nitrophenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-N,2-diphenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H24N4O3
(7S)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-N,2-diphenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23BrN4O2
(7R)-7-(4-bromophenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-chlorophenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClN4O2
(7R)-7-(4-chlorophenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2,5-dimethyl-7-(4-nitrophenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H19N5O3
(7R)-2,5-dimethyl-7-(4-nitrophenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-cyanophenyl)-2,5-dimethyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H19N5O
(7S)-7-(4-cyanophenyl)-2,5-dimethyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3-cyano-N-(2,4-dimethylphenyl)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C24H23N5O3
(7R)-3-cyano-N-(2,4-dimethylphenyl)-7-(4-hydroxy-3-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-bromophenyl)-2,5-dimethyl-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H19BrN4O
(7R)-N-(4-bromophenyl)-2,5-dimethyl-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-2,5-dimethyl-7-(4-nitrophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H18ClN5O3
(7S)-N-(4-chlorophenyl)-2,5-dimethyl-7-(4-nitrophenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-hydroxy-3-methoxyphenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26N4O4
(7R)-7-(4-hydroxy-3-methoxyphenyl)-2-(4-methoxyphenyl)-5-methyl-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-3-cyano-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H18BrN5O2
(7R)-7-(4-bromophenyl)-3-cyano-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[[(1S,2S,4aS,6S,8aS)-1,6-dihydroxy-1,5,5,8a-tetramethyl-3,4,4a,6,7,8-hexahydro-2H-naphthalen-2-yl]methoxy]chromen-2-one —— C24H32O5
7-[[(1S,2S,4aS,6S,8aS)-1,6-dihydroxy-1,5,5,8a-tetramethyl-3,4,4a,6,7,8-hexahydro-2H-naphthalen-2-yl]methoxy]chromen-2-one
—— (7S)-7-(4-cyanophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C23H20N6O3
(7S)-7-(4-cyanophenyl)-6-N-(2-methoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide