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—— (7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21ClN6O3
(7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H22ClN5O3
(7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21N5O3
(7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H20ClN5O3S
(7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H22ClN5O3
(7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(methoxymethyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23N5O4
(7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(methoxymethyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-methylsulfanyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21N5O3S
(7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-methylsulfanyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23N5O3S
(7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21ClN6O3
(7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(methoxymethyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23N5O4
(7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(methoxymethyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H20ClN5O3
(7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21ClN6O3
(7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O3
(7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-phenyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22N6O3
(7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-phenyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(hydroxymethyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21N5O4
(7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(hydroxymethyl)-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23N5O3S
(7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethylsulfanyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H20ClN5O3S
(7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23N5O3
(7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethyl-5-methyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-phenyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22N6O3
(7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-phenyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O3
(7R)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H21ClN6O3
(7S)-N-(4-chlorophenyl)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-phenyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H18F3N5O3
(7S)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-phenyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,5-dimethyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21N5O3
(7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,5-dimethyl-N-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-phenyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H22N6O3
(7R)-7-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-N-phenyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-chloro-3-cyclohexyl-2-[[(2S)-oxolan-2-yl]methylsulfanyl]quinazolin-4-one —— C19H23ClN2O2S
7-chloro-3-cyclohexyl-2-[[(2S)-oxolan-2-yl]methylsulfanyl]quinazolin-4-one
—— 7-[(3-methoxyphenyl)methyl]-N-[(3S)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine —— C20H26N4O2
7-[(3-methoxyphenyl)methyl]-N-[(3S)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine
—— 7-[(3-methoxyphenyl)methyl]-N-[(3R)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine —— C20H26N4O2
7-[(3-methoxyphenyl)methyl]-N-[(3R)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine
—— (7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-(3-methylphenyl)-7,8-dihydro-6H-quinazolin-5-one —— C26H25N5O
(7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-(3-methylphenyl)-7,8-dihydro-6H-quinazolin-5-one
—— 7-[(3R)-3-(2-chlorophenyl)pyrrolidin-1-yl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidine —— C18H19ClN4O
7-[(3R)-3-(2-chlorophenyl)pyrrolidin-1-yl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidine
—— 7-[(3S)-3-(2-chlorophenyl)pyrrolidin-1-yl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidine —— C18H19ClN4O
7-[(3S)-3-(2-chlorophenyl)pyrrolidin-1-yl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidine
—— (7R)-4-amino-2-(furan-2-ylmethylamino)-7-phenyl-7,8-dihydro-6H-quinazolin-5-one —— C19H18N4O2
(7R)-4-amino-2-(furan-2-ylmethylamino)-7-phenyl-7,8-dihydro-6H-quinazolin-5-one
—— 7-[(3S)-3-methoxypyrrolidin-1-yl]-5-propan-2-ylpyrazolo[1,5-a]pyrimidine —— C14H20N4O
7-[(3S)-3-methoxypyrrolidin-1-yl]-5-propan-2-ylpyrazolo[1,5-a]pyrimidine
—— (7R)-7-(2,4-dimethoxyphenyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7,8-dihydro-6H-quinazolin-5-one —— C27H27N5O3
(7R)-7-(2,4-dimethoxyphenyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7,8-dihydro-6H-quinazolin-5-one
—— 7-[(3R)-3-methoxypyrrolidin-1-yl]-5-propan-2-ylpyrazolo[1,5-a]pyrimidine —— C14H20N4O
7-[(3R)-3-methoxypyrrolidin-1-yl]-5-propan-2-ylpyrazolo[1,5-a]pyrimidine
—— (7R)-4-amino-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-7-phenyl-7,8-dihydro-6H-quinazolin-5-one —— C23H22N4O
(7R)-4-amino-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-7-phenyl-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4,7-dimethyl-7,8-dihydro-6H-quinazolin-5-one —— C20H21N5O
(7S)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4,7-dimethyl-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-(2-methylphenyl)-7,8-dihydro-6H-quinazolin-5-one —— C26H25N5O
(7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-(2-methylphenyl)-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-7-(3-chlorophenyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7,8-dihydro-6H-quinazolin-5-one —— C25H22ClN5O
(7S)-7-(3-chlorophenyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-4-amino-2-(furan-2-ylmethylamino)-7-phenyl-7,8-dihydro-6H-quinazolin-5-one —— C19H18N4O2
(7S)-4-amino-2-(furan-2-ylmethylamino)-7-phenyl-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-[(E)-2-phenylethenyl]-7,8-dihydro-6H-quinazolin-5-one —— C27H25N5O
(7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-[(E)-2-phenylethenyl]-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-7-(3-chlorophenyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7,8-dihydro-6H-quinazolin-5-one —— C25H22ClN5O
(7R)-7-(3-chlorophenyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-7-(4-fluorophenyl)-4-methyl-7,8-dihydro-6H-quinazolin-5-one —— C25H22FN5O
(7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-7-(4-fluorophenyl)-4-methyl-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-thiophen-2-yl-7,8-dihydro-6H-quinazolin-5-one —— C23H21N5OS
(7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-thiophen-2-yl-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-4-amino-2-(benzylamino)-7-phenyl-7,8-dihydro-6H-quinazolin-5-one —— C21H20N4O
(7S)-4-amino-2-(benzylamino)-7-phenyl-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4,7-dimethyl-7,8-dihydro-6H-quinazolin-5-one —— C20H21N5O
(7R)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4,7-dimethyl-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-2-[(4,6-dimethylquinazolin-2-yl)amino]-7-(4-fluorophenyl)-4-methyl-7,8-dihydro-6H-quinazolin-5-one —— C25H22FN5O
(7S)-2-[(4,6-dimethylquinazolin-2-yl)amino]-7-(4-fluorophenyl)-4-methyl-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-7-(4-chlorophenyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7,8-dihydro-6H-quinazolin-5-one —— C25H22ClN5O
(7S)-7-(4-chlorophenyl)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-4-amino-2-(cyclohexylamino)-7-phenyl-7,8-dihydro-6H-quinazolin-5-one —— C20H24N4O
(7R)-4-amino-2-(cyclohexylamino)-7-phenyl-7,8-dihydro-6H-quinazolin-5-one
—— (7R)-4-amino-2-[(3R)-3-methylpiperidin-1-yl]-7-phenyl-7,8-dihydro-6H-quinazolin-5-one —— C20H24N4O
(7R)-4-amino-2-[(3R)-3-methylpiperidin-1-yl]-7-phenyl-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-thiophen-2-yl-7,8-dihydro-6H-quinazolin-5-one —— C23H21N5OS
(7S)-2-[(4,6-dimethylquinazolin-2-yl)amino]-4-methyl-7-thiophen-2-yl-7,8-dihydro-6H-quinazolin-5-one