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—— 7-[(2-Methyl-1-prop-2-enylindol-3-yl)methyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H29N5O2
7-[(2-Methyl-1-prop-2-enylindol-3-yl)methyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— [7-(Ethoxycarbonylamino)-2-oxochromen-4-yl]methyl-(3-propan-2-yloxypropyl)azanium —— C19H27N2O5+
[7-(Ethoxycarbonylamino)-2-oxochromen-4-yl]methyl-(3-propan-2-yloxypropyl)azanium
—— 7-[[(2S)-3,4-dihydro-2H-pyran-2-yl]methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H28N4O2
7-[[(2S)-3,4-dihydro-2H-pyran-2-yl]methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(5-bromofuran-2-yl)methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H23BrN4O3
7-[(5-bromofuran-2-yl)methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(6-Methylpyridin-2-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H23N5O
7-[(6-Methylpyridin-2-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Propan-2-ylbenzimidazol-2-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N6O
7-[(1-Propan-2-ylbenzimidazol-2-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-bromothiophen-2-yl)methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H23BrN4O2S
7-[(4-bromothiophen-2-yl)methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(6-methyl-4-oxochromen-3-yl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H28N4O3
7-[(6-methyl-4-oxochromen-3-yl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2H-chromen-3-ylmethyl)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H28N4O3
7-(2H-chromen-3-ylmethyl)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(Cyclohexylmethyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H32N4O
7-(Cyclohexylmethyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[(1R,2S)-2,4-dimethylcyclohex-3-en-1-yl]methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H34N4O2
7-[[(1R,2S)-2,4-dimethylcyclohex-3-en-1-yl]methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[(2R)-3,4-dihydro-2H-pyran-2-yl]methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H26N4O2
7-[[(2R)-3,4-dihydro-2H-pyran-2-yl]methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3-Methylthiophen-2-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H22N4OS
7-[(3-Methylthiophen-2-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[(2S)-3,4-dihydro-2H-pyran-2-yl]methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H26N4O2
7-[[(2S)-3,4-dihydro-2H-pyran-2-yl]methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(5-Methylfuran-2-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H22N4O2
7-[(5-Methylfuran-2-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(furan-2-ylmethyl)-2-[(3R)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H24N4O2
7-(furan-2-ylmethyl)-2-[(3R)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2R)-3-(1,3-benzodioxol-5-yl)-2-methylpropyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H32N4O3
7-[(2R)-3-(1,3-benzodioxol-5-yl)-2-methylpropyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— [7-(Ethoxycarbonylamino)-2-oxochromen-4-yl]methyl-(3-morpholin-4-ium-4-ylpropyl)azanium —— C20H29N3O5+2
[7-(Ethoxycarbonylamino)-2-oxochromen-4-yl]methyl-(3-morpholin-4-ium-4-ylpropyl)azanium
—— 7-[[(1R,2S)-2,4-dimethylcyclohex-3-en-1-yl]methyl]-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H34N4O2
7-[[(1R,2S)-2,4-dimethylcyclohex-3-en-1-yl]methyl]-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[1-(4-Methylpyridin-2-yl)pyrrol-2-yl]methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H26N6O
7-[[1-(4-Methylpyridin-2-yl)pyrrol-2-yl]methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2H-chromen-3-ylmethyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H28N4O2
7-(2H-chromen-3-ylmethyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(furan-2-ylmethyl)-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H24N4O2
7-(furan-2-ylmethyl)-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclohexylmethyl)-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H32N4O2
7-(cyclohexylmethyl)-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— [7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl-[[(2R)-oxolan-2-yl]methyl]azanium —— C18H23N2O5+
[7-(ethoxycarbonylamino)-2-oxochromen-4-yl]methyl-[[(2R)-oxolan-2-yl]methyl]azanium
—— 7-[(1,5-dimethylpyrazol-4-yl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H28N6O
7-[(1,5-dimethylpyrazol-4-yl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Prop-2-ynylindol-3-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O
7-[(1-Prop-2-ynylindol-3-yl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Ethyl-4-methyl-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one —— C11H11N3O2
7-Ethyl-4-methyl-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one
—— 7-Ethyl-4-methyl-10-(2-morpholin-4-yl-2-oxoethyl)-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one —— C17H20N4O4
7-Ethyl-4-methyl-10-(2-morpholin-4-yl-2-oxoethyl)-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one
—— 7-ethyl-4-methyl-10-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one —— C19H24N4O3
7-ethyl-4-methyl-10-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one
—— 7-ethyl-4-methyl-10-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one —— C19H24N4O3
7-ethyl-4-methyl-10-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one
—— 7-Ethyl-10-[(3-fluorophenyl)methyl]-4-methyl-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one —— C18H16FN3O2
7-Ethyl-10-[(3-fluorophenyl)methyl]-4-methyl-3-oxa-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one
—— 7-[(2-methylsulfanylbenzoyl)amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate —— C18H16NO5S-
7-[(2-methylsulfanylbenzoyl)amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate
—— 7-Ethyl-4-methyl-10-prop-2-ynyl-3-thia-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one —— C14H13N3OS
7-Ethyl-4-methyl-10-prop-2-ynyl-3-thia-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one
—— 7-[(2-chlorobenzoyl)amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate —— C17H13ClNO5-
7-[(2-chlorobenzoyl)amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate
—— 7-[(4-Fluorophenyl)methyl]-4-methyl-10-(2-pyrrolidin-1-ylethyl)-3-thia-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one —— C22H23FN4OS
7-[(4-Fluorophenyl)methyl]-4-methyl-10-(2-pyrrolidin-1-ylethyl)-3-thia-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one
—— 7-[(3-Methoxyphenyl)methyl]-4-methyl-10-(2-pyrrolidin-1-ylethyl)-3-thia-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one —— C23H26N4O2S
7-[(3-Methoxyphenyl)methyl]-4-methyl-10-(2-pyrrolidin-1-ylethyl)-3-thia-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one
—— [7-(Difluoromethyl)-5-methylpyrazolo[1,5-a]pyrimidin-3-yl]-[4-(5-pyridin-4-ylpyrimidin-4-yl)piperidin-1-yl]methanone —— C23H21F2N7O
[7-(Difluoromethyl)-5-methylpyrazolo[1,5-a]pyrimidin-3-yl]-[4-(5-pyridin-4-ylpyrimidin-4-yl)piperidin-1-yl]methanone
—— 7-[(3-Methoxyphenyl)methyl]-4-methyl-10-propan-2-yl-3-thia-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one —— C20H21N3O2S
7-[(3-Methoxyphenyl)methyl]-4-methyl-10-propan-2-yl-3-thia-7,10,11-triazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),4,11-tetraen-9-one
—— 7-[(2,4-dimethoxybenzoyl)amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate —— C19H18NO7-
7-[(2,4-dimethoxybenzoyl)amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate
—— 7-[[2-(difluoromethoxy)benzoyl]amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate —— C18H14F2NO6-
7-[[2-(difluoromethoxy)benzoyl]amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate
—— 7-[(2-methylsulfonylbenzoyl)amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate —— C18H16NO7S-
7-[(2-methylsulfonylbenzoyl)amino]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxylate
—— (7R)-N-(5-chloro-2-methoxyphenyl)-3-(4-methoxyphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C21H19ClN4O4
(7R)-N-(5-chloro-2-methoxyphenyl)-3-(4-methoxyphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(5-chloro-2-methoxyphenyl)-2-(4-chlorophenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C20H16Cl2N4O3
(7S)-N-(5-chloro-2-methoxyphenyl)-2-(4-chlorophenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C22H22N4O3
(7S)-N-(2,4-dimethylphenyl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C22H22N4O3
(7R)-N-(2,4-dimethylphenyl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(4-bromophenyl)-2-(4-methylphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C20H17BrN4O2
(7R)-N-(4-bromophenyl)-2-(4-methylphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-2-[(2,4-difluorophenyl)sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H16F2N2OS2
(7S)-2-[(2,4-difluorophenyl)sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-N-(4-methoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C15H16N4O3
(7R)-N-(4-methoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(2,5-dimethoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C16H18N4O4
(7R)-N-(2,5-dimethoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(5-chloro-2-methoxyphenyl)-3-(4-methoxyphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide —— C21H19ClN4O4
(7S)-N-(5-chloro-2-methoxyphenyl)-3-(4-methoxyphenyl)-5-oxo-6,7-dihydro-1H-pyrazolo[1,5-a]pyrimidine-7-carboxamide