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—— (7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(4,6-dimethyl-2-methylsulfanylpyrimidin-5-yl)propanoate —— C17H19N5O3S2
(7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(4,6-dimethyl-2-methylsulfanylpyrimidin-5-yl)propanoate
—— (7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(2-methylpropan-2-yl)oxycarbonylamino]benzoate —— C19H20N4O5S
(7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(2-methylpropan-2-yl)oxycarbonylamino]benzoate
—— (7-hydroxy-2-oxo-2H-chromen-4-yl)methyl acetate —— C12H10O5
(7-hydroxy-2-oxo-2H-chromen-4-yl)methyl acetate
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate —— C20H16N2O6S
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate
—— (7,8-Dimethyl-2-oxochromen-4-yl)methyl acetate —— C14H14O4
(7,8-Dimethyl-2-oxochromen-4-yl)methyl acetate
—— (7,8-Dimethyl-2-oxochromen-4-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate —— C21H18N2O5S
(7,8-Dimethyl-2-oxochromen-4-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate
—— (7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate —— C19H16N4O4S
(7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)propanoate
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 2-(3,4-dichlorophenyl)acetate —— C18H12Cl2O5
(7-Hydroxy-2-oxochromen-4-yl)methyl 2-(3,4-dichlorophenyl)acetate
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 2,6-dichlorobenzoate —— C17H10Cl2O5
(7-Hydroxy-2-oxochromen-4-yl)methyl 2,6-dichlorobenzoate
—— (7-Ethyl-2-oxochromen-4-yl)methyl 2,6-dichlorobenzoate —— C19H14Cl2O4
(7-Ethyl-2-oxochromen-4-yl)methyl 2,6-dichlorobenzoate
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2,6-dichlorobenzoate —— C18H12Cl2O5
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2,6-dichlorobenzoate
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 2,5-dichlorobenzoate —— C17H10Cl2O5
(7-Hydroxy-2-oxochromen-4-yl)methyl 2,5-dichlorobenzoate
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2,5-dichlorobenzoate —— C18H12Cl2O5
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2,5-dichlorobenzoate
—— 7-[(3R)-3-propoxypiperidin-1-yl]-5-propylpyrazolo[1,5-a]pyrimidine —— C17H26N4O
7-[(3R)-3-propoxypiperidin-1-yl]-5-propylpyrazolo[1,5-a]pyrimidine
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2-cyclopentylacetate —— C18H20O5
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2-cyclopentylacetate
—— 7-[(3S)-3-propoxypiperidin-1-yl]-5-propylpyrazolo[1,5-a]pyrimidine —— C17H26N4O
7-[(3S)-3-propoxypiperidin-1-yl]-5-propylpyrazolo[1,5-a]pyrimidine
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 2-cyclopentylacetate —— C17H18O5
(7-Hydroxy-2-oxochromen-4-yl)methyl 2-cyclopentylacetate
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2-(2-chloro-6-fluorophenyl)acetate —— C19H14ClFO5
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2-(2-chloro-6-fluorophenyl)acetate
—— (7S)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-7-methyl-6,7,8,9-tetrahydro-[1,2,4]triazolo[1,5-a]quinazoline —— C19H20N4O2
(7S)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-7-methyl-6,7,8,9-tetrahydro-[1,2,4]triazolo[1,5-a]quinazoline
—— (7R)-2-[(3,4-difluorophenyl)sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H16F2N2OS2
(7R)-2-[(3,4-difluorophenyl)sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28N6O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H27N5O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(4-methoxyphenyl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O3
(7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O4
(7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H29N5O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-ethyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(4-methylphenyl)-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26N6O3
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(4-methylphenyl)-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O4S
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(2-methylphenyl)-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H27N5O3
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(2-methylphenyl)-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O3
(7R)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H20ClN5O3
(7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-7-methyl-6,7,8,9-tetrahydro-[1,2,4]triazolo[1,5-a]quinazoline —— C19H20N4O2
(7R)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-7-methyl-6,7,8,9-tetrahydro-[1,2,4]triazolo[1,5-a]quinazoline
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-methoxyphenyl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26N6O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-methoxyphenyl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-methoxyphenyl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H27N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-methoxyphenyl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H24ClN5O4
(7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(4-methylphenyl)-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H25N5O3S
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-N-(4-methylphenyl)-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H19ClF3N5O3
(7R)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-N-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H27N5O4S
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-ethylsulfanyl-N-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-methoxyphenyl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26N6O4
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-methoxyphenyl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClN6O3
(7S)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-3-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClN6O3
(7R)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O3
(7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2,5-dimethyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H21ClF3N5O3
(7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H26ClN5O4
(7S)-N-(3-chloro-4-methylphenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(methoxymethyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H29N5O4S
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H22ClN5O3S
(7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-methylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23ClN6O3
(7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-pyridin-4-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H19ClF3N5O3
(7R)-N-(2-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H29N5O4
(7S)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-N-(2-ethoxyphenyl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H24ClN5O3
(7S)-N-(3-chlorophenyl)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5-methyl-2-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H25N5O5
(7R)-7-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-(hydroxymethyl)-N-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide