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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-Methyl-4-(pyridin-3-ylmethyl)-12,14-dioxa-2,4,5-triazatetracyclo[7.7.0.02,6.011,15]hexadeca-1(16),5,7,9,11(15)-pentaen-3-one —— C18H14N4O3
7-Methyl-4-(pyridin-3-ylmethyl)-12,14-dioxa-2,4,5-triazatetracyclo[7.7.0.02,6.011,15]hexadeca-1(16),5,7,9,11(15)-pentaen-3-one
—— 7-[2-(2-Methylbenzimidazol-1-yl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H24N6O2
7-[2-(2-Methylbenzimidazol-1-yl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3,4-dichlorophenyl)methyl]-2-[(2R)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24Cl2N4O
7-[(3,4-dichlorophenyl)methyl]-2-[(2R)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-(3-Methoxyphenyl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N4O3
7-[2-(3-Methoxyphenyl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-Hydroxy-3-methoxyphenyl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N4O3
7-[(4-Hydroxy-3-methoxyphenyl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3-methoxyphenyl)methyl]-2-[(2R)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N4O2
7-[(3-methoxyphenyl)methyl]-2-[(2R)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(5-Methyl-1-propylpyrazole-4-carbonyl)-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H28N6O2
7-(5-Methyl-1-propylpyrazole-4-carbonyl)-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3,5-dimethoxyphenyl)methyl]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N4O4
7-[(3,5-dimethoxyphenyl)methyl]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,5-dimethoxyphenyl)methyl]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N4O4
7-[(2,5-dimethoxyphenyl)methyl]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(5-chloro-2-hydroxyphenyl)methyl]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25ClN4O3
7-[(5-chloro-2-hydroxyphenyl)methyl]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(6-hydroxy-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8-trien-7-yl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C26H35N5O2
7-[(6-hydroxy-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8-trien-7-yl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-(2-Methoxyphenyl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N4O3
7-[2-(2-Methoxyphenyl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,4-dimethoxyphenyl)methyl]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N4O4
7-[(2,4-dimethoxyphenyl)methyl]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-Morpholin-4-ylphenyl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H29N5O2
7-[(4-Morpholin-4-ylphenyl)methyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(Furan-2-carbonyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H22N4O3
7-(Furan-2-carbonyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-Methoxyphenyl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N4O2
7-[(2-Methoxyphenyl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-Ethoxyphenyl)methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N4O2
7-[(4-Ethoxyphenyl)methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[3-(3,5-Dimethylpyrazol-1-yl)propanoyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H30N6O2
7-[3-(3,5-Dimethylpyrazol-1-yl)propanoyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,5-dimethoxyphenyl)methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N4O4
7-[(2,5-dimethoxyphenyl)methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-(2-Chlorophenyl)acetyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H21ClN4O3
7-[2-(2-Chlorophenyl)acetyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2H-chromene-3-carbonyl)-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H22N4O4
7-(2H-chromene-3-carbonyl)-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Methyl-12,14-dioxa-2,4,5-triazatetracyclo[7.7.0.02,6.011,15]hexadeca-1(16),5,7,9,11(15)-pentaen-3-one —— C12H9N3O3
7-Methyl-12,14-dioxa-2,4,5-triazatetracyclo[7.7.0.02,6.011,15]hexadeca-1(16),5,7,9,11(15)-pentaen-3-one
—— 7-Methoxy-4-methyl-2-(pyridin-3-ylmethyl)-[1,2,4]triazolo[4,3-a]quinolin-1-one —— C18H16N4O2
7-Methoxy-4-methyl-2-(pyridin-3-ylmethyl)-[1,2,4]triazolo[4,3-a]quinolin-1-one
—— 7-(furan-2-carbonyl)-2-[(2S)-2-methylpiperidin-1-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H22N4O3
7-(furan-2-carbonyl)-2-[(2S)-2-methylpiperidin-1-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-(3-Hydroxyphenyl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H22N4O3
7-[2-(3-Hydroxyphenyl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3,4-Dimethoxyphenyl)methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N4O3
7-[(3,4-Dimethoxyphenyl)methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3,5-dimethoxyphenyl)methyl]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N4O4
7-[(3,5-dimethoxyphenyl)methyl]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-(dimethylamino)phenyl]methyl]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H31N5O2
7-[[4-(dimethylamino)phenyl]methyl]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(1-Ethyl-3-methylpyrazole-4-carbonyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H28N6O2
7-(1-Ethyl-3-methylpyrazole-4-carbonyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Methoxy-4-methyl-2-(pyridin-2-ylmethyl)-[1,2,4]triazolo[4,3-a]quinolin-1-one —— C18H16N4O2
7-Methoxy-4-methyl-2-(pyridin-2-ylmethyl)-[1,2,4]triazolo[4,3-a]quinolin-1-one
—— 7-(furan-2-carbonyl)-2-[(2R)-2-methylpiperidin-1-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H22N4O3
7-(furan-2-carbonyl)-2-[(2R)-2-methylpiperidin-1-yl]-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(Pyrazolo[1,5-a]pyrimidine-3-carbonyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H19N7O2
7-(Pyrazolo[1,5-a]pyrimidine-3-carbonyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-(Benzotriazol-1-yl)acetyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H23N7O2
7-[2-(Benzotriazol-1-yl)acetyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(5-Methyl-1-propylpyrazole-4-carbonyl)-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H26N6O3
7-(5-Methyl-1-propylpyrazole-4-carbonyl)-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-(4-Methoxyphenyl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N4O3
7-[2-(4-Methoxyphenyl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[5-(Piperidin-1-ylmethyl)furan-2-carbonyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H29N5O3
7-[5-(Piperidin-1-ylmethyl)furan-2-carbonyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(Pyridine-2-carbonyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H19N5O2
7-(Pyridine-2-carbonyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[4-(Dimethylamino)benzoyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O2
7-[4-(Dimethylamino)benzoyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(3,4-Dimethoxybenzoyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O4
7-(3,4-Dimethoxybenzoyl)-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(3-Phenylpropanoyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N4O2
7-(3-Phenylpropanoyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(1-Ethylpyrazole-4-carbonyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H22N6O2
7-(1-Ethylpyrazole-4-carbonyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-Fluorobenzoyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H19FN4O2
7-(2-Fluorobenzoyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Ethyl-4-(pyridin-4-ylmethyl)-12,14-dioxa-2,4,5-triazatetracyclo[7.7.0.02,6.011,15]hexadeca-1(16),5,7,9,11(15)-pentaen-3-one —— C19H16N4O3
7-Ethyl-4-(pyridin-4-ylmethyl)-12,14-dioxa-2,4,5-triazatetracyclo[7.7.0.02,6.011,15]hexadeca-1(16),5,7,9,11(15)-pentaen-3-one
—— 7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H28N6O2
7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-(4-oxo-3H-phthalazin-1-yl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H22N6O3
7-[2-(4-oxo-3H-phthalazin-1-yl)acetyl]-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(1H-pyrazole-5-carbonyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C15H18N6O2
7-(1H-pyrazole-5-carbonyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-Methylpropanoyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C15H22N4O2
7-(2-Methylpropanoyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-Cyclopentylacetyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H26N4O2
7-(2-Cyclopentylacetyl)-2-pyrrolidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3R)-1-benzyl-5-oxopyrrolidine-3-carbonyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H27N5O4
7-[(3R)-1-benzyl-5-oxopyrrolidine-3-carbonyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-(2-Ethylbenzimidazol-1-yl)acetyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H26N6O3
7-[2-(2-Ethylbenzimidazol-1-yl)acetyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one