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—— 7-[(2S)-1-[2-(1H-indol-3-yl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C24H25N5O3
7-[(2S)-1-[2-(1H-indol-3-yl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(cyclopentanecarbonyl)piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C20H26N4O3
7-[(3R)-1-(cyclopentanecarbonyl)piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-(cyclopentanecarbonyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C20H26N4O3
7-[(2R)-1-(cyclopentanecarbonyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C21H23FN4O2
7-[(2R)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3S)-1-(cyclopropylmethyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C19H23F3N4O2
7-[(3S)-1-(cyclopropylmethyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-(cyclopentanecarbonyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C20H26N4O3
7-[(2S)-1-(cyclopentanecarbonyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H23FN4O3
7-[(2R)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C18H25N5O3
7-[(2S)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-(4-methoxyphenyl)sulfonylpiperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine —— C19H21N5O3S
7-[(2S)-1-(4-methoxyphenyl)sulfonylpiperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(2R)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C18H25N5O3
7-[(2R)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(cyclopropylmethyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C19H23F3N4O2
7-[(3R)-1-(cyclopropylmethyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C21H25N5O4
7-[(2S)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H23FN4O3
7-[(2S)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine —— C18H18FN5O2S
7-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(2S)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C24H28N4O4
7-[(2S)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-(4-methoxyphenyl)sulfonylpiperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine —— C19H21N5O3S
7-[(2R)-1-(4-methoxyphenyl)sulfonylpiperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(2R)-1-[2-(1H-indol-3-yl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C24H25N5O3
7-[(2R)-1-[2-(1H-indol-3-yl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-[2-(4-fluorophenoxy)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H23FN4O4
7-[(2S)-1-[2-(4-fluorophenoxy)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C24H28N4O4
7-[(2R)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C20H21FN4O4S
7-[(2S)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[[2-(2-methoxyphenyl)phenyl]methyl]-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C23H27N5O
7-[[2-(2-methoxyphenyl)phenyl]methyl]-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-methyl-3-[(2S)-1-methylpiperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C12H21N5
7-methyl-3-[(2S)-1-methylpiperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(4-methoxy-2,5-dimethylphenyl)sulfonyl-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C18H25N5O3S
7-(4-methoxy-2,5-dimethylphenyl)sulfonyl-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[[2-(2-methoxyphenyl)phenyl]methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C23H27N5O
7-[[2-(2-methoxyphenyl)phenyl]methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[[4-(3-fluorophenyl)phenyl]methyl]-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C23H26FN5
7-[[4-(3-fluorophenyl)phenyl]methyl]-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(2-methylphenyl)methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C18H25N5
7-[(2-methylphenyl)methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[[4-(3-fluorophenyl)phenyl]methyl]-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C22H24FN5
7-[[4-(3-fluorophenyl)phenyl]methyl]-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(4-methoxy-2,5-dimethylphenyl)sulfonyl-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C18H25N5O3S
7-(4-methoxy-2,5-dimethylphenyl)sulfonyl-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(2-methoxy-4-methylphenyl)methyl]-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H27N5O
7-[(2-methoxy-4-methylphenyl)methyl]-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(4,6-dimethylpyrimidin-2-yl)-3-[(2R)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C16H23N7
7-(4,6-dimethylpyrimidin-2-yl)-3-[(2R)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C21H29N5O
7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-methyl-3-[(2S)-1-(2-phenylethylsulfonyl)piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H27N5O2S
7-methyl-3-[(2S)-1-(2-phenylethylsulfonyl)piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(2-phenylethyl)-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C18H25N5
7-(2-phenylethyl)-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C22H31N5O
7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[[4-(3-fluorophenyl)phenyl]methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C22H24FN5
7-[[4-(3-fluorophenyl)phenyl]methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C22H31N5O
7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(2-phenylethyl)-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C18H25N5
7-(2-phenylethyl)-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[[2-(2-fluorophenyl)phenyl]methyl]-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C23H26FN5
7-[[2-(2-fluorophenyl)phenyl]methyl]-3-[(2R)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-methyl-3-[(2S)-1-[(3-methylphenyl)methylsulfonyl]piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H27N5O2S
7-methyl-3-[(2S)-1-[(3-methylphenyl)methylsulfonyl]piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(2-methoxy-4-methylphenyl)methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H27N5O
7-[(2-methoxy-4-methylphenyl)methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[[4-(3-fluorophenyl)phenyl]methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C23H26FN5
7-[[4-(3-fluorophenyl)phenyl]methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-methyl-3-[(2R)-1-methylpiperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C12H21N5
7-methyl-3-[(2R)-1-methylpiperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(4,6-dimethylpyrimidin-2-yl)-3-[(2S)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C16H23N7
7-(4,6-dimethylpyrimidin-2-yl)-3-[(2S)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[[2-(2-fluorophenyl)phenyl]methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C23H26FN5
7-[[2-(2-fluorophenyl)phenyl]methyl]-3-[(2S)-piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(4-fluoro-3-methylphenyl)sulfonyl-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C16H20FN5O2S
7-(4-fluoro-3-methylphenyl)sulfonyl-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H25N5O3
7-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-methyl-3-[(2R)-1-[(3-methylphenyl)methylsulfonyl]piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H27N5O2S
7-methyl-3-[(2R)-1-[(3-methylphenyl)methylsulfonyl]piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-methyl-3-[(2R)-1-(2-phenylethylsulfonyl)piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H27N5O2S
7-methyl-3-[(2R)-1-(2-phenylethylsulfonyl)piperidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C21H29N5O
7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2S)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(2-piperidin-1-ylphenyl)methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C21H30N6
7-[(2-piperidin-1-ylphenyl)methyl]-3-[(2R)-pyrrolidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine