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—— (7R)-2-[(1R)-1-[(2-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H24FN3OS
(7R)-2-[(1R)-1-[(2-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-[methyl-[(2-methylphenyl)methyl]amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3OS
(7R)-7-methyl-2-[(1R)-1-[methyl-[(2-methylphenyl)methyl]amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1S)-1-(3-oxopiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H23N4O2S+
(7S)-7-methyl-2-[(1S)-1-(3-oxopiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1S)-1-[methyl(thiophen-2-ylmethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H23N3OS2
(7R)-7-methyl-2-[(1S)-1-[methyl(thiophen-2-ylmethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1S)-1-[methyl-[(4-methylphenyl)methyl]amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3OS
(7R)-7-methyl-2-[(1S)-1-[methyl-[(4-methylphenyl)methyl]amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-[methyl(thiophen-2-ylmethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H23N3OS2
(7R)-7-methyl-2-[(1R)-1-[methyl(thiophen-2-ylmethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-[(2-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H24FN3OS
(7S)-2-[(1R)-1-[(2-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1S)-1-(3-oxopiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H23N4O2S+
(7R)-7-methyl-2-[(1S)-1-(3-oxopiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1R)-1-[methyl(thiophen-2-ylmethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H23N3OS2
(7S)-7-methyl-2-[(1R)-1-[methyl(thiophen-2-ylmethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-(3-oxopiperazin-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H22N4O2S
(7R)-7-methyl-2-[(1R)-1-(3-oxopiperazin-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-(3-oxopiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H23N4O2S+
(7R)-7-methyl-2-[(1R)-1-(3-oxopiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1R)-1-[(3-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H24FN3OS
(7R)-2-[(1R)-1-[(3-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-[(3-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H24FN3OS
(7R)-2-[(1S)-1-[(3-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-[(3-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H24FN3OS
(7S)-2-[(1R)-1-[(3-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-(2,3-dihydro-1H-inden-5-ylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H25N3OS
(7R)-2-[(1S)-1-(2,3-dihydro-1H-inden-5-ylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1S)-1-[(4-methylphenyl)methylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H25N3OS
(7S)-7-methyl-2-[(1S)-1-[(4-methylphenyl)methylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1R)-1-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H27N3O3S
(7R)-2-[(1R)-1-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-[2-(4-methylphenoxy)ethylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S
(7R)-7-methyl-2-[(1R)-1-[2-(4-methylphenoxy)ethylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-Ethyl-4-[(4-pyrrolidin-1-ylanilino)methyl]chromen-2-one —— C22H24N2O2
7-Ethyl-4-[(4-pyrrolidin-1-ylanilino)methyl]chromen-2-one
—— (7S)-7-methyl-2-[(1S)-1-[methyl(2-phenoxyethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S
(7S)-7-methyl-2-[(1S)-1-[methyl(2-phenoxyethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-Hydroxy-8-methyl-4-[(4-pyrrolidin-1-ylanilino)methyl]chromen-2-one —— C21H22N2O3
7-Hydroxy-8-methyl-4-[(4-pyrrolidin-1-ylanilino)methyl]chromen-2-one
—— (7R)-2-[(1S)-1-[(3-methoxyphenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S
(7R)-2-[(1S)-1-[(3-methoxyphenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-[2-(2-methoxyphenoxy)ethylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O3S
(7S)-2-[(1R)-1-[2-(2-methoxyphenoxy)ethylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-(2,3-dihydro-1H-inden-5-ylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H25N3OS
(7S)-2-[(1R)-1-(2,3-dihydro-1H-inden-5-ylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-Methyl-2-[(4-pyrrolidin-1-ylanilino)methyl]pyrido[1,2-a]pyrimidin-4-one —— C20H22N4O
7-Methyl-2-[(4-pyrrolidin-1-ylanilino)methyl]pyrido[1,2-a]pyrimidin-4-one
—— (7R)-2-[(1R)-1-[(3-methoxyphenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S
(7R)-2-[(1R)-1-[(3-methoxyphenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H27N3O3S
(7S)-2-[(1R)-1-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-(2,3-dihydro-1H-inden-5-ylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H25N3OS
(7S)-2-[(1S)-1-(2,3-dihydro-1H-inden-5-ylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1S)-1-[2-(4-methylphenoxy)ethylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S
(7S)-7-methyl-2-[(1S)-1-[2-(4-methylphenoxy)ethylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-(thiophen-2-ylmethylamino)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H21N3OS2
(7R)-7-methyl-2-[(1R)-1-(thiophen-2-ylmethylamino)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-(3,4-diethoxyanilino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H29N3O3S
(7S)-2-[(1R)-1-(3,4-diethoxyanilino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-[(3-methoxyphenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S
(7S)-2-[(1R)-1-[(3-methoxyphenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1S)-1-[methyl(thiophen-2-ylmethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H23N3OS2
(7S)-7-methyl-2-[(1S)-1-[methyl(thiophen-2-ylmethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-[methyl(2-phenoxyethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S
(7R)-7-methyl-2-[(1R)-1-[methyl(2-phenoxyethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1S)-1-(thiophen-2-ylmethylamino)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H21N3OS2
(7S)-7-methyl-2-[(1S)-1-(thiophen-2-ylmethylamino)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-[(3-methoxyphenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S
(7S)-2-[(1S)-1-[(3-methoxyphenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1R)-1-(4-pyrrolidin-1-ylanilino)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H28N4OS
(7S)-7-methyl-2-[(1R)-1-(4-pyrrolidin-1-ylanilino)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7,8-Dimethyl-4-[(4-pyrrolidin-1-ylanilino)methyl]chromen-2-one —— C22H24N2O2
7,8-Dimethyl-4-[(4-pyrrolidin-1-ylanilino)methyl]chromen-2-one
—— (7S)-7-methyl-2-[(1R)-1-[methyl(2-phenoxyethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H27N3O2S
(7S)-7-methyl-2-[(1R)-1-[methyl(2-phenoxyethyl)amino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1S)-1-(thiophen-2-ylmethylamino)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H21N3OS2
(7R)-7-methyl-2-[(1S)-1-(thiophen-2-ylmethylamino)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1S)-1-(3-oxopiperazin-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H22N4O2S
(7R)-7-methyl-2-[(1S)-1-(3-oxopiperazin-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-[(4-methylphenyl)methylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H25N3OS
(7R)-7-methyl-2-[(1R)-1-[(4-methylphenyl)methylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1R)-1-(3-chloro-4-methoxyanilino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H22ClN3O2S
(7R)-2-[(1R)-1-(3-chloro-4-methoxyanilino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1S)-1-[(4-methylphenyl)methylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H25N3OS
(7R)-7-methyl-2-[(1S)-1-[(4-methylphenyl)methylamino]ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1S)-1-(4-pyridin-1-ium-2-ylpiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H29N5OS+2
(7S)-7-methyl-2-[(1S)-1-(4-pyridin-1-ium-2-ylpiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1R)-1-[2-(4-fluorophenyl)ethylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H24FN3OS
(7R)-2-[(1R)-1-[2-(4-fluorophenyl)ethylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-[[(2S)-1-methoxypropan-2-yl]amino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H25N3O2S
(7R)-2-[(1S)-1-[[(2S)-1-methoxypropan-2-yl]amino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-(cyclopentylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H25N3OS
(7S)-2-[(1S)-1-(cyclopentylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-(3-ethylanilino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H25N3OS
(7S)-2-[(1S)-1-(3-ethylanilino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-(3-ethoxypropylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H27N3O2S
(7R)-2-[(1S)-1-(3-ethoxypropylamino)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one