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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-[4-(4-Methoxyphenyl)piperazin-1-yl]-5,6-dimethyl-2-(1-methylimidazol-2-yl)pyrazolo[1,5-a]pyrimidine —— C23H27N7O
7-[4-(4-Methoxyphenyl)piperazin-1-yl]-5,6-dimethyl-2-(1-methylimidazol-2-yl)pyrazolo[1,5-a]pyrimidine
—— 7-[(4-fluorophenyl)methyl]-N-(3-propan-2-yloxypropyl)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C25H30FN5O
7-[(4-fluorophenyl)methyl]-N-(3-propan-2-yloxypropyl)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— [7-(difluoromethyl)-5-methylpyrazolo[1,5-a]pyrimidin-3-yl]-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C21H19F2N7O
[7-(difluoromethyl)-5-methylpyrazolo[1,5-a]pyrimidin-3-yl]-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— [7-(difluoromethyl)-5-methylpyrazolo[1,5-a]pyrimidin-3-yl]-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C21H19F2N7O
[7-(difluoromethyl)-5-methylpyrazolo[1,5-a]pyrimidin-3-yl]-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— 7-[(1-Benzyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H26N6O
7-[(1-Benzyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[3-(3,5-Dimethylpyrazol-1-yl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[[3-(3,5-Dimethylpyrazol-1-yl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-Hydroxy-3-(piperidin-1-ylmethyl)phenyl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H29N5O2
7-[[4-Hydroxy-3-(piperidin-1-ylmethyl)phenyl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Acetylindol-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H21N5O2
7-[(1-Acetylindol-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,5-Dimethyl-1-pyridin-2-ylpyrrol-3-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[(2,5-Dimethyl-1-pyridin-2-ylpyrrol-3-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Methylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H18N6O
7-[(1-Methylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,5-Dimethoxy-4-pyrrolidin-1-ylphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H29N5O3
7-[(2,5-Dimethoxy-4-pyrrolidin-1-ylphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N6O
7-[(1-Ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Benzylbenzimidazol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C27H24N6O
7-[(1-Benzylbenzimidazol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(4-Ethylpiperazin-1-yl)-5,6-dimethyl-2-(oxan-4-yl)pyrazolo[1,5-a]pyrimidine —— C19H29N5O
7-(4-Ethylpiperazin-1-yl)-5,6-dimethyl-2-(oxan-4-yl)pyrazolo[1,5-a]pyrimidine
—— 7-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H19ClN6O
7-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(7-ethyl-1H-indol-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H23N5O
7-[(7-ethyl-1H-indol-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-Methoxy-3-(pyrazol-1-ylmethyl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O2
7-[[4-Methoxy-3-(pyrazol-1-ylmethyl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-fluorophenyl)methyl]-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C18H22FN5
7-[(4-fluorophenyl)methyl]-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-[[3-(3,5-Dimethylpyrazol-1-yl)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[[3-(3,5-Dimethylpyrazol-1-yl)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-Methoxy-3-(morpholin-4-ylmethyl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H29N5O3
7-[[4-Methoxy-3-(morpholin-4-ylmethyl)phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Methylpyrrol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H19N5O
7-[(1-Methylpyrrol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-(Diethylamino)-2-methoxyphenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H29N5O2
7-[[4-(Diethylamino)-2-methoxyphenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Benzyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H26N6O
7-[(1-Benzyl-3,5-dimethylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-pyridin-3-ylpyrrol-2-yl)methyl]-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C21H25N7
7-[(1-pyridin-3-ylpyrrol-2-yl)methyl]-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-[(2-Methyl-4-morpholin-4-ylphenyl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27N5O2
7-[(2-Methyl-4-morpholin-4-ylphenyl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,7-Dimethoxyquinolin-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H23N5O3
7-[(2,7-Dimethoxyquinolin-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-Methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H29N5O2
7-[[4-Methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Ethyl-5-methoxyindol-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H25N5O2
7-[(1-Ethyl-5-methoxyindol-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[1-(4-Fluorophenyl)pyrazol-4-yl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H19FN6O
7-[[1-(4-Fluorophenyl)pyrazol-4-yl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(6-Bromo-1,3-benzodioxol-5-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H17BrN4O3
7-[(6-Bromo-1,3-benzodioxol-5-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[1-(4-Methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C26H27N5O2
7-[[1-(4-Methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27N5O
7-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-Hydroxy-3-[(4-methylpiperazin-1-yl)methyl]phenyl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H30N6O2
7-[[4-Hydroxy-3-[(4-methylpiperazin-1-yl)methyl]phenyl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3-Benzylimidazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H22N6O
7-[(3-Benzylimidazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3,4-difluorophenyl)methyl]-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C18H21F2N5
7-[(3,4-difluorophenyl)methyl]-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-[[4-[(2-Fluorophenyl)methoxy]phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C26H23FN4O2
7-[[4-[(2-Fluorophenyl)methoxy]phenyl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,5-Dimethoxy-4-pyrrolidin-1-ylphenyl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H29N5O3
7-[(2,5-Dimethoxy-4-pyrrolidin-1-ylphenyl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[1-(2-Methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C26H27N5O2
7-[[1-(2-Methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1,5-Dimethylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H20N6O
7-[(1,5-Dimethylpyrazol-4-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-(Azepan-1-yl)-2-oxoethyl]-5-(2-methylphenyl)-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one —— C23H28N6O2
7-[2-(Azepan-1-yl)-2-oxoethyl]-5-(2-methylphenyl)-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one
—— 7-[(4,5-Dimethylfuran-2-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N4O2
7-[(4,5-Dimethylfuran-2-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-Propan-2-ylindol-3-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H25N5O
7-[(1-Propan-2-ylindol-3-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-3,4-dihydro-2H-pyrimido[1,2-c]quinazolin-6-one —— C20H26N4O2
7-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-3,4-dihydro-2H-pyrimido[1,2-c]quinazolin-6-one
—— 7-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one —— C23H28N6O2
7-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one
—— 7-[2-[(2R,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one —— C23H28N6O2
7-[2-[(2R,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one
—— 7-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one —— C22H26N6O2
7-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one
—— 7-Benzyl-4-(1-ethylpiperidin-4-yl)oxy-5,6-dimethylpyrrolo[2,3-d]pyrimidine —— C22H28N4O
7-Benzyl-4-(1-ethylpiperidin-4-yl)oxy-5,6-dimethylpyrrolo[2,3-d]pyrimidine
—— 7-[(1,3-Dimethylpyrazol-4-yl)methyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H24N6O2
7-[(1,3-Dimethylpyrazol-4-yl)methyl]-2-morpholin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-Aminopyrimidin-5-yl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H25N7O
7-[(2-Aminopyrimidin-5-yl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(5-Methylfuran-2-yl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H26N4O2
7-[(5-Methylfuran-2-yl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one