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—— 7-[[4-(3-fluorophenyl)phenyl]methyl]-3-piperidin-4-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C23H26FN5
7-[[4-(3-fluorophenyl)phenyl]methyl]-3-piperidin-4-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-methylsulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C20H30N4O3S
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-methylsulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O2
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-methylsulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C20H30N4O3S
7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-methylsulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-2-[1-(3-methoxypropanoyl)piperidin-4-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O4
7-[(3-methoxyphenyl)methyl]-2-[1-(3-methoxypropanoyl)piperidin-4-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(2S)-1-[3-(2-methylimidazol-1-yl)propanoyl]pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H28N6O2
7-benzyl-4-methyl-2-[(2S)-1-[3-(2-methylimidazol-1-yl)propanoyl]pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2R)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N6O2
7-(cyclopropylmethyl)-2-[(2R)-1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H28N4O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H34N4O3
7-(cyclohexylmethyl)-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H29FN4O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O4
7-[(4-methoxyphenyl)methyl]-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H29FN4O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C22H25FN4O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-propanoylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— (7-Methoxy-2-oxochromen-4-yl)methyl 2-[(2-chlorophenyl)methylsulfanyl]acetate —— C20H17ClO5S
(7-Methoxy-2-oxochromen-4-yl)methyl 2-[(2-chlorophenyl)methylsulfanyl]acetate
—— 7-[(2,5-dimethoxyphenyl)methyl]-3-[(3S)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C20H29N5O2
7-[(2,5-dimethoxyphenyl)methyl]-3-[(3S)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-(2-methoxyphenyl)sulfonyl-3-[(3R)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C18H25N5O3S
7-(2-methoxyphenyl)sulfonyl-3-[(3R)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-[(3-methoxy-5,6,7,8-tetrahydronaphthalen-2-yl)methyl]-3-[(3S)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C23H33N5O
7-[(3-methoxy-5,6,7,8-tetrahydronaphthalen-2-yl)methyl]-3-[(3S)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-methyl-3-[(3S)-1-(4-methylphenyl)sulfonylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C19H27N5O2S
7-methyl-3-[(3S)-1-(4-methylphenyl)sulfonylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-[(3-methoxy-5,6,7,8-tetrahydronaphthalen-2-yl)methyl]-3-[(3R)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C23H33N5O
7-[(3-methoxy-5,6,7,8-tetrahydronaphthalen-2-yl)methyl]-3-[(3R)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-[(2,5-dimethoxyphenyl)methyl]-3-[(3R)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C20H29N5O2
7-[(2,5-dimethoxyphenyl)methyl]-3-[(3R)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-(2-methoxyphenyl)sulfonyl-3-[(3S)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C18H25N5O3S
7-(2-methoxyphenyl)sulfonyl-3-[(3S)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-methyl-3-[(3R)-1-(4-methylphenyl)sulfonylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C19H27N5O2S
7-methyl-3-[(3R)-1-(4-methylphenyl)sulfonylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— (7-Methoxy-2-oxochromen-4-yl)methyl 2-[2-oxo-5-(trifluoromethyl)pyridin-1-yl]acetate —— C19H14F3NO6
(7-Methoxy-2-oxochromen-4-yl)methyl 2-[2-oxo-5-(trifluoromethyl)pyridin-1-yl]acetate
—— (7S)-7-methyl-2-[2-oxo-2-(1H-pyrrol-2-yl)ethyl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H21N3O2S2
(7S)-7-methyl-2-[2-oxo-2-(1H-pyrrol-2-yl)ethyl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[2-oxo-2-(1H-pyrrol-2-yl)ethyl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H21N3O2S2
(7R)-7-methyl-2-[2-oxo-2-(1H-pyrrol-2-yl)ethyl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7-Acetamido-2-oxochromen-4-yl)methyl 4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C21H19NO5S
(7-Acetamido-2-oxochromen-4-yl)methyl 4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— 7-(1-Pyrazin-2-ylpiperidin-4-yl)-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine —— C16H15F3N6
7-(1-Pyrazin-2-ylpiperidin-4-yl)-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine
—— 7-(1-Pyrimidin-2-ylpiperidin-4-yl)-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine —— C16H15F3N6
7-(1-Pyrimidin-2-ylpiperidin-4-yl)-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine
—— 7-methyl-3-(1-pyrazin-2-ylpiperidin-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C15H21N7
7-methyl-3-(1-pyrazin-2-ylpiperidin-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-(1-Methylsulfonylpiperidin-4-yl)-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine —— C13H15F3N4O2S
7-(1-Methylsulfonylpiperidin-4-yl)-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine
—— 7-Ethyl-4-[[(1-morpholin-4-ylcyclohexyl)methylamino]methyl]chromen-2-one —— C23H32N2O3
7-Ethyl-4-[[(1-morpholin-4-ylcyclohexyl)methylamino]methyl]chromen-2-one
—— (7-acetamido-2-oxochromen-4-yl)methyl 5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylate —— C20H17NO5S
(7-acetamido-2-oxochromen-4-yl)methyl 5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylate
—— 7-[(3S)-1-(2-methoxyethyl)piperidin-3-yl]-2,3,5-trimethylimidazo[5,1-b][1,3]thiazole —— C16H25N3OS
7-[(3S)-1-(2-methoxyethyl)piperidin-3-yl]-2,3,5-trimethylimidazo[5,1-b][1,3]thiazole
—— 7-[(3R)-1-(2-methoxyethyl)piperidin-3-yl]-2,3,5-trimethylimidazo[5,1-b][1,3]thiazole —— C16H25N3OS
7-[(3R)-1-(2-methoxyethyl)piperidin-3-yl]-2,3,5-trimethylimidazo[5,1-b][1,3]thiazole
—— 7-(1-Propan-2-ylpiperidin-4-yl)-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine —— C15H19F3N4
7-(1-Propan-2-ylpiperidin-4-yl)-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine
—— 7-bromo-1-[[(3S)-3-hydroxypiperidin-1-yl]methyl]indole-2,3-dione —— C14H15BrN2O3
7-bromo-1-[[(3S)-3-hydroxypiperidin-1-yl]methyl]indole-2,3-dione
—— 7-bromo-1-[[(3R)-3-hydroxypiperidin-1-ium-1-yl]methyl]indole-2,3-dione —— C14H16BrN2O3+
7-bromo-1-[[(3R)-3-hydroxypiperidin-1-ium-1-yl]methyl]indole-2,3-dione
—— 7-bromo-1-[[(3S)-3-hydroxypiperidin-1-ium-1-yl]methyl]indole-2,3-dione —— C14H16BrN2O3+
7-bromo-1-[[(3S)-3-hydroxypiperidin-1-ium-1-yl]methyl]indole-2,3-dione
—— 7-bromo-1-[[(3R)-3-hydroxypiperidin-1-yl]methyl]indole-2,3-dione —— C14H15BrN2O3
7-bromo-1-[[(3R)-3-hydroxypiperidin-1-yl]methyl]indole-2,3-dione
—— 7-methyl-3-[2-[5-(trifluoromethyl)pyridin-2-yl]hydrazinyl]indol-2-one —— C15H11F3N4O
7-methyl-3-[2-[5-(trifluoromethyl)pyridin-2-yl]hydrazinyl]indol-2-one
—— (7-Methyl-2-oxochromen-4-yl)methyl 5-methyl-2-phenyl-1,3-oxazole-4-carboxylate —— C22H17NO5
(7-Methyl-2-oxochromen-4-yl)methyl 5-methyl-2-phenyl-1,3-oxazole-4-carboxylate
—— 7-(2-Methylphenyl)-1-(2-methylpropyl)-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C19H18F3N3O2
7-(2-Methylphenyl)-1-(2-methylpropyl)-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[[2-(4-Methylphenyl)-1,3-thiazol-4-yl]methoxy]chromen-2-one —— C20H15NO3S
7-[[2-(4-Methylphenyl)-1,3-thiazol-4-yl]methoxy]chromen-2-one
—— 7-[2-(4-acetyl-3,5-dimethyl-1H-pyrrol-2-yl)-2-oxoethoxy]-4-phenylchromen-2-one —— C25H21NO5
7-[2-(4-acetyl-3,5-dimethyl-1H-pyrrol-2-yl)-2-oxoethoxy]-4-phenylchromen-2-one
—— (7S)-3-[(6-chloro-4H-1,3-benzodioxin-8-yl)methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H19ClN2O3S
(7S)-3-[(6-chloro-4H-1,3-benzodioxin-8-yl)methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-[(2-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H24FN3OS
(7R)-2-[(1S)-1-[(2-fluorophenyl)methyl-methylamino]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1R)-1-(3-oxopiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H23N4O2S+
(7S)-7-methyl-2-[(1R)-1-(3-oxopiperazin-1-ium-1-yl)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one