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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-[4-(3-chlorophenyl)piperazine-1-carbonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C20H20ClN3O2S
7-[4-(3-chlorophenyl)piperazine-1-carbonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (7-hydroxy-8-methyl-2-oxochromen-4-yl)methyl 3-[[(E)-3-phenylprop-2-enoyl]amino]propanoate —— C23H21NO6
(7-hydroxy-8-methyl-2-oxochromen-4-yl)methyl 3-[[(E)-3-phenylprop-2-enoyl]amino]propanoate
—— (7S)-2-[(Z)-1-chloro-2-(3-fluoro-4-methoxyphenyl)ethenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H18ClFN2O2S
(7S)-2-[(Z)-1-chloro-2-(3-fluoro-4-methoxyphenyl)ethenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(Z)-1-chloro-2-quinoxalin-2-ylethenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H17ClN4OS
(7S)-2-[(Z)-1-chloro-2-quinoxalin-2-ylethenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(Z)-1-chloro-2-quinoxalin-2-ylethenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H17ClN4OS
(7R)-2-[(Z)-1-chloro-2-quinoxalin-2-ylethenyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H19N3O3S
7-[[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-[[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H19N3O3S
7-[[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-oxo-2H-isoquinoline-3-carboxylate —— C20H15N3O4
(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-oxo-2H-isoquinoline-3-carboxylate
—— (7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-(2,2-dimethylpropanoyl)piperidine-4-carboxylate —— C21H27N3O4
(7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-(2,2-dimethylpropanoyl)piperidine-4-carboxylate
—— (7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 5-(4-fluorophenyl)thiophene-2-carboxylate —— C21H15FN2O3S
(7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 5-(4-fluorophenyl)thiophene-2-carboxylate
—— 7-[4-(4-fluorophenyl)piperazine-1-carbonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C20H20FN3O2S
7-[4-(4-fluorophenyl)piperazine-1-carbonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— 7-Methoxy-4-[2-(1-methylpyrazol-4-yl)ethoxy]quinoline —— C16H17N3O2
7-Methoxy-4-[2-(1-methylpyrazol-4-yl)ethoxy]quinoline
—— (7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(2-methylphenoxy)propanoate —— C17H17N3O4S
(7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(2-methylphenoxy)propanoate
—— 7-[(6-Bromo-1,3-benzodioxol-5-yl)methoxy]-4-methylchromen-2-one —— C18H13BrO5
7-[(6-Bromo-1,3-benzodioxol-5-yl)methoxy]-4-methylchromen-2-one
—— 7-[[(3R)-3-(5-methylfuran-2-yl)thiomorpholin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H17N3O2S2
7-[[(3R)-3-(5-methylfuran-2-yl)thiomorpholin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-[[(3S)-3-(5-methylfuran-2-yl)thiomorpholin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H17N3O2S2
7-[[(3S)-3-(5-methylfuran-2-yl)thiomorpholin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-Methyl-2-[(3-oxo-5,6,7,8-tetrahydrocinnolin-2-yl)methyl]pyrido[1,2-a]pyrimidin-4-one —— C18H18N4O2
7-Methyl-2-[(3-oxo-5,6,7,8-tetrahydrocinnolin-2-yl)methyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-[[(2S)-3-oxo-2-thiophen-2-ylpiperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H14N4O2S2
7-[[(2S)-3-oxo-2-thiophen-2-ylpiperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-[[(2R)-3-oxo-2-thiophen-2-ylpiperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H14N4O2S2
7-[[(2R)-3-oxo-2-thiophen-2-ylpiperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C22H25N3O3S
7-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 4-phenoxybutanoate —— C17H17N3O4S
(7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 4-phenoxybutanoate
—— (7-hydroxy-2-oxochromen-4-yl)methyl (E)-3-[4-(trifluoromethoxy)phenyl]prop-2-enoate —— C20H13F3O6
(7-hydroxy-2-oxochromen-4-yl)methyl (E)-3-[4-(trifluoromethoxy)phenyl]prop-2-enoate
—— (7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(4-methylphenoxy)propanoate —— C17H17N3O4S
(7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(4-methylphenoxy)propanoate
—— 7-chloro-2-[[[(2R)-2-(1,3-thiazol-2-yl)butan-2-yl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one —— C16H17ClN4OS
7-chloro-2-[[[(2R)-2-(1,3-thiazol-2-yl)butan-2-yl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-chloro-2-[[[(2S)-2-(1,3-thiazol-2-yl)butan-2-yl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one —— C16H17ClN4OS
7-chloro-2-[[[(2S)-2-(1,3-thiazol-2-yl)butan-2-yl]amino]methyl]pyrido[1,2-a]pyrimidin-4-one
—— (7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(1,3-dioxoisoindol-2-yl)propanoate —— C18H14N4O5S
(7-Methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-(1,3-dioxoisoindol-2-yl)propanoate
—— (7S)-7-methyl-2-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H27N3O2S
(7S)-7-methyl-2-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-Methyl-2-[(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)sulfanylmethyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C18H17N5OS3
7-Methyl-2-[(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)sulfanylmethyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— (7S)-N-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-N,2-dimethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-amine —— C16H18N4O2S
(7S)-N-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-N,2-dimethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-amine
—— 7-(4-phenylpiperazine-1-carbonyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C20H21N3O2S
7-(4-phenylpiperazine-1-carbonyl)-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (7R)-N-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-N,2-dimethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-amine —— C16H18N4O2S
(7R)-N-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-N,2-dimethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-7-amine
—— 7-chloro-N-[2-(3-fluorophenyl)ethyl]-1,3-benzodioxole-5-carboxamide —— C16H13ClFNO3
7-chloro-N-[2-(3-fluorophenyl)ethyl]-1,3-benzodioxole-5-carboxamide
—— 7-Methyl-2-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanylmethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C16H13N5OS3
7-Methyl-2-(7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9,11-tetraen-12-ylsulfanylmethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 7-[[4-Amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C17H16N6O2S2
7-[[4-Amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-Methyl-2-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-ylsulfanylmethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C17H15N5OS3
7-Methyl-2-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-ylsulfanylmethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— (7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-(2-fluorophenyl)cyclopentane-1-carboxylate —— C22H21FN2O3
(7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-(2-fluorophenyl)cyclopentane-1-carboxylate
—— 7-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one —— C21H23N3O3S
7-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-3,5-dihydro-2H-1,5-benzothiazepin-4-one
—— (7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(5-chlorothiophen-2-yl)-4-oxobutanoate —— C18H15ClN2O4S
(7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-(5-chlorothiophen-2-yl)-4-oxobutanoate
—— (7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate —— C18H18N4O5S
(7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate
—— (7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate —— C18H18N4O5S
(7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]propanoate
—— (7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate —— C18H20N4O5S
(7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(3aR,7aR)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate
—— (7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate —— C18H20N4O5S
(7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-[(3aS,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]propanoate
—— (7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-pyrrol-1-yl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C23H21N3O3S
(7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-pyrrol-1-yl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (7S)-7-methyl-3-[2-(1-methyl-2-oxo-3H-indol-5-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H21N3O3S
(7S)-7-methyl-3-[2-(1-methyl-2-oxo-3H-indol-5-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-chloro-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]-1,3-benzodioxole-5-carboxamide —— C16H16ClNO3S
7-chloro-N-[(1S)-2-methyl-1-thiophen-2-ylpropyl]-1,3-benzodioxole-5-carboxamide
—— (7S)-7-methyl-3-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H16N4O2S2
(7S)-7-methyl-3-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-3-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H16N4O2S2
(7R)-7-methyl-3-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-3-[2-(1-methyl-2-oxo-3H-indol-5-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H21N3O3S
(7R)-7-methyl-3-[2-(1-methyl-2-oxo-3H-indol-5-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-(cyclopropylmethyl)-2-[(2R)-2-(hydroxymethyl)-2,5-dihydropyrrole-1-carbonyl]-6-(4-methoxyphenyl)imidazo[1,2-a]pyrazin-8-one —— C23H24N4O4
7-(cyclopropylmethyl)-2-[(2R)-2-(hydroxymethyl)-2,5-dihydropyrrole-1-carbonyl]-6-(4-methoxyphenyl)imidazo[1,2-a]pyrazin-8-one
—— 7-(cyclopropylmethyl)-2-[(2S)-2-(hydroxymethyl)-2,5-dihydropyrrole-1-carbonyl]-6-(4-methoxyphenyl)imidazo[1,2-a]pyrazin-8-one —— C23H24N4O4
7-(cyclopropylmethyl)-2-[(2S)-2-(hydroxymethyl)-2,5-dihydropyrrole-1-carbonyl]-6-(4-methoxyphenyl)imidazo[1,2-a]pyrazin-8-one