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—— (7-Bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-amino-5-chlorobenzoate —— C16H11BrClN3O3
(7-Bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-amino-5-chlorobenzoate
—— (7-Methoxy-2-oxochromen-4-yl)methyl 2-amino-5-chlorobenzoate —— C18H14ClNO5
(7-Methoxy-2-oxochromen-4-yl)methyl 2-amino-5-chlorobenzoate
—— 7-benzyl-2-methyl-N-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C20H21N5
7-benzyl-2-methyl-N-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-benzyl-2-methyl-N-pyrazin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C19H20N6
7-benzyl-2-methyl-N-pyrazin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-(benzenesulfonyl)-2-methyl-N-pyrazin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C18H18N6O2S
7-(benzenesulfonyl)-2-methyl-N-pyrazin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-(benzenesulfonyl)-2-methyl-N-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C19H19N5O2S
7-(benzenesulfonyl)-2-methyl-N-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— (7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C17H13N5O3S
(7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(1H-pyrazole-5-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H30N6O2
7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(1H-pyrazole-5-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— (7-methoxy-2-oxochromen-4-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C21H16N2O5
(7-methoxy-2-oxochromen-4-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H31N5O2
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(1H-pyrazole-5-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H30N6O2
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(1H-pyrazole-5-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— (7-hydroxy-8-methyl-2-oxochromen-4-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C21H16N2O5
(7-hydroxy-8-methyl-2-oxochromen-4-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 1-benzyl-3,5-dimethylpyrazole-4-carboxylate —— C23H20N2O5
(7-Hydroxy-2-oxochromen-4-yl)methyl 1-benzyl-3,5-dimethylpyrazole-4-carboxylate
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H31N5O2
7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— (7-ethyl-2-oxochromen-4-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C22H18N2O4
(7-ethyl-2-oxochromen-4-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— 7-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(2-phenylacetyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H28N4O2
7-(cyclopropylmethyl)-4-methyl-2-[(2S)-1-(2-phenylacetyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— (7,8-dimethyl-2-oxochromen-4-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate —— C22H18N2O4
(7,8-dimethyl-2-oxochromen-4-yl)methyl 3-phenyl-1H-pyrazole-5-carboxylate
—— (7R)-7-methyl-2-[[5-(2-methylpropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H23N5OS3
(7R)-7-methyl-2-[[5-(2-methylpropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C16H19N5OS3
(7R)-2-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1R)-1-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H21N5OS3
(7R)-2-[(1R)-1-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H21N5OS3
(7R)-2-[(1S)-1-[[5-(ethylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[(2R)-1-(2-amino-2-oxoethyl)pyrrolidin-2-yl]-N,N-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H20N6O2
7-[(2R)-1-(2-amino-2-oxoethyl)pyrrolidin-2-yl]-N,N-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-[(2S)-1-(2-hydroxyethyl)pyrrolidin-2-yl]-N,N-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H21N5O2
7-[(2S)-1-(2-hydroxyethyl)pyrrolidin-2-yl]-N,N-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-[(2S)-1-acetylpyrrolidin-2-yl]-N,N-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H19N5O2
7-[(2S)-1-acetylpyrrolidin-2-yl]-N,N-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-[(2R)-1-acetylpyrrolidin-2-yl]-N,N-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C15H19N5O2
7-[(2R)-1-acetylpyrrolidin-2-yl]-N,N-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-[2-(Azepan-1-yl)-2-oxoethoxy]-2-methyl-3-phenoxychromen-4-one —— C24H25NO5
7-[2-(Azepan-1-yl)-2-oxoethoxy]-2-methyl-3-phenoxychromen-4-one
—— 7-[(3S)-1-(quinolin-4-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C23H21F3N6
7-[(3S)-1-(quinolin-4-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(2R)-1-(1-acetylpiperidine-4-carbonyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H29N5O4
7-[(2R)-1-(1-acetylpiperidine-4-carbonyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-[3-(4-fluorophenyl)propanoyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H25FN4O3
7-[(2R)-1-[3-(4-fluorophenyl)propanoyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(quinolin-4-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C23H21F3N6
7-[(3R)-1-(quinolin-4-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(2S)-1-(1-acetylpiperidine-4-carbonyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H29N5O4
7-[(2S)-1-(1-acetylpiperidine-4-carbonyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-[(4-methoxyphenyl)methyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H26N4O3
7-[(2R)-1-[(4-methoxyphenyl)methyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-[3-(4-fluorophenyl)propanoyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H25FN4O3
7-[(2S)-1-[3-(4-fluorophenyl)propanoyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H26N4O4
7-[(2R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H26N4O4
7-[(2S)-1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2R)-1-(4-fluorobenzoyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C21H21FN4O3
7-[(2R)-1-(4-fluorobenzoyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-[(4-methoxyphenyl)methyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H26N4O3
7-[(2S)-1-[(4-methoxyphenyl)methyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-(4-fluorobenzoyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C21H21FN4O3
7-[(2S)-1-(4-fluorobenzoyl)piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— (7-ethyl-2-oxochromen-4-yl)methyl (3aR)-4-oxo-2,3,3a,5-tetrahydro-1H-pyrrolo[1,2-a]quinoxaline-7-carboxylate —— C24H22N2O5
(7-ethyl-2-oxochromen-4-yl)methyl (3aR)-4-oxo-2,3,3a,5-tetrahydro-1H-pyrrolo[1,2-a]quinoxaline-7-carboxylate
—— (7-ethyl-2-oxochromen-4-yl)methyl (3aS)-4-oxo-2,3,3a,5-tetrahydro-1H-pyrrolo[1,2-a]quinoxaline-7-carboxylate —— C24H22N2O5
(7-ethyl-2-oxochromen-4-yl)methyl (3aS)-4-oxo-2,3,3a,5-tetrahydro-1H-pyrrolo[1,2-a]quinoxaline-7-carboxylate
—— 7-(4-methoxyphenyl)sulfonyl-N-methyl-2-[(2R)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C20H27N5O3S
7-(4-methoxyphenyl)sulfonyl-N-methyl-2-[(2R)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-(4-methoxyphenyl)sulfonyl-N-methyl-2-[(2S)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine —— C20H27N5O3S
7-(4-methoxyphenyl)sulfonyl-N-methyl-2-[(2S)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-amine
—— 7-Chloro-2-[[5-(furan-2-yl)-1,2-oxazol-3-yl]methylsulfanyl]-3-propylquinazolin-4-one —— C19H16ClN3O3S
7-Chloro-2-[[5-(furan-2-yl)-1,2-oxazol-3-yl]methylsulfanyl]-3-propylquinazolin-4-one
—— 7-Chloro-3-propyl-2-[(1-propyltetrazol-5-yl)methylsulfanyl]quinazolin-4-one —— C16H19ClN6OS
7-Chloro-3-propyl-2-[(1-propyltetrazol-5-yl)methylsulfanyl]quinazolin-4-one
—— (7-methylimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-[6-methyl-4-[(3-methylpyridin-2-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone —— C26H28N6O
(7-methylimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-[6-methyl-4-[(3-methylpyridin-2-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone
—— (7-methylimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-[6-methyl-4-[(3-methylpyridin-2-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone —— C26H28N6O
(7-methylimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-[6-methyl-4-[(3-methylpyridin-2-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone
—— 7-[(2R)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C21H25N5O4
7-[(2R)-1-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine —— C19H20FN5
7-[(2S)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(2S)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C21H23FN4O2
7-[(2S)-1-[(4-fluorophenyl)methyl]piperidin-2-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2S)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine —— C18H18FN5O2S
7-[(2S)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]pyrido[2,3-d]pyrimidin-4-amine