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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-propyl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C15H13F3N4O
7-propyl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-pyridin-4-yl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C17H10F3N5O
7-pyridin-4-yl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-pyridin-3-yl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C17H10F3N5O
7-pyridin-3-yl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-(methoxymethyl)-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C14H11F3N4O2
7-(methoxymethyl)-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-ethyl-5-(4-fluorophenyl)-8-methyl-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C14H13FN4O
7-ethyl-5-(4-fluorophenyl)-8-methyl-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-ethyl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C14H11F3N4O
7-ethyl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-phenyl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C18H11F3N4O
7-phenyl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-[[2-(Trifluoromethyl)quinazolin-4-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H9F3N4OS2
7-[[2-(Trifluoromethyl)quinazolin-4-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7,8-dimethyl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C14H11F3N4O
7,8-dimethyl-5-[4-(trifluoromethyl)phenyl]-2H-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-Methyl-2-[(3-methylphenyl)methyl]-5-[4-(trifluoromethyl)phenyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C21H17F3N4O
7-Methyl-2-[(3-methylphenyl)methyl]-5-[4-(trifluoromethyl)phenyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-[(2S)-2-ethylpiperidin-1-yl]-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H25N5O
7-[(2S)-2-ethylpiperidin-1-yl]-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-Methyl-5-(3-methylanilino)-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C21H21N5O
7-Methyl-5-(3-methylanilino)-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-(4-Chlorophenyl)-5-methyl-3-[(3-methylphenyl)methyl]pyrrolo[3,2-d]pyrimidin-4-one —— C21H18ClN3O
7-(4-Chlorophenyl)-5-methyl-3-[(3-methylphenyl)methyl]pyrrolo[3,2-d]pyrimidin-4-one
—— 7-Anilino-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C19H17N5O
7-Anilino-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-(4-Methoxyphenyl)-5-methyl-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C21H20N4O2
7-(4-Methoxyphenyl)-5-methyl-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H25N5O
7-[(2R)-2-ethylpiperidin-1-yl]-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[4-(3-Methoxyphenyl)piperazin-1-yl]-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C24H26N6O2
7-[4-(3-Methoxyphenyl)piperazin-1-yl]-2-[(3-methylphenyl)methyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-methyl-3-[(3-methylphenyl)methylsulfanyl]-2H-1,4-benzoxazine —— C17H17NOS
7-methyl-3-[(3-methylphenyl)methylsulfanyl]-2H-1,4-benzoxazine
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H25N5O2
7-[(2R)-2-ethylpiperidin-1-yl]-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C19H22FN5O
7-[(2R)-2-ethylpiperidin-1-yl]-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C21H22FN7O2
7-[(2R)-2-ethylpiperidin-1-yl]-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H24FN5O2
7-[(2R)-2-ethylpiperidin-1-yl]-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C26H25FN8O2
7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2S)-2-ethylpiperidin-1-yl]-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H25N5O
7-[(2S)-2-ethylpiperidin-1-yl]-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C25H28N6O
7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2S)-2-ethylpiperidin-1-yl]-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H24FN5O2
7-[(2S)-2-ethylpiperidin-1-yl]-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C25H25FN6O2
7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2S)-2-ethylpiperidin-1-yl]-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C22H25N7O2S
7-[(2S)-2-ethylpiperidin-1-yl]-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H22FN5O2
7-[(2R)-2-ethylpiperidin-1-yl]-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C23H26N6O2
7-[(2R)-2-ethylpiperidin-1-yl]-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C22H22F3N7O2
7-[(2R)-2-ethylpiperidin-1-yl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C28H29N7O2
7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C25H27FN6O2
7-[4-(2,3-Dimethylphenyl)piperazin-1-yl]-2-[(3-fluoro-4-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2S)-2-ethylpiperidin-1-yl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C22H22F3N7O2
7-[(2S)-2-ethylpiperidin-1-yl]-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2S)-2-ethylpiperidin-1-yl]-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H25N5O2
7-[(2S)-2-ethylpiperidin-1-yl]-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C22H25N7O2S
7-[(2R)-2-ethylpiperidin-1-yl]-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2S)-2-ethylpiperidin-1-yl]-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C19H22FN5O
7-[(2S)-2-ethylpiperidin-1-yl]-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-[(2S)-2-ethylpiperidin-1-yl]-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H22FN5O2
7-[(2S)-2-ethylpiperidin-1-yl]-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— (7R)-7-(1,3-benzodioxol-5-yl)-5-(4-fluorophenyl)-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C19H12F4N4O2
(7R)-7-(1,3-benzodioxol-5-yl)-5-(4-fluorophenyl)-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7S)-7-(4-butoxyphenyl)-5-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C22H24N4O
(7S)-7-(4-butoxyphenyl)-5-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-[(2R)-2-ethylpiperidin-1-yl]-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C20H25N5O
7-[(2R)-2-ethylpiperidin-1-yl]-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— (7S)-7-(1,3-benzodioxol-5-yl)-5-(4-fluorophenyl)-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C19H12F4N4O2
(7S)-7-(1,3-benzodioxol-5-yl)-5-(4-fluorophenyl)-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-[(2S)-2-ethylpiperidin-1-yl]-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C23H26N6O2
7-[(2S)-2-ethylpiperidin-1-yl]-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-Pyrrolidin-1-yl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C19H16F3N7O2
7-Pyrrolidin-1-yl-2-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-(4-Fluoroanilino)-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C18H13F2N5O
7-(4-Fluoroanilino)-2-[(3-fluorophenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-(4-Fluoroanilino)-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C21H16FN7O2S
7-(4-Fluoroanilino)-2-[[3-(4-methylsulfanylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-(4-Fluoroanilino)-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C19H13F2N5O2
7-(4-Fluoroanilino)-2-[2-(4-fluorophenyl)-2-oxoethyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-(4-Fluoroanilino)-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C19H16FN5O2
7-(4-Fluoroanilino)-2-[(3-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— 7-(4-Fluoroanilino)-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one —— C19H16FN5O
7-(4-Fluoroanilino)-2-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidin-3-one
—— (7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-ethoxy-3-nitrobenzoate —— C19H17N3O6
(7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 4-ethoxy-3-nitrobenzoate