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—— (7S)-7-(3-methoxyphenyl)-2-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C20H23N5O3
(7S)-7-(3-methoxyphenyl)-2-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— 7-[[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C19H19N3O4
7-[[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C19H19N3O4
7-[[(2S)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7S)-2-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-7-(4-fluorophenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C18H18FN5OS
(7S)-2-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-7-(4-fluorophenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-7-(3-methoxyphenyl)-2-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C20H23N5O3
(7R)-7-(3-methoxyphenyl)-2-[(5-propan-2-yl-1,2,4-oxadiazol-3-yl)methyl]-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7S)-7-(4-chlorophenyl)-5-(3,4-dichlorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C17H11Cl3N4
(7S)-7-(4-chlorophenyl)-5-(3,4-dichlorophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-[(2S)-3,3,3-trifluoro-2-hydroxypropanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C10H11F3N4O3
7-[(2S)-3,3,3-trifluoro-2-hydroxypropanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— 7-[(2R)-1-methylsulfonylpyrrolidine-2-carbonyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C13H19N5O4S
7-[(2R)-1-methylsulfonylpyrrolidine-2-carbonyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— 7-[(2S)-1-methylsulfonylpyrrolidine-2-carbonyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C13H19N5O4S
7-[(2S)-1-methylsulfonylpyrrolidine-2-carbonyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— 7-[(2R)-3,3,3-trifluoro-2-hydroxypropanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C10H11F3N4O3
7-[(2R)-3,3,3-trifluoro-2-hydroxypropanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— 7-[(3S)-3-(4-ethyl-5-oxo-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-3-methylquinazolin-4-one —— C19H22N6O3
7-[(3S)-3-(4-ethyl-5-oxo-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-3-methylquinazolin-4-one
—— 7-[(3R)-3-(4-ethyl-5-oxo-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-3-methylquinazolin-4-one —— C19H22N6O3
7-[(3R)-3-(4-ethyl-5-oxo-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-3-methylquinazolin-4-one
—— 7-methoxy-3-[[methyl-[2-[(2R)-oxan-2-yl]ethyl]amino]methyl]-1H-quinolin-2-one —— C19H26N2O3
7-methoxy-3-[[methyl-[2-[(2R)-oxan-2-yl]ethyl]amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[methyl-[2-[(2S)-oxan-2-yl]ethyl]amino]methyl]-1H-quinolin-2-one —— C19H26N2O3
7-methoxy-3-[[methyl-[2-[(2S)-oxan-2-yl]ethyl]amino]methyl]-1H-quinolin-2-one
—— [7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone —— C19H20ClN3O4
[7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone
—— [7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-morpholin-2-yl]methanone —— C19H20ClN3O4
[7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-morpholin-2-yl]methanone
—— 7-methoxy-3-[[(3S)-3-(methoxymethyl)pyrrolidin-1-yl]methyl]-1H-quinolin-2-one —— C17H22N2O3
7-methoxy-3-[[(3S)-3-(methoxymethyl)pyrrolidin-1-yl]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[(3R)-3-(methoxymethyl)pyrrolidin-1-yl]methyl]-1H-quinolin-2-one —— C17H22N2O3
7-methoxy-3-[[(3R)-3-(methoxymethyl)pyrrolidin-1-yl]methyl]-1H-quinolin-2-one
—— [7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone —— C19H19ClN2O4
[7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone
—— 7-methoxy-3-[[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]methyl]-1H-quinolin-2-one —— C20H27N3O3
7-methoxy-3-[[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]methyl]-1H-quinolin-2-one —— C20H27N3O3
7-methoxy-3-[[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]methyl]-1H-quinolin-2-one
—— (7S)-7-(3-methoxyphenyl)-2-[5-(2-methylpropyl)-1,2,4-oxadiazol-3-ylidene]-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one —— C20H23N5O3
(7S)-7-(3-methoxyphenyl)-2-[5-(2-methylpropyl)-1,2,4-oxadiazol-3-ylidene]-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one
—— (7R)-7-(3-methoxyphenyl)-2-[5-(2-methylpropyl)-1,2,4-oxadiazol-3-ylidene]-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one —— C20H23N5O3
(7R)-7-(3-methoxyphenyl)-2-[5-(2-methylpropyl)-1,2,4-oxadiazol-3-ylidene]-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4-one
—— [(7S)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-(3-aminophenyl)methanone —— C21H21N5O
[(7S)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-(3-aminophenyl)methanone
—— 7-methoxy-3-[[methyl-[(1R)-1-(1,3-thiazol-2-yl)ethyl]amino]methyl]-1H-quinolin-2-one —— C17H19N3O2S
7-methoxy-3-[[methyl-[(1R)-1-(1,3-thiazol-2-yl)ethyl]amino]methyl]-1H-quinolin-2-one
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-oxolan-2-yl]methanone —— C20H20ClNO4
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-oxolan-2-yl]methanone
—— 7-[(2R)-2-prop-2-enylsulfanylpropanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C13H18N4O2S
7-[(2R)-2-prop-2-enylsulfanylpropanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— [(7R)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-(3-aminophenyl)methanone —— C21H21N5O
[(7R)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-(3-aminophenyl)methanone
—— 7-methoxy-3-[[methyl-[(1S)-1-(1,3-thiazol-2-yl)ethyl]amino]methyl]-1H-quinolin-2-one —— C17H19N3O2S
7-methoxy-3-[[methyl-[(1S)-1-(1,3-thiazol-2-yl)ethyl]amino]methyl]-1H-quinolin-2-one
—— 7-[(2S)-2-pyrazol-1-ylbutanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C14H18N6O2
7-[(2S)-2-pyrazol-1-ylbutanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— 7-[(2S)-2-prop-2-enylsulfanylpropanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C13H18N4O2S
7-[(2S)-2-prop-2-enylsulfanylpropanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone —— C20H20ClNO4
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone
—— 7-(3-chlorophenyl)-4-[2-[(3S)-oxolan-3-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C21H24ClNO3
7-(3-chlorophenyl)-4-[2-[(3S)-oxolan-3-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-[(2R)-2-pyrazol-1-ylbutanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C14H18N6O2
7-[(2R)-2-pyrazol-1-ylbutanoyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— [(7R)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-cyclopentylmethanone —— C20H24N4O
[(7R)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-cyclopentylmethanone
—— [(7S)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-cyclopentylmethanone —— C20H24N4O
[(7S)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-cyclopentylmethanone
—— 7-(5-chloropyridin-2-yl)-4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C21H26ClN3O2
7-(5-chloropyridin-2-yl)-4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-(5-chloropyridin-2-yl)-4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C21H26ClN3O2
7-(5-chloropyridin-2-yl)-4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-[(2R)-1-[4-(difluoromethoxy)phenyl]-1-oxopropan-2-yl]oxychromen-2-one —— C19H14F2O5
7-[(2R)-1-[4-(difluoromethoxy)phenyl]-1-oxopropan-2-yl]oxychromen-2-one
—— 7-[(3-Morpholin-4-ylsulfonylphenyl)methoxy]chromen-2-one —— C20H19NO6S
7-[(3-Morpholin-4-ylsulfonylphenyl)methoxy]chromen-2-one
—— 7-[(1R)-1-(2-chlorophenyl)ethoxy]chromen-2-one —— C17H13ClO3
7-[(1R)-1-(2-chlorophenyl)ethoxy]chromen-2-one
—— 7-[(2S)-1-(4-ethoxyphenyl)-1-oxopropan-2-yl]oxychromen-2-one —— C20H18O5
7-[(2S)-1-(4-ethoxyphenyl)-1-oxopropan-2-yl]oxychromen-2-one
—— 7-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethoxy]chromen-2-one —— C17H19NO4
7-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethoxy]chromen-2-one
—— 7-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethoxy]chromen-2-one —— C17H19NO5
7-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethoxy]chromen-2-one
—— 7-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethoxy]chromen-2-one —— C17H19NO5
7-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethoxy]chromen-2-one
—— 7-(2-Oxo-2-thiophen-2-ylethoxy)chromen-2-one —— C15H10O4S
7-(2-Oxo-2-thiophen-2-ylethoxy)chromen-2-one
—— 7-[(1S)-1-(2-chlorophenyl)ethoxy]chromen-2-one —— C17H13ClO3
7-[(1S)-1-(2-chlorophenyl)ethoxy]chromen-2-one
—— 7-[2-[1-(3-Methoxypropyl)-2,5-dimethylpyrrol-3-yl]-2-oxoethoxy]chromen-2-one —— C21H23NO5
7-[2-[1-(3-Methoxypropyl)-2,5-dimethylpyrrol-3-yl]-2-oxoethoxy]chromen-2-one
—— 7-[(2R)-1-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]oxychromen-2-one —— C21H17NO4
7-[(2R)-1-(2-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]oxychromen-2-one
—— 7-[(2S)-1-[4-(difluoromethoxy)phenyl]-1-oxopropan-2-yl]oxychromen-2-one —— C19H14F2O5
7-[(2S)-1-[4-(difluoromethoxy)phenyl]-1-oxopropan-2-yl]oxychromen-2-one