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—— [(7S)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-(3-amino-1H-pyrazol-5-yl)methanone —— C18H19N7O
[(7S)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-(3-amino-1H-pyrazol-5-yl)methanone
—— (7R)-2-benzylsulfanyl-N-(2-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C20H19N5O2S
(7R)-2-benzylsulfanyl-N-(2-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(2,5-dimethoxyphenyl)-7-(3-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5O4
(7S)-N-(2,5-dimethoxyphenyl)-7-(3-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,4-dimethoxyphenyl)-7-(4-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5O4
(7R)-N-(2,4-dimethoxyphenyl)-7-(4-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,5-dimethoxyphenyl)-7-(3-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5O4
(7R)-N-(2,5-dimethoxyphenyl)-7-(3-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-ethoxy-4-methoxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O3
(7S)-7-(3-ethoxy-4-methoxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-ethoxy-4-methoxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O3
(7R)-7-(3-ethoxy-4-methoxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,4-dimethoxyphenyl)-7-(3-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5O4
(7R)-N-(2,4-dimethoxyphenyl)-7-(3-hydroxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-[[(2R)-oxolan-2-yl]methylamino]-7-phenyl-7,8-dihydro-6H-quinazolin-5-one —— C19H21N3O2
(7R)-2-[[(2R)-oxolan-2-yl]methylamino]-7-phenyl-7,8-dihydro-6H-quinazolin-5-one
—— (7S)-2-[[(2R)-oxolan-2-yl]methylamino]-7-phenyl-7,8-dihydro-6H-quinazolin-5-one —— C19H21N3O2
(7S)-2-[[(2R)-oxolan-2-yl]methylamino]-7-phenyl-7,8-dihydro-6H-quinazolin-5-one
—— 7-methoxy-4-methyl-2-[(5S)-2-methyl-2,7-diazaspiro[4.5]decan-7-yl]quinazoline —— C19H26N4O
7-methoxy-4-methyl-2-[(5S)-2-methyl-2,7-diazaspiro[4.5]decan-7-yl]quinazoline
—— 7-(3-nitrophenyl)-1,2,4-triazolo<1,5-a>pyrimidine —— C11H7N5O2
7-(3-nitrophenyl)-1,2,4-triazolo<1,5-a>pyrimidine
—— (7R)-2-benzylsulfanyl-N-(3-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C20H19N5O2S
(7R)-2-benzylsulfanyl-N-(3-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(1,3-benzodioxol-5-yl)-2-methylsulfanyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C14H13N5O4S
(7R)-N-(1,3-benzodioxol-5-yl)-2-methylsulfanyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(1,3-benzodioxol-5-yl)-2-methylsulfanyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C14H13N5O4S
(7S)-N-(1,3-benzodioxol-5-yl)-2-methylsulfanyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-2-benzylsulfanyl-N-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C20H19N5O3S
(7R)-2-benzylsulfanyl-N-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-2-methylsulfanyl-5-oxo-N-[2-(trifluoromethyl)phenyl]-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C14H12F3N5O2S
(7R)-2-methylsulfanyl-5-oxo-N-[2-(trifluoromethyl)phenyl]-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-2-benzylsulfanyl-N-(3-fluorophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C19H16FN5O2S
(7R)-2-benzylsulfanyl-N-(3-fluorophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-2-benzylsulfanyl-N-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C20H19N5O3S
(7S)-2-benzylsulfanyl-N-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-2-methyl-N-(2-methyl-5-nitrophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C14H14N6O4
(7S)-2-methyl-N-(2-methyl-5-nitrophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(4-fluorophenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C13H12FN5O2
(7R)-N-(4-fluorophenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-2-benzylsulfanyl-5-oxo-N-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C19H17N5O2S
(7R)-2-benzylsulfanyl-5-oxo-N-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-methylsulfanyl-3-[[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-quinolin-2-one —— C20H21N3OS
7-methylsulfanyl-3-[[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-quinolin-2-one
—— (7R)-2-methyl-N-(2-methyl-5-nitrophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C14H14N6O4
(7R)-2-methyl-N-(2-methyl-5-nitrophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-2-benzylsulfanyl-5-oxo-N-(4-propan-2-ylphenyl)-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C22H23N5O2S
(7R)-2-benzylsulfanyl-5-oxo-N-(4-propan-2-ylphenyl)-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-methylsulfanyl-3-[[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-quinolin-2-one —— C20H21N3OS
7-methylsulfanyl-3-[[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-quinolin-2-one
—— 7-methyl-N-(4-methylphenyl)-2-[4-(morpholin-4-yl)phenyl]imidazo[1,2-a]pyridin-3-amine —— C25H26N4O
7-methyl-N-(4-methylphenyl)-2-[4-(morpholin-4-yl)phenyl]imidazo[1,2-a]pyridin-3-amine
—— 7-[[(3S)-3-propylmorpholin-4-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C18H22N2O4
7-[[(3S)-3-propylmorpholin-4-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-chloro-3-[[(3S)-3-(diethylamino)pyrrolidin-1-yl]methyl]-1H-quinolin-2-one —— C18H24ClN3O
7-chloro-3-[[(3S)-3-(diethylamino)pyrrolidin-1-yl]methyl]-1H-quinolin-2-one
—— (7S)-2-(2-methylpropyl)-N-(4-nitrophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C16H18N6O4
(7S)-2-(2-methylpropyl)-N-(4-nitrophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-2-methyl-N-(2-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C14H15N5O2
(7S)-2-methyl-N-(2-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-chloro-2-(5-methylfuran-2-yl)-N-(2-methylphenyl)imidazo[2,1-b][1,3]benzothiazol-3-amine —— C21H16ClN3OS
7-chloro-2-(5-methylfuran-2-yl)-N-(2-methylphenyl)imidazo[2,1-b][1,3]benzothiazol-3-amine
—— (7R)-2-methyl-N-(2-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C14H15N5O2
(7R)-2-methyl-N-(2-methylphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-[[(3R)-3-propylmorpholin-4-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C18H22N2O4
7-[[(3R)-3-propylmorpholin-4-yl]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-2-(2-methylpropyl)-N-(4-nitrophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C16H18N6O4
(7R)-2-(2-methylpropyl)-N-(4-nitrophenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-(3-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C20H22ClNO3
7-(3-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-[[methyl-[(1S)-1-pyrimidin-4-ylethyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C18H18N4O3
7-[[methyl-[(1S)-1-pyrimidin-4-ylethyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-methoxy-3-[[(2R)-4-methyl-3-oxo-2-propan-2-ylpiperazin-1-yl]methyl]-1H-quinolin-2-one —— C19H25N3O3
7-methoxy-3-[[(2R)-4-methyl-3-oxo-2-propan-2-ylpiperazin-1-yl]methyl]-1H-quinolin-2-one
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(1S)-2,2-dimethylcyclopropyl]methanone —— C22H22N2O3S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(1S)-2,2-dimethylcyclopropyl]methanone
—— 7-[2-[(3S)-3-phenylpyrrolidin-1-yl]acetyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C19H23N5O2
7-[2-[(3S)-3-phenylpyrrolidin-1-yl]acetyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— 7-[2-[[(2R)-oxan-2-yl]methoxy]acetyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C15H22N4O4
7-[2-[[(2R)-oxan-2-yl]methoxy]acetyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— 7-[2-[(3R)-3-phenylpyrrolidin-1-yl]acetyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C19H23N5O2
7-[2-[(3R)-3-phenylpyrrolidin-1-yl]acetyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— 7-methyl-N-(2-methylphenyl)-2-[4-(morpholin-4-yl)phenyl]imidazo[1,2-a]pyridin-3-amine —— C25H26N4O
7-methyl-N-(2-methylphenyl)-2-[4-(morpholin-4-yl)phenyl]imidazo[1,2-a]pyridin-3-amine
—— 7-methyl-3-[[methyl-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]amino]methyl]-1H-quinolin-2-one —— C21H25N3O
7-methyl-3-[[methyl-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]amino]methyl]-1H-quinolin-2-one
—— (7-Hydroxy-5,6-dimethyl[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)(morpholin-4-yl)methanone —— C12H15N5O3
(7-Hydroxy-5,6-dimethyl[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)(morpholin-4-yl)methanone
—— 7-methoxy-3-[[(2S)-4-methyl-3-oxo-2-propan-2-ylpiperazin-1-yl]methyl]-1H-quinolin-2-one —— C19H25N3O3
7-methoxy-3-[[(2S)-4-methyl-3-oxo-2-propan-2-ylpiperazin-1-yl]methyl]-1H-quinolin-2-one
—— 7-[2-[[(2S)-oxan-2-yl]methoxy]acetyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide —— C15H22N4O4
7-[2-[[(2S)-oxan-2-yl]methoxy]acetyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine-3-carboxamide
—— [(7R)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-(3-methylpyridin-2-yl)methanone —— C21H21N5O
[(7R)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-(3-methylpyridin-2-yl)methanone
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-oxolan-3-yl]methanone —— C21H20N2O4S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-oxolan-3-yl]methanone
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-oxolan-3-yl]methanone —— C21H20N2O4S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-oxolan-3-yl]methanone