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—— (7R)-N-(2-methoxy-5-methylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C15H17N5O3
(7R)-N-(2-methoxy-5-methylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(2,4-dimethoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C15H17N5O4
(7R)-N-(2,4-dimethoxyphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C15H17N5O2
(7R)-N-(2,4-dimethylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(3,5-dimethylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C15H17N5O2
(7S)-N-(3,5-dimethylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(4-chlorophenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C13H12ClN5O2
(7S)-N-(4-chlorophenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-(1-benzothiophen-3-yl)-4-[[(2R)-1,4-dioxan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H23NO4S
7-(1-benzothiophen-3-yl)-4-[[(2R)-1,4-dioxan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— (7R)-N-(3,5-dimethylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C15H17N5O2
(7R)-N-(3,5-dimethylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-[[[(R)-cyclopropyl(pyridin-2-yl)methyl]-methylamino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C21H21N3O3
7-[[[(R)-cyclopropyl(pyridin-2-yl)methyl]-methylamino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-(1-benzothiophen-3-yl)-4-[[(2S)-1,4-dioxan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H23NO4S
7-(1-benzothiophen-3-yl)-4-[[(2S)-1,4-dioxan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— (7S)-2-methylsulfanyl-5-oxo-N-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C13H13N5O2S
(7S)-2-methylsulfanyl-5-oxo-N-phenyl-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C14H11ClF3N5O2
(7S)-N-[4-chloro-3-(trifluoromethyl)phenyl]-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(5-chloro-2-methylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C14H14ClN5O2
(7R)-N-(5-chloro-2-methylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7R)-N-(4-chlorophenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C13H12ClN5O2
(7R)-N-(4-chlorophenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-[[[(S)-cyclopropyl(pyridin-2-yl)methyl]-methylamino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C21H21N3O3
7-[[[(S)-cyclopropyl(pyridin-2-yl)methyl]-methylamino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C15H15N5O4
(7R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— (7S)-N-(2-methoxy-5-methylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C15H17N5O3
(7S)-N-(2-methoxy-5-methylphenyl)-2-methyl-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-[[(1S,4aR,6R,8aS)-6-hydroxy-2,5,5,8a-tetramethyl-1,4,4a,6,7,8-hexahydronaphthalen-1-yl]methoxy]chromen-2-one —— C24H30O4
7-[[(1S,4aR,6R,8aS)-6-hydroxy-2,5,5,8a-tetramethyl-1,4,4a,6,7,8-hexahydronaphthalen-1-yl]methoxy]chromen-2-one
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-spiro[2.3]hexan-2-yl]methanone —— C22H22ClNO3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-spiro[2.3]hexan-2-yl]methanone
—— (7R)-7-bromo-6-methyl-2,3-diphenyl-7,9-dihydroimidazo[1,2-b][1,2,4]triazepin-8-one —— C19H15BrN4O
(7R)-7-bromo-6-methyl-2,3-diphenyl-7,9-dihydroimidazo[1,2-b][1,2,4]triazepin-8-one
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-spiro[2.3]hexan-2-yl]methanone —— C22H22ClNO3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-spiro[2.3]hexan-2-yl]methanone
—— 7-[(E)-but-2-enyl]-3-methyl-8-[(2E)-2-[(E)-4-phenylbut-3-en-2-ylidene]hydrazinyl]purine-2,6-dione —— C20H22N6O2
7-[(E)-but-2-enyl]-3-methyl-8-[(2E)-2-[(E)-4-phenylbut-3-en-2-ylidene]hydrazinyl]purine-2,6-dione
—— 7-[(E)-but-2-enyl]-3-methyl-8-[2-[1-(6-oxocyclohexa-2,4-dien-1-ylidene)ethyl]hydrazinyl]purine-2,6-dione —— C18H20N6O3
7-[(E)-but-2-enyl]-3-methyl-8-[2-[1-(6-oxocyclohexa-2,4-dien-1-ylidene)ethyl]hydrazinyl]purine-2,6-dione
—— (7R,7aR)-9,9-diethyl-7-methyl-7,7a,8,10-tetrahydronaphtho[1,2-f]isoindol-9-ium —— C21H26N+
(7R,7aR)-9,9-diethyl-7-methyl-7,7a,8,10-tetrahydronaphtho[1,2-f]isoindol-9-ium
—— 7-Methyl-3-morpholin-4-yl-1-piperidin-1-yl-5,6,7,8-tetrahydro-2,7-naphthyridine-2,7-diium-4-carbonitrile —— C19H29N5O+2
7-Methyl-3-morpholin-4-yl-1-piperidin-1-yl-5,6,7,8-tetrahydro-2,7-naphthyridine-2,7-diium-4-carbonitrile
—— 7-methyl-4-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]thieno[3,2-d]pyrimidine —— C15H17N5S
7-methyl-4-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]thieno[3,2-d]pyrimidine
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-pyrrolidin-3-yl]methanone —— C20H21ClN2O3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-pyrrolidin-3-yl]methanone
—— 7-methyl-4-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]thieno[3,2-d]pyrimidine —— C15H17N5S
7-methyl-4-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]thieno[3,2-d]pyrimidine
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone —— C20H21ClN2O3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone —— C21H21N3O4S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-morpholin-2-yl]methanone —— C21H21N3O4S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-morpholin-2-yl]methanone
—— 7-chloro-3-[[(2S)-4-ethyl-2-methyl-3-oxopiperazin-1-yl]methyl]-1H-quinolin-2-one —— C17H20ClN3O2
7-chloro-3-[[(2S)-4-ethyl-2-methyl-3-oxopiperazin-1-yl]methyl]-1H-quinolin-2-one
—— 7-chloro-3-[[(2R)-4-ethyl-2-methyl-3-oxopiperazin-1-yl]methyl]-1H-quinolin-2-one —— C17H20ClN3O2
7-chloro-3-[[(2R)-4-ethyl-2-methyl-3-oxopiperazin-1-yl]methyl]-1H-quinolin-2-one
—— 7-(3-chlorophenyl)-4-[(2S)-2-hydroxybutyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C19H22ClNO3
7-(3-chlorophenyl)-4-[(2S)-2-hydroxybutyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-[[methyl-[(1R)-1-pyridin-3-ylethyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C19H19N3O3
7-[[methyl-[(1R)-1-pyridin-3-ylethyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[methyl-[(1S)-1-pyridin-3-ylethyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C19H19N3O3
7-[[methyl-[(1S)-1-pyridin-3-ylethyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— (7-methylimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl]methanone —— C25H31N5O
(7-methylimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl]methanone
—— 7-chloro-4-methyl-2-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]quinoline —— C18H19ClN4
7-chloro-4-methyl-2-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]quinoline
—— (7-methylimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl]methanone —— C25H31N5O
(7-methylimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl]methanone
—— 7-chloro-4-methyl-2-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]quinoline —— C18H19ClN4
7-chloro-4-methyl-2-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]quinoline
—— (7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(5-methylfuran-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H21N5O2
(7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(5-methylfuran-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-hydroxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H19N5O2
(7R)-7-(4-hydroxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— [7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone —— C22H21NO4S
[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone
—— (7S)-7-(4-hydroxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H19N5O2
(7S)-7-(4-hydroxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(2,5-dimethoxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O3
(7R)-7-(2,5-dimethoxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-benzyl-7-(2,5-dimethoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O3
(7S)-N-benzyl-7-(2,5-dimethoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(2,5-dimethoxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O3
(7S)-7-(2,5-dimethoxyphenyl)-5-methyl-N-(2-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(5-methylfuran-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H21N5O2
(7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(5-methylfuran-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chlorophenyl)-5-methyl-7-(2-nitrophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H15ClN6O3
(7S)-N-(4-chlorophenyl)-5-methyl-7-(2-nitrophenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-N-(2-methylphenyl)-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H17N5OS
(7S)-5-methyl-N-(2-methylphenyl)-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-(2-methylphenyl)-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H17N5OS
(7R)-5-methyl-N-(2-methylphenyl)-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide