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—— 7-Methyl-2-[[5-(4-methylphenyl)tetrazol-2-yl]methyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C15H13N7OS
7-Methyl-2-[[5-(4-methylphenyl)tetrazol-2-yl]methyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 7-[[4-(1,3-Benzothiazol-2-yl)piperidin-1-yl]methyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C20H21N5OS2
7-[[4-(1,3-Benzothiazol-2-yl)piperidin-1-yl]methyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 7-[[4-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-2-ethyl-8H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-4-ium-5-one —— C20H22N5OS2+
7-[[4-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-2-ethyl-8H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-4-ium-5-one
—— 7-methyl-3-[(3S)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C12H21N5
7-methyl-3-[(3S)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-methyl-3-[(3R)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C12H21N5
7-methyl-3-[(3R)-piperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine
—— 7-[(2S)-piperidin-2-yl]-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine —— C12H13F3N4
7-[(2S)-piperidin-2-yl]-5-(trifluoromethyl)imidazo[1,2-a]pyrimidine
—— 7-[[(3,4-Dichlorophenyl)methyl-methylamino]methyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C16H16Cl2N4OS
7-[[(3,4-Dichlorophenyl)methyl-methylamino]methyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— (7R)-2-[(1R)-1-(4-methoxyphenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H22N2O2S2
(7R)-2-[(1R)-1-(4-methoxyphenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— [7-[4-(6-methylpyridin-3-yl)-5-pyridin-4-ylpyrimidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl]methanol —— C21H20N8O
[7-[4-(6-methylpyridin-3-yl)-5-pyridin-4-ylpyrimidin-2-yl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-3-yl]methanol
—— (7R)-2-[(1S)-1-(4-methoxyphenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H22N2O2S2
(7R)-2-[(1S)-1-(4-methoxyphenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-(4-methoxyphenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H22N2O2S2
(7S)-2-[(1R)-1-(4-methoxyphenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-(4-methoxyphenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H22N2O2S2
(7S)-2-[(1S)-1-(4-methoxyphenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(2-nitrophenoxy)methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H17N3O4S
(7S)-7-methyl-2-[(2-nitrophenoxy)methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(2-nitrophenoxy)methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H17N3O4S
(7R)-7-methyl-2-[(2-nitrophenoxy)methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1R)-1-(4-nitrophenoxy)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H19N3O4S
(7S)-7-methyl-2-[(1R)-1-(4-nitrophenoxy)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(4-nitrophenoxy)methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H17N3O4S
(7R)-7-methyl-2-[(4-nitrophenoxy)methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1S)-1-(4-nitrophenoxy)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H19N3O4S
(7R)-7-methyl-2-[(1S)-1-(4-nitrophenoxy)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7-Hydroxy-2-oxochromen-4-yl)methyl 2-(methanesulfonamido)benzoate —— C18H15NO7S
(7-Hydroxy-2-oxochromen-4-yl)methyl 2-(methanesulfonamido)benzoate
—— (7S)-7-methyl-2-[(1S)-1-(4-nitrophenoxy)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H19N3O4S
(7S)-7-methyl-2-[(1S)-1-(4-nitrophenoxy)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(1R)-1-(4-nitrophenoxy)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H19N3O4S
(7R)-7-methyl-2-[(1R)-1-(4-nitrophenoxy)ethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(4-nitrophenoxy)methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H17N3O4S
(7S)-7-methyl-2-[(4-nitrophenoxy)methyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-methoxy-1'-[(3,4,5-trimethoxyphenyl)methyl]spiro[5H-pyrrolo[1,2-a]quinoxaline-4,4'-piperidine] —— C26H31N3O4
7-methoxy-1'-[(3,4,5-trimethoxyphenyl)methyl]spiro[5H-pyrrolo[1,2-a]quinoxaline-4,4'-piperidine]
—— 7-Benzyl-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one —— C20H16N2O4
7-Benzyl-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one
—— 7-[[(2R)-oxolan-2-yl]methyl]-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one —— C18H18N2O5
7-[[(2R)-oxolan-2-yl]methyl]-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one
—— 7-[[(2S)-oxolan-2-yl]methyl]-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one —— C18H18N2O5
7-[[(2S)-oxolan-2-yl]methyl]-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one
—— 7-(Furan-2-ylmethyl)-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one —— C18H14N2O5
7-(Furan-2-ylmethyl)-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one
—— 7-[(2-Methoxyphenyl)methyl]-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one —— C21H18N2O5
7-[(2-Methoxyphenyl)methyl]-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one
—— (7R)-2-[(1S)-1-[[5-(cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H21N5OS3
(7R)-2-[(1S)-1-[[5-(cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-(2-Methoxyethyl)-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one —— C16H16N2O5
7-(2-Methoxyethyl)-4,14,16-trioxa-2,7-diazatetracyclo[9.7.0.03,9.013,17]octadeca-1,3(9),10,12,17-pentaen-6-one
—— (7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(3-cyano-4-methyl-6-oxo-1H-pyridin-2-yl)sulfanyl]acetate —— C19H16N4O4S
(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(3-cyano-4-methyl-6-oxo-1H-pyridin-2-yl)sulfanyl]acetate
—— (7S)-2-[(4-methoxy-2-nitrophenoxy)methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H19N3O5S
(7S)-2-[(4-methoxy-2-nitrophenoxy)methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-[[5-(cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H21N5OS3
(7S)-2-[(1S)-1-[[5-(cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1S)-1-(4-methoxy-2-nitrophenoxy)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H21N3O5S
(7R)-2-[(1S)-1-(4-methoxy-2-nitrophenoxy)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[1-[(2S)-3-(4-chloropyrazol-1-yl)-2-methylpropanoyl]piperidin-4-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C22H23ClF3N5O2
7-[1-[(2S)-3-(4-chloropyrazol-1-yl)-2-methylpropanoyl]piperidin-4-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— (7R)-2-[(1R)-1-[[5-(cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H21N5OS3
(7R)-2-[(1R)-1-[[5-(cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[(3S)-1-(3,4-dimethoxybenzoyl)piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C24H24F3N3O4
7-[(3S)-1-(3,4-dimethoxybenzoyl)piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— (7R)-2-[[5-(cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C17H19N5OS3
(7R)-2-[[5-(cyclopropylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(4-methoxy-2-nitrophenoxy)methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H19N3O5S
(7R)-2-[(4-methoxy-2-nitrophenoxy)methyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1R)-1-(4-methoxy-2-nitrophenoxy)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H21N3O5S
(7S)-2-[(1R)-1-(4-methoxy-2-nitrophenoxy)ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[1-[(2R)-3-(4-chloropyrazol-1-yl)-2-methylpropanoyl]piperidin-4-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C22H23ClF3N5O2
7-[1-[(2R)-3-(4-chloropyrazol-1-yl)-2-methylpropanoyl]piperidin-4-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3R)-1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C24H24F3N3O4
7-[(3R)-1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3R)-1-(3,4-dimethoxybenzoyl)piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C24H24F3N3O4
7-[(3R)-1-(3,4-dimethoxybenzoyl)piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3S)-1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C24H24F3N3O4
7-[(3S)-1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— (7-fluoro-1H-indol-2-yl)-[(3S)-3-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C22H19F4N5O
(7-fluoro-1H-indol-2-yl)-[(3S)-3-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— (7-fluoro-1H-indol-2-yl)-[(3R)-3-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C22H19F4N5O
(7-fluoro-1H-indol-2-yl)-[(3R)-3-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— 7-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidine-1-carbonyl]-2-(2-methoxyethyl)-3H-isoindol-1-one —— C22H24FN3O4
7-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidine-1-carbonyl]-2-(2-methoxyethyl)-3H-isoindol-1-one
—— 7-(5-pyrazin-2-yl-4-thiophen-2-ylpyrimidin-2-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C17H14N8S
7-(5-pyrazin-2-yl-4-thiophen-2-ylpyrimidin-2-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7,7-dimethyl-3-phenyl-2,6-dihydro-1H-azepin-5-one —— C14H17NO
7,7-dimethyl-3-phenyl-2,6-dihydro-1H-azepin-5-one
—— 7-[4-(4-Methoxyphenyl)piperazin-1-yl]-5-methyl-2-(1-methylimidazol-2-yl)pyrazolo[1,5-a]pyrimidine —— C22H25N7O
7-[4-(4-Methoxyphenyl)piperazin-1-yl]-5-methyl-2-(1-methylimidazol-2-yl)pyrazolo[1,5-a]pyrimidine
—— 7-[4-(2-Methoxyethyl)piperazin-1-yl]-5-methyl-2-(1-methylimidazol-2-yl)pyrazolo[1,5-a]pyrimidine —— C18H25N7O
7-[4-(2-Methoxyethyl)piperazin-1-yl]-5-methyl-2-(1-methylimidazol-2-yl)pyrazolo[1,5-a]pyrimidine