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—— 5-[(R)-(3-chlorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H24ClN5OS
5-[(R)-(3-chlorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(3,4-difluorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H21F2N5OS
5-[(S)-(3,4-difluorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(4-benzylpiperazine-1,4-diium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C22H27N5O2S+2
5-[(S)-(4-benzylpiperazine-1,4-diium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3,4-difluorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H21F2N4O2S+
5-[(S)-(3,4-difluorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-7-methyl-2-[4-(tetrazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C14H22N6O2
(5S)-7-methyl-2-[4-(tetrazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(benzimidazol-1-ylmethyl)-N-[(2R)-1-thiophen-3-ylpropan-2-yl]-1H-pyrazole-3-carboxamide —— C19H19N5OS
5-(benzimidazol-1-ylmethyl)-N-[(2R)-1-thiophen-3-ylpropan-2-yl]-1H-pyrazole-3-carboxamide
—— (5R)-5-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethylamino)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H25N3O4
(5R)-5-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethylamino)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(R)-(3-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H21ClN4O2S
5-[(R)-(3-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(3-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H21ClN4O2S
5-[(S)-(3-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(3-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22ClN4O2S+
5-[(R)-(3-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H24ClN5O2S
5-[(R)-(3-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(4-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H24FN4O2S+
5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(4-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5R)-5-(4-methoxycarbonylpiperidin-1-yl)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C18H25N3O4
(5R)-5-(4-methoxycarbonylpiperidin-1-yl)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-5-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethylamino)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H25N3O4
(5S)-5-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethylamino)-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— 5-[(R)-(3,4-dimethoxyphenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H26N4O4S
5-[(R)-(3,4-dimethoxyphenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(4-benzylpiperazine-1,4-diium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C22H27N5O2S+2
5-[(R)-(4-benzylpiperazine-1,4-diium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H24ClN5O2S
5-[(S)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(2-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22ClN4O2S+
5-[(S)-(2-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22ClN4O2S+
5-[(S)-(4-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-ethoxyphenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H29N5O2S+2
5-[(R)-(4-ethoxyphenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3,4-difluorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H23F2N5OS+2
5-[(R)-(3,4-difluorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-chlorophenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H26ClN5OS+2
5-[(R)-(2-chlorophenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H24ClN5O2S
5-[(R)-(4-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(3,4-difluorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H23F2N5OS
5-[(R)-(3,4-difluorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(3,4-dimethoxyphenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O4S+
5-[(S)-(3,4-dimethoxyphenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-chlorophenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H26ClN5OS+2
5-[(S)-(4-chlorophenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H24ClN5O2S
5-[(R)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(4-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H21ClN4O2S
5-[(S)-(4-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(4-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H24ClN5O2S
5-[(S)-(4-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[(2R)-4-methylpentan-2-yl]-1,2-oxazole-3-carboxamide —— C17H29N3O3
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[(2R)-4-methylpentan-2-yl]-1,2-oxazole-3-carboxamide
—— 5-[(R)-(4-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H21ClN4O2S
5-[(R)-(4-chlorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(3,4-difluorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H21F2N4O2S+
5-[(R)-(3,4-difluorophenyl)-(4-hydroxypiperidin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H26ClN5O2S+2
5-[(S)-(4-chlorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-benzylpiperazin-1-ium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C22H25N5O2S
5-[(S)-(4-benzylpiperazin-1-ium-1-yl)-(furan-2-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(4-chlorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H24ClN5OS
5-[(S)-(4-chlorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(4-chlorophenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H26ClN5OS+2
5-[(R)-(4-chlorophenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3-chlorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H24ClN5OS+2
5-[(S)-(3-chlorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3,4-dimethoxyphenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H27N5O3S
5-[(S)-(3,4-dimethoxyphenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(2,4-dichlorophenyl)-morpholin-4-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H18Cl2N4O2S
5-[(R)-(2,4-dichlorophenyl)-morpholin-4-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3,4-dimethoxyphenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H29N5O3S+2
5-[(S)-(3,4-dimethoxyphenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-ethoxyphenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H27N5O2S
5-[(R)-(4-ethoxyphenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(3-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H23FN4O2S
5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(3-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(2-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H23FN4O2S
5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(2-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3,4-dimethoxyphenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H27N5O3S
5-[(R)-(3,4-dimethoxyphenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(3-methoxyphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O3S
5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-(3-methoxyphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-chlorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H24ClN5OS
5-[(R)-(4-chlorophenyl)-(4-ethylpiperazin-1-ium-1-yl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(4-methylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H27N4O3S+
5-[(S)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(4-methylphenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(3-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H23FN4O3S
5-[(R)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(3-fluorophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-nitrophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H25N5O3S
5-[(R)-[(3S,5R)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-nitrophenyl)methyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(3-chlorophenyl)-morpholin-4-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H19ClN4O2S
5-[(S)-(3-chlorophenyl)-morpholin-4-ylmethyl]-2-ethyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol