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—— (5R)-1-ethyl-5-(6-oxa-9-azaspiro[4.5]decan-9-yl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C18H27N3O3
(5R)-1-ethyl-5-(6-oxa-9-azaspiro[4.5]decan-9-yl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— [5-(benzimidazol-1-ylmethyl)-1H-pyrazol-3-yl]-[(2S)-2-(4-fluorophenyl)azetidin-1-yl]methanone —— C21H18FN5O
[5-(benzimidazol-1-ylmethyl)-1H-pyrazol-3-yl]-[(2S)-2-(4-fluorophenyl)azetidin-1-yl]methanone
—— 5-methyl-N-[2-[(3S)-1-[(2-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl]ethyl]pyrazine-2-carboxamide —— C18H26N6O
5-methyl-N-[2-[(3S)-1-[(2-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl]ethyl]pyrazine-2-carboxamide
—— [5-[(3,5-dimethylpyrazol-1-yl)methyl]-1H-pyrazol-3-yl]-[(2S)-2-(2-methylphenyl)pyrrolidin-1-yl]methanone —— C21H25N5O
[5-[(3,5-dimethylpyrazol-1-yl)methyl]-1H-pyrazol-3-yl]-[(2S)-2-(2-methylphenyl)pyrrolidin-1-yl]methanone
—— (5R)-N-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-propan-2-yl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H20N4O3
(5R)-N-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-propan-2-yl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-propan-2-yl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H20N4O3
(5S)-N-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-propan-2-yl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(3R)-1-(3-azaspiro[5.5]undecan-9-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole —— C22H31N5O
5-[(3R)-1-(3-azaspiro[5.5]undecan-9-yl)piperidin-3-yl]-3-pyridin-3-yl-1,2,4-oxadiazole
—— (5S)-5-[3-(trifluoromethyl)phenoxy]-1-azabicyclo[3.2.1]octane —— C14H16F3NO
(5S)-5-[3-(trifluoromethyl)phenoxy]-1-azabicyclo[3.2.1]octane
—— (5S)-5-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-1-(2-methylpropyl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C21H27N3O3
(5S)-5-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-1-(2-methylpropyl)-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5R)-5-[3-(trifluoromethyl)phenoxy]-1-azabicyclo[3.2.1]octane —— C14H16F3NO
(5R)-5-[3-(trifluoromethyl)phenoxy]-1-azabicyclo[3.2.1]octane
—— 5-[(3S)-1-(1,3-benzothiazole-5-carbonyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C18H21N5O2S
5-[(3S)-1-(1,3-benzothiazole-5-carbonyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-[(3R)-1-[2-(benzotriazol-2-yl)acetyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C18H23N7O2
5-[(3R)-1-[2-(benzotriazol-2-yl)acetyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— [5-[(3-fluorophenoxy)methyl]-1H-pyrazol-3-yl]-[(3R)-3-phenylpiperazin-1-yl]methanone —— C21H21FN4O2
[5-[(3-fluorophenoxy)methyl]-1H-pyrazol-3-yl]-[(3R)-3-phenylpiperazin-1-yl]methanone
—— 5-[(3R)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C18H29N7O
5-[(3R)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]hexanamide —— C13H26N2O
5-methyl-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]hexanamide
—— 5-[(3S)-1-[2-(benzotriazol-2-yl)acetyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C18H23N7O2
5-[(3S)-1-[2-(benzotriazol-2-yl)acetyl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-[4-[(3R)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C21H30N4O3
5-[4-[(3R)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— 5-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]hexanamide —— C13H26N2O
5-methyl-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]hexanamide
—— (5R,6S)-5-(4-fluorophenyl)-2-[(3R)-3-methylpiperidin-1-yl]-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile —— C20H20FN5O2
(5R,6S)-5-(4-fluorophenyl)-2-[(3R)-3-methylpiperidin-1-yl]-4,7-dioxo-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile
—— (5R)-5-[4-(3-propan-2-yl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrrolidin-2-one —— C16H24N4O2
(5R)-5-[4-(3-propan-2-yl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrrolidin-2-one
—— (5R,6S)-2-[(3S)-3-methylpiperidin-1-yl]-4,7-dioxo-5-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile —— C20H21N5O2
(5R,6S)-2-[(3S)-3-methylpiperidin-1-yl]-4,7-dioxo-5-phenyl-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile
—— 5-(furan-2-yl)-2-[(3S)-3-methylpiperidin-1-yl]-3H-pyrido[2,3-d]pyrimidin-4-one —— C17H18N4O2
5-(furan-2-yl)-2-[(3S)-3-methylpiperidin-1-yl]-3H-pyrido[2,3-d]pyrimidin-4-one
—— (5S)-5-[4-(3-propan-2-yl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrrolidin-2-one —— C16H24N4O2
(5S)-5-[4-(3-propan-2-yl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrrolidin-2-one
—— 5-nitro-2-(1H-pyrrol-1-yl)phenol —— C10H8N2O3
5-nitro-2-(1H-pyrrol-1-yl)phenol
—— 5-[(3S)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C18H29N7O
5-[(3S)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— (5E)-5-[(4-chlorophenyl)methylidene]-4,6-diimino-1-(3-methylphenyl)-2-oxopiperidine-3-carbonitrile —— C20H15ClN4O
(5E)-5-[(4-chlorophenyl)methylidene]-4,6-diimino-1-(3-methylphenyl)-2-oxopiperidine-3-carbonitrile
—— (5S)-5-benzyl-2-[4-(4-methylphenyl)piperazin-1-yl]-4,5-dihydro-1,3-thiazole —— C21H25N3S
(5S)-5-benzyl-2-[4-(4-methylphenyl)piperazin-1-yl]-4,5-dihydro-1,3-thiazole
—— [5-[(3-fluorophenoxy)methyl]-1H-pyrazol-3-yl]-[(3S)-3-phenylpiperazin-1-yl]methanone —— C21H21FN4O2
[5-[(3-fluorophenoxy)methyl]-1H-pyrazol-3-yl]-[(3S)-3-phenylpiperazin-1-yl]methanone
—— (5R,6S)-2-[(3R)-3-methylpiperidin-1-yl]-4,7-dioxo-5-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile —— C20H21N5O2
(5R,6S)-2-[(3R)-3-methylpiperidin-1-yl]-4,7-dioxo-5-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile
—— (5E)-5-[(4-bromophenyl)methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one —— C16H17BrN2O2S
(5E)-5-[(4-bromophenyl)methylidene]-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one
—— (5S,7S)-N-[(2S)-butan-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H23F3N4O2
(5S,7S)-N-[(2S)-butan-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5E)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-5-[(4-hydroxyphenyl)methylidene]-1,3-thiazol-4-one —— C16H18N2O3S
(5E)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-5-[(4-hydroxyphenyl)methylidene]-1,3-thiazol-4-one
—— (5R,6S)-5-(4-fluorophenyl)-2-[(3S)-3-methylpiperidin-1-yl]-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile —— C20H20FN5O2
(5R,6S)-5-(4-fluorophenyl)-2-[(3S)-3-methylpiperidin-1-yl]-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile
—— (5R)-5-tert-butyl-3-(1,1,2,2,3,3,3-heptafluoropropyl)-5-hydroxy-4H-pyrazole-1-carbaldehyde —— C11H13F7N2O2
(5R)-5-tert-butyl-3-(1,1,2,2,3,3,3-heptafluoropropyl)-5-hydroxy-4H-pyrazole-1-carbaldehyde
—— 5-[[(6R)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]amino]-5-oxopentanoate —— C15H19N2O4S-
5-[[(6R)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]amino]-5-oxopentanoate
—— (5S,7R)-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxylate —— C12H8ClF3N3O2S-
(5S,7R)-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxylate
—— (5S,6S)-5-(2-fluorophenyl)-2-[(3S)-3-methylpiperidin-1-yl]-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile —— C20H20FN5O2
(5S,6S)-5-(2-fluorophenyl)-2-[(3S)-3-methylpiperidin-1-yl]-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-6-carbonitrile
—— (5-Bromo-2,4-dimethoxyphenyl)methyl-pentan-3-ylazanium —— C14H23BrNO2+
(5-Bromo-2,4-dimethoxyphenyl)methyl-pentan-3-ylazanium
—— [(5R)-3-(4-chlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-phenylmethanone —— C17H12ClF3N2O2
[(5R)-3-(4-chlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-phenylmethanone
—— 5-[(4-Methylpiperazine-1,4-diium-1-yl)methyl]-6-phenylimidazo[2,1-b][1,3]thiazole —— C17H22N4S+2
5-[(4-Methylpiperazine-1,4-diium-1-yl)methyl]-6-phenylimidazo[2,1-b][1,3]thiazole
—— (5E)-2-(4-ethylpiperazin-4-ium-1-yl)-5-[(4-hydroxy-3-methoxyphenyl)methylidene]-1,3-thiazol-4-one —— C17H22N3O3S+
(5E)-2-(4-ethylpiperazin-4-ium-1-yl)-5-[(4-hydroxy-3-methoxyphenyl)methylidene]-1,3-thiazol-4-one
—— [(5S)-3-(4-chlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-phenylmethanone —— C17H12ClF3N2O2
[(5S)-3-(4-chlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-phenylmethanone
—— 5-(Furan-2-yl)-2-(2-hydroxyethyliminomethyl)cyclohexane-1,3-dione —— C13H15NO4
5-(Furan-2-yl)-2-(2-hydroxyethyliminomethyl)cyclohexane-1,3-dione
—— (5Z)-1-(4-fluorophenyl)-5-[4-(propan-2-yloxy)benzylidene]-2-thioxodihydropyrimidine-4,6(1H,5H)-dione —— C20H17FN2O3S
(5Z)-1-(4-fluorophenyl)-5-[4-(propan-2-yloxy)benzylidene]-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
—— (5Z)-5-[(5-chloro-2-hydroxy-3-methoxyphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C11H9ClN2O3S
(5Z)-5-[(5-chloro-2-hydroxy-3-methoxyphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5R)-2-naphthalen-1-ylsulfonyl-2,9-diazaspiro[4.5]decane —— C18H22N2O2S
(5R)-2-naphthalen-1-ylsulfonyl-2,9-diazaspiro[4.5]decane
—— 5-(benzimidazol-1-ylmethyl)-N-[(2S)-1-imidazol-1-ylbutan-2-yl]-1,2-oxazole-3-carboxamide —— C19H20N6O2
5-(benzimidazol-1-ylmethyl)-N-[(2S)-1-imidazol-1-ylbutan-2-yl]-1,2-oxazole-3-carboxamide
—— (5R)-5-[methyl-[(2-methyl-1,3-thiazol-4-yl)methyl]amino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid —— C17H22N4O2S
(5R)-5-[methyl-[(2-methyl-1,3-thiazol-4-yl)methyl]amino]-1-prop-2-enyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid
—— (5S)-5-(4-methoxyanilino)-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C16H14N2O2S2
(5S)-5-(4-methoxyanilino)-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[2-[[(5R)-1-azabicyclo[3.2.1]octan-5-yl]oxy]-5-methylphenyl]-1,2-oxazole —— C17H20N2O2
5-[2-[[(5R)-1-azabicyclo[3.2.1]octan-5-yl]oxy]-5-methylphenyl]-1,2-oxazole