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—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3R)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate —— C18H14FN3O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3R)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate
—— 5-methoxy-1,3-dimethyl-N-[(2R)-2-phenoxybutyl]pyrazole-4-carboxamide —— C17H23N3O3
5-methoxy-1,3-dimethyl-N-[(2R)-2-phenoxybutyl]pyrazole-4-carboxamide
—— 5-methyl-3-[(2R)-1-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C14H20N4O2
5-methyl-3-[(2R)-1-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-methoxy-1,3-dimethyl-N-[(2S)-2-phenoxybutyl]pyrazole-4-carboxamide —— C17H23N3O3
5-methoxy-1,3-dimethyl-N-[(2S)-2-phenoxybutyl]pyrazole-4-carboxamide
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (3R)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate —— C20H16FN3O4
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (3R)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate
—— [5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (3S)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate —— C18H14FN3O5
[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (3S)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3S)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate —— C18H14FN3O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (3S)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate
—— 5-(4-fluorophenyl)-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-5-oxopentanamide —— C17H23FN2O2
5-(4-fluorophenyl)-N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-5-oxopentanamide
—— (5-acetyl-2-methoxyphenyl)methyl (3S)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate —— C21H20FNO5
(5-acetyl-2-methoxyphenyl)methyl (3S)-1-(2-fluorophenyl)-5-oxopyrrolidine-3-carboxylate
—— 5-(4-fluorophenyl)-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-5-oxopentanamide —— C17H23FN2O2
5-(4-fluorophenyl)-N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-5-oxopentanamide
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(4-fluorophenoxy)-2-methylpropanoate —— C19H17FN2O4
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(4-fluorophenoxy)-2-methylpropanoate
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 4-(2,3-dihydro-1H-inden-5-yl)-4-oxobutanoate —— C20H18N2O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 4-(2,3-dihydro-1H-inden-5-yl)-4-oxobutanoate
—— (5S)-N-[(1R)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C19H23N5O2
(5S)-N-[(1R)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 5-[(1S)-1-(4-fluorophenoxy)ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C17H12F4N2O2
5-[(1S)-1-(4-fluorophenoxy)ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— 5-propan-2-yl-3-[(2R)-1-pyrimidin-2-ylpyrrolidin-2-yl]-1,2,4-oxadiazole —— C13H17N5O
5-propan-2-yl-3-[(2R)-1-pyrimidin-2-ylpyrrolidin-2-yl]-1,2,4-oxadiazole
—— (5R)-N-[(1S)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C19H23N5O2
(5R)-N-[(1S)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 5,6-dimethyl-3-[[(2R,3R)-3-pyrazol-1-ylbutan-2-yl]amino]pyridazine-4-carbonitrile —— C14H18N6
5,6-dimethyl-3-[[(2R,3R)-3-pyrazol-1-ylbutan-2-yl]amino]pyridazine-4-carbonitrile
—— (5R)-N-[(1R)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C19H23N5O2
(5R)-N-[(1R)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-fluorophenoxy)-2-methylpropanoate —— C17H15FN2O5
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-fluorophenoxy)-2-methylpropanoate
—— 5-propan-2-yl-3-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]-1,2,4-oxadiazole —— C13H17N5O
5-propan-2-yl-3-[(2S)-1-pyrimidin-2-ylpyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5,6-dimethyl-3-[[(2S,3S)-3-pyrazol-1-ylbutan-2-yl]amino]pyridazine-4-carbonitrile —— C14H18N6
5,6-dimethyl-3-[[(2S,3S)-3-pyrazol-1-ylbutan-2-yl]amino]pyridazine-4-carbonitrile
—— (5R)-2-(4-chlorophenyl)-4,5-dihydro-1H-imidazole-5-carbonitrile —— C10H8ClN3
(5R)-2-(4-chlorophenyl)-4,5-dihydro-1H-imidazole-5-carbonitrile
—— 5-chloro-6-[(2S)-2-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carboxamide —— C15H18ClN5O2
5-chloro-6-[(2S)-2-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carboxamide
—— (5S)-N-[(1S)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C19H23N5O2
(5S)-N-[(1S)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)-2-methylpropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 5-chloro-6-[(2R)-2-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carboxamide —— C15H18ClN5O2
5-chloro-6-[(2R)-2-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carboxamide
—— 5-[(1R)-1-(4-fluorophenoxy)ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C17H12F4N2O2
5-[(1R)-1-(4-fluorophenoxy)ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl 4-(2,3-dihydro-1H-inden-5-yl)-4-oxobutanoate —— C22H20N2O4
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl 4-(2,3-dihydro-1H-inden-5-yl)-4-oxobutanoate
—— 5-chloro-6-[(2S)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carboxamide —— C14H16ClN5O2
5-chloro-6-[(2S)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)pyrrolidin-1-yl]pyridine-3-carboxamide
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2,3-dihydro-1H-indene-5-carboxylate —— C19H18N2O4
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2,3-dihydro-1H-indene-5-carboxylate
—— (5S)-2-(4-chlorophenyl)-4,5-dihydro-1H-imidazole-5-carbonitrile —— C10H8ClN3
(5S)-2-(4-chlorophenyl)-4,5-dihydro-1H-imidazole-5-carbonitrile
—— 5,6-dimethyl-3-[[(2S,3R)-3-pyrazol-1-ylbutan-2-yl]amino]pyridazine-4-carbonitrile —— C14H18N6
5,6-dimethyl-3-[[(2S,3R)-3-pyrazol-1-ylbutan-2-yl]amino]pyridazine-4-carbonitrile
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 3-(2-methylpropoxy)benzoate —— C18H18N2O4S
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 3-(2-methylpropoxy)benzoate
—— 5,6-dimethyl-3-[[(2R,3S)-3-pyrazol-1-ylbutan-2-yl]amino]pyridazine-4-carbonitrile —— C14H18N6
5,6-dimethyl-3-[[(2R,3S)-3-pyrazol-1-ylbutan-2-yl]amino]pyridazine-4-carbonitrile
—— 5-tert-butyl-3-[[4-[(1R)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]methyl]-1,2,4-oxadiazole —— C18H30N6O2
5-tert-butyl-3-[[4-[(1R)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[[(2S)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole —— C14H19ClN4O
5-[[(2S)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole
—— 5-tert-butyl-3-[[4-[(1S)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]methyl]-1,2,4-oxadiazole —— C18H30N6O2
5-tert-butyl-3-[[4-[(1S)-1-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)ethyl]piperazin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-Bromo-6-[(4-methoxyphenyl)sulfanylmethyl]-1,3-benzodioxole —— C15H13BrO3S
5-Bromo-6-[(4-methoxyphenyl)sulfanylmethyl]-1,3-benzodioxole
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3-(2-methylpropoxy)benzoate —— C20H20N2O4
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 3-(2-methylpropoxy)benzoate
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 3-(2-methylpropoxy)benzoate —— C18H18N2O5
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 3-(2-methylpropoxy)benzoate
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 3-(methoxymethyl)-1-benzofuran-2-carboxylate —— C20H18N2O6
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 3-(methoxymethyl)-1-benzofuran-2-carboxylate
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 3,5-dimethyl-1,2-oxazole-4-carboxylate —— C16H13ClN2O4
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 3,5-dimethyl-1,2-oxazole-4-carboxylate
—— 5-[(4-Methoxyphenyl)sulfanylmethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C14H12N2O2S2
5-[(4-Methoxyphenyl)sulfanylmethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-[[5-(4-ethylphenyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C17H15N5OS2
5-[[5-(4-ethylphenyl)-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-[[(2R)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C15H22ClN5O2
5-[[(2R)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-(4-chlorophenyl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazole —— C18H13ClN4OS
5-(4-chlorophenyl)-2-[(5-phenyl-1H-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-oxazole
—— 5-cyclopropyl-3-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H23N5O2
5-cyclopropyl-3-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[[(2R)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-2-methyl-1,3-thiazole —— C14H19ClN4S
5-[[(2R)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-2-methyl-1,3-thiazole
—— 5-[[(2S)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C15H22ClN5O2
5-[[(2S)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-[[(2R)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(furan-3-yl)-1,2,4-oxadiazole —— C16H18ClN5O2
5-[[(2R)-2-(5-chloro-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(furan-3-yl)-1,2,4-oxadiazole
—— 5-chloro-4-[(2R)-1-[(1-ethylimidazol-2-yl)methyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole —— C15H22ClN5
5-chloro-4-[(2R)-1-[(1-ethylimidazol-2-yl)methyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole