N2-(4-(((2-amino-4-oxo-3,4-dihydropteridin-6-yl)methyl)amino)benzoyl)-N5-(4-(3,4 -diaminophenoxy)butyl)glutamine 、
2,5-bis<(3-ethyl-5-formyl-4-methylpyrrol-2-yl)methyl>-3,4-diethylpyrrole 在
盐酸 作用下,
以
甲醇 为溶剂,
反应 0.5h,
生成 N2-(4-(((2-amino-4-oxo-3,4-dihydropteridin-6-yl)methyl)amino)benzoyl)-N5-(4-(((6E,9E)-13,33, 34,53-tetraethyl-14,54-dimethyl-31H-11l2,51l2-1l2,51l2,7,9-tetraaza-1,3,5(2,5)-tripyrrolidine-8(1,2)-benzocyclodecane-6,9-diene-84-yl)oxy)butyl)glutamine