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—— 6-[[(1S)-1-cyclopropylethyl]-(2-methoxyethyl)amino]pyridazine-3-carboxylic acid —— C13H19N3O3
6-[[(1S)-1-cyclopropylethyl]-(2-methoxyethyl)amino]pyridazine-3-carboxylic acid
—— 6-benzyl-2-[(4-bromophenyl)-hydroxymethyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C23H20BrN5O3
6-benzyl-2-[(4-bromophenyl)-hydroxymethyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-[1-hydroxy-3-(5-methylfuran-2-yl)butyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C25H27N5O4
6-benzyl-2-[1-hydroxy-3-(5-methylfuran-2-yl)butyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-cyclohexyl-2-[hydroxy-(3,4,5-trimethoxyphenyl)methyl]-1-(4-methoxyanilino)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C30H37N3O7
6-cyclohexyl-2-[hydroxy-(3,4,5-trimethoxyphenyl)methyl]-1-(4-methoxyanilino)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-[[(1R)-1-cyclopropylethyl]-(2-methoxyethyl)amino]pyridazine-3-carboxylic acid —— C13H19N3O3
6-[[(1R)-1-cyclopropylethyl]-(2-methoxyethyl)amino]pyridazine-3-carboxylic acid
—— 6-benzyl-2-(1-hydroxy-2-phenylethyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C24H23N5O3
6-benzyl-2-(1-hydroxy-2-phenylethyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-cyclohexyl-2-[furan-2-yl(hydroxy)methyl]-1-(4-methoxyanilino)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C25H29N3O5
6-cyclohexyl-2-[furan-2-yl(hydroxy)methyl]-1-(4-methoxyanilino)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-(1-hydroxy-2-phenylpropyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C25H25N5O3
6-benzyl-2-(1-hydroxy-2-phenylpropyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-(chloromethyl)-N-[(1S)-1-cyclopropylethyl]-N-(2-methoxyethyl)pyridazin-3-amine —— C13H20ClN3O
6-(chloromethyl)-N-[(1S)-1-cyclopropylethyl]-N-(2-methoxyethyl)pyridazin-3-amine
—— 6-cyclohexyl-2-[hydroxy-(4-methoxy-3-phenylmethoxyphenyl)methyl]-1-(4-methoxyanilino)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C35H39N3O6
6-cyclohexyl-2-[hydroxy-(4-methoxy-3-phenylmethoxyphenyl)methyl]-1-(4-methoxyanilino)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-[hydroxy-(4-methoxynaphthalen-1-yl)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C28H25N5O4
6-benzyl-2-[hydroxy-(4-methoxynaphthalen-1-yl)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-(2-ethyl-1-hydroxyhexyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C24H31N5O3
6-benzyl-2-(2-ethyl-1-hydroxyhexyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-[cyclohex-3-en-1-yl(hydroxy)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C23H25N5O3
6-benzyl-2-[cyclohex-3-en-1-yl(hydroxy)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-[(4-fluorophenyl)-hydroxymethyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C23H20FN5O3
6-benzyl-2-[(4-fluorophenyl)-hydroxymethyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-[hydroxy(naphthalen-1-yl)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C27H23N5O3
6-benzyl-2-[hydroxy(naphthalen-1-yl)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-[[3,5-bis(trifluoromethyl)phenyl]-hydroxymethyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C25H19F6N5O3
6-benzyl-2-[[3,5-bis(trifluoromethyl)phenyl]-hydroxymethyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-[hydroxy(phenyl)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C23H21N5O3
6-benzyl-2-[hydroxy(phenyl)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-(1-hydroxyundecyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C27H37N5O3
6-benzyl-2-(1-hydroxyundecyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-(1-hydroxypentyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C21H25N5O3
6-benzyl-2-(1-hydroxypentyl)-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-oxo-1-propyl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]pyridazine-3-carboxamide —— C17H18F3N3O2
6-oxo-1-propyl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]pyridazine-3-carboxamide
—— 6-[[(1R)-1-cyclopropylethyl]-(2-methoxyethyl)amino]pyridine-3-carbothioamide —— C14H21N3OS
6-[[(1R)-1-cyclopropylethyl]-(2-methoxyethyl)amino]pyridine-3-carbothioamide
—— 6-benzyl-2-[1-hydroxy-3-(4-nitrophenyl)prop-2-enyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C25H22N6O5
6-benzyl-2-[1-hydroxy-3-(4-nitrophenyl)prop-2-enyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— (6R,13R)-13-benzyl-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotetradec-8-ene-5,14-dione —— C33H42N2O5
(6R,13R)-13-benzyl-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotetradec-8-ene-5,14-dione
—— 6-benzyl-2-[(5-bromo-2,4-dimethoxyphenyl)-hydroxymethyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C25H24BrN5O5
6-benzyl-2-[(5-bromo-2,4-dimethoxyphenyl)-hydroxymethyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-benzyl-2-[hydroxy-(4-methoxy-3-phenylmethoxyphenyl)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione —— C31H29N5O5
6-benzyl-2-[hydroxy-(4-methoxy-3-phenylmethoxyphenyl)methyl]-1-(1,2,4-triazol-4-yl)-4a,7a-dihydro-2H-pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-oxo-1-propyl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]pyridazine-3-carboxamide —— C17H18F3N3O2
6-oxo-1-propyl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]pyridazine-3-carboxamide
—— (6R,13R)-13-benzyl-6-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotetradec-8-ene-5,14-dione —— C28H40N2O5
(6R,13R)-13-benzyl-6-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotetradec-8-ene-5,14-dione
—— (6R,13R)-13-benzyl-6-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl]-1-oxa-4-azacyclotetradec-8-ene-5,14-dione —— C26H36N2O5
(6R,13R)-13-benzyl-6-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl]-1-oxa-4-azacyclotetradec-8-ene-5,14-dione
—— (6R)-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotetradec-8-ene-5,14-dione —— C26H36N2O5
(6R)-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotetradec-8-ene-5,14-dione
—— 6-[2-[(2S)-2-(4-methoxyphenyl)azepan-1-yl]-2-oxoethoxy]-3,4-dihydro-1H-quinolin-2-one —— C24H28N2O4
6-[2-[(2S)-2-(4-methoxyphenyl)azepan-1-yl]-2-oxoethoxy]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(2R)-2-methylmorpholin-4-yl]sulfonyl-4H-1,4-benzoxazin-3-one —— C13H16N2O5S
6-[(2R)-2-methylmorpholin-4-yl]sulfonyl-4H-1,4-benzoxazin-3-one
—— (6R,12R)-12-benzyl-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotridec-8-ene-5,13-dione —— C32H40N2O5
(6R,12R)-12-benzyl-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotridec-8-ene-5,13-dione
—— (6R,12R)-12-benzyl-6-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotridec-8-ene-5,13-dione —— C27H38N2O5
(6R,12R)-12-benzyl-6-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotridec-8-ene-5,13-dione
—— (6R)-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotridec-8-ene-5,13-dione —— C25H34N2O5
(6R)-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-3,3-dimethyl-1-oxa-4-azacyclotridec-8-ene-5,13-dione
—— (6R,12R)-12-benzyl-6-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl]-1-oxa-4-azacyclotridec-8-ene-5,13-dione —— C25H34N2O5
(6R,12R)-12-benzyl-6-[2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl]-1-oxa-4-azacyclotridec-8-ene-5,13-dione
—— (6R)-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-1-oxa-4-azacyclotridec-8-ene-5,13-dione —— C23H30N2O5
(6R)-6-[2-[(3S)-3-(hydroxymethyl)-3,4-dihydro-1H-isoquinolin-2-yl]-2-oxoethyl]-1-oxa-4-azacyclotridec-8-ene-5,13-dione
—— 6-[[(2R)-butan-2-yl]-butylamino]pyridine-3-carboxylic acid —— C14H22N2O2
6-[[(2R)-butan-2-yl]-butylamino]pyridine-3-carboxylic acid
—— 6-[2-methoxyethyl-[(2S)-1-methoxypropan-2-yl]amino]pyridazine-3-carboxylic acid —— C12H19N3O4
6-[2-methoxyethyl-[(2S)-1-methoxypropan-2-yl]amino]pyridazine-3-carboxylic acid
—— 6-chloro-N-methyl-N-[(1R,2S)-2-methylcyclohexyl]-3-nitropyridin-2-amine —— C13H18ClN3O2
6-chloro-N-methyl-N-[(1R,2S)-2-methylcyclohexyl]-3-nitropyridin-2-amine
—— [6-[[(2S)-butan-2-yl]-butylamino]-3-chloropyridin-2-yl]methanol —— C14H23ClN2O
[6-[[(2S)-butan-2-yl]-butylamino]-3-chloropyridin-2-yl]methanol
—— 6-[2-methoxyethyl-[(2S)-1-methoxypropan-2-yl]amino]hexan-2-one —— C13H27NO3
6-[2-methoxyethyl-[(2S)-1-methoxypropan-2-yl]amino]hexan-2-one
—— [6-[methyl-[(1R,2S)-2-methylcyclohexyl]amino]pyridin-3-yl]methanol —— C14H22N2O
[6-[methyl-[(1R,2S)-2-methylcyclohexyl]amino]pyridin-3-yl]methanol
—— 6-chloro-N-(2-methoxyethyl)-N-[(2S)-1-methoxypropan-2-yl]pyridazine-3-carboxamide —— C12H18ClN3O3
6-chloro-N-(2-methoxyethyl)-N-[(2S)-1-methoxypropan-2-yl]pyridazine-3-carboxamide
—— [6-[methyl-[(1R,2R)-2-methylcyclohexyl]amino]pyridin-3-yl]methanol —— C14H22N2O
[6-[methyl-[(1R,2R)-2-methylcyclohexyl]amino]pyridin-3-yl]methanol
—— [6-[methyl-[(1S,2R)-2-methylcyclohexyl]amino]pyridazin-3-yl]methanol —— C13H21N3O
[6-[methyl-[(1S,2R)-2-methylcyclohexyl]amino]pyridazin-3-yl]methanol
—— 6-[methyl-[(1R,2R)-2-methylcyclohexyl]amino]pyridine-3-carbothioamide —— C14H21N3S
6-[methyl-[(1R,2R)-2-methylcyclohexyl]amino]pyridine-3-carbothioamide
—— 6-[methyl-[(1S,2R)-2-methylcyclohexyl]amino]pyridine-3-carbothioamide —— C14H21N3S
6-[methyl-[(1S,2R)-2-methylcyclohexyl]amino]pyridine-3-carbothioamide
—— 6-[[(2S)-butan-2-yl]-butylamino]pyridine-3-carbothioamide —— C14H23N3S
6-[[(2S)-butan-2-yl]-butylamino]pyridine-3-carbothioamide
—— [6-[methyl-[(1S,2S)-2-methylcyclohexyl]amino]pyridin-3-yl]methanol —— C14H22N2O
[6-[methyl-[(1S,2S)-2-methylcyclohexyl]amino]pyridin-3-yl]methanol
—— [6-[2-methoxyethyl-[(2S)-1-methoxypropan-2-yl]amino]pyridin-3-yl]methanol —— C13H22N2O3
[6-[2-methoxyethyl-[(2S)-1-methoxypropan-2-yl]amino]pyridin-3-yl]methanol