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—— (6S)-N-(4-chlorophenyl)-2-[(2E)-2-[(4-methoxyphenyl)methylidene]hydrazinyl]-4-oxo-5,6-dihydro-1,3-thiazine-6-carboxamide —— C19H17ClN4O3S
(6S)-N-(4-chlorophenyl)-2-[(2E)-2-[(4-methoxyphenyl)methylidene]hydrazinyl]-4-oxo-5,6-dihydro-1,3-thiazine-6-carboxamide
—— 6-[(Z)-2-phenylethenyl]-2-prop-2-enyl-4,5-dihydropyridazin-3-one —— C15H16N2O
6-[(Z)-2-phenylethenyl]-2-prop-2-enyl-4,5-dihydropyridazin-3-one
—— 6-[(Z)-3-(dimethylamino)prop-2-enoyl]-2-(3-methoxyphenyl)-4-methyl-1,2,4-triazine-3,5-dione —— C16H18N4O4
6-[(Z)-3-(dimethylamino)prop-2-enoyl]-2-(3-methoxyphenyl)-4-methyl-1,2,4-triazine-3,5-dione
—— 6-[(Z)-2-(4-methoxyphenyl)ethenyl]-2-methyl-4,5-dihydropyridazin-3-one —— C14H16N2O2
6-[(Z)-2-(4-methoxyphenyl)ethenyl]-2-methyl-4,5-dihydropyridazin-3-one
—— 6-tert-butyl-3-[(Z)-3-(dimethylamino)prop-2-enoyl]-1H-pyridin-2-one —— C14H20N2O2
6-tert-butyl-3-[(Z)-3-(dimethylamino)prop-2-enoyl]-1H-pyridin-2-one
—— [6-methyl-4-(2-propan-2-yloxyphenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidin-5-yl]-phenylmethanone —— C21H22N2O2S
[6-methyl-4-(2-propan-2-yloxyphenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidin-5-yl]-phenylmethanone
—— 6-[[1-(3-Chlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H20ClN5OS
6-[[1-(3-Chlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-Bromo-2-[[1-(4-chlorophenyl)tetrazol-5-yl]sulfanylmethyl]imidazo[1,2-a]pyridine —— C15H10BrClN6S
6-Bromo-2-[[1-(4-chlorophenyl)tetrazol-5-yl]sulfanylmethyl]imidazo[1,2-a]pyridine
—— 6-[[3-[4-[4-[[4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid —— C42H47ClN2O7
6-[[3-[4-[4-[[4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-6-oxohexanoic acid
—— 6,8-Difluoro-2-[2-(trifluoromethyl)phenyl]quinoline-4-carboxylic acid —— C17H8F5NO2
6,8-Difluoro-2-[2-(trifluoromethyl)phenyl]quinoline-4-carboxylic acid
—— 6-Amino-4-(3-methoxy-4-phenylmethoxyphenyl)-3-(trifluoromethyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C22H17F3N4O3
6-Amino-4-(3-methoxy-4-phenylmethoxyphenyl)-3-(trifluoromethyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-acetamido-N-[[4-[4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide —— C34H42N2O6S
6-acetamido-N-[[4-[4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]hexanamide
—— 6-Amino-4-[4-[(4-cyanophenyl)methoxy]-3-ethoxyphenyl]-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C24H21N5O3
6-Amino-4-[4-[(4-cyanophenyl)methoxy]-3-ethoxyphenyl]-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-Methoxy-2-[3-(2-nitrophenyl)prop-2-enylidene]-3,4-dihydronaphthalen-1-one —— C20H17NO4
6-Methoxy-2-[3-(2-nitrophenyl)prop-2-enylidene]-3,4-dihydronaphthalen-1-one
—— (6R)-N-cyclohexyl-5-[2-(diethylamino)ethyl]-6-methyl-4-oxo-2-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H43N5O2
(6R)-N-cyclohexyl-5-[2-(diethylamino)ethyl]-6-methyl-4-oxo-2-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6E)-2-ethyl-6-[[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H19FN4O3S
(6E)-2-ethyl-6-[[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6,8-dimethyl-1-(4-nitrophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C19H19N3O2
6,8-dimethyl-1-(4-nitrophenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— (6R)-2-tert-butyl-N-cyclohexyl-5-(4-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H31FN4O2
(6R)-2-tert-butyl-N-cyclohexyl-5-(4-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-5-[2-(diethylamino)ethyl]-6-methyl-4-oxo-2-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H43N5O2
(6S)-N-cyclohexyl-5-[2-(diethylamino)ethyl]-6-methyl-4-oxo-2-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-4-oxo-5-[[(2S)-oxolan-2-yl]methyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N4O3
(6R)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-4-oxo-5-[[(2S)-oxolan-2-yl]methyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-tert-butyl-N-cyclohexyl-5-(3-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H31FN4O2
(6R)-2-tert-butyl-N-cyclohexyl-5-(3-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-chloro-1-(4-methoxy-3-methylphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole —— C19H19ClN2O
6-chloro-1-(4-methoxy-3-methylphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
—— (6R)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-4-oxo-5-[[(2R)-oxolan-2-yl]methyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N4O3
(6R)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-4-oxo-5-[[(2R)-oxolan-2-yl]methyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-Amino-4-{3-[(2,4-difluorophenoxy)methyl]-4-methoxyphenyl}-3-propyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C24H22F2N4O3
6-Amino-4-{3-[(2,4-difluorophenoxy)methyl]-4-methoxyphenyl}-3-propyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-acetamido-N-[[3-[3-[4-[[[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-methylamino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C42H51N3O7
6-acetamido-N-[[3-[3-[4-[[[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-methylamino]methyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— (6R)-2-tert-butyl-N-cyclohexyl-5-(3,5-dimethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H36N4O4
(6R)-2-tert-butyl-N-cyclohexyl-5-(3,5-dimethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-Chloro-3-ethyl-2-[1-(furan-2-ylmethylamino)ethyl]quinazolin-4-one —— C17H18ClN3O2
6-Chloro-3-ethyl-2-[1-(furan-2-ylmethylamino)ethyl]quinazolin-4-one
—— 6-methyl-3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-[(1R)-1-phenylethyl]quinolin-2-amine —— C21H20N4O
6-methyl-3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-[(1R)-1-phenylethyl]quinolin-2-amine
—— 6-[8-(3-chloro-4-fluorophenyl)-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid —— C34H31ClF4N2O8
6-[8-(3-chloro-4-fluorophenyl)-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-6a-methyl-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid
—— (6S)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-4-oxo-5-[[(2R)-oxolan-2-yl]methyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N4O3
(6S)-N-cyclohexyl-2-(4-ethylphenyl)-6-methyl-4-oxo-5-[[(2R)-oxolan-2-yl]methyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cyclohexyl-5-(4-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H31FN4O2
(6S)-2-tert-butyl-N-cyclohexyl-5-(4-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cyclohexyl-5-(3-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H31FN4O2
(6S)-2-tert-butyl-N-cyclohexyl-5-(3-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-methyl-N-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-amine —— C14H13N3S
6-methyl-N-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-amine
—— (6S)-N-(4-chlorophenyl)-2-[(2E)-2-[[4-(dimethylamino)phenyl]methylidene]hydrazinyl]-4-oxo-5,6-dihydro-1,3-thiazine-6-carboxamide —— C20H20ClN5O2S
(6S)-N-(4-chlorophenyl)-2-[(2E)-2-[[4-(dimethylamino)phenyl]methylidene]hydrazinyl]-4-oxo-5,6-dihydro-1,3-thiazine-6-carboxamide
—— 6-methyl-N-(3-nitrophenyl)thieno[2,3-d]pyrimidin-4-amine —— C13H10N4O2S
6-methyl-N-(3-nitrophenyl)thieno[2,3-d]pyrimidin-4-amine
—— 6-methyl-3-(5-propyl-1,2,4-oxadiazol-3-yl)-N-[(1S)-1-pyridin-3-ylethyl]quinolin-2-amine —— C22H23N5O
6-methyl-3-(5-propyl-1,2,4-oxadiazol-3-yl)-N-[(1S)-1-pyridin-3-ylethyl]quinolin-2-amine
—— (6E)-5-imino-6-[(3-methoxy-4-phenylmethoxyphenyl)methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H22N4O3S
(6E)-5-imino-6-[(3-methoxy-4-phenylmethoxyphenyl)methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-methyl-3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-[(1S)-1-phenylethyl]quinolin-2-amine —— C21H20N4O
6-methyl-3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-[(1S)-1-phenylethyl]quinolin-2-amine
—— (6S)-2-[(2E)-2-[(4-chlorophenyl)methylidene]hydrazinyl]-N-(4-ethylphenyl)-4-oxo-5,6-dihydro-1,3-thiazine-6-carboxamide —— C20H19ClN4O2S
(6S)-2-[(2E)-2-[(4-chlorophenyl)methylidene]hydrazinyl]-N-(4-ethylphenyl)-4-oxo-5,6-dihydro-1,3-thiazine-6-carboxamide
—— (6E)-3-(4-methylphenyl)-6-[(3-methylphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C19H15N3OS
(6E)-3-(4-methylphenyl)-6-[(3-methylphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— 6-methyl-N-(3-methylphenyl)thieno[2,3-d]pyrimidin-4-amine —— C14H13N3S
6-methyl-N-(3-methylphenyl)thieno[2,3-d]pyrimidin-4-amine
—— 6-amino-8-{4-[(4-chlorobenzyl)oxy]-3-methoxyphenyl}-8H-[1,3]dioxolo[4,5-g]chromene-7-carbonitrile —— C25H19ClN2O5
6-amino-8-{4-[(4-chlorobenzyl)oxy]-3-methoxyphenyl}-8H-[1,3]dioxolo[4,5-g]chromene-7-carbonitrile
—— 6-[(4-bromophenyl)methylsulfanyl]-3-(3,3,5-trimethylcyclohexyl)-2,4-dihydro-1H-1,3,5-triazine —— C19H28BrN3S
6-[(4-bromophenyl)methylsulfanyl]-3-(3,3,5-trimethylcyclohexyl)-2,4-dihydro-1H-1,3,5-triazine
—— 6-chloro-2-[(1R)-1-(4-chloro-3-methylphenoxy)ethyl]-1H-benzimidazole —— C16H14Cl2N2O
6-chloro-2-[(1R)-1-(4-chloro-3-methylphenoxy)ethyl]-1H-benzimidazole
—— (6E)-2-ethyl-6-[[4-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H19FN4O3S
(6E)-2-ethyl-6-[[4-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2-ethyl-6-[[3-[(2-fluorophenyl)methoxy]phenyl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H17FN4O2S
(6E)-2-ethyl-6-[[3-[(2-fluorophenyl)methoxy]phenyl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-benzyl-5-methyl-4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-2-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C27H29N5O2
6-benzyl-5-methyl-4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-2-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— 6-(4-chlorophenyl)-3-pentyl-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine —— C15H17ClN4S
6-(4-chlorophenyl)-3-pentyl-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine
—— 6-(2-Hydroxy-3-prop-2-enoxypropyl)-2-[(3-methylphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H27N3O3
6-(2-Hydroxy-3-prop-2-enoxypropyl)-2-[(3-methylphenyl)methyl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Amino-3-(3-ethoxyphenyl)-4-(3-nitrophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C21H17N5O4
6-Amino-3-(3-ethoxyphenyl)-4-(3-nitrophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile